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ターゲット

阻害剤

天然化合物

リコンビナントタンパク質

カタログ番号	製品名	別名	ターゲット
T10616	BRM/BRG1 ATP Inhibitor-1		Epigenetic Reader Domain
	BRM/BRG1 ATP Inhibitor-1 is an allosteric dual Brahma homolog (BRM)/SWI/SNF related matrix-associated actin-dependent regulator of chromatin subfamily A member 2 (SMARCA2) and BRG1/SMARCA4 ATPase activity inhibitor (IC50...		Epigenetic Reader Domain
T3545	RG13022	RG 13022,Tyrphostin RG13022	EGFR
	RG13022 (Tyrphostin RG13022) is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of the EGF receptor (IC50: 4 μM).		EGFR
T3554	RG14620	Tyrphostin RG14620,RG 14620	EGFR , HER
	RG14620 (Tyrphostin RG14620) is an epidermal growth factor receptor (EGFR) inhibitor.		EGFR , HER
T2038	RG108	N-Phthalyl-L-tryptophan	DNA Methyltransferase
	RG108 (N-Phthalyl-L-tryptophan) is an DNA methyltransferase inhibitor(IC50=115 nM).		DNA Methyltransferase
T78525	IRG1-IN-1		Others
	IRG1-IN-1 is an itaconic acid derivative with the ability to inhibit the activity of Immune Response Gene 1 (IRG1) and is suitable for use in the field of cancer, inflammation and autoimmune disease research.		Others
TP1931L1	[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate	[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base)	cholecystokinin
	[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist ...		cholecystokinin
T60032	BRM/BRG1 ATP Inhibitor-2		Epigenetic Reader Domain
	BRM/BRG1 ATP Inhibitor-2 is an inhibitor of BRG1/BRM ATPase and can be used in studies about the treatment of BAF-related disorders.		Epigenetic Reader Domain
T76446	(D-Arg1,D-Pro2,D-Phe7,D-His9)-Substance P
	(D-Arg1,D-Pro2,D-Phe7,D-His9)-Substance P is a selective NK 1 receptor antagonist [1] .
T83195	Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)
	Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP(1-7)-GRF(8-27) is a selective antagonist [1] for the vasoactive intestinal peptide 1 (VIP 1) receptor.
T75896	[Arg14,Lys15]Nociceptin TFA
	[Arg14,Lys15]Nociceptin TFA is a potent and selective agonist for the NOP receptor (ORL1; OP4), exhibiting an EC50 of 1 nM. It demonstrates significant selectivity against opioid receptors, with IC50 values of 0.32 nM fo...
T83500	[Des-Arg10]-HOE I40
	[Des-Arg10]-HOE 140 is a bioactive peptide that functions as a potent B1 bradykinin receptor antagonist.
T72257	BRM/BRG1 ATP Inhibitor-3
	BRM/BRG1 ATP Inhibitor-3 is a potent inhibitor targeting both BRM and BRG1 components of the BAF complex, exhibiting IC50 values of 10.4 nM for BRM and 19.3 nM for BRG1, respectively. It holds potential for research appl...
T60870	BRG1-IN-1
	BRG1-IN-1 (Compound 11d) is a potent BRG1 inhibitor with better efficacy than PFI-3 in sensitizing GBM cells to the antiproliferative and cell death inducing effects of Temozolomide in vitro. BRG1-IN-1 enhances the inhib...
TP1931	[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
	Broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradyki...
TP1986	[Arg14,Lys15]Nociceptin
	Highly potent and selective NOP receptor agonist (EC50 = 1 nM). Displays > 875-fold selectivity over opioid receptors (IC50 values are 0.32, 280, > 10000 and 1500 for NOP, μ, δ and κ receptors respectively). Longer lasti...
T78656	ARG1-IN-1 hydrochloride		Arginase
	ARG1-IN-1 hydrochloride is a potent inhibitor of human arginase 1, exhibiting an IC50 value of 29 nM [1].		Arginase
T83548	(D-Arg1,D-Pro2,D-Trp7,9,L-Leu11)-Substance P acetate
	(D-Arg1,D-Pro2,D-Trp7,9,L-Leu11)-Substance P (acetate), an antagonist for Substance P and Bombesin, modulates ocular inflammatory responses triggered by antidromic trigeminal nerve stimulation [1].
T83690	[Leu144, Arg147]-PLP (139-151) TFA	[Leu144, Arg147] Proteolipid Peptide (139-151),H-His-Ser-Leu-Gly-Lys-Leu-Leu-Gly-Arg-Pro-Asp-Lys-Phe-OH
	[Leu144,Arg147]-PLP (139-151) is a mutated fragment of the myelin proteolipid protein (PLP), featuring substitutions of tryptophan to leucine and histidine to arginine at positions 144 and 147, respectively. Immunizing m...
T72258	BRM/BRG1 ATP Inhibitor-4
	BRM/BRG1 ATP Inhibitor-4, a potent inhibitor of BRG1/BRM, is utilized in the research of cancers and BAF complex-related disorders.
T76445	(D-Arg1,D-Pro2,D-Trp7,9,L-Leu11)-Substance P
	(D-Arg1,D-Pro2,D-Trp7,9,L-Leu11)-Substance P is a neuropeptide Substance P antagonist [1] .
T39932	ARG1-IN-1	ARG1-IN-1
	ARG1-IN-1 is a human arginase 1 inhibitor with an IC 50 of 29 nM.

Compounds

BRM/BRG1 ATP Inhibitor-1

T10616

Synonym:

Target: Epigenetic Reader Domain

RG13022

T3545

Synonym: RG 13022,Tyrphostin RG13022

Target: EGFR

RG14620

T3554

Synonym: Tyrphostin RG14620,RG 14620

Target: EGFR, HER

RG108

T2038

Synonym: N-Phthalyl-L-tryptophan

Target: DNA Methyltransferase

[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate

TP1931L1

Synonym: [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base)

Target: cholecystokinin

BRM/BRG1 ATP Inhibitor-2

T60032

Synonym:

Target: Epigenetic Reader Domain

(D-Arg1,D-Pro2,D-Phe7,D-His9)-Substance P

T76446

Synonym:

Target:

Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)

T83195

Synonym:

Target:

[Arg14,Lys15]Nociceptin TFA

BRM/BRG1 ATP Inhibitor-3

[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P

TP1931

Synonym:

Target:

[Arg14,Lys15]Nociceptin

TP1986

Synonym:

Target:

ARG1-IN-1 hydrochloride

T78656

Synonym:

Target: Arginase

(D-Arg1,D-Pro2,D-Trp7,9,L-Leu11)-Substance P acetate

T83548

Synonym:

Target:

[Leu144, Arg147]-PLP (139-151) TFA

T83690

Synonym: [Leu144, Arg147] Proteolipid Peptide (139-151),H-His-Ser-Leu-Gly-Lys-Leu-Leu-Gly-Arg-Pro-Asp-Lys-Phe-OH

Target:

BRM/BRG1 ATP Inhibitor-4

T72258

Synonym:

Target:

(D-Arg1,D-Pro2,D-Trp7,9,L-Leu11)-Substance P

カタログ番号	製品名	別名	ターゲット
T2777	Ginsenoside Rg1	Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,Panaxoside A,Ginsenoside A2	Apoptosis , Beta Amyloid , NF-κB
	Ginsenoside Rg1 (Panaxoside Rg1) is a class of steroid glycosides, and triterpene saponins found exclusively in the plant genus Panax (ginseng). It improves spatial learning and increase hippocampal synaptophysin level i...		Apoptosis , Beta Amyloid , NF-κB
T3401	Ginsenoside F1	20(S)-Ginsenoside F1	P450 , Endogenous Metabolite
	Ginsenoside F1 (20(S)-Ginsenoside F1) is an enzymatically modified derivative of ginsenoside Rg1, showing competitive inhibition of the activity of CYP3A4 and a weaker inhibition of the activity of CYP2D6.		P450 , Endogenous Metabolite
T3917	Protopanaxatriol	20(R)-APPT,20(R)-Protopanaxatriol,(20R)-Protopanaxatriol	PPAR
	Protopanaxatriol (20(R)-APPT), a major ginseng constituent, is a novel PPARγ antagonist.		PPAR

天然物製品

Ginsenoside Rg1

T2777

Synonym: Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,Panaxoside A,Ginsenoside A2

Target: Apoptosis, Beta Amyloid, NF-κB

Ginsenoside F1

T3401

Synonym: 20(S)-Ginsenoside F1

Target: P450, Endogenous Metabolite

Protopanaxatriol

T3917

Synonym: 20(R)-APPT,20(R)-Protopanaxatriol,(20R)-Protopanaxatriol

Target: PPAR

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPK-01246	GDF-15 Protein, Mouse, Recombinant (His)	Mouse	E. coli
	Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t...
TMPK-01243	GDF-15 Protein, Rat, Recombinant (His)	Rat	E. coli
	Growth Differentiation Factor 15 (GDF15), also known as NSAID activated gene-1 (NAG-1), is associated with a large number of biological processes and diseases, including cancer and obesity. GDF15 is synthesized as pro-GD...
TMPK-01245	GDF-15 Protein (Primary Amine Labeling), Mouse, Recombinant (hFc), Biotinylated	Mouse	HEK293 Cells
	Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t...
TMPK-00663	GDF-15 Protein, Cynomolgus, Recombinant (hFc)	Cynomolgus	HEK293 Cells
	Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t...
TMPK-00664	GDF-15 Protein (Primary Amine Labeling), Cynomolgus, Recombinant (hFc), Biotinylated	Cynomolgus	HEK293 Cells
	Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t...
TMPK-00198	GDF-15 Protein (Primary Amine Labeling), Human, Recombinant (hFc), Biotinylated	Human	HEK293 Cells
	Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t...
TMPK-00569	GDF-15 Protein, Canine, Recombinant (His)	Canine	E. coli
	Growth Differentiation Factor 15 (GDF15), also known as NSAID activated gene-1 (NAG-1), is associated with a large number of biological processes and diseases, including cancer and obesity. GDF15 is synthesized as pro-GD...
TMPK-00665	GDF-15 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	E. coli
	Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t...
TMPK-00197	GDF-15 Protein (Primary Amine Labeling), Human, Recombinant (H202D, hFc), Biotinylated	Human	HEK293 Cells
	Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t...
TMPK-00196	GDF-15 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	E. coli
	Growth Differentiation Factor 15 (GDF15), also known as NSAID activated gene-1 (NAG-1), is associated with a large number of biological processes and diseases, including cancer and obesity. GDF15 is synthesized as pro-GD...
TMPK-01244	GDF-15 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	Growth and differentiation factor 15 (GDF15) is an inflammation-associated hormone with poorly defined biology. Here, we investigated the role of GDF15 in bacterial and viral infections. Inflammation induced GDF15, and t...
TMPY-04018	LRG1 Protein, Human, Recombinant	Human	HEK293 Cells
	LRG1 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 35.1 kDa and the accession number is AAH34389.1.
TMPY-02168	Arginase 1/ARG1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Arginase 1/ARG1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 36.2 kDa and the accession number is P05089-1.
TMPY-00479	Neuregulin-1/NRG1 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Neuregulin-1/NRG1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 35.5 kDa and the accession number is Q02297-12.
TMPH-02064	SCRG1 Protein, Human, Recombinant (His & SUMO)	Human	E. coli
	SCRG1 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli.
TMPY-03965	LRG1 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	LRG1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 61.3 kDa and the accession number is AAH34389.1.
TMPY-04237	Neuregulin-1/NRG1 Protein, Canine, Recombinant (aa 176-240, His)	Canine	HEK293 Cells
	Neuregulin-1/NRG1 Protein, Canine, Recombinant (aa 176-240, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 9.7 kDa.
TMPK-01128	LRG1 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Diabetic nephropathy (DN) is an important public health concern of increasing proportions and the leading cause of end-stage renal disease (ESRD) in diabetic patients. It is one of the most common long-term microvascular...
TMPK-00750	KLRG1 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	KLRG1 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with N-hFc tag. The predicted molecular weight is 42.3 kDa and the accession number is O88713.
TMPY-03902	Neuregulin-1/NRG1 Protein, Canine, Recombinant (mFc)	Canine	HEK293 Cells
	Neuregulin-1/NRG1 Protein, Canine, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 34 kDa and the accession number is XP_858147.1.
TMPY-02705	NRG1 beta 1 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	NRG1 beta 1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 55.2 kDa and the accession number is Q02297-6.
TMPY-03943	Neuregulin-1/NRG1 Protein, Canine, Recombinant (hFc)	Canine	HEK293 Cells
	Neuregulin-1/NRG1 Protein, Canine, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 50.8 kDa and the accession number is XP_858147.1.
TMPY-02721	NRG1 alpha Protein, Human, Recombinant (His)	Human	HEK293 Cells
	NRG1 alpha Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.5kDa and the accession number is Q02297-1.
TMPH-02524	Arginase-1/ARG1 Protein, Mouse, Recombinant (His)	Mouse	P. pastoris (Yeast)
	Key element of the urea cycle converting L-arginine to urea and L-ornithine, which is further metabolized into metabolites proline and polyamides that drive collagen synthesis and bioenergetic pathways critical for cell ...
TMPH-02525	Arginase-1/ARG1 Protein, Mouse, Recombinant (His & SUMO)	Mouse	E. coli
	Arginase-1/ARG1 Protein, Mouse, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 50.8 kDa and the accession number is Q61176.
TMPY-04685	Arginase 1/ARG1 Protein, Human, Recombinant (His & MYC)	Human	HEK293 Cells
	Arginase 1/ARG1 Protein, Human, Recombinant (His & MYC) is expressed in HEK293 mammalian cells with His and MYC tag. The predicted molecular weight is 36.7 kDa and the accession number is P05089-1.
TMPH-02887	SCRG1 Protein, Mouse, Recombinant (His)	Mouse	E. coli
	N/A. SCRG1 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 15.0 kDa and the accession number is O88745?.
TMPY-04690	Influenza A H3N2 (A/Netherlands/178/1995 (RG145K)) Hemagglutinin/HA Protein (His)	H3N2	Baculovirus Insect Cells
	Influenza A H3N2 (A/Netherlands/178/1995 (RG145K)) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.3 kDa and the accession number is I6V5M4.
TMPH-03447	ERG11 Protein, S. cerevisiae, Recombinant (GST)	Saccharomyces cerevisiae	E. coli
	Catalyzes C14-demethylation of lanosterol which is critical for ergosterol biosynthesis. It transforms lanosterol into 4,4'-dimethyl cholesta-8,14,24-triene-3-beta-ol. ERG11 Protein, S. cerevisiae, Recombinant (GST) is e...
TMPY-03010	NRG1 beta 1 Protein, Human, Recombinant	Human	HEK293 Cells
	NRG1 beta 1 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.8 kDa and the accession number is Q02297-6.
TMPY-03601	PDRG1 Protein, Human, Recombinant (His)	Human	E. coli
	PDRG1, also known as C2orf126, belongs to the prefoldin subunit beta family. It is predominantly expressed in normal testis and exhibits reduced but detectable expression in other organs. PDRG1 may play a role in chapero...
TMPY-02719	NRG1 alpha Protein, Human, Recombinant (EGF Domain, hFc)	Human	HEK293 Cells
	NRG1 alpha Protein, Human, Recombinant (EGF Domain, hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 35.8 kDa and the accession number is Q02297-1.
TMPJ-00448	NRG1 beta 1 Protein, Human, Recombinant (aa 2-246)	Human	E. coli
	Pro-neuregulin-1,Neuregulin-1 beta 1（NRG1） is a single-pass type I membrane protein and belongs to the neuregulin family .It contains 1 EGF-like domain and 1 Ig-like C2-type (immunoglobulin-like) domain. Direct ligand f...
TMPK-01140	KLRG1 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	KLRG1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with N-hFc tag. The predicted molecular weight is 42.8 kDa and the accession number is Q96E93-1.
TMPY-04088	Neuregulin-1/NRG1 Protein, Canine, Recombinant	Canine	HEK293 Cells
	Neuregulin-1/NRG1 Protein, Canine, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 24.7 kDa and the accession number is XP_858147.1.
TMPY-04603	Influenza A H3N2 (A/Netherlands/178/1995 (RG145K)) Hemagglutinin/HA1 Protein (His)	H3N2	HEK293 Cells
	Influenza A H3N2 (A/Netherlands/178/1995 (RG145K)) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is I6V5M4.
TMPY-00031	Neuregulin-1/NRG1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Neuregulin-1/NRG1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.3 kDa and the accession number is Q02297-12.
TMPY-02720	NRG1 alpha Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	NRG1 alpha Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 51 kDa and the accession number is Q02297-1.
TMPY-03443	NDRG1 Protein, Human, Recombinant (His)	Human	E. coli
	NDRG1 gene is a member of the N-Myc downregulated gene family which belongs to the alpha/beta hydrolase superfamily. NDRG1 is a cytoplasmic protein involved in stress responses, hormone responses, cell growth, and differ...
TMPY-03903	Neuregulin-1/NRG1 Protein, Canine, Recombinant (aa 19-240, His)	Canine	HEK293 Cells
	Neuregulin-1/NRG1 Protein, Canine, Recombinant (aa 19-240, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.5 kDa and the accession number is XP_858147.1.
TMPY-03966	LRG1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	LRG1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 35.8 kDa and the accession number is AAH34389.1.
TMPY-05813	Neuregulin-1/NRG1 Protein, Human, Recombinant , Biotinylated	Human	HEK293 Cells
	Neuregulin-1/NRG1 Protein, Human, Recombinant , Biotinylated is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.8 kDa and the accession number is Q02297.
TMPY-02600	NRG1 beta 1 Protein, Human, Recombinant (EGF Domain, hFc)	Human	HEK293 Cells
	NRG1 beta 1 Protein, Human, Recombinant (EGF Domain, hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 36.7 kDa and the accession number is Q02297-6.
TMPJ-00231	LRG1 Protein, Human, Recombinant (hFc & His)	Human	HEK293 Cells
	LRG1 is a secreted protein and contains eight LRR repeats and one LRRCT domain, It can be expressed during granulocyte differentiation. LRG1 has been shown to be involved in protein-protein interaction, signal transducti...
TMPK-00526	LRG1 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Diabetic nephropathy (DN) is an important public health concern of increasing proportions and the leading cause of end-stage renal disease (ESRD) in diabetic patients. It is one of the most common long-term microvascular...