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Search Results for " adrenergic "

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Adrenergic Receptor Adrenergic Receptor

515

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43

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ライブラリー

カタログ番号 製品名 別名 ターゲット
T13016 SR59230A Adrenergic Receptor
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
T37906 Dibenamine hydrochloride Adrenergic Receptor
Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.
T7065 Tizanidine Adrenergic Receptor
Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons.
T7160 Lofexidine Adrenergic Receptor
Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
T7045 Clonidine Nexiclon,Catapres,Kapvay Adrenergic Receptor
Clonidine (Kapvay) is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide-scale use for many years, clonidine has not been l...
T40622 Mapenterol hydrochloride Adrenergic Receptor
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.
T0279 Metaraminol tartrate Metaradrine tartrate,Metaraminol bitartrate Adrenergic Receptor
Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in the treatment of HYPOTENSION.
T8348 Phentolamine Adrenergic Receptor
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
T7728 ACEPROMAZINE MALEATE Dopamine Receptor
ACEPROMAZINE MALEATE is a dopamine receptor antagonist
T8899 Metipranolol Adrenergic Receptor
Metipranolol (Betamann) is a type of β- Adrenergic receptors（ β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta bloc...
T5471 GUANABENZ Adrenergic Receptor
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
T2524 Dexmedetomidine Adrenergic Receptor
Dexmedetomidine is a Central alpha-2 Adrenergic Agonist. The mechanism of action of dexmedetomidine is as an Adrenergic alpha2-Agonist. The physiologic effect of dexmedetomidine is by means of General Anesthesia.
T8580 Bupranolol Adrenergic Receptor
Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.
T21640 Talinolol Adrenergic Receptor
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
T1275 Phentolamine mesylate Phentolamine methanesulfonate,Phentolamine mesilate Adrenergic Receptor
Phentolamine mesylate (Phentolamine methanesulfonate) is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma, vasospasm of RAYNAUD DISEAS...
T5511 L-765314 Adrenergic Receptor
L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the role of α1B receptors in the regulation of blood pressure.
T10830 CL 316243 Adrenergic Receptor
CL316243 is a highly potent selective agonist of β3-adrenoceptor, with a EC50 of 3 nM. CL316243 is an effective stimulant of adipocyte lipolysis and increases brown adipose tissue thermogenesis and metabolic rate. CL3162...
T1584 Terbutaline Sulfate Terbutaline hemisulfate Antibacterial , Adrenergic Receptor , Antibiotic
Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.
T4983 Isoetharine mesylate salt Isoetarine mesilate Others , Adrenergic Receptor
Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
T2320 Indacaterol Adrenergic Receptor
Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.
T8708 Paroxetine Serotonin Transporter
Paroxetine is a inhibitor of serotonin uptake that is effective in the treatment of depression.
T22406 Prazosin Prazosine,Furazosin,Prazocin Adrenergic Receptor
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T6872 L755507 Adrenergic Receptor , CRISPR/Cas9
L755507 is an effective, selective agonist of β3-AR（IC50=35 nM）.
T6641 Rilmenidine Phosphate Apoptosis , Adrenergic Receptor , Autophagy , Imidazoline Receptor
Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.
T11318 Dopexamine hydrochloride FPL60278AR Adrenergic Receptor
Dopexamine hydrochloride (FPL60278AR) is a β2-adrenergic receptor agonist. Dopexamine can attenuate the inflammatory response and protect against organ injury in the absence of significant effects on hemodynamics or regi...
T12829 Salmeterol GR33343X Adrenergic Receptor
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
T19680 Zotepine Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM, 3.3 nM, 7.3 nM, and 8 nM, respectively. Zotepine is a second...
T12402 Penbutolol sulfate (-)-Terbuclomine Adrenergic Receptor
Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.
T3284 Carazolol Conducton,Suacron Adrenergic Receptor
Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
T1132 Nicergoline Nicergolinum,Nimergoline Adrenergic Receptor
Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
T21957 Guanabenz hydrochloride NE56490 Adrenergic Receptor
Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.
T1247 Clonidine hydrochloride Clonidine HCl,Catapres Adrenergic Receptor
Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
T8358 Fenoterol Adrenergic Receptor
Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.
T1012 Acebutolol hydrochloride Acebutolol HCl Adrenergic Receptor
Acebutolol hydrochloride (Acebutolol HCl) acts as a cardioselective beta-adrenergic antagonist with little effect on bronchial receptors and has intrinsic sympathomimetic properties. Acebutolol hydrochloride is the hydro...
T17111 Todralazine hydrochloride Ecarazine hydrochloride Adrenergic Receptor
Todralazine hydrochloride (Ecarazine hydrochloride) is a β2AR blocker and has antioxidant and free radical scavenging activities. Todralazine hydrochloride can be used in anti-hypertensive research.
T22316 Doxazosin UK 33274 Adrenergic Receptor
Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.
T7164 Levalbuterol tartrate Levosalbutamol tartrate Adrenergic Receptor
Levalbuterol tartrate (Levosalbutamol tartrate) is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
T1671 Mirabegron YM178 Adrenergic Receptor
Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
T0394 Moxisylyte hydrochloride Thymoxamine hydrochloride Adrenergic Receptor
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
T0154 Nebivolol hydrochloride R 065824 hydrochloride,Nebivolol HCl,R-65824 Apoptosis , Adrenergic Receptor
Nebivolol hydrochloride (R 065824 hydrochloride) is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR through the endothelial L-arginine/ NITRIC OXIDE system. It is us...
T19654 Guanoclor VATENSOL Others
Guanoclor (VATENSOL) (INN), also known as guanochlor, is a sympatholytic drug. It is known to bind to non-adrenergic sites in pig kidney membranes.
T0993 Methoxamine hydrochloride Methoxamine HCl Adrenergic Receptor
Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
T0397 Tetrahydrozoline Tetryzolin,Tetryzoline Adrenergic Receptor
Tetrahydrozoline (Tetryzoline), an alpha agonist, have an effect on the constriction of conjunctival blood vessels. This contributes to relieve the redness of the eye resulted from minor ocular irritants.
T0165 Urapidil Mediatensyl,Ebrantil,Eupressyl 5-HT Receptor , Adrenergic Receptor
Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
T6766 Atipamezole Antisedan,MPV 1248 Adrenergic Receptor
Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
T6408 Betaxolol Kerlone,SL 75212,Betoptic Adrenergic Receptor
Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
T1139 Salbutamol Albuterol,AH-3365 Adrenergic Receptor
Salbutamol (Albuterol) stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3', 5'-adenosine monophosphate (cAMP). Salbutamol ...
T1050 Prazosin hydrochloride Prazosin hydrochloride,Prazosin HCl,cp-12299-1,Peripress,Vasoflex,Minipress Potassium Channel , MRP , Adrenergic Receptor , ABC , Autophagy
Prazosin hydrochloride (Vasoflex) reduces peripheral resistance and relaxes vascular smooth muscles as a selective adrenergic alpha-1 antagonist by a mechanism not completely known. Prazosin hydrochloride is a synthetic ...
T0210 Tamsulosin hydrochloride Flomax,Flomax hydrochloride Adrenergic Receptor
Tamsulosin hydrochloride (Flomax hydrochloride) is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.
T6647 Rotigotine- Neupro,N-0923,N-0437,SPM 962 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome. Administered as a once-daily transdermal patch, Rotigotine has not been associated with ser...

Compounds

SR59230A
T13016
Synonym:
Target: Adrenergic Receptor
Dibenamine hydrochloride
T37906
Synonym:
Target: Adrenergic Receptor
Tizanidine
T7065
Synonym:
Target: Adrenergic Receptor
Lofexidine
T7160
Synonym:
Target: Adrenergic Receptor
Clonidine
T7045
Synonym: Nexiclon,Catapres,Kapvay
Target: Adrenergic Receptor
Mapenterol hydrochloride
T40622
Synonym:
Target: Adrenergic Receptor
Metaraminol tartrate
T0279
Synonym: Metaradrine tartrate,Metaraminol bitartrate
Target: Adrenergic Receptor
Phentolamine
T8348
Synonym:
Target: Adrenergic Receptor
ACEPROMAZINE MALEATE
T7728
Synonym:
Target: Dopamine Receptor
Metipranolol
T8899
Synonym:
Target: Adrenergic Receptor
GUANABENZ
T5471
Synonym:
Target: Adrenergic Receptor
Dexmedetomidine
T2524
Synonym:
Target: Adrenergic Receptor
Bupranolol
T8580
Synonym:
Target: Adrenergic Receptor
Talinolol
T21640
Synonym:
Target: Adrenergic Receptor
Phentolamine mesylate
T1275
Synonym: Phentolamine methanesulfonate,Phentolamine mesilate
Target: Adrenergic Receptor
L-765314
T5511
Synonym:
Target: Adrenergic Receptor
CL 316243
T10830
Synonym:
Target: Adrenergic Receptor
Terbutaline Sulfate
T1584
Synonym: Terbutaline hemisulfate
Target: Antibacterial, Adrenergic Receptor, Antibiotic
Isoetharine mesylate salt
T4983
Synonym: Isoetarine mesilate
Target: Others, Adrenergic Receptor
Indacaterol
T2320
Synonym:
Target: Adrenergic Receptor
Paroxetine
T8708
Synonym:
Target: Serotonin Transporter
Prazosin
T22406
Synonym: Prazosine,Furazosin,Prazocin
Target: Adrenergic Receptor
L755507
T6872
Synonym:
Target: Adrenergic Receptor, CRISPR/Cas9
Rilmenidine Phosphate
T6641
Synonym:
Target: Apoptosis, Adrenergic Receptor, Autophagy, Imidazoline Receptor
Dopexamine hydrochloride
T11318
Synonym: FPL60278AR
Target: Adrenergic Receptor
Salmeterol
T12829
Synonym: GR33343X
Target: Adrenergic Receptor
Zotepine
T19680
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Penbutolol sulfate
T12402
Synonym: (-)-Terbuclomine
Target: Adrenergic Receptor
Carazolol
T3284
Synonym: Conducton,Suacron
Target: Adrenergic Receptor
Nicergoline
T1132
Synonym: Nicergolinum,Nimergoline
Target: Adrenergic Receptor
Guanabenz hydrochloride
T21957
Synonym: NE56490
Target: Adrenergic Receptor
Clonidine hydrochloride
T1247
Synonym: Clonidine HCl,Catapres
Target: Adrenergic Receptor
Fenoterol
T8358
Synonym:
Target: Adrenergic Receptor
Acebutolol hydrochloride
T1012
Synonym: Acebutolol HCl
Target: Adrenergic Receptor
Todralazine hydrochloride
T17111
Synonym: Ecarazine hydrochloride
Target: Adrenergic Receptor
Doxazosin
T22316
Synonym: UK 33274
Target: Adrenergic Receptor
Levalbuterol tartrate
T7164
Synonym: Levosalbutamol tartrate
Target: Adrenergic Receptor
Mirabegron
T1671
Synonym: YM178
Target: Adrenergic Receptor
Moxisylyte hydrochloride
T0394
Synonym: Thymoxamine hydrochloride
Target: Adrenergic Receptor
Nebivolol hydrochloride
T0154
Synonym: R 065824 hydrochloride,Nebivolol HCl,R-65824
Target: Apoptosis, Adrenergic Receptor
Guanoclor
T19654
Synonym: VATENSOL
Target: Others
Methoxamine hydrochloride
T0993
Synonym: Methoxamine HCl
Target: Adrenergic Receptor
Tetrahydrozoline
T0397
Synonym: Tetryzolin,Tetryzoline
Target: Adrenergic Receptor
Urapidil
T0165
Synonym: Mediatensyl,Ebrantil,Eupressyl
Target: 5-HT Receptor, Adrenergic Receptor
Atipamezole
T6766
Synonym: Antisedan,MPV 1248
Target: Adrenergic Receptor
Betaxolol
T6408
Synonym: Kerlone,SL 75212,Betoptic
Target: Adrenergic Receptor
Salbutamol
T1139
Synonym: Albuterol,AH-3365
Target: Adrenergic Receptor
Prazosin hydrochloride
T1050
Synonym: Prazosin hydrochloride,Prazosin HCl,cp-12299-1,Peripress,Vasoflex,Minipress
Target: Potassium Channel, MRP, Adrenergic Receptor, ABC, Autophagy
Tamsulosin hydrochloride
T0210
Synonym: Flomax,Flomax hydrochloride
Target: Adrenergic Receptor
Rotigotine-
T6647
Synonym: Neupro,N-0923,N-0437,SPM 962
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
1 2 3 4 5 6 7 8 9 10 11
カタログ番号 製品名 別名 ターゲット
T1287 Synephrine Oxedrine Endogenous Metabolite , Adrenergic Receptor
Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
TN1015 Meranzin Adrenergic Receptor , Immunology/Inflammation related
Meranzin, a bioactive compound derived from the Traditional Chinese Medicine (TCM) Chaihu-Shugan-San (CSS) and isolated from Murraya exotica L. leaves, targets the alpha 2-adrenoceptor and engages the AMPA-ERK1/2–BDNF si...
T6688 Synephrine hydrochloride Oxedrine hydrochloride,Synephrine HCl Endogenous Metabolite , Adrenergic Receptor
Synephrine hydrochloride (Oxedrine hydrochloride) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
T6662 Scopine 6,7-Epoxytropine Adrenergic Receptor
Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
T2142 Yohimbine hydrochloride Antagonil,Yohimbine HCl Adrenergic Receptor
Yohimbine hydrochloride (Antagonil) is a plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of ERECTILE DYSFUNCTION.
T6519 Gramine NSC 16892,Donaxine Adiponectin receptor , Reverse Transcriptase , Adrenergic Receptor
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4.2 μM for AdipoR2 and AdipoR1, respectively. Gramine is als...
T8149 Dobutamine hydrochloride Dobutamine (hydrochloride) Adrenergic Receptor
Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
T17310 Phenylephrine L-Phenylephrine,(R)-(-)-Phenylephrine Adrenergic Receptor
Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
TN1465 Cannabigerol NOS , 5-HT Receptor , ROS
Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also binds to the CB2 receptor; it can relieve interocular pressur...
T13655 DL-Norepinephrine hydrochloride Lys,DL-lysine Adrenergic Receptor
DL-Norepinephrine hydrochloride (DL-lysine) is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 μM.
T0076 Paliperidone 9-hydroxyrisperidone Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the primary active metabolite of the older...
T0505 Methyldopa L-(-)-α-Methyldopa,MK-351 Dopamine Receptor , Adrenergic Receptor
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic.
T0453 Phenylephrine hydrochloride NCI-c55641,Phenylephrine HCl,(R)-(-)-Phenylephrine hydrochloride Endogenous Metabolite , Adrenergic Receptor
Phenylephrine hydrochloride (NCI-c55641) is a selective agonist of the α1-adrenergic receptor.
T7044 Norepinephrine Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol MMP , Endogenous Metabolite , Adrenergic Receptor , Autophagy
Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression of vascular endothelial growth factor, matrix metalloprotei...
T0469 Octopamine hydrochloride (±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl Dopamine Receptor , Endogenous Metabolite , Adrenergic Receptor
Octopamine hydrochloride ((±)-p-Octopamine hydrochlorid) is a biogenic monoamine structurally associated with noradrenaline. It can serve as a neurohormone, a neurotransmitter, and a neuromodulator in invertebrates.
T3158 Harmane Loturine,Harman,Aribine Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T2889 Isoferulic acid Isoferulate,Hesperetic acid,3-Hydroxy-4-methoxycinnamic acid,Hesperetate Influenza Virus , Adrenergic Receptor
Isoferulic acid (Hesperetate) exhibits hypoglycemic properties.
T5S2059 Glaucine Calcium Channel , Dopamine Receptor , Influenza Virus , Adrenergic Receptor , PDE
Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 production. Glaucine can inhibit the migration and invasion of h...
TCS2185 Yohimbine Adrenergic Receptor
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
T3232 Higenamine hydrochloride Higenamine HCl,Demethylcoclaurine hydrochloride,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride Adrenergic Receptor
Higenamine hydrochloride (norcoclaurine HCl) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupled receptors, and are the most prominent...
T1064 Norepinephrine bitartrate monohydrate Levophed,Noradrenaline bitartrate monohydrate Endogenous Metabolite , Adrenergic Receptor , Autophagy
Norepinephrine bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator.
T4429 Rauwolscine hydrochloride Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride Adrenergic Receptor
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes b...
T1680 Tolazoline hydrochloride Imidaline hydrochloride,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride) Adrenergic Receptor
Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn.
T7056 Dronedarone SR 33589 P450 , Potassium Channel , Calcium Channel , Sodium Channel , Adrenergic Receptor , AChR , Autophagy
Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
T21066 Norepinephrine bitartrate salt Adrenergic Receptor
Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
T3095 Tyramine 4-hydroxyphenethylamine,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine MAO , Endogenous Metabolite
Tyramine (Uteramine) is an indirect sympathomimetic that occurs naturally in cheese and other foods. Tyramine does not directly activate adrenergic receptors, but it can serve as a substrate for adrenergic uptake systems...
TN7042 N-methyltyramine Adrenergic Receptor
N-methyltyramine is an alkaloid isolated from the leguminous plant Acacia grandiflora.It is an α2-adrenoceptor antagonist that regulates adrenergic receptors through enzymatic adrenergic synthesis.It is used in the study...
T8304 Anisodamine Hydrobromide 6-Hydroxyhyoscyamine Adrenergic Receptor , AChR
Anisodamine Hydrobromide (6-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T6S0627 Mesaconitine TNF
1. Mesaconitine has antiinflammatory activity. 2. Mesaconitine has antinociceptive activity through cyclic AMP and stimulation of the central β-adrenergic system.
T0970 Racanisodamine Anisodamine,7β-Hydroxyhyoscyamine,Raceanisodamine Adrenergic Receptor , AChR
Racanisodamine (7β-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T0783 Mianserin hydrochloride Mianserin HCl,Org GB 94,ORG GB-94 HCl Dopamine Receptor , 5-HT Receptor , Opioid Receptor , Adrenergic Receptor , Histamine Receptor
Mianserin hydrochloride (Org GB 94) is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin receptors. It may cause drowsiness and hematolog...
TN7129 Methyl maslinate Maslinic acid methyl ester,Crategolic acid methyl ester Adrenergic Receptor
T1644 Dopamine hydrochloride Dopamine HCl,ASL279 Ferroptosis , Dopamine Receptor , 5-HT Receptor , Endogenous Metabolite
Dopamine hydrochloride (ASL279) is a naturally occurring catecholamine formed by decarboxylation of dihydroxyphenylalanine and a precursor of norepinephrine and epinephrine. Dopamine hydrochloride binds to alpha-1- and b...
T0266 Quinidine hydrochloride monohydrate Quinidine hydrochloride Potassium Channel , Sodium Channel , Parasite
Quinidine hydrochloride monohydrate is an optical isomer of quinine, extracted from the bark of the Cinchona tree and similar plant species. It prolongs cellular action potential and decreases automaticity. This alkaloid...
T5S1177 Aloin B Isobarbaloin Others
Aloin B (Isobarbaloin) is an isomer of aloin.1. The extract of A. vera and its active ingredient aloin cause melanin aggregation leading to skin lightening via alpha adrenergic receptor stimulation, the result opens new ...
T19910 Corynanthine NSC-407306,NSC407306,NSC 407306
Corynanthe is a plant alkaloid. Corynanthe also has an alpha-2-adrenergic blocking activity.
T75425 Synephrine hemitartrate
Synephrine hemitartrate (Oxedrine), an alkaloid extracted from Citrus aurantium, functions as both an α-adrenergic and β-adrenergic agonist. As a sympathomimetic compound, it has applications in weight loss [1] [2].
TN4882 Quinine HCl Adrenergic Receptor
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T11937 M-Tyramine Others
m-Tyramine has effects on the adrenergic and dopaminergic receptor.m-Tyramine is an endogenous trace amine neuromodulator.
T2S1727 Lycorenine Antifection
Lycorenine may produce a decrease in blood pressure as the result of alpha-adrenergic blockade in conjunction with the reduction of the spontaneous sympathetic nerve activity, and produce bradycardia by modifying vagal a...
T60245 Norepinephrine hydrochloride
Norepinephrine hydrochloride (Levarterenol hydrochloride) is a β1 -selective agonist of the adrenergic receptor with EC 50 of 5.37 μM [1].
TN1797 Isorhoifolin Adrenergic Receptor
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile force by increasing the l-type calcium current and activatin...
TN2001 Oblongine Others
Oblongine chloride may have potential haemodynamic effects, it can cause a dose-dependent reduction of systolic and diastolic blood pressure, and that these effects are not mediated by α²-adrenergic receptor stimulation.

天然物製品

Synephrine
T1287
Synonym: Oxedrine
Target: Endogenous Metabolite, Adrenergic Receptor
Meranzin
TN1015
Synonym:
Target: Adrenergic Receptor, Immunology/Inflammation related
Synephrine hydrochloride
T6688
Synonym: Oxedrine hydrochloride,Synephrine HCl
Target: Endogenous Metabolite, Adrenergic Receptor
Scopine
T6662
Synonym: 6,7-Epoxytropine
Target: Adrenergic Receptor
Yohimbine hydrochloride
T2142
Synonym: Antagonil,Yohimbine HCl
Target: Adrenergic Receptor
Gramine
T6519
Synonym: NSC 16892,Donaxine
Target: Adiponectin receptor, Reverse Transcriptase, Adrenergic Receptor
Dobutamine hydrochloride
T8149
Synonym: Dobutamine (hydrochloride)
Target: Adrenergic Receptor
Phenylephrine
T17310
Synonym: L-Phenylephrine,(R)-(-)-Phenylephrine
Target: Adrenergic Receptor
Cannabigerol
TN1465
Synonym:
Target: NOS, 5-HT Receptor, ROS
DL-Norepinephrine hydrochloride
T13655
Synonym: Lys,DL-lysine
Target: Adrenergic Receptor
Paliperidone
T0076
Synonym: 9-hydroxyrisperidone
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Methyldopa
T0505
Synonym: L-(-)-α-Methyldopa,MK-351
Target: Dopamine Receptor, Adrenergic Receptor
Phenylephrine hydrochloride
T0453
Synonym: NCI-c55641,Phenylephrine HCl,(R)-(-)-Phenylephrine hydrochloride
Target: Endogenous Metabolite, Adrenergic Receptor
Norepinephrine
T7044
Synonym: Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol
Target: MMP, Endogenous Metabolite, Adrenergic Receptor, Autophagy
Octopamine hydrochloride
T0469
Synonym: (±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl
Target: Dopamine Receptor, Endogenous Metabolite, Adrenergic Receptor
Harmane
T3158
Synonym: Loturine,Harman,Aribine
Target: Adrenergic Receptor, Monoamine Oxidase, Imidazoline Receptor
Isoferulic acid
T2889
Synonym: Isoferulate,Hesperetic acid,3-Hydroxy-4-methoxycinnamic acid,Hesperetate
Target: Influenza Virus, Adrenergic Receptor
Glaucine
T5S2059
Synonym:
Target: Calcium Channel, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, PDE
Yohimbine
TCS2185
Synonym:
Target: Adrenergic Receptor
Higenamine hydrochloride
T3232
Synonym: Higenamine HCl,Demethylcoclaurine hydrochloride,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride
Target: Adrenergic Receptor
Norepinephrine bitartrate monohydrate
T1064
Synonym: Levophed,Noradrenaline bitartrate monohydrate
Target: Endogenous Metabolite, Adrenergic Receptor, Autophagy
Rauwolscine hydrochloride
T4429
Synonym: Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride
Target: Adrenergic Receptor
Tolazoline hydrochloride
T1680
Synonym: Imidaline hydrochloride,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)
Target: Adrenergic Receptor
Dronedarone
T7056
Synonym: SR 33589
Target: P450, Potassium Channel, Calcium Channel, Sodium Channel, Adrenergic Receptor, AChR, Autophagy
Norepinephrine bitartrate salt
T21066
Synonym:
Target: Adrenergic Receptor
Tyramine
T3095
Synonym: 4-hydroxyphenethylamine,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine
Target: MAO, Endogenous Metabolite
N-methyltyramine
TN7042
Synonym:
Target: Adrenergic Receptor
Anisodamine Hydrobromide
T8304
Synonym: 6-Hydroxyhyoscyamine
Target: Adrenergic Receptor, AChR
Mesaconitine
T6S0627
Synonym:
Target: TNF
Racanisodamine
T0970
Synonym: Anisodamine,7β-Hydroxyhyoscyamine,Raceanisodamine
Target: Adrenergic Receptor, AChR
Mianserin hydrochloride
T0783
Synonym: Mianserin HCl,Org GB 94,ORG GB-94 HCl
Target: Dopamine Receptor, 5-HT Receptor, Opioid Receptor, Adrenergic Receptor, Histamine Receptor
Methyl maslinate
TN7129
Synonym: Maslinic acid methyl ester,Crategolic acid methyl ester
Target: Adrenergic Receptor
Dopamine hydrochloride
T1644
Synonym: Dopamine HCl,ASL279
Target: Ferroptosis, Dopamine Receptor, 5-HT Receptor, Endogenous Metabolite
Quinidine hydrochloride monohydrate
T0266
Synonym: Quinidine hydrochloride
Target: Potassium Channel, Sodium Channel, Parasite
Aloin B
T5S1177
Synonym: Isobarbaloin
Target: Others
Corynanthine
T19910
Synonym: NSC-407306,NSC407306,NSC 407306
Target:
Synephrine hemitartrate
T75425
Synonym:
Target:
Quinine HCl
TN4882
Synonym:
Target: Adrenergic Receptor
m-Tyramine
T11937
Synonym:
Target: Others
Lycorenine
T2S1727
Synonym:
Target: Antifection
Norepinephrine hydrochloride
T60245
Synonym:
Target:
Isorhoifolin
TN1797
Synonym:
Target: Adrenergic Receptor
Oblongine
TN2001
Synonym:
Target: Others

Recombinant Proteins

Species：
Human (4)
Mouse (2)
Expression System：
E. coli (5)
Baculovirus Insect Cells (1)
Tag：
N-6xHis-SUMO (3)
C-6xHis (1)
His, GST (1)
N-6xHis (1)
カタログ番号 製品名 Species Expression System
TMPY-04562 GRK2 Protein, Human, Recombinant (His & GST) Human Baculovirus Insect Cells
G-protein coupled receptor kinase 2 (GRK2), also referred as Adrenergic, beta, receptor kinase 1 (ADRBK1), is a ubiquitous member of the G protein-coupled receptor kinase (GRK) family that appears to play a central, inte...
TMPJ-00983 ARRB1 Protein, Human, Recombinant (His) Human E. coli
β-Arrestin-1 (ARRB1) is a cytoplasmic protein that belongs to the arrestin family. ARRB1 is expressed at high levels in peripheral blood leukocytes and the central nervous system. ARRB1 regulates agonist-mediated G-prote...
TMPH-02693 GNAI2 Protein, Mouse, Recombinant (His) Mouse E. coli
Guanine nucleotide-binding proteins (G proteins) are involved as modulators or transducers in various transmembrane signaling systems. The G(i) proteins are involved in hormonal regulation of adenylate cyclase: they inhi...
TMPH-01422 GNAS Protein, Human, Recombinant (His & SUMO) Human E. coli
Guanine nucleotide-binding proteins (G proteins) function as transducers in numerous signaling pathways controlled by G protein-coupled receptors (GPCRs). Signaling involves the activation of adenylyl cyclases, resulting...
TMPH-01250 MAP2K3 Protein, Human, Recombinant (His & SUMO) Human E. coli
Dual specificity kinase. Is activated by cytokines and environmental stress in vivo. Catalyzes the concomitant phosphorylation of a threonine and a tyrosine residue in the MAP kinase p38. Part of a signaling cascade that...
TMPH-02540 GRK2 Protein, Mouse, Recombinant (His & SUMO) Mouse E. coli
Specifically phosphorylates the agonist-occupied form of the beta-adrenergic and closely related receptors, probably inducing a desensitization of them. Key regulator of LPAR1 signaling. Competes with RALA for binding to...
カタログ番号 製品名
L2700 Adrenergic Receptor-Targeted Compound Library

193 compounds
A unique collection of 193 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification;
L2610 Neurotransmitter Receptor Compound Library

1513 compounds
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；

ライブラリー

Adrenergic Receptor-Targeted Compound Library
L2700
Compounds: 193
Neurotransmitter Receptor Compound Library
L2610
Compounds: 1513
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