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阻害剤 血管新生 アポトーシス オートファジー 細胞周期・チェックポイント クロマチン・エピジェネティック 細胞骨格シグナル DNA損傷・DNA修復 内分泌・ホルモン GPCR/Gタンパク質 免疫・炎症 JAK・STATシグナル MAPK
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シグナル伝達経路 血管新生 アポトーシス オートファジー 細胞周期・チェックポイント クロマチン・エピジェネティック 細胞骨格シグナル
DNA損傷・DNA修復 内分泌・ホルモン GPCR/Gタンパク質 免疫・炎症 JAK・STATシグナル MAPK 膜輸送体・イオンチャネル
代謝 微生物学・ウィルス学 神経科学 NF-Κb 酸化還元 PI3K/Akt/mTORシグナル プロテアーゼ・プロテアソーム
幹細胞 チロシンキナーゼ・アダプター ユビキチン その他 PROTAC
生物活性化合物ライブラリー ゼネラルバイオウアクティヴライブラリー 承認/再開発 医薬品ライブラリー 疾患別 化合物ライブラリー 標的/経路別 化合物ライブラリー 特徴的な生物活性化合物ライブラリー
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ドラッグライク 化合物ライブラリー ドラッグライクライブラリー
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CD Proteins •   T Cell CD Proteins •   B Cell CD Proteins Immune Checkpoint Proteins •   Co-inhibitory Immune Checkpoint Proteins •   Co-stimulatory Immune Checkpoint Proteins
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Search Results for " Voltage-gated "

ターゲット

TRP/TRPV Channel

127

阻害剤

12

天然化合物

15

リコンビナントタンパク質

1

ライブラリー

カタログ番号 製品名 別名 ターゲット
T19723 AMTB hydrochloride AMTB TRP/TRPV Channel
AMTB hydrochloride (AMTB HCl) is a novel TRPM8 channel blocker and is effective for pain and urinary diseases. AMTB can act on the bladder afferent pathway to attenuate the bladder micturition reflex and nociceptive refl...
T0939 Phenytoin Diphenylhydantoin,5,5-Diphenylhydantoin Virus Protease , Sodium Channel
Phenytoin (5,5-Diphenylhydantoin) is a hydantoin derivative and a non-sedative antiepileptic agent with anticonvulsant activity. Phenytoin potentially acts by promoting sodium efflux from neurons located in the motor cor...
T15260 Evenamide NW-3509 Sodium Channel
Evenamide (NW-3509) is a sodium channel blocker. Which shows efficacy in a broad spectrum of rodent models of psychosis, mania, depression, and aggressiveness.
T4497 Amifampridine 3,4-Pyridinediamine,Pyridine-3,4-Diamine,3,4-Diaminopyridine Others
Amifampridine (3,4-Diaminopyridine) is predominantly in the treatment of a number of rare muscle diseases. Amifampridine works by blocking potassium channel efflux in nerve terminals so that action potential duration is ...
T0008 Phenytoin sodium 5,5-Diphenylhydantoin sodium salt,Diphantoine,Dilantin sodium,Diphenylhydantoin Sodium Virus Protease , Sodium Channel
Phenytoin sodium (Diphantoine) is an inactive stabilizer for voltage-gated sodium channel .
T7806 Licarbazepine ​10,11-hydroxy-10,11 Dihydrocarbamezer Others
Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial seizures and bipolar disorders.
T11990 Meclofenamic acid Meclofenamate Others , Gap Junction Protein
Meclofenamic acid (Meclofenamate) is a non-selective gap-junction blocker and a selective fat mass and obesity-associated (FTO) enzyme inhibitor. Meclofenamic acid has anti-inflammatory activities.
T60010 BTT-266 Calcium Channel
BTT-266 is a blocker of voltage-gated calcium channel for pain management.
T31716 Etidocaine Hydrochloride W-19053,Duranest,W19053,W 19053 Sodium Channel
Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel.
T77712 Calcium Channel antagonist 3 Calcium Channel
Calcium Channel antagonist 3 is a voltage-gated calcium channel inhibitor (IC50 : 5-20 μM).
T77711 Calcium Channel antagonist 4 Calcium Channel
Calcium Channel antagonist 4 is a voltage-gated calcium channel inhibitor (IC50 : 5-20 μM).
T22675 Co 102862 V 102862 Others , Sodium Channel
Co 102862 is a voltage-gated sodium channel blocker. Co 102862 can be used for anticonvulsant studies.
T9751 Transfluthrin Others
Transfluthrin is a volatile pyrethroid insecticide that targets insect voltage-gated sodium channels (VGSC).
T12424 PF-06305591 PF-6305591 Others
T6571 Lomerizine dihydrochloride Terranas,Lomerizine 2HCl,Lomerizine hydrochloride,KB-2796 Calcium Channel
Lomerizine dihydrochloride (KB-2796) is an antagonist of L- and T-type voltage-gated calcium channels used to treat migraine.
T2523 Rufinamide CGP 33101,E 2080,RUF 331 Sodium Channel
Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.
T23497 UK 78282 hydrochloride Potassium Channel
UK 78282 hydrochloride, a novel potent and selective Kv1.3 blocker.UK 78282 hydrochloride inhibits Kv1.3 voltage-gated potassium channels and suppresses human T cell activation.
T12181 NaV1.7 inhibitor-1 Sodium Channel
NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).
T7066 Fosphenytoin disodium Fosphenytoin sodium,ACC-9653 Sodium Channel
Fosphenytoin disodium (ACC-9653) is a prodrug of phenytoin that is rapidly converted to phenytoin, a voltage-gated sodium channel blocker
T12786 RY785 Potassium Channel
RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.
T0024 Primidone Primaclone,Mysoline,NCI-C56360 GABA Receptor , Sodium Channel , GluR , AChR
Primidone (NCI-C56360) is a potent anticonvulsant agent. It is a neuronal voltage-gated sodium channel blocker and has value in the study of epilepsy, essential tremor, and psychiatric disorders.
T6782L Benzocaine xHCl(94-09-7(free base)) Sodium Channel
Benzocaine shares a common receptor with all othe rLAs in the voltage-gated Na+ channel(IC50 of 0.8 mM tested with a potential of +30 mV).
T68073 Flosatidil Calcium Channel
Flosatidil is a small molecule voltage-gated calcium channel complex (VDCCs) blocker for the treatment of neurological disorders and cardiovascular diseases, and can be used in the study of angina pectoris.
T8639 Phenibut (hydrochloride) 3-Amino-4-phenylbutyric acid hydrochloride GABA Receptor
Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing voltage-gated calcium channels, stimulates dopamine receptor...
T77642 1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride Calcium Channel
1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride can be us...
T0796 Prilocaine hydrochloride Prilocaine HCl,Propitocaine hydrochloride,Xylonest ATPase , Sodium Channel
Prilocaine hydrochloride (Prilocaine HCl) is a local anesthetic of the amino amide type, binds to voltage-gated sodium ion channels in the neuronal membrane, thereby preventing the permeability of sodium ions.
T50030 1-(2,4-difluorophenyl)guanidine hydrochloride Others
1-(2,4-difluorophenyl)guanidine hydrochloride is a compound that is a potent and selective inhibitor of the voltage-gated sodium channel Nav1.7, a key player in pain signaling. It is therefore able to reduce pain signali...
T0222 Proparacaine hydrochloride Proparacaine HCl,Proxymetacaine Hydrochloride Apoptosis , Sodium Channel
Proparacaine Hydrochloride is the hydrochloride salt form of proparacaine, a benzoic acid derivative with local anesthetic property. Proparacaine hydrochloride (Proparacaine HCl) stabilizes the neuronal membrane by bindi...
T0018 Procainamide hydrochloride Procapan,Procainamide HCl,Pronestyl,Procanbid DNA Methyltransferase , Sodium Channel , AChR , Autophagy
Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog of procaine. Procainamide hydrochloride reversibly binds to...
T22361 Mepivacaine Carbocaine Sodium Channel
Mepivacaine (Carbocaine) is an amide compound for local anaesthesia that causes transient loss of self-consciousness in humans or animals. mepivacaine acts by binding to specific voltage-gated sodium channels in nerve ce...
T7502 PF 05089771 tosylate Sodium Channel
PF-05089771 is a voltage-gated sodium channel 1.7 (Nav1.7) blocker (IC50: 11, 16, 33, and 20 nM for 5N11S, 5A11L, 5A11S, and 5A11L Nav1.7 splice variants, respectively). It is selective for Nav1.7 over Nav1.1-1.6 and 1.8...
T0802 Procaine hydrochloride Novocaine HCl,Procaine HCl Histone Demethylase , 5-HT Receptor , DNA/RNA Synthesis , Sodium Channel , NMDAR , AChR
Procaine hydrochloride (Novocaine HCl) is the hydrochloride salt form of procaine, a benzoic acid derivative with local anesthetic and antiarrhythmic properties. Procaine binds to and inhibits voltage-gated sodiumchannel...
T1046 Mexiletine hydrochloride KOE-1173 (hydrochloride),Mexiletine HCl,KO1173 AhR , Sodium Channel
Mexiletine hydrochloride (KOE-1173 hydrochloride) is a voltage-gated sodium channel blocker and a Class IB antiarrhythmic drug. Mexiletine hydrochloride exerts antiarrhythmic effects by inhibiting sodium current in myoca...
T26174 SAK3 SAK 3,SAK-3 Calcium Channel , AChR
SAK3 is a novel modulator of nAChR activity that enhances T-type voltage-gated Ca2+ channel (T-VGCC) activity, and has potentiating effects on both Cav3.1 and Cav3.3 T-type Ca2+ channel currents.SAK3 is neuroprotective a...
T4612 NS309 EGFR , Potassium Channel , HER
NS309 is a nonselective activator of small- and intermediate-conductance Ca2+-activated K+ (SK/KCa2 and IK/KCa3.1) channels (EC50s range from 0.12-1.2 µM for SK channels and 10-90 nM for IK channels). It can also activat...
T1496 Amiodarone hydrochloride Amiodar,Amiodarone HCl,Nexterone Potassium Channel , Adrenergic Receptor , Autophagy
Amiodarone hydrochloride (Amiodarone HCl) is an antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action by inhibiting POTASSIUM CHANNELS and VOLTAGE-GATED SODIUM C...
T0267 Zonisamide AD 810,CI 912 Calcium Channel , Sodium Channel , Carbonic Anhydrase
Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures. It may inhibit a carbonic anhydrase although this is not one of the main mechanisms...
T5148 Atosiban acetate RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164 Oxytocin Receptor , Vasopressin Receptor
Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban acetate (RW22164) inhibits...
T22925 Linopirdine dihydrochloride Others
KV7 (KCNQ) voltage-gated potassium channels blocker
T27040 Clathrodin
Clathrodin is a voltage-gated sodium (NaV) channels modulator.
T22887 KC 12291 hydrochloride Others
voltage-gated sodium channel blocker
T13830 Propoxycaine hydrochloride Sodium Channel
Propoxycaine hydrochloride is an inhibit of voltage-gated sodium channels.
T70139 MSD-D
MSD-D is an inhibitor of voltage-gated K(+) (Kv) channels Kv1.5.
T31843 Fomocaine HCl P-652 HCl,Fomocaine,P652 hydrochloride,P-652 hydrochloride,Panacaine hydrochloride,P 652 hydrochloride
Fomocaine is an type of anaesthetic agent blocking voltage-gated Na(+) currents in neurons.
T26319 Vincanol Vincanolum
Vincanol is a potent voltage-gated Na+ channels blocker.
T24137 HENA
HENA is a novel activator of large conductance, voltage- and Ca2+-gated K+ (BK) channels.
T69866 PhotoGBI1
photoGBI1 is a photocontrol inhibitor of the voltage-gated proton channel Hv1.
T68748 Saxitoxinol
Saxitoxinol is an analog of saxitoxin, a known voltage-gated sodium channel blocker.
T33943 PF-04856264 PF-4856264,PF4856264,PF 4856264
PF-04856264 is a potent and selective human Nav1.7 voltage-gated sodium channel inhibitor (IC50 = 28 nM).
T14201 AM-2099 Others

Compounds

AMTB hydrochloride
T19723
Synonym: AMTB
Target: TRP/TRPV Channel
Phenytoin
T0939
Synonym: Diphenylhydantoin,5,5-Diphenylhydantoin
Target: Virus Protease, Sodium Channel
Evenamide
T15260
Synonym: NW-3509
Target: Sodium Channel
Amifampridine
T4497
Synonym: 3,4-Pyridinediamine,Pyridine-3,4-Diamine,3,4-Diaminopyridine
Target: Others
Phenytoin sodium
T0008
Synonym: 5,5-Diphenylhydantoin sodium salt,Diphantoine,Dilantin sodium,Diphenylhydantoin Sodium
Target: Virus Protease, Sodium Channel
Licarbazepine
T7806
Synonym: ​10,11-hydroxy-10,11 Dihydrocarbamezer
Target: Others
Meclofenamic acid
T11990
Synonym: Meclofenamate
Target: Others, Gap Junction Protein
BTT-266
T60010
Synonym:
Target: Calcium Channel
Etidocaine Hydrochloride
T31716
Synonym: W-19053,Duranest,W19053,W 19053
Target: Sodium Channel
Calcium Channel antagonist 3
T77712
Synonym:
Target: Calcium Channel
Calcium Channel antagonist 4
T77711
Synonym:
Target: Calcium Channel
Co 102862
T22675
Synonym: V 102862
Target: Others, Sodium Channel
Transfluthrin
T9751
Synonym:
Target: Others
PF-06305591
T12424
Synonym: PF-6305591
Target: Others
Lomerizine dihydrochloride
T6571
Synonym: Terranas,Lomerizine 2HCl,Lomerizine hydrochloride,KB-2796
Target: Calcium Channel
Rufinamide
T2523
Synonym: CGP 33101,E 2080,RUF 331
Target: Sodium Channel
UK 78282 hydrochloride
T23497
Synonym:
Target: Potassium Channel
NaV1.7 inhibitor-1
T12181
Synonym:
Target: Sodium Channel
Fosphenytoin disodium
T7066
Synonym: Fosphenytoin sodium,ACC-9653
Target: Sodium Channel
RY785
T12786
Synonym:
Target: Potassium Channel
Primidone
T0024
Synonym: Primaclone,Mysoline,NCI-C56360
Target: GABA Receptor, Sodium Channel, GluR, AChR
Benzocaine xHCl(94-09-7(free base))
T6782L
Synonym:
Target: Sodium Channel
Flosatidil
T68073
Synonym:
Target: Calcium Channel
Phenibut (hydrochloride)
T8639
Synonym: 3-Amino-4-phenylbutyric acid hydrochloride
Target: GABA Receptor
1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride
T77642
Synonym:
Target: Calcium Channel
Prilocaine hydrochloride
T0796
Synonym: Prilocaine HCl,Propitocaine hydrochloride,Xylonest
Target: ATPase, Sodium Channel
1-(2,4-difluorophenyl)guanidine hydrochloride
T50030
Synonym:
Target: Others
Proparacaine hydrochloride
T0222
Synonym: Proparacaine HCl,Proxymetacaine Hydrochloride
Target: Apoptosis, Sodium Channel
Procainamide hydrochloride
T0018
Synonym: Procapan,Procainamide HCl,Pronestyl,Procanbid
Target: DNA Methyltransferase, Sodium Channel, AChR, Autophagy
Mepivacaine
T22361
Synonym: Carbocaine
Target: Sodium Channel
PF 05089771 tosylate
T7502
Synonym:
Target: Sodium Channel
Procaine hydrochloride
T0802
Synonym: Novocaine HCl,Procaine HCl
Target: Histone Demethylase, 5-HT Receptor, DNA/RNA Synthesis, Sodium Channel, NMDAR, AChR
Mexiletine hydrochloride
T1046
Synonym: KOE-1173 (hydrochloride),Mexiletine HCl,KO1173
Target: AhR, Sodium Channel
SAK3
T26174
Synonym: SAK 3,SAK-3
Target: Calcium Channel, AChR
NS309
T4612
Synonym:
Target: EGFR, Potassium Channel, HER
Amiodarone hydrochloride
T1496
Synonym: Amiodar,Amiodarone HCl,Nexterone
Target: Potassium Channel, Adrenergic Receptor, Autophagy
Zonisamide
T0267
Synonym: AD 810,CI 912
Target: Calcium Channel, Sodium Channel, Carbonic Anhydrase
Atosiban acetate
T5148
Synonym: RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164
Target: Oxytocin Receptor, Vasopressin Receptor
Linopirdine dihydrochloride
T22925
Synonym:
Target: Others
Clathrodin
T27040
Synonym:
Target:
KC 12291 hydrochloride
T22887
Synonym:
Target: Others
Propoxycaine hydrochloride
T13830
Synonym:
Target: Sodium Channel
MSD-D
T70139
Synonym:
Target:
Fomocaine HCl
T31843
Synonym: P-652 HCl,Fomocaine,P652 hydrochloride,P-652 hydrochloride,Panacaine hydrochloride,P 652 hydrochloride
Target:
Vincanol
T26319
Synonym: Vincanolum
Target:
HENA
T24137
Synonym:
Target:
photoGBI1
T69866
Synonym:
Target:
Saxitoxinol
T68748
Synonym:
Target:
PF-04856264
T33943
Synonym: PF-4856264,PF4856264,PF 4856264
Target:
AM-2099
T14201
Synonym:
Target: Others
1 2 3
カタログ番号 製品名 別名 ターゲット
T2173 Veratridine Sodium Channel
Veratridine is a benzoate-cevane found in Veratrum and Schoenocaulon. It activates sodium channels to stay open longer than normal.
T3013 Catharanthine tartrate Catharanthine hemitartrate Others , Calcium Channel
Catharanthine tartrate (Catharanthine hemitartrate) is an alkaloid from periwinkle that inhibits voltage-gated L-type calcium channels and has antitumor and hypotensive activities.
T3021 Bulleyaconitine A Bulleyaconi cine A Sodium Channel
Bulleyaconitine A (Bulleyaconi cine A), an analgesic and antiinflammatory drug isolated from Aconitum plants, has several potential targets, such as voltage-gated Na+ channels.
TN6713 6-Benzoylheteratisine Heteratisan-14-one, 6-(benzoyloxy)-20-ethyl-8-hydroxy-1-methoxy-4-meth Sodium Channel
6-Benzoylheteratisine (Heteratisan-14-one, 6-(benzoyloxy)-20-ethyl-8-hydroxy-1-methoxy-4-meth) is a Aconitum alkaloid. It can inhibits voltage-gated Na+ channels in rat brain synaptosomes
T4S1869 12-Epinapelline Others
12- Epinapelline is a diterpene alkaloid which displays anaesthetic activity as toxic neurological agents. Similar to aconitine, its suggested that modulation of voltage gated Na+ channels are responsible for these obser...
TN2347 Methylsticin Methysticin Others
Methysticin is a kavalactone isolated from the kava roots. Methylsticin (Methysticin) exhibit osteoclast formation inhibitory activity. It inhibits activation of NF-χB in lung adenocarcinoma tissue, activates Nrf2 in neu...
T8716 Physalin F Apoptosis
Physalin F is a natural blocker of CaV2.3 (R-type) and CaV2.2 (N-type) voltage-gated calcium channels.It is a secosteroid with potent anti-inflammatory and immunomodulatory activities. Physalin F induces apoptosis of PBM...
TN2322 Yangambin Calcium Channel , PAFR
Yangambin is a selective antagonist of the cardiovascular effects of platelet activating factor (PAF); it has hypotensive effect, which is probably due to a peripheral vasodilatation that involves, at least, the inhibiti...
TN1254 3'-Methoxydaidzein Sodium Channel
3'-Methoxydaidzein is a dual isoflavone and Sodium Channel inhibitor. 3'-Methoxydaidzein inhibited NaV1.7, NaV1.8 and NaV1.3 with IC50 of 181 nM, 397 nM and 505 nM, respectively. 3'-Methoxydaidzein was specific for colla...
T10609 Brevetoxin-3 PbTx-3 Others
T27564 Hymenidin 5-HT Receptor
Hymenidin, an alkaloid isolated from the Okinawan sponge Hymeniacidon sp. is a 5-hydroxytryptaminergic receptor antagonist and voltage-gated potassium channel inhibitor with potential antiprotozoal effects.It selectively...
T36068 Brevetoxin B
Brevetoxin B is a polyketide neurotoxin produced by Karenia species and other dinoflagellates. It binds to site 5 on the alpha subunit of voltage-gated sodium channels (IC50 = 15 nM) on neurons at the neuromuscular junct...

天然物製品

Veratridine
T2173
Synonym:
Target: Sodium Channel
Catharanthine tartrate
T3013
Synonym: Catharanthine hemitartrate
Target: Others, Calcium Channel
Bulleyaconitine A
T3021
Synonym: Bulleyaconi cine A
Target: Sodium Channel
6-Benzoylheteratisine
TN6713
Synonym: Heteratisan-14-one, 6-(benzoyloxy)-20-ethyl-8-hydroxy-1-methoxy-4-meth
Target: Sodium Channel
12-Epinapelline
T4S1869
Synonym:
Target: Others
Methylsticin
TN2347
Synonym: Methysticin
Target: Others
physalin F
T8716
Synonym:
Target: Apoptosis
Yangambin
TN2322
Synonym:
Target: Calcium Channel, PAFR
3'-Methoxydaidzein
TN1254
Synonym:
Target: Sodium Channel
Brevetoxin-3
T10609
Synonym: PbTx-3
Target: Others
Hymenidin
T27564
Synonym:
Target: 5-HT Receptor
Brevetoxin B
T36068
Synonym:
Target:

Recombinant Proteins

Species：
Human (13)
Anemonia sulcata (1)
Guinea pig (1)
Expression System：
E. coli (8)
HEK293 Cells (6)
P. pastoris (Yeast) (1)
Tag：
C-hFc (3)
N-6xHis (3)
N-His (3)
C-His (2)
N-10xHis (2)
N-10xHis, C-Myc (1)
N-6xHis-SUMO (1)
カタログ番号 製品名 Species Expression System
TMPY-03697 SCN2B Protein, Human, Recombinant (His) Human HEK293 Cells
SCN2B Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 34.7 kDa and the accession number is O60939.
TMPY-03183 SCN2B Protein, Human, Recombinant (hFc) Human HEK293 Cells
SCN2B Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.2 kDa and the accession number is O60939.
TMPY-02976 SCN3B Protein, Human, Recombinant (His) Human HEK293 Cells
SCN3B Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 17.2 kDa and the accession number is Q9NY72.
TMPY-02722 SCN3B Protein, Human, Recombinant (hFc) Human HEK293 Cells
SCN3B Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.5 kDa and the accession number is Q9NY72.
TMPH-02308 CACNA2D1 Protein, Human, Recombinant (His & SUMO) Human E. coli
The alpha-2/delta subunit of voltage-dependent calcium channels regulates calcium current density and activation/inactivation kinetics of the calcium channel. Plays an important role in excitation-contraction coupling.
TMPH-00780 CACNA1C Protein, Guinea Pig, Recombinant (His) Guinea pig E. coli
Pore-forming, alpha-1C subunit of the voltage-gated calcium channel that gives rise to L-type calcium currents. Mediates influx of calcium ions into the cytoplasm, and thereby triggers calcium release from the sarcoplasm...
TMPY-02245 SNAP-25 Protein, Human, Recombinant (His) Human E. coli
Synaptosomal-associated protein 25, also known as Super protein, Synaptosomal-associated 25 kDa protein, SNAP25 and SNAP, is a cytoplasm and cell membrane protein that belongs to the SNAP-25 family. SNAP25 / SUP contains...
TMPY-03615 CSEN Protein, Human, Recombinant (His) Human E. coli
KCNIP3 (Potassium Voltage-Gated Channel Interacting Protein 3, also known as CSEN) is a Protein Coding gene. CSEN is a member of the family of voltage-gated potassium (Kv) channel-interacting proteins, which belong to th...
TMPH-01609 LGI1 Protein, Human, Recombinant (His & Myc) Human E. coli
Regulates voltage-gated potassium channels assembled from KCNA1, KCNA4 and KCNAB1. It slows down channel inactivation by precluding channel closure mediated by the KCNAB1 subunit. Ligand for ADAM22 that positively regula...
TMPH-03751 CYBB Protein, Human, Recombinant (His) Human E. coli
Critical component of the membrane-bound oxidase of phagocytes that generates superoxide. It is the terminal component of a respiratory chain that transfers single electrons from cytoplasmic NADPH across the plasma membr...
TMPH-01744 NOX1 Protein, Human, Recombinant (His) Human E. coli
NOH-1S is a voltage-gated proton channel that mediates the H(+) currents of resting phagocytes and other tissues. It participates in the regulation of cellular pH and is blocked by zinc. NOH-1L is a pyridine nucleotide-d...
TMPH-01394 GRIN1 Protein, Human, Recombinant (His) Human E. coli
Component of NMDA receptor complexes that function as heterotetrameric, ligand-gated ion channels with high calcium permeability and voltage-dependent sensitivity to magnesium. Channel activation requires binding of the ...
TMPJ-00587 NRCAM Protein, Human, Recombinant (hFc) Human HEK293 Cells
Neuronal cell adhesion molecule(NRCAM) is a single-pass type I membrane protein ,containing 5 fibronectin type-III domains and 6 Ig-like C2-type (immunoglobulin-like) domains.It belongs to the immunoglobulin superfamily....
TMPH-00056 Delta-AITX-Avd1c Protein, Anemonia sulcata, Recombinant (His) Anemonia sulcata P. pastoris (Yeast)
Binds specifically to voltage-gated sodium channels (Nav) (site 3), thereby delaying their inactivation. Has a strong effect on crustaceans and insects (DmNav1) and a weaker effect on mammals. This toxin is highly potent...
TMPY-01854 DPP10 Protein, Human, Recombinant (His) Human HEK293 Cells
Inactive dipeptidyl peptidase 1, also known as Dipeptidyl peptidase IV-related protein 3, Dipeptidyl peptidase X, Dipeptidyl peptidase-like protein 2, DPRP-3, DPL2 and DPP1, is a single-pass type II membrane protein w...
カタログ番号 製品名
L7400 Sodium Channel Blocker Library

118 compounds
A unique collection of 118 sodium channel blockers and agonists for high throughput and high content screening;

ライブラリー

Sodium Channel Blocker Library
L7400
Compounds: 118
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