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カタログ番号 | 製品名 | 別名 | ターゲット |
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T50077 | M-Nisoldipine | 3-methyl 5-(2-methylpropyl) 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate | Others |
m-Nisoldipine (3-methyl 5-(2-methylpropyl) 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate) is a dihydropyridine calcium channel blocker, a derivative of nisoldipine, that blocks L-type calcium chann... | |||
T11074 | Dolutegravir intermediate-1 | 1-(2,2-dimethoxyethyl)-5-methoxy-6-methoxycarbonyl-4-oxopyridine-3-carboxylic acid,1-(2,2-dimethoxyethyl)-5-methoxy-6-(methoxycarbonyl)-4-oxo-1,4-dihydropyridine-3-carboxylic acid | HIV Protease |
Dolutegravir intermediate-1 (1-(2,2-dimethoxyethyl)-5-methoxy-6-(methoxycarbonyl)-4-oxo-1,4-dihydropyridine-3-carboxylic acid) is a new synthetic Dolutegravir intermediate. Dolutegravir is an integrase inhibitor develope... | |||
T1385 | Amlodipine | UK-48340 | Calcium Channel |
Amlodipine (UK-48340) is a synthetic dihydropyridine and a calcium channel blocker with antihypertensive and antianginal properties. | |||
T0231 | Amlodipine Besylate | Amlodipine benzenesulfonate | Calcium Channel |
Amlodipine Besylate(Amlodipine benzenesulfonate) is a long-lasting calcium channel blocker. | |||
T0343 | Nimodipine | BAY-e 9736 | Glucocorticoid Receptor , AhR , Calcium Channel , Autophagy |
Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells. | |||
T0145 | Felodipine | CGH-869 | Calcium Channel , Autophagy |
Felodipine (CGH-869) is a longlasting 1, 4-dihydropyridine calcium channel repressor. | |||
T0388 | Cilnidipine | FRC-8653 | Calcium Channel |
Cilnidipine (FRC-8653)(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity. | |||
T67605 | 4-(2,3-Dichlorophenyl)-5-(methoxycarbonyl)-2,6-dimethyl-1,4-dihydropyridine-3-carboxylic acid | ||
4-(2,3-Dichlorophenyl)-5-(methoxycarbonyl)-2,6-dimethyl-1,4-dihydropyridine-3-carboxylic acid is a useful organic compound for research related to life sciences. The catalog number is T67605 and the CAS number is 123853-... | |||
T0957 | Isradipine | PN 200-110 | Calcium Channel , Autophagy |
Isradipine (PN 200-110) is a dihydropyridine calcium channel blockers with antihypertensive and vasodilator activities. Isradipine blocks the calcium entry through the calcium ion channels of coronary and peripheral vasc... | |||
T67592 | 5-(Methoxycarbonyl)-2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3-carboxylic acid | ||
5-(Methoxycarbonyl)-2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3-carboxylic acid is a useful organic compound for research related to life sciences. The catalog number is T67592 and the CAS number is 74936-72-4. | |||
T0999 | Clevidipine | Clevidipine butyrate,Cleviprex | Calcium Channel , AChR |
Clevidipine (Clevidipine butyrate) is a dihydropyridine L-type calcium channel blocker that is selective for vascular smooth muscle and is indicated for blood pressure reduction when oral therapy is not an option. | |||
T15053 | Darodipine | PY-108068,PY 108-068 | Calcium Channel |
Darodipine (PY-108068) is a dihydropyridine type Ca+2 antagonist. | |||
T0121 | Azelnidipine | CS 905,UR-12592 | Calcium Channel |
Azelnidipine (UR-12592) is a dihydropyridine used as calcium channel blocker. | |||
T2323 | Efonidipine | (±)-Efonidipine,NZ-105 | Calcium Channel |
Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels. | |||
T6874 | Lercanidipine hydrochloride | Corifeo,Carmen,Cardiovasc | Calcium Channel |
Lercanidipine hydrochloride (Corifeo) is a calcium channel blocker of the dihydropyridine class. | |||
T6577 | Manidipine | Iperten,Franidipine,Artedil | Calcium Channel |
Manidipine (Iperten), a calcium channel blocker, which is dihydropyridine type. It is utilized | |||
T2519 | Lercanidipine | Masnidipine | Calcium Channel |
Lercanidipine (Masnidipine) is a calcium channel blocker of the dihydropyridine class. | |||
T6227 | Benidipine hydrochloride | (±)-Benidipine,Benidipine HCl,KW-3049,Coniel | EGFR , Calcium Channel , Src |
Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel. | |||
T0163 | Nisoldipine | BAY-k 5552 | Calcium Channel , Reactive Oxygen Species |
Nisoldipine (BAY-k 5552) is a dihydropyridine calcium channel antagonist that acts as a potent arterial vasodilator and antihypertensive agent. | |||
T21263 | Amlodipine maleate | Amlodipine (+-)-form maleate,Amvaz | Calcium Channel |
Amlodipine maleate (Amvaz) is an orally active dihydropyridine calcium channel blocker that inhibits calcium inward flow by blocking voltage-dependent L-type calcium channels.Amlodipine maleate is used in the study of hy... | |||
T24932 | Vatanidipine | AE-0047,AE 0047,AE0047 | Calcium Channel |
Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lasting hypotensive action was observed in various experimental hypertensi... | |||
T21454 | Nicardipine | Cardene,Dagan,Antagonil,Flusemide | Calcium Channel |
Nicardipine (Cardene), a calcium channel blockers belonging to the dihydropyridine class, is a drug used to treat angina and high blood pressure. | |||
TQ0145 | (R)-(+)-Bay-K-8644 | (R)-(+)-Bay K 8644 | Calcium Channel , PPAR |
T5856 | Barnidipine hydrochloride | YM-09730-5 hydrochloride,Mepirodipine (hydrochloride) | Calcium Channel |
Barnidipine hydrochloride (YM-09730-5 hydrochloride) is a dihydropyridine calcium channel blocker that has an IC50 value of 0.35 nM in potassium-induced tonic contraction of pig coronary artery | |||
T1439 | Lacidipine | SN-305,GX-1048,GR-43659X | Apoptosis , Calcium Channel , Reactive Oxygen Species |
Lacidipine (SN-305) is a lipophilic dihydropyridine calcium antagonist with an intrinsically slow onset of activity. Due to its long duration of action, lacidipine does not lead to reflex tachycardia. It displays specifi... | |||
T16571 | Pranidipine | OPC-13340 | Calcium Channel |
Pranidipine (OPC-13340) is a novel, long-acting 1,4-dihydropyridine calcium channel blocker. It prolongs acetylcholine-induced relaxation in presence of endothelium as well as nitroglycerin-induced relaxation in absence ... | |||
T1545 | Levamlodipine | (S)-Amlodipine,S-amlodipine | Calcium Channel |
Levamlodipine (S-amlodipine) belongs to the dihydropyridine group of calcium channel blockers. Levamlodipine, also known as S-amlodipine, is a pharmacologically active enantiomer of amlodipine, an antihypertensive and an... | |||
T4284 | Levamlodipine besylate | (S)-Amlodipine Besylate (103129-82-4(free base)) | Calcium Channel |
Levamlodipine besylate ((S)-Amlodipine Besylate (103129-82-4(free base))) , also known as S-amlodipine, is a pharmacologically active enantiomer of amlodipine, an antihypertensive and anti-anginal medication. Levamlodipi... | |||
T1146 | Nifedipine | BAY-a-1040,Procardia XL,Procardia,Adalat | CaMK , Potassium Channel , Calcium Channel , Autophagy |
Nifedipine (Procardia) is a dihydropyridine calcium channel blocking agent. Nifedipine inhibits the transmembrane influx of extracellular calcium ions into myocardial and vascular smooth muscle cells, causing dilatation ... | |||
T68123 | Oxodipine | Calcium Channel | |
Oxodipine, a dihydropyridine-type calcium antagonist , inhibited KCl-induced aortic contraction in rabbits and reduced cardiac force in less potent rat ventricular test-paper contractions. In rat cultured neonatal ventri... | |||
T15733 | Lemildipine | NB-818,NPK-1886 | Others |
Lemildipine is a new blocker of dihydropyridine calcium entry. | |||
T33466 | Modipafant | ||
Modipaafant is a potent dihydropyridine PAF (platelet activating factor) antagonist. | |||
T34460 | S 16317 | S-16317,S16317 | |
S 16317 is a dihydropyridine derivatives with low calcium channel affinity. | |||
T32997 | LY 249933 | LY249933,LY-249933 | |
LY 249933 is a cardioselective 1, 4-dihydropyridine with positive inotropic activity. | |||
T69157 | H 160-51 | ||
H 160-51 is a calcium agonistic 1,4-dihydropyridine. | |||
T17277 | YS-201 | Others | |
YS-201 is an antagonist of dihydropyridine-type calcium channel. | |||
T13812 | PCA50941 | Others | |
PCA50941 is a 1,4-dihydropyridine derivative, treatment for cardiovascular disease. | |||
T69001 | Perindopril arginine | ||
Perindopril arginine is an angiotensin converting enzyme inhibitor, and amlodipine, a dihydropyridine calcium channel blocker, and is indicated for the treatment of hypertension, to lower blood pressure. | |||
T0112L2 | Diltiazem malate | Tiamate,UNII-14Y6444DRP,MK-793 | |
Diltiazem malate is an ACE inhibitor and non-dihydropyridine calcium channel blocker used in the treatment of hypertension. | |||
T70963 | S 11568 | ||
S 11568 is a dihydropyridine calcium channel antagonist. | |||
T15021 | CV-159 | Others | |
T23710 | Watanidipine dihydrochloride | ||
Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions. | |||
T68263 | MDL-72567 | ||
MDL-72567 is a dihydropyridine calcium antagonist that causes vasodilation and direct sinus bradycardia. | |||
T68404 | Azidopine | ||
Azidopine is a photoactive dihydropyridine channel blocker which may also act as a multidrug resistant (MDR) modulator. | |||
T39770 | UK-59811 hydrochloride | ||
UK-59811 hydrochloride is a potent inhibitor of the Ca V Ab voltage-gated calcium channels in bacterial homotetrameric models. It is derived from Br-dihydropyridine, possessing significant inhibitory properties with an I... | |||
T25691 | Levamlodipine gentisate | (S)-Amlodipine gentisate,(S)-(-)-Amlodipine gentisate | |
Levamlodipine gentisate is a pharmacologically active enantiomer of amlodipine. Amlodipine is the dihydropyridine calcium channel blocker used as an antihypertensive and antianginal drug. | |||
T25669 | Lercanidipine, (S)- | (S)-Lercanidipine,(+)-Lercanidipine | |
Lercanidipine, (S)- is an isomer of Lercanidipine, an antihypertensive compound.Lercanidipine is a dihydropyridine calcium channel blocker with long-lasting antihypertensive and nephroprotective effects. | |||
T0112L | Diltiazem | Diltiazem free base,Dilticard,CRD-401,CRD401,Dilzen,CRD 401 | |
Diltiazem is a non-dihydropyridine (non-DHP) calcium channel blocker that relaxes the smooth muscle in arterial walls, thus opening (dilating) arteries, allowing easier blood flow, and lowering blood pressure, and is use... | |||
T71583 | Amlodipine hydrochloride, (R)- | ||
Amlodipine hydrochloride, (R)-, is a medication used to lower blood pressure and prevent chest pain. It belongs to a group of medications known as dihydropyridine-type calcium channel blockers. By widening of blood vess... | |||
T28321 | PD 122860 | PD-122860,PD122860 | |
PD 122860 is a dihydropyridine with calcium channel blocking and sodium channel stimulating properties. In the rat heart, PD 122860 increased left ventricular contractility, decreased coronary resistance and altered the ... |
カタログ番号 | 製品名 | 別名 | ターゲット |
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T6981 | 1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid | Nudifloric Acid | Others |
1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid (Nudifloric Acid) is from Cordyceps bassiana. Nudifloric Acid targets to block AP-1-mediated luciferase activity, implying it has an anti-inflammatory function. | |||
T8150 | Nudifloramide | 1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide | PARP , Endogenous Metabolite |
Nudifloramide (1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide) is one of the end degradation products of nicotinamide-adenine dinucleotide (NAD). |