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Search Results for " Artemisinin "

阻害剤

天然化合物

リコンビナントタンパク質

ライブラリー

カタログ番号	製品名	別名	ターゲット
T70595	Artemisinin B
	Artemisinin B is a drug which may improve spatial memory in dementia patients and alter the levels of inflammatory cytokines in the hippocampus and the cortex. Artemisinin B may inhibit neuroinflammation and exert neurop...
T131541	Artemisinin (Arteannuin, Qinghaosu, Qing Hau Sau)
	Artemisinin (Arteannuin, Qinghaosu, Qing Hau Sau) is a useful organic compound for research related to life sciences and the catalog number is T131541.
T7744	Piperaquine tetraphosphate tetrahydrate		Parasite
	Piperaquine tetraphosphate tetrahydrate is a potent anti-parasites agent.		Parasite
T7532	Piperaquine		Parasite
	Piperaquine is a bis-quinoline compound that inhibits the ex vivo growth of P. falciparum isolates from malaria-infected patients with IC50s ranging from 11.8-217.3 nM.		Parasite
T64399	Dihydroartemisinin (mixture of α and β isomers)
	Dihydroartemisinin (mixture of α and β isomers) is a useful organic compound for research related to life sciences. The catalog number is T64399 and the CAS number is 131175-87-6.
T10378	Artelinic acid		Parasite
	Artelinic acid is a water-soluble artemisinin analog with antimalarial activity and is used for the treatment of multi-drug resistant strains of Plasmodium falciparum.		Parasite
T38723	β-Aminoarteether	β-Aminoarteether,SM934 free base	Others
	β-Aminoarteether (SM934 free base), an orally active derivative of Artemisinin, serves a pivotal role in the research of inflammation and autoimmune disorders, including those related to lupus diseases.		Others
T9741	INE963		Others
	INE963 demonstrates potent cellular activity against Pf 3D7 (EC50 = 6 nM) and achieves "artemisinin-like" kill kinetics in vitro with a parasite clearance time of <24 h. INE963 is also potent against P. falciparum and P....		Others
T8826	3-AMINO-1,2,4-TRIAZINE		Others
	3-AMINO-1,2,4-TRIAZINE is an aromatic bioactive compound. It has been used to synthesize a variety of drugs, including the antifungal drug fluconazole, the anti-inflammatory drug ibuprofen and the anticancer drug paclita...		Others
T10377	Artefenomel	OZ439	Others
	Artefenomel (OZ439) is a synthetic antimalarial agent with the artemisinin pharmacophore.		Others
T61917	TCMDC-125457
	TCMDC-125457 can effectively induce calcium redistribution, but has little effect on inhibiting heme crystallization. When TCMDC-125457 is combined with artesunate, it can effectively treat tightly synchronized artemisin...
T78805	AD4		Others , PROTACs
	AD4, an artemisinin derivative functioning as a proteolytic targeting chimera (PROTAC) for PCLAF, effectively degrades PCLAF in RS4;11 cells with an IC50 of 0.6 nM. This degradation activates the p21/Rb axis, resulting i...		Others , PROTACs

Compounds

Artemisinin (Arteannuin, Qinghaosu, Qing Hau Sau)

T131541

Synonym:

Target:

Piperaquine tetraphosphate tetrahydrate

Dihydroartemisinin (mixture of α and β isomers)

Synonym: β-Aminoarteether,SM934 free base

3-AMINO-1,2,4-TRIAZINE

Target: Others, PROTACs

カタログ番号	製品名	別名	ターゲット
T0392	Artemisinin	Qinghaosu,Artemisinine,Qinghaosu,NSC 369397,Artemisinine	HCV Protease , Ferroptosis , Akt , Parasite
	Artemisinin (Qinghaosu) is an ancient Chinese herbal therapy for malarial fevers which has been recently found to have potent activity against many forms of malarial organisms, including chloroquine-resistant Plasmodium ...		HCV Protease , Ferroptosis , Akt , Parasite
TN2449	Anhydro Dihydro Artemisinin		Others
	Anhydro Dihydro Artemisinin is a natural product from Artemisia carvifolia Buch.-Ham. ex Roxb.		Others
T0607	Dihydroartemisinin	β-Dihydroartemisinin,Dihydroqinghaosu,Artenimol,DHA	Apoptosis , NF-κB , Parasite , Autophagy
	Dihydroartemisinin (Artenimol) is a metabolite of artemisinin.		Apoptosis , NF-κB , Parasite , Autophagy
T7059	α-Dihydroartemisinin	α-Artenimol,α-Dihydroqinghaosu	Parasite
	α-Dihydroartemisinin (α-Dihydroqinghaosu) is an intermediate of artemisinin-based antimalarial compounds with good antimalarial and anticancer activity, and can be used in the study of lupus erythematosus.		Parasite
TN1568	Deoxyartemisinin	2-deoxyartemisinin	Antifection
	Deoxyartemisinin (2-deoxyartemisinin), a compound derived from Artemisia annua, has anti-inflammatory and anti-ulcer effects and is used in the study of malaria.		Antifection
T21065	Artemisitene		Others
	Artemisitene is the oxidized form of Artemisinin and is an antimalarial agent. Artemisinin precursors are the important basic substances for biosynthesis of Artemisinin, including Artemisinin B, Artemisitene, Artemisini...		Others
T0433	Artesunate	WR-256283	Virus Protease , Ferroptosis , STAT , Parasite
	Artesunate (WR-256283) is part of the artemisinin group of drugs that treat malaria. It is a semi-synthetic derivative of artemisinin that is water-soluble and may therefore be given by injection. It is on the World Heal...		Virus Protease , Ferroptosis , STAT , Parasite
TJS1159	Chrysosplenetin	Chrysosptertin B	P450 , Ferroptosis , P-gp
	Chrysosplenetin is a metabolic inhibitor of artemisinin.		P450 , Ferroptosis , P-gp
THS1455	DihydroarteMisinic acid	Dihydro-Artmisinic Acid	Ferroptosis , Parasite
	DihydroarteMisinic acid (Dihydro-Artmisinic Acid) is a natural product from Artemisia annua and the main direct precursor of artemisinin, which is a medicinal herb that is widely used to treat Malaria.		Ferroptosis , Parasite
T4S1452	Artemisic acid	(+)-Artemisinic Acid,Artemisinic acid	Antibacterial
	1. Artemisic acid ((+)-Artemisinic Acid) shows antibacterial activity. 2. Artemisinic acid is a major precursor of artemisinin (an antimalaric compound), isolated as the active principles of the medicinal plant Artemisia...		Antibacterial

天然物製品

Artemisinin

T0392

Synonym: Qinghaosu,Artemisinine,Qinghaosu,NSC 369397,Artemisinine

Target: HCV Protease, Ferroptosis, Akt, Parasite

Anhydro Dihydro Artemisinin

Synonym: β-Dihydroartemisinin,Dihydroqinghaosu,Artenimol,DHA

Target: Apoptosis, NF-κB, Parasite, Autophagy

α-Dihydroartemisinin

T7059

Synonym: α-Artenimol,α-Dihydroqinghaosu

Target: Parasite

Deoxyartemisinin

TN1568

Synonym: 2-deoxyartemisinin

Target: Virus Protease, Ferroptosis, STAT, Parasite

Chrysosplenetin

TJS1159

Synonym: Chrysosptertin B

Target: P450, Ferroptosis, P-gp

DihydroarteMisinic acid

THS1455

Synonym: Dihydro-Artmisinic Acid

Target: Ferroptosis, Parasite

Artemisic acid

T4S1452

Synonym: (+)-Artemisinic Acid,Artemisinic acid

Target: Antibacterial

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-03509	TCTP/TPT1 Protein, Human, Recombinant (His)	Human	E. coli
	Tumor protein, also known as TPT1, is a highly conserved protein among many eukaryotic organisms. Tumor protein is involved in a variety of cellular activities, including microtubule stabilization, calcium-binding activi...

TCTP/TPT1 Protein, Human, Recombinant (His)

TMPY-03509

Species: Human

Expression System: E. coli

カタログ番号	製品名
L6500	Microbial Natural Product Library	550 compounds
	A unique collection of 550 microbial natural products for high throughput screening (HTS) and high content screening (HCS);
L4600	Selected Plant-Sourced Compound Library	3048 compounds
	A unique collection of 3048 plant-sourced compounds that derived from 277 plant species for high throughput screening (HTS) and high content screening (HCS);
L6810	Traditional Chinese Medicine Monomer Library	2755 compounds
	A unique collection of 2755 compounds (TCM monomers) sourcing from traditional Chinese Medicines, is a powerful tool for drug discovery and research in mechanism；
L6020	Selectable Natural Product Library	16627 compounds
	A unique collection of 16627 pure natural products with diverse structures and sources covering various plant, animal, and microbe species;
L6800	Chinese Pharmacopoeia Natural Product Library	2051 compounds
	A unique collection of 2051 natural products included in Chinese Pharmacopoeia (CP), a powerful tool for drug development and pharmacological study;

ライブラリー

Microbial Natural Product Library

L6500

Compounds: 550

Selected Plant-Sourced Compound Library

L4600

Compounds: 3048

Traditional Chinese Medicine Monomer Library

L6810

Compounds: 2755

Selectable Natural Product Library

L6020

Compounds: 16627

Chinese Pharmacopoeia Natural Product Library

L6800

Compounds: 2051