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カタログ番号 | 製品名 | 別名 | ターゲット |
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T50032 | 5-(2-furyl)-N-propylisoxazole-3-carboxamide | Others | |
5-(2-furyl)-N-propylisoxazole-3-carboxamide is a compound used as a molecular structural unit and is thought to be a modulator of NMDA receptors, and has been shown to be protective against glutamate-induced excitotoxici... | |||
T8502 | N-(1-benzyl-4-piperidyl)adamantane-1-carboxamide | Influenza Virus | |
N-(1-benzyl-4-piperidyl)adamantane-1-carboxamide inhibiting the entry of Ebola virus in host cells by binding to the surface glycoprotein, the compound inhibited the Ebola virus with EC50 of 3.9 μM. | |||
T1120 | Dacarbazine | Imidazole Carboxamide,DTIC-Dome | Apoptosis , Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis |
Dacarbazine (DTIC-Dome) is an antineoplastic agent. It has significant activity against melanomas. | |||
T25175 | BRD 9757 | BRD9757,N-Hydroxy-1-cyclopentene-1-carboxamide,BRD-9757 | HDAC |
BRD 9757 (N-Hydroxy-1-cyclopentene-1-carboxamide) is a selective inhibitor of HDAC6 (IC50 = 30 nM). | |||
T22009 | CB2 receptor agonist 2 | ZINC72105556,4-Quinolone-3-Carboxamide Furan CB2 Agonist | Cannabinoid Receptor |
CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2. | |||
T8501 | 3-Phenyl-N-[1-(phenylmethyl)-4-piperidinyl]-tricyclo[3.3.1.13,7]decane-1-carboxamide | Influenza Virus | |
3- Phenyl- N- [1- (phenylmethyl) - 4- piperidinyl] -tricyclo[3.3.1.13, 7] decane- 1- carboxamide with antiviral activity against Ebola virus that targets the surface-exposed glycoprotein and inhibits viral entry into hos... | |||
T22988 | MK-4827 Racemate | Niraparib Racemate,2-(4-piperidin-3-ylphenyl)indazole-7-carboxamide | PARP |
MK-4827 Racemate (Niraparib Racemate) is a selective PARP1 and PARP2 inhibitor with IC50s of 3.8 nM and 2.1 nM, respectively, over 330-fold selectivity for PARP3, V-PARP and Tank1. | |||
T19214 | Bredinin aglycone | 5-Hydroxy-1H-imidazole-4-carboxamide,SM-108 | Others |
Bredinin aglycone (SM-108) is a purine nucleotide analog. It can be used to examine the efficiency of catalysts for the preparation of purine nucleotide analogs. | |||
T9679 | N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)pyrazine-2-carboxamide | Antibacterial | |
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)pyrazine-2-carboxamide exhibit an inhibitory effect on bacterial DNA helicases, nucleases, or helicase-nuclease enzyme complexes, such as, for example, one or more enzym... | |||
T6833 | Favipiravir | T-705,6-Fluoro-3-oxo-3,4-dihydropyrazine-2-carboxamide | Others , SARS-CoV , Influenza Virus , DNA/RNA Synthesis |
Favipiravir (T-705) (T-705), an effective and selective RNA-dependent RNA polymerase inhibitor, are applied to treat influenza virus infections. | |||
T60041 | N-[2-(5-Chloro-1H-indol-3-yl)ethyl]-4'-cyanobiphenyl-2-carboxaMide | Microtubule Associated | |
N-[2-(5-Chloro-1H-indol-3-yl)ethyl]-4'-cyanobiphenyl-2-carboxaMide, a TAU cytotoxicity inhibitor, inhibits LDH leakage of M17-TAU P301L cells with EC50 of 325nM. | |||
T60087 | CFMS Receptor Inhibitor IV | 5-cyano-N-(2,5-di(piperidin-1-yl)phenyl)furan-2-carboxamide | c-Fms |
cFMS Receptor Inhibitor IV is an inhibitor of c-Fms tyrosine kinase. | |||
T16109 | ML402 | ZINC3671497,N-[2-(4-chloro-2-methylphenoxy)ethyl]thiophene-2-carboxamide | Potassium Channel |
ML402 (ZINC3671497) is an activator of TREK-1 and TREK-2 with EC50s of 13.7 μM and 5.9 μM. | |||
T16950 | Sudoxicam | 4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide | COX |
Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema, and antipyretic properties. | |||
T5962 | TRPM8 antagonist WS-3 | Cyclohexanecarboxamide,N-Ethyl-p-menthane-3-carboxamide,N-Ethyl-2-isopropyl-5-methylcyclohexanecarboxamide | TRP/TRPV Channel |
TRPM8 antagonist WS-3 (Cyclohexanecarboxamide) is an agonist of TRPM8( EC50 : 3.7 μM). | |||
T9578 | ELOVL1-IN-1 | 1-(2-Fluorophenyl)-N-(1-(2-fluoropyridin-4-YL)-1H-pyrazol-3-YL)cyclopropane-1-carboxamide | Others |
ELOVL1-IN-1 (1-(2-Fluorophenyl)-N-(1-(2-fluoropyridin-4-YL)-1H-pyrazol-3-YL)cyclopropane-1-carboxamide) is an ELOVL1 inhibitor. ELOVL1-IN-1 can reduce the levels of very long chain fatty acids. ELOVL1-IN-1 can be used in... | |||
T9137 | SN-011 | [1,1'-Biphenyl]-4-carboxamide, N-[3-[[(4-fluorophenyl)sulfonyl]amino]-4-hydroxyphenyl]-,GUN35901 | STING |
SN-011 (GUN35901) is a STING inhibitor, which inhibited the activation of the STING signal pathway and to prevent or treat a STING- mediated disease. It is a demethyl analogue of DUN99845. | |||
T8579 | Nav1.8-IN-1 | 5-(4-Chlorophenyl)-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]pyridine-3-carboxamide,CHEMBL1270208 | Sodium Channel |
Nav1.8-IN-1 (CHEMBL1270208) is an inhibitor of human NaV1.8 | |||
T16922 | SPOP-IN-6b | 2-Imino-10-methyl-N-(3-morpholinopropyl)-5-oxo-1-phenethyl-1,5-dihydro-2H-dipyrido[1,2-a:2',3'-d]pyrimidine-3-carboxamide | Others |
SPOP-IN-6b is an effective inhibitor of speckle-type POZ protein (SPOP) with an IC50 of 3.58 μM and can be used in stuides about the treatment of renal cancer. | |||
T20942 | De(5-carboxamide)oxcarbazepine | Oxcarbazepine related compound E,Oxcarbazepine impurity C | |
De(5-carboxamide)oxcarbazepine is used for organic synthesis. | |||
T67699L | ALK/ROS1 inhibitor 2e HCL | (R)-1-(2-((2-methoxy-4-(piperazin-1-yl)phenyl)amino)pyridin-4-yl)-N-(4-(trifluoromethoxy)benzyl)piperidine-3-carboxamide hydrochloride(2365497-12-5 Free base) | Apoptosis |
ALK/ROS1 inhibitor 2e HCL possesses anti-apoptotic, anti-proliferative and anti-tumour activities. | |||
T21658 | ARN14974 | Others | |
ARN14974 is a benzoxazolone carboxamide. ARN14974 is a potent inhibitor of acid ceramidase with IC50 of 79 nM[1]. | |||
T67888 | Iso-Samidorphan | (9ξ,13ξ,14ξ)-17-(Cyclopropylmethyl)-4,14-dihydroxy-6-oxomorphinan-3-carboxamide | Others |
Iso-Samidorphan is a biochemical reagent that can be used in biological experiments. | |||
TNU0298 | Adenosine-2-carboxamide | ||
Adenosine-2-carboxamide is a Nucleoside Derivative - 2-Modified purine nucleoside. | |||
T29625 | Acridine-9-carboxamide, 1,2,3,4-tetrahydro-N,N-diethyl- | O=C(C1=C(CCCC2)C2=NC3=CC=CC=C31)N(CC)CC | |
Acridine-9-carboxamide, 1,2,3,5-tetrahydro-N,N-diethyl- is a biochemcial. | |||
T31664 | Lysergamide, N-cyclopropyl-, maleate | Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate | |
Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate is a bioactive chemical. | |||
T31663 | Lysergamide, N-cycloheptyl-, maleate | Ergoline-8-beta-carboxamide, N-cycloheptyl-9,10-didehydro-6-methyl-, maleate | |
Lysergamide, N-cycloheptyl-, maleate can be used in related research in the field of life sciences. Its product number is T31663 and CAS number is 103070-86-6. | |||
T66387 | 3,6-Difluoropyrazine-2-carboxamide | ||
3,6-Difluoropyrazine-2-carboxamide is a useful organic compound for research related to life sciences and the catalog number is T66387. | |||
T4348 | Syk Inhibitor II | 5-HT Receptor , Syk | |
Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM). | |||
T60000 | STING (WT/R232) activity regulator 126 | STING | |
STING (WT/R232) activity regulator 126 is a STING modulator with antibacterial and antiviral effects. | |||
T67652 | (S)-Pyrrolidine-2-carboxamide hydrochloride | ||
(S)-Pyrrolidine-2-carboxamide hydrochloride is a useful organic compound for research related to life sciences. The catalog number is T67652 and the CAS number is 42429-27-6. | |||
T50083 | Cell-cell interaction 1 | Others | |
12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide available as a molecular structural unit, it is used in the synthesis of various compounds. | |||
T60186 | (S)-4-methyl-N-(3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-2-(pyrimidin-5-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide | Discoidin Domain Receptor (DDR) | |
MitoBloCK-6 is an effective inhibitor of Erv1/ALR with IC50 values of 900 nM and 700 nM, respectively. Additionally, MitoBloCK-6 inhibits Erv2 (IC50=1.4 μM). It induces apoptosis in hESCs by promoting the release of cyto... | |||
T66159 | 6-Bromo-3-hydroxypyrazine-2-carboxamide | ||
6-Bromo-3-hydroxypyrazine-2-carboxamide is a useful organic compound for research related to life sciences. The catalog number is T66159 and the CAS number is 259793-88-9. | |||
T67506 | 3-Amino-1H-pyrazole-4-carboxamide | ||
3-Amino-1H-pyrazole-4-carboxamide is a useful organic compound for research related to life sciences. The catalog number is T67506 and the CAS number is 5334-31-6. | |||
T66158 | 6-Chloro-3-hydroxypyrazine-2-carboxamide | ||
6-Chloro-3-hydroxypyrazine-2-carboxamide is a useful organic compound for research related to life sciences. The catalog number is T66158 and the CAS number is 259793-90-3. | |||
T64465 | 5-Chloro-N-methylthiophene-2-carboxamide | ||
5-Chloro-N-methylthiophene-2-carboxamide is a useful organic compound for research related to life sciences. The catalog number is T64465 and the CAS number is 97799-98-9. | |||
T67488 | 5-Amino-1H-imidazole-4-carboxamide hydrochloride | ||
5-Amino-1H-imidazole-4-carboxamide hydrochloride is a useful organic compound for research related to life sciences. The catalog number is T67488 and the CAS number is 72-40-2. | |||
T60194 | N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(N-ethylcyclopropanecarboxamido)-4-methyl-4′-morpholino-[1,1′-biphenyl]-3-carboxamide | Histone Methyltransferase | |
N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(N-ethylcyclopropanecarboxamido)-4-methyl-4′-morpholino-[1,1′-biphenyl]-3-carboxamide is a potent and selective Enhancer of Zeste Homolog 2 (EZH2) inhibitor with I... | |||
T60075 | Dopamine D2 receptor agonist-2 | Dopamine D2 Receptor | Dopamine Receptor |
Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor. | |||
T67228 | (2S,5R)-5-((Benzyloxy)amino)piperidine-2-carboxamide | ||
(2S,5R)-5-((Benzyloxy)amino)piperidine-2-carboxamide is a useful organic compound for research related to life sciences. The catalog number is T67228 and the CAS number is 1416134-49-0. | |||
T6561 | Laquinimod | LAQ,ABR-215062 | Apoptosis , Others , NF-κB |
Laquinimod (LAQ) is an effective immunomodulator, which is currently under development in phase III trials for the treatment of multiple sclerosis as an oral therapy. | |||
T60162 | 1H-Pyrazole-5-carboxamide, 4-(5-chloro-2-furanyl)-1,3-bis(2,4-difluorophenyl)-4,5-dihydro-5-methyl-N-[(4-methyl-2-morpholinyl)methyl] | Others | |
1H-Pyrazole-5-carboxamide, 4-(5-chloro-2-furanyl)-1,3-bis(2,4-difluorophenyl)-4,5-dihydro-5-methyl-N-[(4-methyl-2-morpholinyl)methyl] is an antifibrotic agent. | |||
T64535 | (R)-N-(2,6-Dimethylphenyl)-1-propylpiperidine-2-carboxamide hydrochloride | ||
(R)-N-(2,6-Dimethylphenyl)-1-propylpiperidine-2-carboxamide hydrochloride is a useful organic compound for research related to life sciences and the catalog number is T64535. | |||
T66988 | 10-Bromo-5H-dibenzo[b,f]azepine-5-carboxamide | ||
10-Bromo-5H-dibenzo[b,f]azepine-5-carboxamide is a useful organic compound for research related to life sciences. The catalog number is T66988 and the CAS number is 59690-97-0. | |||
T77670 | (1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid | Somatostatin | |
(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist. | |||
T64886 | 5-(2-Thioxo-2,3-dihydrothiazol-4-yl)thiophene-2-carboxamide | ||
5-(2-Thioxo-2,3-dihydrothiazol-4-yl)thiophene-2-carboxamide is a useful organic compound for research related to life sciences and the catalog number is T64886. | |||
T65317 | 2-Methyl-6-oxo-1,6-dihydro-[3,4'-bipyridine]-5-carboxamide | ||
2-Methyl-6-oxo-1,6-dihydro-[3,4'-bipyridine]-5-carboxamide is a useful organic compound for research related to life sciences. The catalog number is T65317 and the CAS number is 80047-24-1. | |||
T66252 | N-(4-Cyano-3-(trifluoromethyl)phenyl)-2-methyloxirane-2-carboxamide | ||
N-(4-Cyano-3-(trifluoromethyl)phenyl)-2-methyloxirane-2-carboxamide is a useful organic compound for research related to life sciences. The catalog number is T66252 and the CAS number is 90357-51-0. | |||
T65742 | 1-Methyl-4-nitro-3-propyl-(1H)-pyrazole-5-carboxamide | ||
1-Methyl-4-nitro-3-propyl-(1H)-pyrazole-5-carboxamide is a useful organic compound for research related to life sciences. The catalog number is T65742 and the CAS number is 139756-01-7. |
カタログ番号 | 製品名 | 別名 | ターゲット |
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T1705 | 5-Amino-3H-imidazole-4-Carboxamide | 4-Amino-5-imidazolecarboxamide,AICA,5-Aminoimidazole-4-carboxamide | Endogenous Metabolite |
5-Amino-3H-imidazole-4-Carboxamide (AICA) is an imidazole derivative which is a metabolite of the antineoplastic agents BIC and DIC. By itself, or as the ribonucleotide, it is used as a condensation agent in the preparat... | |||
T37009 | Oxychlororaphine | phenazine-1-carboxamide | Antibacterial |
Oxychlororaphine (phenazine-1-carboxamide) inhibits strongly the growth of Streptomyces sp. 441. | |||
T5233 | N-Methylnicotinamide | N'-Methylnicotinamide,Nicotinic Acid Methylamide,N-Methylpyridine-3-carboxamide | Others , Endogenous Metabolite |
N-Methylnicotinamide (Nicotinic Acid Methylamide) is a metabolite of niacin (or nicotinamide) and is commonly found in human urine. However low levels of urinary excretion of N-Methylnicotinamide (Nicotinic Acid Methylam... | |||
TN7142 | N-methyl-1H-indole-2-carboxamide | 1H-indole-2-carboxylic acid methylamide,ZINC35137534 | Others |
N-methyl-1H-indole-2-carboxamide (ZINC35137534) is a marine derived natural products found in Neosartorya pseudofischeri. | |||
T8150 | Nudifloramide | 1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide | PARP , Endogenous Metabolite |
Nudifloramide (1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide) is one of the end degradation products of nicotinamide-adenine dinucleotide (NAD). | |||
T13108 | Pamufetinib | H2OL3Q4XRD,4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide,TAS-115 | VEGFR , c-Met/HGFR |
Pamufetinib (TAS-115) is a potent inhibitor of VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase(IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively). | |||
T4853 | TRIA-662 | 3-Carbamoyl-1-methylpyridinium Chloride,1-Methylnicotinamide chloride,1-methylpyridin-1-ium-3-carboxamide hydrochloride,Nicotinamide Chloromethylate | Others , Endogenous Metabolite |
TRIA-662 (Nicotinamide Chloromethylate) is a niacin metabolite excreted via the urinary system. |
カタログ番号 | 製品名 | Species | Expression System |
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TMPH-03181 | LaaA Protein, Pseudomonas azotoformans, Recombinant (His & Myc & SUMO) | Pseudomonas azotoformans | E. coli |
Hydrolyzes L-prolinamide, L-proline-p-nitroanilide, L-alaninamide, L-methioninamide, piperidine-2-carboxamide and piperazine-2-carboxamide. Has a much lower activity towards piperazine-2-tert-butylcarboxamide. Does not h... | |||
TMPY-02552 | Adenylosuccinate Lyase Protein, Human, Recombinant (His) | Human | E. coli |
Adenylosuccinate lyase, also known as adenylosuccinase, ADSL or ASL, is an enzyme implicated in the reaction of adenylosuccinat converting to AMP and fumarate as part of the purine nucleotide cycle. The two substates of ... |