|
T10140 |
4-Diethylaminobenzaldehyde
|
|
Dehydrogenase
|
|
4-Diethylaminobenzaldehyde is a reversible aldehyde dehydrogenase (ALDH) inhibitor (Ki: 4 nM for ALDH1). It displays a potent anti-androgenic effect (IC50: 1.71μM). |
|
T0488 |
Finasteride
|
MK-906 |
Reductase
|
|
Finasteride (MK-906) is an oral inhibitor of active testosterone 5-alpha-reductase and Ki value is 10 nM. |
|
T19213 |
Boldenone Cypionate
|
|
Others
,
Androgen Receptor
|
|
Boldenone Cypionate is an androgenic anabolic steroid. |
|
T14843 |
Bifluranol
|
BX341 |
Androgen Receptor
|
|
Bifluranol (BX341) has anti-androgenic activity and has shown significant anti-prostatic activity in in vivo studies for the treatment of benign prostatic hyperplasia (BPH). |
|
T11410L |
GLPG0492
|
|
Androgen Receptor
|
|
GLPG0492 is a novel selective androgen receptor modulator. After oral dosing, it showed anabolic activity on muscle, strongly dissociated from the androgenic activity on the prostate. |
|
T1514 |
Norethindrone
|
Norethisterone |
Estrogen/progestogen Receptor
,
Progesterone Receptor
|
|
Norethindrone (Norethisterone) is a synthetic progestational hormone with actions similar to those of PROGESTERONE but functioning as a more potent inhibitor of ovulation. It has weak estrogenic and androgenic properties... |
|
T10889 |
CRTh2 antagonist 2
|
|
GPR
|
|
CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 can be used to study the direction of androgenic alopecia. |
|
T30161 |
EN3356
|
AS N001,ASN-001 |
P450
|
|
EN3356 is an orally available and selective inhibitor of steroidal 17-alpha-hydroxylase/C17,20 cleavage enzyme (CYP17A1 or CYP17), a non-steroidal cleavage enzyme-selective compound with potential anti-androgenic and ant... |
|
T2556 |
Nandrolone decanoate
|
19-Nortestosterone decanoate |
Others
,
HIV Protease
|
|
Nandrolone decanoate (19-Nortestosterone decanoate) is the decanoate salt form of nandrolone, an anabolic steroid analog of testosterone with androgenic, anabolic, and erythropoietin stimulating effects. Nandrolone enter... |
|
T25961 |
Piperophos
|
Rilof |
|
|
Piperophos is an organophosphate with anti-androgenic activities. |
|
T40809 |
2α-Methyl androsterone
|
|
|
|
2α-Methyl androsterone, a metabolite of mesterolone and drostanolone, is classified as an anabolic androgenic steroid. |
|
T19195 |
Androstenediol 17-acetate
|
|
Others
|
|
Androstenediol 17-acetate is a synthetic anabolic-androgenic steroid and an androgen ester. |
|
T25304 |
Demegestone
|
R-2453,Lutionex,R 2453,RU 2453,R2453 |
|
|
Demegestone is a progestin, or a synthetic progestogen, and hence is a progesterone receptor agonist, the biological target of progestogens like progesterone. It has no androgenic activity. Previously used to treat lutea... |
|
T2195L |
Epiandrosterone Sulfate
|
Epiandrosterone 16-bromo,Epiandrosterone |
|
|
Epiandrosterone sulfate is a steroid hormone with weak androgenic activity. Epiandrosterone is naturally produced by the enzyme 5α-reductase of the adrenal hormone DHEA. |
|
T73671 |
7β-Hydroxy-epi-androsterone
|
|
|
|
7β-Hydroxy-epi-androsterone (7β-Hydroxy-EpiA) is an endogenous androgenic derivative of dehydroepiandrosterone that possesses the ability to bind to ERβ, offering both anti-inflammatory and neuroprotective properties [1]... |
|
T81662 |
N-Nitrosodicyclohexylamine
|
NDCHA |
Androgen Receptor
|
|
N-Nitrosodicyclohexylamine (NDCHA), an N-nitrosocompound, exhibits anti-androgenic activity by competitively binding to the androgen receptor (AR) in opposition to 5α-dihydrotestosterone and reducing AR protein levels [1... |
|
T61029 |
TP0427736 hydrochloride
|
|
|
|
TP0427736 hydrochloride can be used in the androgenic alopecia (AGA) research. TP0427736 hydrochloride inhibits the phosphorylation of Smad2/3 in A549 cells induced by TGF-β1 with an IC50 value of 8.68 nM. TP0427736 hydr... |
|
T41331 |
Cyprodinil
|
|
|
|
Cyprodinil, an anilinopyrimidine broad-spectrum fungicide, inhibits methionine biosynthesis in phytopathogenic fungi, effectively limiting cell growth of B. cinerea, P. herpotrichoides, and H. oryzae on amino acid-free m... |
|
T21668 |
Finasteride acetate
|
|
|
|
Finasteride (MK-906) acetate is a potent and competitive 5α-reductase inhibitor, with an IC 50 of 4.2 nM for type II 5α-reductase. The affinity of Finasteride acetate for type II 5α-reductase enzyme was approximately 100... |
|
T84319 |
5α-Dihydrotestosterone
|
Stanolone,DHT,Dihydrotestosterone,Androstanolone |
|
|
Dihydrotestosterone(DHT) is an endogenous androgenic steroid and hormone that acts as an agonist for androgen receptors. DHT promotes the release of erythropoietin (EPO) from the kidneys. Stimulates the proliferation and... |
|
T71142 |
Tebuconazole-d9
|
|
|
|
Tebuconazole-d9 is intended for use as an internal standard for the quantification of tebuconazole by GC- or LC-MS. Tebuconazole is a triazole fungicide that is active against both seed and foliar fungi. It inhibits 14α-... |
