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カタログ番号	製品名	別名	ターゲット
T9741	INE963		Others
	INE963 demonstrates potent cellular activity against Pf 3D7 (EC50 = 6 nM) and achieves "artemisinin-like" kill kinetics in vitro with a parasite clearance time of <24 h. INE963 is also potent against P. falciparum and P....		Others
T1491	Atovaquone	Atavaquone	Others , P450 , Dehydrogenase , Antibiotic , Parasite
	Atovaquone (Atavaquone) is a hydroxynaphthoquinone that has antimicrobial activity and is being used in antimalarial protocols.		Others , P450 , Dehydrogenase , Antibiotic , Parasite
T8767	PfDHODH-IN-2		Dehydrogenase , Parasite
	PfDHODH-IN-2 is a dihydrothiophenone derivative, is a potent Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH, IC50 : 1.11 μM) inhibitor . It is used an antimalarial agent and can be used for the research of m...		Dehydrogenase , Parasite
T12909	SID 26681509		Cysteine Protease , Parasite
			Cysteine Protease , Parasite
T4264	Takinib	EDHS-206	Apoptosis , MAPK
	Takinib (EDHS-206) is a specific and effective TAK1 inhibitor(IC50= 9.5 nM).		Apoptosis , MAPK
T0850	Primaquine diphosphate	Primaquine phosphate,Primaquine bisphosphate	Antibiotic , Parasite
	Primaquine diphosphate is the phosphate salt form of primaquine, a synthetic, 8-aminoquinoline derivative with antimalarial properties. Although its mechanism of action is unclear, primaquine bind to and alter the proper...		Antibiotic , Parasite
T12908	SIBA	5'-Deoxy-5'-isobutylthioadenosine,5'-Isobutylthioadenosine	Nucleoside Antimetabolite/Analog , HSV
	SIBA (5'-Deoxy-5'-isobutylthioadenosine) is a synthetic analogue of SAH, acts as an inhibitor of S-adenosylmethionine-mediated transmethylation. SIBA can interfere with a variety of enzymatic activities in vitro, such as...		Nucleoside Antimetabolite/Analog , HSV
T16269	Nanaomycin A		DNA Methyltransferase , Dehydrogenase , Parasite
	Nanaomycin A is the first selective DNMT3B inhibitor (IC50: 500 nM). Nanaomycin A inhibits in vitro growth of the human malaria parasite Plasmodium falciparum (IC80: 33.1 nM). Nanaomycin A is quinone antibiotics, reactiv...		DNA Methyltransferase , Dehydrogenase , Parasite
T79535	Antimalarial agent 30		Parasite
	Antimalarial agent 30 has anti-Plasmodium berghei liver stage parasite activity and antimalarial activity for the study of malarial infections.		Parasite
T10336	Antimalarial agent 1		Parasite
	Antimalarial agent 1 is an effective antimalarial agent.		Parasite
T9984	Antimalarial agent 13	N2-(3-chlorophenyl)-N4-(furan-2-ylmethyl)quinazoline-2,4-diamine	Parasite
	Antimalarial agent 13 (N2-(3-chlorophenyl)-N4-(furan-2-ylmethyl)quinazoline-2,4-diamine) is a potent antimalarial agent.		Parasite
T22381	Antimalarial agent 14	4-hydroxy-3-phenyl-naphthalene-1,2-dione,2-Hydroxy-3-phenyl-1,4-naphthoquinone	Others
	Antimalarial agent 14 (NSC-102533) is a bioactive chemical.		Others
T62936	Antimalarial agent 8
	Antimalarial agent 8 (Compound 7e) is a novel, orally active antimalarial agent that is effective against P. falciparum in vitro and effective orally in an in vivo mouse model of malaria (40 mg/kg).
T63043	Antimalarial agent 2
	Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.
T78952	Antimalarial agent 26		Parasite
	Antimalarial agent 26, a derivative of 1,4-naphthoquinones, demonstrates antimalarial properties through oral administration. It exhibits cytotoxic effects on P. falciparum while maintaining selectivity against mammalian...		Parasite
T72416	Antimalarial agent 18
	Antimalarial agent 18, a powerful antimalarial compound characterized by its electronic, highly lipophilic, and siderophoric properties, falls within the acyloxymethyl series, acting as a fosmidomycin surrogate. It effec...
T72396	Antimalarial agent 20
	Antimalarial agent 20, exhibiting potent efficacy with an IC50 value of 0.6 nM against the P. falciparum NF54 parasite strain within the NF54 albumax assay, serves as a significant antimalarial compound.
T63655	Antimalarial agent 9
	Antimalarial agent 9 is an effective antimalarial agent, a quinoline-imidazole derivative compound. antimalarial agent 9 showed significant in vitro antimalarial effects against CQ-susceptible strains (IC50-0.14 μM) and ...
T63595	Antimalarial agent 16
	Antimalarial agent 16 is a parasite inhibitor that exhibits antimalarial effects and inhibits the growth of Plasmodium falciparum with an IC50 value of 2.0 nM.
T62537	Antimalarial agent 7
	Antimalarial agent 7 is a potent and effective inhibitor of PfATP4. Antimalarial agent 7 has potential for the study of the human plasmodium falciparum.
T62300	Antimalarial agent 11
	Antimalarial agent 11 (compound 1) is a potent antimalarial agent, a spirocyclic chromane. Antimalarial agent 11 is able to act on D6 (EC50: 1.48 μM) and ARC08-022 (EC50: 1.81 μM).
T78951	Antimalarial agent 24		Parasite
	Compound 24 (Compound 7), an in vitro antimalarial agent, demonstrates inhibitory activity against the Plasmodium falciparum W2 strain with an IC50 of 0.81 μM and exhibits a cytotoxicity threshold (CC50) exceeding 200 μM...		Parasite
T79534	Antimalarial agent 29		Parasite
	Compound 29 (also known as Compound 16) is an antimalarial agent that demonstrates inhibition of the P. berghei liver stage parasite load, exhibiting an effective concentration (EC50) of 5.2 μM [1].		Parasite
T75067	Antimalarial agent 19		Parasite
	Antimalarial agent 19 (compound 6e) exhibits antimalarial activity against the blood stages of P. falciparum K1 and P. berghei, with EC50 values of 0.3 µM and 15.3 µM, respectively. It demonstrates good aqueous solubilit...		Parasite
T74845	Antimalarial agent 23
	Antimalarial agent 23, a benzimidazole-based compound, exhibits potent antimalarial activity, demonstrated by its low IC50 values of 0.08 μM for PfNF54 and 0.10 μM for PfK1, respectively. This compound effectively inhibi...
T79335	Antimalarial agent 31		Parasite
	Compound 31 (compound 7k) is an orally active inhibitor of Plasmodium falciparum aspartic protease, plasmepsin X (PMX), with antimalarial properties [1].		Parasite
T61200	Antimalarial agent 3
	Antimalarial agent 3, an antimalarial agent, exhibits potent activity against Plasmodium with an IC50 of 0.035 μM. Furthermore, it demonstrates an exceptionally high selectivity index in relation to mammalian cells.
T83044	Antimalarial agent 33		Parasite
	Antimalarial agent 33 (compound 5g) exhibits antiplasmodial activity targeting both erythrocytic and hepatic stages of Plasmodium, with an effective concentration (EC50) of 1.1 μM against the K1 strain of P. falciparum. ...		Parasite
T74695	Antimalarial agent 17
	Antimalarial agent 17, functioning both as an antimalarial agent and a herbicide, inhibits photosystem II and demonstrates post-emergence herbicidal efficacy comparable to commercial herbicides [1].
T78936	Antimalarial agent 27		Parasite
	Antimalarial agent 27 (compound 11a) potently inhibits P. falciparum with an IC50 of 0.37 μM and targets the parasite's 1-deoxy-D-xylulose-5-phosphate reductoisomerase (DXR) enzyme with an IC50 of 0.11 μM, indicating its...		Parasite
T79460	Antimalarial agent 28		Parasite
	Antimalarial agent 28 (Compound 2i) acts as an antiplasmodial agent, exhibiting inhibition of P. berghei with IC50 values of 0.561 μM for the liver stage, 0.14 μM for early gametocytes, and 4.34 μM for the ring stages of...		Parasite
T63052	Antimalarial agent 10
	Antimalarial agent 10 (Compound 17b) is an amino alcohol-quinoline compound. Antimalarial agent 10 is also an antimalarial agent capable of acting on Pf3D7 (IC50: 14.9 nM) and PfW2 (IC50: 11 nM) with a selectivity index ...
T63456	Antimalarial agent 12
	Antimalarial agent 12 is an effective antimalarial agent that inhibits the growth of Plasmodium falciparum strains Dd2 and 3D7 with EC50 values of 155 nM and 136 nM, respectively. antimalarial agent 12 has a MIC >250,000...
T63413	Antimalarial agent 15
	Antimalarial agent 15 is a parasite inhibitor that exhibits antimalarial effects and inhibits the growth of Plasmodium falciparum 3D7 with an IC50 value of 20 nM.
T17313	(+)-SJ733	SJ000557733	ATPase , Parasite
	(+)-SJ733 (SJ000557733) is a potent Na+-ATPase PfATP4 inhibitor with antimalarial activity for the study of malaria.		ATPase , Parasite
T74696	SpdSyn binder-1		Parasite
	SpdSyn binder-1 is a weak binding agent that binds to the active site of Plasmodium falciparum spermidine synthase, which is partially inhibitory to malaria and can be used to study malaria.		Parasite
T9004	TM2-115		Parasite
	TM2-115 is a inhibitor of malaria parasite histone methyltransferases that results in rapid and irreversible parasite death [1].		Parasite
T35903	N-acetyl Dapsone		Antibacterial , Parasite
	N-acetyl Dapsone is an anti-inflammatory and antimicrobial compound widely used in the treatment of leprosy, malaria, acne and various immune disorders.		Antibacterial , Parasite
T0860	Mefloquine hydrochloride	Mefloquin hydrochloride,Mefloquine HCl	Potassium Channel , SARS-CoV , Reactive Oxygen Species , Parasite , Autophagy
	Mefloquine hydrochloride (Mefloquin hydrochloride) is a quinoline derivative used for the prevention and therapy of P. falciparum malaria.
T8381	Amodiaquine		Others , Histone Methyltransferase , Parasite
	Amodiaquine is a synthetic aminoquinoline, used to treat malaria.		Others , Histone Methyltransferase , Parasite
T5916	Fmoc-N-Me-Phe-OH	Fmoc-N-methyl-L-phenylalanine	Others , Parasite
	Fmoc-N-Me-Phe-OH (Fmoc-N-methyl-L-phenylalanine) is a Malaria Parasite inhibitor.		Others , Parasite
T5493	Pyronaridine		Others
	Pyronaridine is an orally active, mannitol-containing anti-malarial compound that acts by interfering with the replication of the malaria parasite (Plasmodium) within red blood cells. Pyronaridine is often used in combin...		Others
T0026	Sulfalene	Sulfalene(SMPZ),Sulfalen,SMP2,Butadiene sulfone,AS-18908,Sulfametopyrazine,3-Sulfolene	Antibacterial , Antibiotic , Parasite , Autophagy
	Sulfalene (SMP2), a long-acting sulfonamide antibiotic, is used for the therapy of chronic bronchitis, urinary tract infections, and malaria.		Antibacterial , Antibiotic , Parasite , Autophagy
T15173	DSM265	PfSPZ	Dehydrogenase , Parasite
	DSM265 (PfSPZ) is a dihydroorotic acid dehydrogenase inhibitor with antimalarial activity (IC50: 8.9 nM).DSM265 inhibits the growth of Pf3D7 parasites and can be used for the treatment and prophylaxis of malaria infectio...		Dehydrogenase , Parasite
T7195	GSK369796 Dihydrochloride	N-tert-butylisoquine	Potassium Channel , Parasite
	GSK369796 Dihydrochloride (N-tert-butylisoquine),is an anti-malaria drug candidate. is an affordable and effective antimalarial and inhibits hERG potassium ion channel repolarization(IC50 of 7.5 μM)		Potassium Channel , Parasite
T77684	4-(2-Aminoethyl)amino-7-chloroquinoline	N1-(7-Chloroquinolin-4-yl)ethane-1,2-diamine	Parasite
	4-(2-Aminoethyl)amino-7-chloroquinoline (N1-(7-Chloroquinolin-4-yl)ethane-1,2-diamine) has potential anthelmintic and antitumor activity for the study of malaria.		Parasite
T67694	ZY-19489		Parasite
	ZY-19489 is an antimalarial compound that is a potential single-dose cure for Plasmodium falciparum and Plasmodium vivax malaria. It has received orphan drug designation from the FDA.		Parasite
T4382	Proguanil hydrochloride	Paludrine hydrochloride,Chlorguanide hydrochloride,Chloroquanil	Others , Dehydrogenase , DNA/RNA Synthesis , Antifolate , Parasite
	Proguanil hydrochloride (Chloroquanil) is a biguanide compound which metabolizes in the body to form cycloguanil, an anti-malaria agent.Upon hydrolysis, Proguanil hydrochloride is converted to its active cyclic triazine ...
T27214	DSM421	DSM 421,DSM-421	Dehydrogenase
	DSM421 (DSM-421) is a dihydrodehydrogenase inhibitor (DHODH) that is in preclinical development as a potential treatment option for malaria and has shown activity against field isolates of both P. falciparum and P. vivax...		Dehydrogenase
T0860L	Mefloquine	Ro215998,WR 142490,Ro-215998,Lariam,Ro 215998	Others
	Mefloquine (Ro 215998), a quinoline antimalarial agent, is an anti-SARS-CoV-2 entry inhibitor. Mefloquine is also a K+ channel (KvQT1/minK) antagonist with an IC50 of ~1 μM. Mefloquine can be used for malaria, systemic l...		Others

Compounds

Target: Others, P450, Dehydrogenase, Antibiotic, Parasite

PfDHODH-IN-2

T8767

Synonym:

Target: Dehydrogenase, Parasite

SID 26681509

T12909

Synonym:

Target: Cysteine Protease, Parasite

Takinib

T4264

Synonym: EDHS-206

Target: Apoptosis, MAPK

Primaquine diphosphate

T0850

Synonym: Primaquine phosphate,Primaquine bisphosphate

Target: Antibiotic, Parasite

SIBA

T12908

Synonym: 5'-Deoxy-5'-isobutylthioadenosine,5'-Isobutylthioadenosine

Target: Nucleoside Antimetabolite/Analog, HSV

Nanaomycin A

T16269

Synonym:

Target: DNA Methyltransferase, Dehydrogenase, Parasite

Antimalarial agent 30

Antimalarial agent 13

T9984

Synonym: N2-(3-chlorophenyl)-N4-(furan-2-ylmethyl)quinazoline-2,4-diamine

Target: Parasite

Antimalarial agent 14

T22381

Synonym: 4-hydroxy-3-phenyl-naphthalene-1,2-dione,2-Hydroxy-3-phenyl-1,4-naphthoquinone

Antimalarial agent 26

T78952

Synonym:

Target: Parasite

Antimalarial agent 18

T72416

Synonym:

Target:

Antimalarial agent 20

Antimalarial agent 16

Antimalarial agent 11

T62300

Synonym:

Target:

Antimalarial agent 24

T78951

Synonym:

Target: Parasite

Antimalarial agent 29

T79534

Synonym:

Target: Parasite

Antimalarial agent 19

T75067

Synonym:

Target: Parasite

Antimalarial agent 23

T74845

Synonym:

Target:

Antimalarial agent 31

Antimalarial agent 33

T83044

Synonym:

Target: Parasite

Antimalarial agent 17

T74695

Synonym:

Target:

Antimalarial agent 27

T78936

Synonym:

Target: Parasite

Antimalarial agent 28

T79460

Synonym:

Target: Parasite

Antimalarial agent 10

T63052

Synonym:

Target:

Antimalarial agent 12

T63456

Synonym:

Target:

Antimalarial agent 15

Target: ATPase, Parasite

Target: Antibacterial, Parasite

Mefloquine hydrochloride

T0860

Synonym: Mefloquin hydrochloride,Mefloquine HCl

Target: Potassium Channel, SARS-CoV, Reactive Oxygen Species, Parasite, Autophagy

Amodiaquine

T8381

Synonym:

Target: Others, Histone Methyltransferase, Parasite

Fmoc-N-Me-Phe-OH

T5916

Synonym: Fmoc-N-methyl-L-phenylalanine

Target: Others, Parasite

Synonym: Sulfalene(SMPZ),Sulfalen,SMP2,Butadiene sulfone,AS-18908,Sulfametopyrazine,3-Sulfolene

Target: Antibacterial, Antibiotic, Parasite, Autophagy

DSM265

T15173

Synonym: PfSPZ

Target: Dehydrogenase, Parasite

GSK369796 Dihydrochloride

T7195

Synonym: N-tert-butylisoquine

Target: Potassium Channel, Parasite

4-(2-Aminoethyl)amino-7-chloroquinoline

T77684

Synonym: N1-(7-Chloroquinolin-4-yl)ethane-1,2-diamine

Proguanil hydrochloride

T4382

Synonym: Paludrine hydrochloride,Chlorguanide hydrochloride,Chloroquanil

Target: Others, Dehydrogenase, DNA/RNA Synthesis, Antifolate, Parasite

DSM421

T27214

Synonym: DSM 421,DSM-421

Target: Dehydrogenase

Mefloquine

T0860L

Synonym: Ro215998,WR 142490,Ro-215998,Lariam,Ro 215998

Target: Others

カタログ番号	製品名	別名	ターゲット
T0690	Quinine		Potassium Channel , Platelet aggregation , Parasite
	Quinine is a natural cinchona alkaloid that has been used for centuries in the prevention and therapy of malaria. Quinine is also used for idiopathic muscle cramps. Quinine therapy has been associated with rare instances...		Potassium Channel , Platelet aggregation , Parasite
T7938	Quinidine		Parasite
	Quinidine is a stereoisomer of the antimalarial agent quinine and a class Ia antiarrhythmic agent. for the treatment of abnormal heart rhythms and also malaria.		Parasite
T6447	Clindamycin	Clinimycin,Sobelin,Chlolincocin	Antibacterial , Antibiotic
	Clindamycin (Sobelin) dissociates peptidyl-tRNA from the bacterial ribosome, thereby disrupting bacterial protein synthesis. Clindamycin is a semisynthetic broad-spectrum antibiotic produced by chemical modification of t...		Antibacterial , Antibiotic
T8689	Chloroquine	CQ	SARS-CoV , TLR , HIV Protease , Antibiotic , Parasite , Autophagy
	Chloroquine is a Toll-like receptor inhibitor that inhibits autophagy. Chloroquine has anti-malarial and anti-inflammatory activity and is widely used in the treatment of malaria and rheumatoid arthritis. Chloroquine als...
T0194	Chloroquine phosphate	Chloroquine diphosphate,Aralen phosphate,Chingamin phosphate	SARS-CoV , TLR , HIV Protease , Antibiotic , Parasite , Autophagy
	Chloroquine phosphate (Aralen phosphate) is an aminoquinoline antimalarial and also is widely used as an autophagy inhibitor. Chloroquine also is an inhibitor of toll-like receptors (TLRs).
T8125	Quinidine sulfate dihydrate	Chinidin Sodium,β-quinine Sodium,Pitayine Sodium,Quinidine sulfate	P450
	Quinidine sulfate dihydrate (Pitayine Sodium) is a potent and selective cytochrome P450db inhibitor		P450
T6631	Quinine hydrochloride dihydrate	Quinine HCl Dihydrate	Potassium Channel , Parasite
	Quinine hydrochloride dihydrate (Quinine HCl Dihydrate) is a white crystalline K+ channel blocker, used to treat malaria.		Potassium Channel , Parasite
TN1012L	Febrifugine dihydrochloride	ISF-2123,Propyldazine hydrochloride,Atensil,(+)-Febrifugine dihydrochloride,Pildralazine dihydrochloride	Parasite
	Febrifugine dihydrochloride (Propyldazine hydrochloride) is a biochemical with therapeutic activity regarding malaria, cancer, fibrosis and inflammatory diseases.		Parasite
T1323	Artemether	SM224,Dihydroartemisinin methyl ether,Dihydroqinghaosu methyl ether,CGP 56696	Antibiotic , Parasite
	Artemether (CGP 56696) is an antimalarial agent used to treat acute uncomplicated malaria.		Antibiotic , Parasite
T4S1519	Pseudoginsenoside RT5		Others
	1. Pseudoginsenoside RT5 has anti-epilepsy, anti-depressant activity by promoting nerve growth and improve cognitive ability. 2. Pseudoginsenoside RT5 has anti-bacterial, anti-tumor and anti-malaria activities.		Others
TN1568	Deoxyartemisinin	2-deoxyartemisinin	Antifection
	Deoxyartemisinin (2-deoxyartemisinin), a compound derived from Artemisia annua, has anti-inflammatory and anti-ulcer effects and is used in the study of malaria.		Antifection
T20754	Deltamethrin	Butoss,RU-22974,Esbecythrin,K-Othrin,Decamethrin,RU 22974	Others
	Deltamethrin (RU 22974), a neurotoxic pyrethroid insecticide, produces a reversible sequence of motor symptoms in rats involving hind limb rigidity and choreoathetosis.Deltamethrin is globally used in crop protection, co...		Others
THS1455	DihydroarteMisinic acid	Dihydro-Artmisinic Acid	Ferroptosis , Parasite
	DihydroarteMisinic acid (Dihydro-Artmisinic Acid) is a natural product from Artemisia annua and the main direct precursor of artemisinin, which is a medicinal herb that is widely used to treat Malaria.		Ferroptosis , Parasite
TN7082	Demethyldaphnoretin-7-O-glucoside		Others
	Demethyldaphnoretin-7-O-glucoside is a natural product that is isolated from Daphne oleoides Schreber subsp. kurdica (DOK). In Turkish traditional medicine, the aerial parts of DOK have been used to treat malaria, rheuma...		Others
T0433	Artesunate	WR-256283	Virus Protease , Ferroptosis , STAT , Parasite
	Artesunate (WR-256283) is part of the artemisinin group of drugs that treat malaria. It is a semi-synthetic derivative of artemisinin that is water-soluble and may therefore be given by injection. It is on the World Heal...		Virus Protease , Ferroptosis , STAT , Parasite
TN7225	2'-Hydroxy-3,4-dimethoxychalcone		Antioxidant , Parasite
	2'-Hydroxy-3,4-dimethoxychalcone, a chalcone compound isolated from the roots of Sophora japonica, has antioxidant activity and inhibited the intracellular survival of Lactobacillus donovani Parasite EC.50 Values ranged ...		Antioxidant , Parasite
T9279	Nerolidol acetate		Others
	Nerolidol acetate is a natural sesquiterpene with anti-cancer, anti-inflammatory, antibacterial and anti-insect activities. Nerolidol acetate can inhibit parasite activity and inhibit schistosomiasis, nematodes, malaria,...		Others
TN3151	6-Acetonyl-N-methyl-dihydrodecarine		Antifection
	6-Acetonyl- N -methyl-dihydrodecarine has mosquito larvicidal activity against the malaria vector Anopheles gambiae.		Antifection
TN4314	Isonardoperoxide		Antifection
	Isonardoperoxide shows strong antimalarial activity against Plasmodium falciparum malaria (6.0 × 10-7 M).		Antifection
TN5327	11(13)-Dehydroivaxillin
	11(13)-Dehydroivaxillin possesses a promising antiplasmodial activity, which can be exploited in malaria therapy.
T10685	Carpaine		Others
	Carpaine, an alkaloid isolated from Carica papaya Linn, has anti-thrombocytopenic activity. It has the anti-plasmodial activity to prevent malaria.		Others
T25579	Kijanimicin	Kijanimicin sodium salt
	Kijanimicin is an antitumor and antibiotic. It is a unique, large acid enol antibiotic and possesses an unusual in vitro spectrum of activity against some Gram-positive and anaerobic microorganisms. It has also shown int...
TN4666	Norcaesalpinin E		Antifection
	Norcaesalpinin E shows antimalarial activity against the malaria parasite Plasmodium falciparum FCR-3/A2 clone in vitro, with an IC50 value of 0.090 microM.		Antifection
T11802	L-Canaline		Others
	L-Canaline, a nonprotein amino acid found in many leguminous plants, exhibits potent anticancer and antiproliferative effects. It effectively inhibits the growth of the malaria parasite Plasmodium falciparum with an IC50...		Others
T21266	Quinine sulfate
	Quinidine is an antiarrhythmic agent. Quinidine is a potent, orally active, selective cytochrome P450db inhibitor. Quinidine is also a blocker of K + channel with an IC 50 of 19.9 μM. Quinidine has potential to be used ...

天然物製品

Quinine

T0690

Synonym:

Target: Potassium Channel, Platelet aggregation, Parasite

Synonym: Clinimycin,Sobelin,Chlolincocin

Target: Antibacterial, Antibiotic

Chloroquine

T8689

Synonym: CQ

Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy

Chloroquine phosphate

T0194

Synonym: Chloroquine diphosphate,Aralen phosphate,Chingamin phosphate

Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy

Quinidine sulfate dihydrate

T8125

Synonym: Chinidin Sodium,β-quinine Sodium,Pitayine Sodium,Quinidine sulfate

Target: P450

Quinine hydrochloride dihydrate

T6631

Synonym: Quinine HCl Dihydrate

Target: Potassium Channel, Parasite

Febrifugine dihydrochloride

TN1012L

Synonym: ISF-2123,Propyldazine hydrochloride,Atensil,(+)-Febrifugine dihydrochloride,Pildralazine dihydrochloride

Target: Parasite

Artemether

T1323

Synonym: SM224,Dihydroartemisinin methyl ether,Dihydroqinghaosu methyl ether,CGP 56696

Target: Antibiotic, Parasite

Pseudoginsenoside RT5

Synonym: 2-deoxyartemisinin

Target: Antifection

Deltamethrin

T20754

Synonym: Butoss,RU-22974,Esbecythrin,K-Othrin,Decamethrin,RU 22974

Target: Others

DihydroarteMisinic acid

THS1455

Synonym: Dihydro-Artmisinic Acid

Target: Ferroptosis, Parasite

demethyldaphnoretin-7-O-glucoside

Target: Virus Protease, Ferroptosis, STAT, Parasite

2'-Hydroxy-3,4-dimethoxychalcone

TN7225

Synonym:

Target: Antioxidant, Parasite

6-Acetonyl-N-methyl-dihydrodecarine

11(13)-Dehydroivaxillin

Synonym: Kijanimicin sodium salt

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-04180	PfLDH Protein, P. falciparum, Recombinant (His)	P. falciparum	E. coli
	Plasmodium falciparum lactate dehydrogenase (PfLDH) is a key enzyme for energy generation of malarial parasites and is considered to be a potential antimalarial target. The ability of PfLDH- or PfIDEh-based immuno-PCR as...
TMPY-01445	CD36 Protein, Mouse, Recombinant (His)	Mouse	HEK293
	The cluster of differentiation (CD) system is commonly used as cell markers in Immunophenotyping. Different kinds of cells in the immune system can be identified through the surface CD molecules associating with the immu...
TMPY-01282	CD36 Protein, Human, Recombinant (His)	Human	HEK293
	The cluster of differentiation (CD) system is commonly used as cell markers in Immunophenotyping. Different kinds of cells in the immune system can be identified through the surface CD molecules associating with the immu...
TMPY-04765	PKLR Protein, Human, Recombinant (His)	Human	E. coli
	Pyruvate kinase (PKLR) is a critical erythrocyte enzyme that is required for glycolysis and production of ATP. Pyruvate kinase deficiency (PKD) is the most frequent red blood cell enzyme abnormality of the glycolytic pat...
TMPY-02696	IgG3 Protein, Mouse, Recombinant	Mouse	HEK293
	IGHG3 (Immunoglobulin Heavy Constant Gamma 3 (G3m Marker), also known as IgG3) is a Protein Coding gene. Ig gamma-3 chain C region is a protein that in humans is encoded by the IGHG3 gene. Immunoglobulins, also known as ...
TMPY-03399	KLHL2 Protein, Human, Recombinant (GST)	Human	E. coli
	KLHL2 (Kelch Like Family Member 2) is a Protein Coding gene. 3 alternatively spliced human isoforms have been reported. KLHL2 contains 1 BTB (POZ) domain and 6 Kelch repeats. It is widely expressed in the brain, esophagu...
TMPY-03985	Adenosine Deaminase Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	Adenosine Desaminase (ADA) deficiency, is a purine metabolic disorder that cause severe combined immunodeficiency (SCID) due to the accumulation of toxic metabolites that primarily affects development, differentiation a...
TMPY-02895	IgG3 Protein, Human, Recombinant	Human	HEK293
	IGHG3 (Immunoglobulin Heavy Constant Gamma 3 (G3m Marker), also known as IgG3) is a Protein Coding gene. Ig gamma-3 chain C region is a protein that in humans is encoded by the IGHG3 gene. Immunoglobulins, also known as ...
TMPY-01449	CD36 Protein, Mouse, Recombinant (His & hFc)	Mouse	HEK293
	The cluster of differentiation (CD) system is commonly used as cell markers in Immunophenotyping. Different kinds of cells in the immune system can be identified through the surface CD molecules associating with the immu...
TMPY-03479	CD36 Protein, Rhesus, Recombinant (hFc)	Rhesus	HEK293
	The cluster of differentiation (CD) system is commonly used as cell markers in Immunophenotyping. Different kinds of cells in the immune system can be identified through the surface CD molecules associating with the immu...
TMPY-03242	CD36 Protein, Rat, Recombinant (hFc)	Rat	HEK293
	The cluster of differentiation (CD) system is commonly used as cell markers in Immunophenotyping. Different kinds of cells in the immune system can be identified through the surface CD molecules associating with the immu...
TMPY-06951	CD36 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293
	The cluster of differentiation (CD) system is commonly used as cell markers in Immunophenotyping. Different kinds of cells in the immune system can be identified through the surface CD molecules associating with the immu...
TMPY-03243	CD36 Protein, Rat, Recombinant (His)	Rat	HEK293
	The cluster of differentiation (CD) system is commonly used as cell markers in Immunophenotyping. Different kinds of cells in the immune system can be identified through the surface CD molecules associating with the immu...

PfLDH Protein, P. falciparum, Recombinant (His)

TMPY-04180

Species: P. falciparum

Expression System: E. coli

CD36 Protein, Mouse, Recombinant (His)

TMPY-01445

Species: Mouse

Expression System: HEK293

CD36 Protein, Human, Recombinant (His)

TMPY-01282

Species: Human

Expression System: HEK293

PKLR Protein, Human, Recombinant (His)

TMPY-04765

Species: Human

Expression System: E. coli

IgG3 Protein, Mouse, Recombinant

TMPY-02696

Species: Mouse

Expression System: HEK293

KLHL2 Protein, Human, Recombinant (GST)

TMPY-03399

Species: Human

Expression System: E. coli

Adenosine Deaminase Protein, Human, Recombinant (His)

TMPY-03985

Species: Human

Expression System: Baculovirus-Insect Cells

IgG3 Protein, Human, Recombinant

TMPY-02895

Species: Human

Expression System: HEK293

CD36 Protein, Mouse, Recombinant (His & hFc)

TMPY-01449

Species: Mouse

Expression System: HEK293

CD36 Protein, Rhesus, Recombinant (hFc)

TMPY-03479

Species: Rhesus

Expression System: HEK293

CD36 Protein, Rat, Recombinant (hFc)

TMPY-03242

Species: Rat

Expression System: HEK293

CD36 Protein, Human, Recombinant (His & Avi), Biotinylated

TMPY-06951

Species: Human

Expression System: HEK293

CD36 Protein, Rat, Recombinant (His)

TMPY-03243

Species: Rat

Expression System: HEK293

カタログ番号	製品名
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	419 well-chosen unique anti-parasitic small molecules;
L6001	Mini Fungal Metabolite Natural Product Screening Library	Inquiry

L1100	Protease Inhibitor Library	343 compounds
	A unique collection of 343 protease and proteasome inhibitors for research in chemical genomics, and drug screening;
L4600	Selected Plant-Sourced Compound Library	3048 compounds
	A unique collection of 3048 plant-sourced compounds that derived from 277 plant species for high throughput screening (HTS) and high content screening (HCS);
L6020	Selectable Natural Product Library	16627 compounds
	A unique collection of 16627 pure natural products with diverse structures and sources covering various plant, animal, and microbe species;
L6620	Antiparasitic Natural Product Library	253 compounds
	A unique collection of 253 natural products with antiparasitic activity, a powerful tool for high throughput screening (HTS) and high content screening (HCS);