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カタログ番号	製品名	別名	ターゲット
T2550	Tolmetin	Tolectin	COX
	Tolmetin (Tolectin) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of tolmetin is as a Cyclooxygenase Inhibitor. The chemical classification of tolmetin is Nonsteroidal Anti-inflammatory Compounds.		COX
T11399	Giredestrant	GDC-9545	Estrogen Receptor/ERR , Estrogen/progestogen Receptor
	Giredestrant (GDC-9545) potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has anti-tumor activity. Giredestrant, a non-steroidal ER ligand,...		Estrogen Receptor/ERR , Estrogen/progestogen Receptor
T0380	Bicalutamide	ICI-176334	Androgen Receptor , Autophagy
	Bicalutamide (ICI-176334), a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the receptor binding of androgens.		Androgen Receptor , Autophagy
T6737	Zaltoprofen	CN100,Soleton	COX
	Zaltoprofen (Soleton) is a Cox-1 and Cox-2 inhibitor, which is used for the treatment of arthritis.		COX
T22371	Mivacurium dichloride	Mivacurium chloride	AChR
	Mivacurium dichloride (Mivacurium chloride) is a non-depolarising, rapid neuromuscular blocker of short duration, used therefore as anesthetic, to provide skeletal muscle relaxation in minor surgical operations, in emerg...		AChR
T0383	Fenspiride hydrochloride	Fenspiride HCl,Pneumorel,Fluiden,Decaspiride	Adrenergic Receptor , PDE , Histamine Receptor
	Fenspiride hydrochloride (Decaspiride) , an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use in Russia for the therapy of chronic and acute inflammatory ...		Adrenergic Receptor , PDE , Histamine Receptor
T26539	AC-262536	AC262536	Androgen Receptor
	AC-262536 is a selective androgen receptor (SAR) modulator. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone.		Androgen Receptor
T4602	Hydrocortisone hemisuccinate	Hydrocortisone 21-he,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate	Glucocorticoid Receptor , Others , Interleukin
	Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.		Glucocorticoid Receptor , Others , Interleukin
T61444	Nonsteroidal aromatase inhibitor 1
	Nonsteroidal aromatase inhibitor 1 (Compound 13h) effectively inhibits the enzyme CYP19A1 with an IC50 value of 0.09 nM. Due to its potent inhibitory activity, Nonsteroidal aromatase inhibitor 1 holds promise for researc...
T26109	Robenacoxib	Onsior	COX
	Robenacoxib (Onsior) is a non-steroidal compound with strong selectivity for cyclooxygenase-2 and anti-inflammatory activity.		COX
T21740	RD162		Androgen Receptor
	RD162 is a non-steroidal antiandrogen (NSAA) specifically binding to the androgen receptor (AR).		Androgen Receptor
T7839	Lasofoxifene Tartrate	CP-336156	Estrogen Receptor/ERR
	Lasofoxifene Tartrate (CP-336156) is a third-generation, non-steroidal selective estrogen receptor modulator.		Estrogen Receptor/ERR
T14546	Bermoprofen	AD-1590,AJ-1590	Others
	Bermoprofen (AD-1590) is an orally active non-steroidal anti-inflammatory compound with anti-inflammatory and analgesic activity used in the study of gastric ulcers.		Others
T27209	Droxicam	Droxicamum	Others
	Droxicam (Droxicamum) is a non-steroidal anti-inflammatory compound and can be used for research on the relief of inflammation and pain in musculoskeletal disorders.		Others
T0321	Indoprofen	(±)-Indoprofe	COX
	Indoprofen ((±)-Indoprofe) is a non-steroidal anti-inflammatory drug.		COX
T19679	Benoxaprofen	NSC 299582,LY-90459,Benoxaphen. Compound 90459	COX
	Benoxaprofen (NSC-299582) is a non-steroidal anti-inflammatory drug.		COX
T25985	Prifelone	R-830,R830,S-16820,S 16820,R 830
	Prifelone (R 830) is a non-steroidal anti-inflammatory compound with antioxidant activity.
T15246	Esaxerenone	XL-550,CS-3150	Glucocorticoid Receptor
	Esaxerenone (XL-550) is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor.		Glucocorticoid Receptor
T6498	Fenoprofen calcium hydrate	Feprona dihydrate,Fenoprofen calcium salt dihydrate,Progesic dihydrate	Apoptosis , Others , COX
	Fenoprofen calcium hydrate (Progesic dihydrate) is a non-steroidal anti-inflammatory drug (NSAID).		Apoptosis , Others , COX
T6540	Ibuprofen Lysine	Neoprofen	COX
	Ibuprofen Lysine (Neoprofen) is a non-steroidal anti-inflammatory drug.		COX
T27798	Lapisteride	CS891B,CS-891,CS-891B,CS891	Others
	Lapisteride (CS-891) a steroidal 5α-reductase inhibitor is used to treat benign prostatic hyperplasia (BPH) and androgenetic alopecia and may be effective in preventing or treating AGA .		Others
T27254	Eltenac	B78820,B 78820,B-78820,BY-820,BY820,BY 820	COX
	Eltenac (B78820) is a non-steroidal anti-inflammatory, COX inhibitor with analgesic activity.Eltenac inhibits COX-1 and COX-2 and is used in the study of Acute Respiratory Distress Syndrome (ARDS).		COX
T0184	Fenoprofen calcium dihydrate		COX
	Fenoprofen calcium is a propionic acid derivative that is used as a non-steroidal anti-inflammatory agent.		COX
T0463	Loxoprofen	Loxoprofene,Loxoprofeno,Koloxo	COX
	Loxoprofen (Koloxo) is an anti-inflammatory non-steroidal medicine.		COX
T19694	Hydronidone	F351,F-351,F 351	Others
	Hydronidone (F-351) is Non-Steroidal Antiinflammatory Drugs. It potentially for the treatment of hepatic fibrosis.		Others
T7389	G15		Estrogen Receptor/ERR
	G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)		Estrogen Receptor/ERR
T1720	Amfenac Sodium Hydrate	Amfenac Sodium Monohydrate	COX
	Amfenac Sodium Hydrate is a non-steroidal analgesic anti-inflammatory drug with acetic acid moiety.		COX
T17217	Vamorolone	VBP15	Glucocorticoid Receptor , NF-κB
	Vamorolone (VBP15) is an orally active dissociative steroidal anti-inflammatory drug and membrane-stabilizer. Vamorolone improves muscular dystrophy without side effects. Vamorolone displays effective NF-κB inhibition an...		Glucocorticoid Receptor , NF-κB
T30150	AS-601811	AS601811,AS 601811,UNII-LIV8A6AE5F	Androgen Receptor
	AS-601811 is a steroidal 5α-reductase inhibitor and androgen receptor modulator used to study hair loss and acne.		Androgen Receptor
T27635	Isoxepac	Olopatadine USP Related Compound C	Others
	Isoxepac (Olopatadine USP Related Compound C) is a non-steroidal anti-antiphlogistic agent and analgesic.		Others
T0637	2-Acetyl-6-methoxynaphthalene		Others
	2-Acetyl-6-methoxynaphthalene, the key intermediate of naphthalene tome and naproxen, is used in synthetic non-steroidal anti-inflammatory analgesic medicine and.		Others
T4542	Clonixin	Clonixic acid	Others
	Clonixin (Clonixic acid) is a non-steroidal anti-inflammatory drug (NSAID) with analgesic properties. This compound has been reported to block prostaglandin synthesis, and to block inward calcium currents.		Others
T4561	Tiaprofenic acid	Tiaprofensaeure,Acido tiaprofenico,Surgam	Others , COX
	Tiaprofenic acid (Acido tiaprofenico) is a non-steroidal anti-inflammatory drug used to treat pain, especially arthritic pain.		Others , COX
T1258	Nabumetone	BRL14777	COX , Glutathione Peroxidase
	Nabumetone (BRL14777)(BRL14777) is a non-steroidal anti-inflammatory drug and its active metabolite 6MNA inhibits the enzymes cyclo-oxygenase I and II.		COX , Glutathione Peroxidase
T30161	EN3356	AS N001,ASN-001	P450
	EN3356 is an orally available and selective inhibitor of steroidal 17-alpha-hydroxylase/C17,20 cleavage enzyme (CYP17A1 or CYP17), a non-steroidal cleavage enzyme-selective compound with potential anti-androgenic and ant...		P450
T0767	Sulfapyridine	Sulfidine,Sulfidin,2-Sulfapyridine	Antibacterial , Antibiotic , Autophagy
	Sulfapyridine (2-Sulfapyridine) is a short-acting sulfonamide antibiotic and by-product of the non-steroidal anti-inflammatory drug sulfasalazine.		Antibacterial , Antibiotic , Autophagy
T21412	Ketorolac	Toradol,Sprix,Acuvail,Macril,Acular	COX
	Ketorolac (Acuvail) is a non-steroidal anti-inflammatory drug (NSAID) in the family of heterocyclic acetic acid derivatives. It acts by inhibiting the bodily synthesis of prostaglandins.		COX
T22307	Diclofenac Epolamine	diclofenac hydroxyethylpyrrolidine,DHEP,DIEP	Others
	Diclofenac Epolamine (DHEP) is a non-steroidal anti-inflammatory agent (NSAID) with analgesic and antipyretic actions.		Others
T11340	Furprofen		Prostaglandin Receptor
	Furprofen is a non-steroidal anti-inflammatory agent that inhibits prostate (PGE) synthesis and is used in the study of rheumatoid arthritis and osteoarthritis.		Prostaglandin Receptor
T0448	(S)-(+)-Ibuprofen	Dexibuprofen,(S)-Ibuprofen	BCL , Thrombin , Cysteine Protease , COX , PPAR
	(S)-(+)-Ibuprofen (Dexibuprofen) , is a non-steroidal anti-inflammatory drug (NSAID), inhibiting cyclooxygenase (COX).		BCL , Thrombin , Cysteine Protease , COX , PPAR
T7313	Enclomiphene citrate	Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate	Estrogen Receptor/ERR
	Enclomiphene citrate (trans-Clomiphene citrate) is a non-steroidal estrogen receptor antagonist,with antioestrogenic property		Estrogen Receptor/ERR
T21361	Alclometasone dipropionate	Vaderm,Sch 22219,Aclovate,Delonal	Others
	Alclometasone dipropionate （Sch 22219） is a synthetic glucocorticoid, a steroidal compound with antiproliferative, anti-inflammatory, anti-allergic, antipruritic, and vasoconstrictive properties, which is used in the stu...		Others
T14666	BL-1249		Potassium Channel
	BL-1249 is a selective and potent non-steroidal potassium channel activator with anti-inflammatory activity that activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2).		Potassium Channel
T1421	Aceclofenac	Preservex,Airtal	COX
	Aceclofenac (Preservex) is a non-steroidal anti-inflammatory drug (NSAID) with marked anti-inflammatory and analgesic properties.		COX
T0890	Mefenamic acid	CN-35355,CI 473	COX
	Mefenamic acid (CN-35355) is a non-steroidal anti-inflammatory agent with analgesic, anti-inflammatory, and antipyretic properties. It is an inhibitor of cyclooxygenase.		COX
T0285	Isoxicam	Isoxicamum,Isoxicamo,Maxicam	COX
	Isoxicam (Isoxicamum) is a non-steroidal anti-inflammatory drug that is not marketed in the United States.		COX
T7293	EC330		Others
	EC330, a novel steroidal LIF inhibitor showed cytotoxicity in various cancer cell lines and NCI-60 cell line panel at low nano-molar range.		Others
T12361	Parcetasal	MR-897	Others
	Parcetasal (MR-897) is a non-steroidal anti-inflammatory agent that can be used in pain relief studies.		Others
T2567	Etonogestrel	3-Oxodesogestrel,3-keto-Desogestrel,Nexplanon,Implanon	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Progesterone Receptor , Endogenous Metabolite
	Etonogestrel (Implanon) is a steroidal progestin used as hormonal contraceptives.
T0319	Suxibuzone	Calibene,Suxibuzonum,Suxibuzona	COX
	Suxibuzone (Suxibuzona) is a drug used for joint and muscular pain. It is a prodrug of the non steroidal anti inflammatory drug phenylbutazone, and is commonly used in horses.		COX

Compounds

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor

Bicalutamide

T0380

Synonym: ICI-176334

Target: Androgen Receptor, Autophagy

Zaltoprofen

T6737

Synonym: CN100,Soleton

Target: COX

Mivacurium dichloride

T22371

Synonym: Mivacurium chloride

Target: AChR

Fenspiride hydrochloride

T0383

Synonym: Fenspiride HCl,Pneumorel,Fluiden,Decaspiride

Target: Adrenergic Receptor, PDE, Histamine Receptor

AC-262536

T26539

Synonym: AC262536

Target: Androgen Receptor

Hydrocortisone hemisuccinate

T4602

Synonym: Hydrocortisone 21-he,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate

Target: Glucocorticoid Receptor, Others, Interleukin

Nonsteroidal aromatase inhibitor 1

Target: Androgen Receptor

Lasofoxifene Tartrate

T7839

Synonym: CP-336156

Target: Estrogen Receptor/ERR

Bermoprofen

T14546

Synonym: AD-1590,AJ-1590

Synonym: (±)-Indoprofe

Target: COX

Benoxaprofen

T19679

Synonym: NSC 299582,LY-90459,Benoxaphen. Compound 90459

Target: COX

Prifelone

T25985

Synonym: R-830,R830,S-16820,S 16820,R 830

Target:

Esaxerenone

T15246

Synonym: XL-550,CS-3150

Target: Glucocorticoid Receptor

Fenoprofen calcium hydrate

T6498

Synonym: Feprona dihydrate,Fenoprofen calcium salt dihydrate,Progesic dihydrate

Target: Apoptosis, Others, COX

Synonym: CS891B,CS-891,CS-891B,CS891

Target: Others

Eltenac

T27254

Synonym: B78820,B 78820,B-78820,BY-820,BY820,BY 820

Target: COX

Fenoprofen calcium dihydrate

Synonym: Loxoprofene,Loxoprofeno,Koloxo

Target: COX

Hydronidone

T19694

Synonym: F351,F-351,F 351

Target: Estrogen Receptor/ERR

Amfenac Sodium Hydrate

T1720

Synonym: Amfenac Sodium Monohydrate

Target: Glucocorticoid Receptor, NF-κB

AS-601811

T30150

Synonym: AS601811,AS 601811,UNII-LIV8A6AE5F

Target: Androgen Receptor

Isoxepac

T27635

Synonym: Olopatadine USP Related Compound C

Target: Others

2-Acetyl-6-methoxynaphthalene

Synonym: Clonixic acid

Target: Others

Tiaprofenic acid

T4561

Synonym: Tiaprofensaeure,Acido tiaprofenico,Surgam

Target: COX, Glutathione Peroxidase

EN3356

T30161

Synonym: AS N001,ASN-001

Target: P450

Sulfapyridine

T0767

Synonym: Sulfidine,Sulfidin,2-Sulfapyridine

Target: Antibacterial, Antibiotic, Autophagy

Ketorolac

T21412

Synonym: Toradol,Sprix,Acuvail,Macril,Acular

Target: COX

Diclofenac Epolamine

T22307

Synonym: diclofenac hydroxyethylpyrrolidine,DHEP,DIEP

Target: Prostaglandin Receptor

(S)-(+)-Ibuprofen

T0448

Synonym: Dexibuprofen,(S)-Ibuprofen

Target: BCL, Thrombin, Cysteine Protease, COX, PPAR

Enclomiphene citrate

T7313

Synonym: Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate

Target: Estrogen Receptor/ERR

Alclometasone dipropionate

T21361

Synonym: Vaderm,Sch 22219,Aclovate,Delonal

Target: Potassium Channel

Aceclofenac

T1421

Synonym: Preservex,Airtal

Target: COX

Mefenamic acid

T0890

Synonym: CN-35355,CI 473

Target: COX

Isoxicam

T0285

Synonym: Isoxicamum,Isoxicamo,Maxicam

Synonym: 3-Oxodesogestrel,3-keto-Desogestrel,Nexplanon,Implanon

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Progesterone Receptor, Endogenous Metabolite

Suxibuzone

T0319

Synonym: Calibene,Suxibuzonum,Suxibuzona

Target: COX

カタログ番号	製品名	別名	ターゲット
T3901	Solasonine		Others
	Solasonine exerts leishmanicidal activity against promastigote forms of L. amazonensis.		Others
T4035	Khasianine		Others
	Khasianine has strong activity against liver damage induced by CCl4.		Others
T3S0509	Gaultherin		COX
	Gaultherin has analgesic, and anti-inflammatory activities.Gaultherin lacks gastric ulcerogenic effect, because of it released salicylate in intestine slowly, not in stomach and it left the cyclooxygenase-1 unaffected, w...		COX
T3S1251	Neoruscogenin		ROR
	1. Neoruscogenin represents a universal pharmacological tool for RORα research due to its specific selectivity profile versus other nuclear receptors.		ROR
T3S1265	Liriopesides B	Nolinospiroside F	Others
	Liriopesides B (Nolinospiroside F) exhibited potential anticancer activity against human ovarian cancer A2780 cells.		Others
T7024	Qingyangshengenin	Qingyangshengenin A,Cynanchagenin	Others
	Qingyangshengenin (Cynanchagenin) is a steroid used in the preparation of antiepileptic agents.		Others
T0301	Ethisterone	17α-Ethynyltestosterone,Pregneninolone	Estrogen Receptor/ERR , Estrogen/progestogen Receptor
	Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.		Estrogen Receptor/ERR , Estrogen/progestogen Receptor
T4036	Solasodine	Solancarpidine,Purapuridine,Solasodin	Apoptosis , Others , E1/E2/E3 Enzyme , Antifungal
	Solasodine (Purapuridine)(Purapuridine) is a poisonous alkaloid chemical compound that occurs in plants of the Solanaceae family. Solasodine showed selective cytotoxicity against cervical cancer cell line (HeLa) and huma...		Apoptosis , Others , E1/E2/E3 Enzyme , Antifungal
T2S0250	Pseudoprotogracillin		Others
	Pseudoprotogracillin is a steroidal saponin extracted from Dioscoreae.		Others
T8094	16-Dehydroprogesterone	16-Dehydroprogesterone	Endogenous Metabolite
	16-Dehydroprogesterone is a endogenous Metabolite. 16-Dehydroprogesterone is a steroidal progestin.		Endogenous Metabolite
T2S2295	Timosaponin A1		Others
	Timosaponin A1 is a coprostane type steroidal saponin found in Rhizoma Anemarrhenae.		Others
T2321	Protodioscin	Furostanol I	Androgen Receptor , Endogenous Metabolite
	Protodioscin (Furostanol I) is a major steroidal saponin in dioscoreae rhizome, with anti-hyperlipidemia, anti-cancer properties.		Androgen Receptor , Endogenous Metabolite
T2S1749	Protogracillin		Others
	Protogracillin may have inhibitions on platelet aggregation (PAG) and thrombosis.		Others
T10233	Acetylarenobufagin		HIF
	Acetylarenobufagin is a steroidal hypoxia-inducible factor-1 (HIF-1) modulator.		HIF
TN2329	Zingiberen newsaponin	Zingiberensis saponin I	PARP , PAFR , Caspase
	Zingiberen newsaponin is a steroidal saponin from Dioscorea zingiberensis.		PARP , PAFR , Caspase
TN6712	Yibeissine		Others
	Yibeissine is a natural steroidal alkaloid isolated from the bulb of Fritillaria pallioiflora Schren.		Others
T5751	Tigogenin		Others
	Tigogenin is one of steroidal sapogenins which is widely used for synthesizing steroid drugs. It might have protective effect on bone and be helpful in preventing the development of osteoporosis.		Others
T2825	Cyclopamine	11-Deoxojervine	Hedgehog/Smoothened , Endogenous Metabolite , Smo
	Cyclopamine (11-Deoxojervine), a Smoothened (Smo) antagonist (IC50: 46 nM in TM3Hh12 cells), belongs to the group of steroidal jerveratrum alkaloids.		Hedgehog/Smoothened , Endogenous Metabolite , Smo
TN2282	Trans-Stilbene	1,2-Diphenylethylene (trans),(E)-Stilbene	Others
	trans-Stilbene (1,2-Diphenylethylene (trans)) is a natural product used in the manufacture of dye lasers, optical brighteners, and non-steroidal synthetic estrogens.		Others
T3150	Caudatin		Apoptosis , Others
	Caudatin is one of the species of C-21 steroidal glycosides mainly isolated from the root of Cynanchum bungei Decne and exhibits potent anticancer activities.		Apoptosis , Others
TN1383	Timosaponin B III	Anemarsaponin BIII	Others , Platelet aggregation
	Timosaponin B III (Anemarsaponin BIII) is a bioactive steroidal saponin isolated from Anemarrhena asphodeloides Bge. Timosaponin B III possesses anti-inflammatory, anti-platelet aggregative and anti-depressive effects.		Others , Platelet aggregation
T1048	Estradiol	E2,17β-Estradiol,17β-Oestradiol,β-Estradiol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	Estradiol (E2) is a naturally occurring steroidal sex hormone that is essential for female fertility and maintenance of secondary sexual characteristics. Estradiol upregulates IL-6 expression through estrogen receptor be...
T20712	Conessine	Conessinum,Wrightine,Roquessine,Neriine,Konessin	Histamine Receptor
	Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.		Histamine Receptor
T16338	Norgestimate metabolite Norelgestromin	17-Deacetyl norgestimate,17-Deacylnorgestimate	Drug Metabolite
	Norgestimate metabolite Norelgestromin (17-Deacylnorgestimate) is one of the active metabolites of norgestimate.It is a steroidal progestin used in contraceptive patches, where it is combined with the estrogen ethinyl es...		Drug Metabolite
T4034	Solamargine	Solamargin,δ-Solanigrine	Apoptosis , p38 MAPK , P-gp , STAT
	Solamargine (δ-Solanigrine) is a major steroidal alkaloid glycoside extracted from a traditional Chinese medicine herb, Solanum nigrum L. (SNL); has been shown to inhibit growth and induce apoptosis of various cancer cel...		Apoptosis , p38 MAPK , P-gp , STAT
T2733	Sarsasapogenin	Parigenin,Sarsagenin	Apoptosis , NF-κB , Endogenous Metabolite
	Sarsasapogenin (Parigenin) is a steroidal sapogenin, that is the aglycosidic portion of a plant saponin. It is named after sarsaparilla (Smilax sp.), a family of climbing plants found in subtropical regions. It was one o...		Apoptosis , NF-κB , Endogenous Metabolite
TMS1461	Qingyangshengenin B	Otophylloside B	Beta Amyloid
	Qingyangshengenin B (Otophylloside B) is a C-21 steroidal glycoside isolated from Qingyangshen. Qingyangshengenin B protects against Aβ toxicity, which decreases Aβ deposition by decreasing the expression of Aβ at the mR...		Beta Amyloid
T4000	(±)-Equol	Equol,(R,S)-Equol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Drug Metabolite
	(±)-Equol ((R,S)-Equol) is a non-steroidal estrogen produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora. The estrogen receptor (ER) agonist activity of the naturally occu...
T6491	(-)-(S)-Equol	(−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	(-)-(S)-Equol (4',7-Dihydroxyisoflavan) is an orally bioavailable, non-steroidal estrogen naturally produced by the metabolism of the isoflavonoid daidzein by human intestinal microflora, with potential chemoprotective a...
T33926	Penupogenin
	Penupogenin is a steroidal aglycone isolated from the roots of Cynanchum auriculatum.
T40890	Proprotogracillin
	Proprotogracillin is a steroidal glycoside isolated from the bulbs of lilium speciosum.
T34584	Scillaren A	Transvaalin,Scillaglykosid A
	Scillaren A is a a crystalline steroidal glycoside from Scilla maritima.
T32610	Laxogenin	6-Oxotigogenin
	Laxogenin is a new steroidal sapogenin extracted from Smilax sieboldi Miq.
T13757	Lirioprolioside B		Others
	Lirioprolioside B is a steroidal glycoside isolated from the underground organs of Liriope spicata var. prolifera.		Others
T2S2321	Pennogenin		Others
	Pennogenin steroidal saponins could be utilized to develop anticancer medicines.		Others
T30170	Aspafilioside A
	Aspafilioside A is a steroidal saponin isolated from the root of Asparagus filicinus.
T10913	Cyclobuxine D		Others
	Cyclobuxine D is a steroidal alkaloid extracted from Buxus microphylla. Cyclostatin D has obvious bradycardia effect on rat heart, and inhibits acetylcholine and Ba ++ induced longitudinal muscle contraction isolated fro...		Others
T13805	Ophiopogonin C	Ophiopogonin C	Others
	Ophiopogonin C is a natural product isolated from the tubers of Ophiopogon japonicus, is a rare naturally occurring C29 steroidal glycoside.		Others
T13577	β-Zearalenol		Others
	β-Zearalenol, a non-steroidal estrogenic mycotoxin synthesized by Fusarium species, potentially influences transcription and affects gene expression on the translational level.		Others
T81093	Sterebin F
	Sterebin F, a steroidal compound extracted from Stevia rebaudiana leaves, exhibits hypoglycemic activity [1].
T39854	Cycloposine
	Cycloposine, a steroidal alkaloid present in the roots and rhizomes of Veratrum californicum, is known to possess teratogenic properties.
T81097	Stauntoside M
	Stauntoside M, a steroidal glycoside, is isolated from the roots of Cynanchum stauntonii [1].
T40193	Ebeiedinone
	Ebeiedinone, a steroidal alkaloid derived from Fritillaria species, effectively inhibits the activity of human whole blood cholinesterase (ChE) at a concentration of 0.1 mM, resulting in a significant inhibitory effect o...
T81545	Parisyunnanoside H
	Parisyunnanoside H, a steroidal saponin, has been isolated from the variety yunnanensis of Paris polyphylla Smith [1].
T82480	Elephanoside D
	Elephanoside D (compound 8), a steroidal saponin, has been isolated from the stems of Yucca elephantipes Regel.
T13641	Dehydrotomatine		Others
	Dehydrolycopene is a major steroidal sugar alkaloid (SGAs), which is mainly found in mature green fruits, leaves and flowers of tomatoes. Dehydrotomato is targeted at bacteria, fungi, insects and animals.		Others
T82544	Disporoside C
	Disporoside C, a steroidal saponin, can be isolated from Disporopsis pernyi [1].
T83259	6β-Hydroxystigmasta-4,22-dien-3-one
	6β-Hydroxystigmasta-4,22-dien-3-one is a steroidal compound that can be isolated from the plant Hedychium coronarium [1].
T82549	Diosgenin-3-O-rhamnosyl(1→2)[glucosyl(1→6)]glucoside
	Diosgenin-3-O-rhamnosyl(1→2)[glucosyl(1→6)]glucoside (compound 9), a steroidal saponin, is isolated from the variety yunnanensis of Paris polyphylla, commonly known as Yunnan pine [1].
T83568	(25R)-Ruscogenin-3-yl α-L-rhamnopyranosyl-(1→2)-[β-D-xylopyranosyl-(1→4)]-β-D-glucopyranoside
	Compound 1, (25R)-Ruscogenin-3-yl α-L-rhamnopyranosyl-(1→2)-[β-D-xylopyranosyl-(1→4)]-β-D-glucopyranoside, is a steroidal saponin that can be isolated from the roots of Ophiopogon japonicus [1].
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天然物製品

Synonym: Nolinospiroside F

Target: Others

Qingyangshengenin

T7024

Synonym: Qingyangshengenin A,Cynanchagenin

Target: Others

Ethisterone

T0301

Synonym: 17α-Ethynyltestosterone,Pregneninolone

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor

Solasodine

T4036

Synonym: Solancarpidine,Purapuridine,Solasodin

Target: Apoptosis, Others, E1/E2/E3 Enzyme, Antifungal

16-Dehydroprogesterone

T8094

Synonym: 16-Dehydroprogesterone

Target: Endogenous Metabolite

Synonym: Furostanol I

Target: Androgen Receptor, Endogenous Metabolite

Zingiberen newsaponin

TN2329

Synonym: Zingiberensis saponin I

Target: PARP, PAFR, Caspase

Synonym: 11-Deoxojervine

Target: Hedgehog/Smoothened, Endogenous Metabolite, Smo

trans-Stilbene

TN2282

Synonym: 1,2-Diphenylethylene (trans),(E)-Stilbene

Target: Apoptosis, Others

Timosaponin B III

TN1383

Synonym: Anemarsaponin BIII

Target: Others, Platelet aggregation

Estradiol

T1048

Synonym: E2,17β-Estradiol,17β-Oestradiol,β-Estradiol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite

Conessine

T20712

Synonym: Conessinum,Wrightine,Roquessine,Neriine,Konessin

Target: Histamine Receptor

Norgestimate metabolite Norelgestromin

T16338

Synonym: 17-Deacetyl norgestimate,17-Deacylnorgestimate

Target: Drug Metabolite

Solamargine

T4034

Synonym: Solamargin,δ-Solanigrine

Target: Apoptosis, p38 MAPK, P-gp, STAT

Sarsasapogenin

T2733

Synonym: Parigenin,Sarsagenin

Target: Apoptosis, NF-κB, Endogenous Metabolite

Qingyangshengenin B

TMS1461

Synonym: Otophylloside B

Target: Beta Amyloid

(±)-Equol

T4000

Synonym: Equol,(R,S)-Equol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Drug Metabolite

(-)-(S)-Equol

T6491

Synonym: (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite

Synonym: Transvaalin,Scillaglykosid A

Target:

Laxogenin

T32610

Synonym: 6-Oxotigogenin

Synonym: Ophiopogonin C

6β-Hydroxystigmasta-4,22-dien-3-one

T83259

Synonym:

Target:

Diosgenin-3-O-rhamnosyl(1→2)[glucosyl(1→6)]glucoside

T82549

Synonym:

Target:

(25R)-Ruscogenin-3-yl α-L-rhamnopyranosyl-(1→2)-[β-D-xylopyranosyl-(1→4)]-β-D-glucopyranoside

T83568

Synonym:

Target:

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Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPH-01640	MRGPRX2 Protein, Human, Recombinant (His)	Human	E. coli
	Mast cell-specific receptor for basic secretagogues, i.e. cationic amphiphilic drugs, as well as endo- or exogenous peptides, consisting of a basic head group and a hydrophobic core. Recognizes and binds small molecules ...

MRGPRX2 Protein, Human, Recombinant (His)

TMPH-01640

Species: Human

Expression System: E. coli

カタログ番号	製品名
L4710	Nonsteroidal Anti-Inflammatory Compound Library	530 compounds
	530 non-steroidal anti-inflammatory compounds for high-throughput and high-content screening.
L6710	Anti-Inflammatory Traditional Chinese Medicine Compound Library	1246 compounds
	A collection of 1246 TCM monomers with anti-inflammatory activity or targeting molecular therapeutic targets in inflammation, a powerful tool for drug discovery and mechanism study；
L4700	Immunology/Inflammation Compound Library	4720 compounds
	A unique collection of 4720 anti-inflammation compounds effective for high throughput screening and high content screening.

ライブラリー

Nonsteroidal Anti-Inflammatory Compound Library

L4710

Compounds: 530

Anti-Inflammatory Traditional Chinese Medicine Compound Library

L6710

Compounds: 1246

Immunology/Inflammation Compound Library

L4700

Compounds: 4720