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ターゲット

380

阻害剤

天然化合物

331

リコンビナントタンパク質

カタログ番号	製品名	別名	ターゲット
T18184	m-PEG3-SH	M-PEG3-Thiol,2-(2-(2-Methoxyethoxy)Ethoxy)Ethanethiol	Others , PROTAC Linker
	m-PEG3-SH (M-PEG3-Thiol) is a PEG-based PROTAC linker. m-PEG3-SH can be used in the synthesis of PROTACs.		Others , PROTAC Linker
T18161	m-PEG2-Br		Others , PROTAC Linker
	m-PEG2-Br is a PEG-based PROTAC linker. m-PEG2-Br can be used in the synthesis of PROTACs.		Others , PROTAC Linker
T8607	M084	M-084 hydrochloride,1H-Benzimidazol-2-amine,N-butyl-(9CI),N-Butyl-1H-benzimidazol-2-amine	TRP/TRPV Channel
	M084 (N-Butyl-1H-benzimidazol-2-amine) is a blocker of TRPC4/5 channel, with antidepressant and anxiolytic effects.		TRP/TRPV Channel
T15904	m-PEG6-2-methylacrylate		Others
	m-PEG6-2-methylacrylate is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome ...		Others
T33131	m-(2-Phenoxyethoxy)phenol
	m-(2-Phenoxyethoxy)phenol is a biaoctive chemical.
T15887	m-PEG5-2-methylacrylate		Others
	m-PEG5-2-methylacrylate is a polyethylene glycol (PEG)- and alkyl/ester-based PROTAC linker employed for the synthesis of proteolysis-targeting chimeras (PROTACs)[1].		Others
T29351	2-Hexyl-m-cresol
	2-Hexyl-m-cresol is a bioactive chemical.
T33147	m-Acetophenetidide, 2-iodo-
	m-Acetophenetidide, 2-iodo- is a bioactive chemical.
T33141	m-Acetanisidide, 2-iodo-
	m-Acetanisidide, 2-iodo- is a bioactive chemical.
T33146	m-Acetophenetidide, 2-chloro-
	m-Acetophenetidide, 2-chloro- is a bioactive chemical.
T8741	MitoBloCK-10	3-fluoro-N'-[(E)-(5-nitrothiophen-2-yl)m	Others
	MitoBloCK-10 (3-fluoro-N'-[(E)-(5-nitrothiophen-2-yl)m) inhibits Tim44 binding to the precursor and to Hsp70.MitoBloCK-10 is the first small molecule modulator to attenuate protein-associated motor (PAM) complex activity...		Others
T18571	m-PEG12-2-methylacrylate	Propargyl-PEG13-alcohol	Others
	Propargyl-PEG13-alcohol is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs[1].		Others
T30063	Aniline, m-(2-(2-(diethylamino)ethoxy)ethyl)-
	Aniline, m-(2-(2-(diethylamino)ethoxy)ethyl)- is a bioactive chemical.
T34002	Phenol, m-(2-(dipropylamino)ethyl)-, hydrobromide
	Phenol, m-(2-(dipropylamino)ethyl)-, hydrobromide is a bioactive chemical.
T34003	Phenol, m-(2-(methylamino)ethyl)-, hydrochloride
	Phenol, m-(2-(methylamino)ethyl)-, hydrochloride is a biaoctive chemical.
T29370	2-Propynyl m-hydroxycarbanilate methylcarbamate
	2-Propynyl m-hydroxycarbanilate methylcarbamate is a bioactive chemical.
T33990	Phenol, m-(1,3-dithiolan-2-yl)-
	Phenol, m-(1,3-dithiolan-2-yl)- is a bioactive chemical.
T34001	Phenol, m-(2-(dimethylaminomethyl)-1-hydroxycyclopentyl)-
	Phenol, m-(2-(dimethylaminomethyl)-1-hydroxycyclopentyl)- is a bioactive chemical.
T33253	m-Dioxan-5-ol, 2-(2-furyl)-
	m-Dioxan-5-ol, 2-(2-furyl)- is a bioactive chemical.
T10198	8-M-PDOT	8-Methoxy-2-propionamidotetralin,AH-002	MT Receptor
			MT Receptor
T34006	Phenol, m-(2-(phenethylamino)ethyl)-, hydrochloride
	Phenol, m-(2-(phenethylamino)ethyl)-, hydrochloride can be used in related research in the field of life sciences. Its product number is T34006 and CAS number is 70045-20-4.
T33149	m-Acetotoluidide, 2-chloro-N-(2-ethoxyethyl)-
	m-Acetotoluidide, 2-chloro-N-(2-ethoxyethyl)- is a bioactive chemical.
T33140	m-Acetanisidide, 2-chloro-N-(2-ethoxyethyl)-
	m-Acetanisidide, 2-chloro-N-(2-ethoxyethyl)- is a bioactive chemical.
T4282	S-methyl-KE-298		MMP , Drug Metabolite
	S-methyl-KE-298 is the second main metabolite in plasma,is a methyl conjugate of deacetyl-KE-298.KE-298 inhibits matrix metalloproteinase (MMP-1) production from rheumatoid arthritis (RA) synovial cells.		MMP , Drug Metabolite
T29432	4-Chloro-2-nitro-m-cresol
	4-Chloro-2-nitro-m-cresol is a biaoctive chemical.
T33150	m-Acetotoluidide, 2-fluoro-N-methyl-
	m-Acetotoluidide, 2-fluoro-N-methyl- is a bioactive chemical.
T33254	m-Dioxane, 2-hexyl-2,4-dimethyl-
	m-Dioxane, 2-hexyl-2,4-dimethyl- is a bioactive chemical.
T33139	m-Acetanisidide, 2-(diethylamino)-4'-(octyloxy)-
	m-Acetanisidide, 2-(diethylamino)-4'-(octyloxy)- is a bioactive chemical.
T34005	Phenol, m-(2-(N-methylphenethylamino)ethyl)-, hydrobromide
	Phenol, m-(2-(N-methylphenethylamino)ethyl)-, hydrobromide is a bioactive chemical.
T30403	Benzoic acid, m-iodo-, 2-phenylhydrazide
	Benzoic acid, m-iodo-, 2-phenylhydrazide is a bioactive chemical.
T33195	m-Anisidine, 4-(2-ethylbutoxy)-, hydrobromide
	m-Anisidine, 4-(2-ethylbutoxy)-, hydrobromide is a bioactive chemical.
T10220	LSN2839567	Abemaciclib metabolite M2	CDK
	LSN2839567 (Abemaciclib metabolite M2) is the active metabolite of Abemaciclib, a potent CDK4 and CDK6 inhibitor (IC50s: 1-3 nM) with anticancer activity.LSN2839567 inhibits CDK9.LSN2839567 inhibits cell growth and cell ...		CDK
T33249	m-Dioxan-5-amine, 2-(p-chlorophenyl)-
	m-Dioxan-5-amine, 2-(p-chlorophenyl)- is a bioactive chemical.
T30721	Carbanilic acid, m-(2-methoxyethoxy)-, 2-(diethylamino)ethyl ester
	Carbanilic acid, m-(2-methoxyethoxy)-, 2-(diethylamino)ethyl ester is a bioactive chemical.
T50077	m-Nisoldipine	3-methyl 5-(2-methylpropyl) 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate	Others
	m-Nisoldipine (3-methyl 5-(2-methylpropyl) 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate) is a dihydropyridine calcium channel blocker, a derivative of nisoldipine, that blocks L-type calcium chann...		Others
T33156	m-Acetotoluidide, N-benzyl-2-(diethylamino)-, monohydrochloride
	m-Acetotoluidide, N-benzyl-2-(diethylamino)-, monohydrochloride is a bioactive chemical.
T33256	m-Dioxane, 5-ethyl-2-(2-furyl)-4-propyl-
	m-Dioxane, 5-ethyl-2-(2-furyl)-4-propyl- is a bioactive chemical.
T33255	m-Dioxane, 5,5-bis(chloromethyl)-2-phenyl-
	m-Dioxane, 5,5-bis(chloromethyl)-2-phenyl- is a bioactive chemical.
T30396	Benzoic acid, m-(2-methyl-5-phenylpyrrol-1-yl)-
	Benzoic acid, m-(2-methyl-5-phenylpyrrol-1-yl)- is a bioactive chemical.
T33257	m-Dioxane, 5-ethyl-5-nitro-2-propyl-
	m-Dioxane, 5-ethyl-5-nitro-2-propyl- is a bioactive chemical.
T33252	m-Dioxan-5-amine, 5-benzylaminomethyl-2-phenyl-
	m-Dioxan-5-amine, 5-benzylaminomethyl-2-phenyl- is a bioactive chemical.
T30392	Benzoic acid, m-(2-(p-bromophenyl)-5-methylpyrrol-1-yl)-
	Benzoic acid, m-(2-(p-bromophenyl)-5-methylpyrrol-1-yl)- is a bioactive chemical.
T33251	m-Dioxan-5-amine, 2-(p-chlorophenyl)-5-methyl-
	m-Dioxan-5-amine, 2-(p-chlorophenyl)-5-methyl- is a bioactive chemical.
T33250	m-Dioxan-5-amine, 2-(p-chlorophenyl)-5-ethyl-
	m-Dioxan-5-amine, 2-(p-chlorophenyl)-5-ethyl- is a bioactive chemical.
T34004	Phenol, m-(2-(N-ethylphenethylamino)ethyl)-, fumarate (1:1)
	Phenol, m-(2-(N-ethylphenethylamino)ethyl)-, fumarate (1:1) is a bioactive chemical.
T33995	Phenol, m-(1-methyl-3-(2-methylbutyl)-3-pyrrolidinyl)-
	Phenol, m-(1-methyl-3-(2-methylbutyl)-3-pyrrolidinyl)- is a bioactive chemical.
T34009	Phenol, m-(2-ethyl-1-methyl-3-propyl-3-pyrrolidinyl)-
	Phenol, m-(2-ethyl-1-methyl-3-propyl-3-pyrrolidinyl)- is a bioactive chemical.
T30358	N,N-Bis(2-chloroethyl)-m-iodobenzylamine	Benzenemethanamine, N,N-bis(2-chloroethyl)-3-iodo- (9CI)
	Benzenemethanamine, N,N-bis(2-chloroethyl)-3-iodo- (9CI) is a bioactive chemical.
T33142	m-Acetanisidide, N-(2-(diethylamino)ethyl)-2-(p-ethoxyphenoxy)-, monopicrate
	m-Acetanisidide, N-(2-(diethylamino)ethyl)-2-(p-ethoxyphenoxy)-, monopicrate is a bioactive chemical.
T30720	Carbanilic acid, m-((pentyloxy)methyl)-, 2-piperidinoethyl ester, hydrochloride
	Carbanilic acid, m-((pentyloxy)methyl)-, 2-piperidinoethyl ester, hydrochloride is a bioactive chemical.

Compounds

m-PEG3-SH

T18184

Synonym: M-PEG3-Thiol,2-(2-(2-Methoxyethoxy)Ethoxy)Ethanethiol

Target: Others, PROTAC Linker

m-PEG2-Br

T18161

Synonym:

Target: Others, PROTAC Linker

M084

T8607

Synonym: M-084 hydrochloride,1H-Benzimidazol-2-amine,N-butyl-(9CI),N-Butyl-1H-benzimidazol-2-amine

Target: TRP/TRPV Channel

m-PEG6-2-methylacrylate

T15904

Synonym:

Target: Others

m-(2-Phenoxyethoxy)phenol

T33131

Synonym:

Target:

m-PEG5-2-methylacrylate

m-Acetophenetidide, 2-iodo-

T33147

Synonym:

Target:

m-Acetanisidide, 2-iodo-

T33141

Synonym:

Target:

m-Acetophenetidide, 2-chloro-

Synonym: 3-fluoro-N'-[(E)-(5-nitrothiophen-2-yl)m

Target: Others

m-PEG12-2-methylacrylate

T18571

Synonym: Propargyl-PEG13-alcohol

Target: Others

Aniline, m-(2-(2-(diethylamino)ethoxy)ethyl)-

T30063

Synonym:

Target:

Phenol, m-(2-(dipropylamino)ethyl)-, hydrobromide

T34002

Synonym:

Target:

Phenol, m-(2-(methylamino)ethyl)-, hydrochloride

T34003

Synonym:

Target:

2-Propynyl m-hydroxycarbanilate methylcarbamate

T29370

Synonym:

Target:

Phenol, m-(1,3-dithiolan-2-yl)-

T33990

Synonym:

Target:

Phenol, m-(2-(dimethylaminomethyl)-1-hydroxycyclopentyl)-

T34001

Synonym:

Target:

m-Dioxan-5-ol, 2-(2-furyl)-

Synonym: 8-Methoxy-2-propionamidotetralin,AH-002

Target: MT Receptor

Phenol, m-(2-(phenethylamino)ethyl)-, hydrochloride

T34006

Synonym:

Target:

m-Acetotoluidide, 2-chloro-N-(2-ethoxyethyl)-

T33149

Synonym:

Target:

m-Acetanisidide, 2-chloro-N-(2-ethoxyethyl)-

Target: MMP, Drug Metabolite

4-Chloro-2-nitro-m-cresol

T29432

Synonym:

Target:

m-Acetotoluidide, 2-fluoro-N-methyl-

T33150

Synonym:

Target:

m-Dioxane, 2-hexyl-2,4-dimethyl-

T33254

Synonym:

Target:

m-Acetanisidide, 2-(diethylamino)-4'-(octyloxy)-

T33139

Synonym:

Target:

Phenol, m-(2-(N-methylphenethylamino)ethyl)-, hydrobromide

T34005

Synonym:

Target:

Benzoic acid, m-iodo-, 2-phenylhydrazide

T30403

Synonym:

Target:

m-Anisidine, 4-(2-ethylbutoxy)-, hydrobromide

Synonym: Abemaciclib metabolite M2

Target: CDK

m-Dioxan-5-amine, 2-(p-chlorophenyl)-

T33249

Synonym:

Target:

Carbanilic acid, m-(2-methoxyethoxy)-, 2-(diethylamino)ethyl ester

Synonym: 3-methyl 5-(2-methylpropyl) 2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate

Target: Others

m-Acetotoluidide, N-benzyl-2-(diethylamino)-, monohydrochloride

T33156

Synonym:

Target:

m-Dioxane, 5-ethyl-2-(2-furyl)-4-propyl-

T33256

Synonym:

Target:

m-Dioxane, 5,5-bis(chloromethyl)-2-phenyl-

T33255

Synonym:

Target:

Benzoic acid, m-(2-methyl-5-phenylpyrrol-1-yl)-

T30396

Synonym:

Target:

m-Dioxane, 5-ethyl-5-nitro-2-propyl-

T33257

Synonym:

Target:

m-Dioxan-5-amine, 5-benzylaminomethyl-2-phenyl-

T33252

Synonym:

Target:

Benzoic acid, m-(2-(p-bromophenyl)-5-methylpyrrol-1-yl)-

T30392

Synonym:

Target:

m-Dioxan-5-amine, 2-(p-chlorophenyl)-5-methyl-

T33251

Synonym:

Target:

m-Dioxan-5-amine, 2-(p-chlorophenyl)-5-ethyl-

T33250

Synonym:

Target:

Phenol, m-(2-(N-ethylphenethylamino)ethyl)-, fumarate (1:1)

T34004

Synonym:

Target:

Phenol, m-(1-methyl-3-(2-methylbutyl)-3-pyrrolidinyl)-

T33995

Synonym:

Target:

Phenol, m-(2-ethyl-1-methyl-3-propyl-3-pyrrolidinyl)-

T34009

Synonym:

Target:

N,N-Bis(2-chloroethyl)-m-iodobenzylamine

T30358

Synonym: Benzenemethanamine, N,N-bis(2-chloroethyl)-3-iodo- (9CI)

Target:

m-Acetanisidide, N-(2-(diethylamino)ethyl)-2-(p-ethoxyphenoxy)-, monopicrate

T33142

Synonym:

Target:

Carbanilic acid, m-((pentyloxy)methyl)-, 2-piperidinoethyl ester, hydrochloride

T30720

Synonym:

Target:

カタログ番号	製品名	別名	ターゲット
T2764	(S)-10-Hydroxycamptothecin	10-Hydroxycamptothecin,10-HCPT	Apoptosis , Topoisomerase
	(S)-10-Hydroxycamptothecin (10-HCPT) is a DNA topoisomerase I inhibitor, utilized as a clinical therapy agent against hepatoma.		Apoptosis , Topoisomerase
T13535	Aflatoxin M2		Others
	Aflatoxin M2 is a major metabolite of Aflatoxin B1. It is a mycotoxin produced by the fungi Aspergillus flavus and Aspergillus parasiticus.		Others
TN1708	Gomisin M2		HIV Protease
	Gomisin M2 is an anti-HIV agent.		HIV Protease
TL0016	Sulforaphene		Apoptosis , ERK , EGFR , NF-κB
	Sulforaphene is a natural product isolated from radish seeds, exhibits an ED50 against velvetleaf seedlings approximately 2 x 10 -4 M. Sulforaphene promotes cancer cells apoptosis and inhibits migration via inhibiting EG...		Apoptosis , ERK , EGFR , NF-κB
T4709	(2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride	D-Mannosamine hydrochloride	Others , Endogenous Metabolite
	(2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride (D-Mannosamine hydrochloride) is a pharmaceutical compound used in the development of mannosylated liposomes for bioadhesive oral drug delivery via M cells ...		Others , Endogenous Metabolite
T6S0109	Sipeimine	Kashmirine,Imperialine	Others
	1. Sipeimine (Kashmirine) has antiasthmatic effect, on tracheal M receptor antagonist. 2. Sipeimine can make Kaba cholinergic induced contraction of tracheal strips of the dose-response curve to the right.		Others
T4S1335	Daphnoretin	Dephnoretin,Thymelol	Influenza Virus , Caspase , PKC
	1. Daphnoretin (Thymelol) has strong antiviral activity, mainly on the later phase of the replication cycle. 2. Daphnoretin has anticancer effects on leukemia, osteosarcoma and uterine cervix cancer cells, might through ...		Influenza Virus , Caspase , PKC
TN2254	Taccalonolide A		Apoptosis , Microtubule Associated
	Taccalonolide A is the first microtubule stabilizing agent to be discovered from a plant since identification of the mechanism of action of paclitaxel and it is the first natural product steroid identified to have these ...		Apoptosis , Microtubule Associated
T6S0071	Fraxinellone		HIF/HIF Prolyl-Hydroxylase , STAT , PD-1/PD-L1
	1. Fraxinellone significantly reduced weight loss and diarrhea in mice and alleviated the macroscopic and microscopic signs of the disease. 2. Fraxinellone exhibited a variety of insecticidal activities including feeding...		HIF/HIF Prolyl-Hydroxylase , STAT , PD-1/PD-L1
T3S0081	Oxypeucedanin	(+-)-Oxypeucedanin,Oxypeucadanin	Potassium Channel
	1. Oxypeucedanin ((+-)-Oxypeucedanin) has novel anticancer effect, mediated via induction of G2-M cell cycle arrest and apoptosis in human prostate carcinoma DU145 cells. 2. Oxypeucedanin is a kind of open-channel blocke...		Potassium Channel
T5S1607	Morusin	Mulberrochromene	NF-κB , Antibacterial , STAT
	1. Morusin (Mulberrochromene) possesses antitumor effects of cell lines including HT-29, A549, MCF-7, and MDA-MB-231, through suppressing STAT3 and NFκB attenuation mediated apoptosis induction. 2. Morusin possesses anti...		NF-κB , Antibacterial , STAT
T2966	Beta-Sitosterol	Cupreol,Beta-Sitosterol,β-Sitosterol,Azuprostat,SKF 14463,22,23-Dihydrostigmasterol,Betaprost	Apoptosis , Lipase , Endogenous Metabolite
	Beta-Sitosterol (SKF 14463) has recently been shown to induce G2/M arrest, endoreduplication, and apoptosis through the Bcl-2 and PI3K/Akt signaling pathways. Beta-Sitosterol (SKF 14463) , a main dietary phytosterol foun...		Apoptosis , Lipase , Endogenous Metabolite
T5S0106	Peimisine	Ebeiensine	RAAS , AChR
	1. Peimisine (Ebeiensine) can affect M-receptor, excit β-receptor, restrain the release of internal calcium, and promote to releaseing nitrogen monoxidum in order to relax tracheal smooth muscle and relieve asthma. 2. Pe...		RAAS , AChR
T3824	Jaceosidin		Apoptosis , BCL , COX , UGT
	Jaceosidin has anti-oxidative activity. Jaceosidin has anti-inflammatory activity, also a microglial inhibitor with anti-neuroinflammation activity. aceosidin has anticancer activity, modulates the ERK/ATM/Chk1/2 pathway...		Apoptosis , BCL , COX , UGT
T5S0055	Chelidonine	Helidonine,Khelidonin,Stylophorin	Apoptosis , Others , Influenza Virus
	1. Chelidonine (Stylophorin) isolated from Chelidonium majus efficiently induced apoptosis in HeLa cells through possible alteration of p38-p53 and AKT/PI3 kinase signalling pathways. 2. Chelidonine is a promising model ...		Apoptosis , Others , Influenza Virus
T3895	Polyphyllin I		Apoptosis , Akt , JNK , PDK , mTOR , Autophagy
	Polyphyllin D induces apoptosis via the mitochondrial apoptotic pathway as evidenced by decreased Bcl-2 expression levels, disruption of MMP and increased Bax, cytochrome C, and cleaved-caspase-3 levels. Polyphyllin D ha...		Apoptosis , Akt , JNK , PDK , mTOR , Autophagy
T0186	Docetaxel trihydrate	RP-56976 (Trihydrate),RP56976 (NSC 628503) Trihydrate	Apoptosis , BCL , Microtubule Associated
			Apoptosis , BCL , Microtubule Associated
T5S0661	Koumine		Others
	1. Koumine can treat the diabetic neuropathy. 2. Koumine has antineoplastic effect, may be a future breast cancer chemotherapeutic agent. 3. Koumine has a significant analgesic effect in rodent behavioral models of infla...		Others
T3779	Crocin II	Crocin 2,Crocetin gentiobiosylglucosyl ester,Tricrocin,Crocin B	Caspase , COX , NO Synthase
	Crocin II (Crocetin gentiobiosylglucosyl ester) has anti-inflammatory and anti-apoptotic effects against gastric ischemia-reperfusion injury in rats, the effect of crocin is mainly mediated by reducing the protein expres...		Caspase , COX , NO Synthase
T38019	Nybomycin
	Nybomycin is a fungal metabolite originally isolated from Streptomyces sp. A717 and has antibacterial activity. It is active against B. subtilis, B. cereus, B. mycoides, M. smegmatis, and K. pneumoniae (MICs = 0.025, 2, ...
T78479	Manool
	Manool, a diterpene derived from Salvia officinalis, demonstrates selective cytotoxicity in cancer cells and causes cell cycle arrest at the G(2)/M phase [1] [2].
TN2116	Pteropodine		BCL , Calcium Channel , 5-HT Receptor
	Pteropodine acts as a positive modulator of muscarinic M(1) and 5-HT(2) receptors. Pteropodine shows antigenotoxic, antioxidant and lymphocyte induction effects, it also shows strong apoptotic effect on acute leukaemic l...		BCL , Calcium Channel , 5-HT Receptor
T79947	10-Hydroxyaloin A		SARS-CoV
	Hydroxyaloin A (10-10-Hydroxyaloin A) is a potent inhibitor of SARS-CoV-2, demonstrating significant efficacy in binding to the active site of the SARS-CoV-2 main protease (M^pro) [1].		SARS-CoV
T72581	SARS-CoV MPro-IN-2
	SARS-CoV MPro-IN-2 effectively inhibits the SARS-CoV-2 main protease (M pro), crucial for the virus's replication and transcription in host cells, with an IC50 value of 72.07 nM. Given its significant role in processing ...
T81991	Kaempferol-3-O-[2″,6″-di-O-E-p-coumaroyl]-β-D-glucopyranoside
	Kaempferol-3-O-[2″,6″-di-O-E-p-coumaroyl]-β-D-glucopyranoside, an acylated kaempferol glucoside, can be extracted from the leaves of O. dentata and functions as a repellent to the fouling organism, the blue mussel M. edu...
T36931	Penicillide
	Penicillide is a fungal metabolite originally isolated from Penicillium that has diverse biological activities. It is an inhibitor of calpain 2/m-calpain (IC50 = 7.1 μM) and acyl-coenzyme A:cholesterol acyltransferase (A...
TN6059	Demethoxyfumitremorgin C
	Demethoxyfumitremorgin C and tryprostatin B are fungal inhibitors of mammalian cell cycle progression at the G(2)/M transition. Demethoxyfumitremorgin C inhibits the proliferation of PC3 human prostate cancer cells via t...
T75602	Albanol B
	Albanol B, an arylbenzofuran derivative, is extracted from mulberries and demonstrates multifarious biological activities, including anti-Alzheimer's, anti-bacterial, and antioxidant effects. It inhibits the proliferatio...
T14121	Actinonin	(-)-Actinonin	Aminopeptidase
			Aminopeptidase
T35609	19-O-Acetylchaetoglobosin A
	19-O-Acetylchaetoglobosin A is a fungal metabolite originally isolated fromC. globosumthat has actin polymerization inhibitory and cytotoxic activities.1,2It inhibits actin polymerization in a cell-free assay when used a...
T38330	Collinin
	Collinin is a coumarin that has been found in Z. schinifolium and has diverse biological activities.1,2,3,4 It is active against drug-susceptible and -resistant strains of M. tuberculosis (MIC50s = 3.13-6.25 μg/ml).1 Col...
T36417	Nargenicin	Antibiotic 47444
	Nargenicin is a macrolide antibiotic that selectively inhibits the growth of S. aureus, methicilin resistant S. aureus (MRSA), and M. luteus (MICs = 0.6, 0.3, and 2.5 μg/ml, respectively) over a panel of 11 Gram-positive...
T37690	Phenylpyropene A
	Phenylpyropene A is a fungal metabolite originally isolated from P. griseofulvum that has enzyme inhibitory and insecticidal activities.1,2,3 It inhibits acyl-coenzyme A:cholesterol acyltransferase (ACAT; IC50 = 0.8 μM)....
T35667	Napyradiomycin A1	Napyradiomycin A1
	Napyradiomycin A1is a fungal metabolite originally isolated fromC. rubraand has diverse biological activities.1,2It is active againstS. aureus,M. luteus,B. anthracis,C. bovis, andM. smegmatis(MICs = 1.56-12.5 μg/ml).1Nap...
T36791	Lysophosphatidylcholine 18:2
	1-Linoleoyl-2-hydroxy-sn-glycero-3-PC (LGPC) is a lysophospholipid containing linoleic acid at thesn-1 position that has been found in mouse heart, lung, liver, spleen, kidney, plasma, and serum.1Serum levels of LGPC dec...
T35752	Xanthoquinodin A1	Xanthoquinodin A1
	Xanthoquinodin A1 is a fungal metabolite that has been found inHumicolaand has diverse biological activities.1,2It inhibitsE. tenellaschizont formation in BHK-21 cells with a minimum effective concentration (MEC) value o...
T37451	Stachybotrysin B
	Stachybotrysin B is a fungal metabolite originally isolated from S. chartarum and has antiviral and anticancer activities.1,2 It has antiviral activity against HIV in SupT1 cells (IC50 = 19.2 μM).1 Stachybotrysin B is cy...
T36915	21-Deoxycortisol
	21-Deoxycortisol is a corticosteroid metabolite of 17-hydroxyprogesterone produced in the adrenal glandvia11-hydroxylation by 11β-hydroxylase.1,2Serum levels of 21-deoxycortisol are elevated in patients with congenital a...
T36295	Echistatin TFA
	Echistatin TFA, the smallest active RGD protein belonging to the family of disintegrins that are derived from snake venoms, is a potent inhibitor of platelet aggregation. Echistatin is a potent inhibitor of bone resorpti...
T35741	Gliovirin
	Gliovirin is a fungal metabolite that has been found inT. harzianumand has fungicidal, antimicrobial and anti-inflammatory activities.1It is active against the plant pathogenic fungusP. ultimum(MIC = 60 ng/ml) and the pa...
T36179	Aspulvinone O
	Aspulvinone O is a fungal metabolite that has been found in P. variotti and has antioxidant and anticancer activities.1,2 It scavenges 2,2-diphenyl-1-picrylhydrazyl radicals in a cell-free assay (IC50 = 11.6 μM).1 Aspulv...
T36563	(E)-Guggulsterone
	Bile acids are essential for solubilization and transport of dietary lipids, are the major products of cholesterol catabolism, and are physiological ligands for farnesoid X receptor (FXR), a nuclear receptor that regulat...
T37272	9(S),12(S),13(S)-TriHOME
	9(S),12(S),13(S)-TriHOME is a linoleic acid-derived oxylipin that has diverse biological activities.1,2,3,4It has been found in various plants and is produced in human eosinophils in a 15-lipoxygenase-dependent, soluble ...
T38069	Aquastatin A
	Aquastatin A is a fungal metabolite originally isolated fromF. aquaeductuumthat has diverse biological activities.1It is active againstS. aureus(MIC = 32 μg/ml) and inhibits enoyl-acyl carrier protein reductase (Fabl; IC...
T36348	Cerebroside C
	Cerebroside C is a fungal metabolite and glycosphingolipid that has been found in the rice pathogenic fungusM. grisea.1It induces production of the phytoalexin momilactone A when applied to wounded rice leaves, indicatin...
T35779	Oosporein
	Oosporein is a mycotoxin that has been found inBeauveriaand has diverse biological activities.1,2It is cytotoxic to Sf9 and Sf21 insect cells with 50% cytotoxic concentration (CC50) values of 4.23 and 10.43 μM, respectiv...

天然物製品

(S)-10-Hydroxycamptothecin

T2764

Synonym: 10-Hydroxycamptothecin,10-HCPT

Target: Apoptosis, Topoisomerase

Target: Apoptosis, ERK, EGFR, NF-κB

(2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride

T4709

Synonym: D-Mannosamine hydrochloride

Target: Others, Endogenous Metabolite

Sipeimine

T6S0109

Synonym: Kashmirine,Imperialine

Target: Others

Daphnoretin

T4S1335

Synonym: Dephnoretin,Thymelol

Target: Influenza Virus, Caspase, PKC

Taccalonolide A

TN2254

Synonym:

Target: Apoptosis, Microtubule Associated

Fraxinellone

T6S0071

Synonym:

Target: HIF/HIF Prolyl-Hydroxylase, STAT, PD-1/PD-L1

Oxypeucedanin

T3S0081

Synonym: (+-)-Oxypeucedanin,Oxypeucadanin

Target: Potassium Channel

Morusin

T5S1607

Synonym: Mulberrochromene

Target: NF-κB, Antibacterial, STAT

Beta-Sitosterol

T2966

Synonym: Cupreol,Beta-Sitosterol,β-Sitosterol,Azuprostat,SKF 14463,22,23-Dihydrostigmasterol,Betaprost

Target: Apoptosis, Lipase, Endogenous Metabolite

Target: Apoptosis, BCL, COX, UGT

Chelidonine

T5S0055

Synonym: Helidonine,Khelidonin,Stylophorin

Target: Apoptosis, Others, Influenza Virus

Polyphyllin I

T3895

Synonym:

Target: Apoptosis, Akt, JNK, PDK, mTOR, Autophagy

Docetaxel trihydrate

T0186

Synonym: RP-56976 (Trihydrate),RP56976 (NSC 628503) Trihydrate

Target: Apoptosis, BCL, Microtubule Associated

Synonym: Crocin 2,Crocetin gentiobiosylglucosyl ester,Tricrocin,Crocin B

Target: Caspase, COX, NO Synthase

Target: BCL, Calcium Channel, 5-HT Receptor

Kaempferol-3-O-[2″,6″-di-O-E-p-coumaroyl]-β-D-glucopyranoside

Demethoxyfumitremorgin C

Synonym: (-)-Actinonin

Target: Aminopeptidase

19-O-Acetylchaetoglobosin A

Synonym: Antibiotic 47444

Synonym: Napyradiomycin A1

Target:

Lysophosphatidylcholine 18:2

Synonym: Xanthoquinodin A1

9(S),12(S),13(S)-TriHOME

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPH-01031	CAPN2 Protein, Human, Recombinant (His)	Human	E. coli
	Calcium-regulated non-lysosomal thiol-protease which catalyzes limited proteolysis of substrates involved in cytoskeletal remodeling and signal transduction. Proteolytically cleaves MYOC at 'Arg-226'. Proteolytically cle...
TMPH-03474	Beta-lactamase CTX-M-2 Protein, Salmonella typhimurium, Recombinant	Salmonella typhimurium	E. coli
	Has cefotaxime-hydrolyzing activity. Beta-lactamase CTX-M-2 Protein, Salmonella typhimurium, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 28.4 kDa and the accession number is P...
TMPY-01037	CSF1R Protein (Met1-Glu512), Human, Recombinant (His)	Human	HEK293 Cells
	CSF1R Protein (Met1-Glu512), Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 56 kDa and the accession number is P07333-1.
TMPY-02630	B2M/beta 2-Microglobulin Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	B2M/beta 2-Microglobulin Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 13 kDa and the accession number is P01887.
TMPY-04764	PCK2 Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	PCK2 promotes tumor initiation by lowering acetyl-CoA level through reducing the mitochondrial tricarboxylic acid (TCA) cycle. The levels of phosphoenolpyruvate carboxykinase isoform 2 (PCK2) are critical for the metabol...
TMPY-01563	PMP2 Protein, Human, Recombinant (His)	Human	E. coli
	Myelin P2 protein, also known as PMP2, is a cytosolic protein found primarily in peripheral nerves. It Belongs to the calycin superfamily. Fatty-acid binding protein (FABP) family. PMP2 is a small, basic, and cytoplasmic...
TMPH-03088	Arginine kinase/AK Protein, Penaeus monodon, Recombinant (His & SUMO)	Penaeus monodon	E. coli
	N/A. Arginine kinase/AK Protein, Penaeus monodon, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 56.0 kDa and the accession number is C7E3T4.
TMPK-00415	M-CSFR/CSF1R/CD115 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	M-CSFR/CSF1R/CD115 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 57.4 kDa and the accession number is P07333-1.
TMPK-00656	M-CSFR/CSF1R/CD115 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	M-CSFR/CSF1R/CD115 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 56.3 kDa and the accession number is G7P8P1.
TMPK-00414	M-CSFR/CSF1R/CD115 Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	M-CSFR/CSF1R/CD115 Protein, Human, Recombinant (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 57.4 kDa and the accession number is P07333-1.
TMPY-05436	CSF1R Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	CSF1R Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 81.9 kDa and the accession number is P09581.
TMPY-01833	CSF1R Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	CSF1R Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 56.8 kDa and the accession number is P09581.
TMPY-04938	CSF1R Protein, Mouse, Recombinant (His), Biotinylated	Mouse	HEK293 Cells
	CSF1R Protein, Mouse, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 56.8 kDa and the accession number is P09581.
TMPK-01062	RGMC Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	RGM gene family ('Repulsive Axonal Guidance molecules' A, B and C),both RGM A and B are mostly expressed in central nervous system, while RGM C is exclusively expressed in all striated muscle and in the myocardium. RGM A...
TMPY-02128	Serpin B1 Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	SerpinB1 is an endogenous inhibitor of serine proteases recognized for its anti-inflammatory and host-protective properties. Serum SerpinB1 levels are elevated in patients with type 2 diabetes compared with that in healt...
TMPJ-00395	SEMA4D Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	SEMA4D is a member of the semaphorin family,contains one Ig-like C2-type domain, one PSI domain and one Sema domain. SEMA4D is strongly expressed in lymphoid tissues, especially in the thymus, as well as in the nervous t...
TMPY-05513	CSF1R Protein (Ala299-Glu512), Human, Recombinant (His)	Human	HEK293 Cells
	CSF1R Protein (Ala299-Glu512), Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.3 kDa and the accession number is P07333-1.
TMPY-04358	CSF1R Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	CSF1R Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 76 kDa and the accession number is P07333-1.
TMPY-06384	CSF1R Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	CSF1R Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 57.76 kDa and the accession number is P07333-1.
TMPY-05264	CSF1R Protein, Human, Recombinant (mFc)	Human	HEK293 Cells
	CSF1R Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 81.5 kDa and the accession number is P07333-1.
TMPY-06389	CSF1R Protein, Human, Recombinant (hFc & Avi), Biotinylated	Human	HEK293 Cells
	CSF1R Protein, Human, Recombinant (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with hFc and Avi tag. The predicted molecular weight is 83.04 kDa and the accession number is P07333-1.
TMPY-05045	CSF1R Protein, Human, Recombinant (Domain I&II&III, His)	Human	HEK293 Cells
	CSF1R Protein, Human, Recombinant (Domain I&II&III, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 31.1 kDa and the accession number is P07333-1.
TMPY-05429	CSF1R Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	CSF1R Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 81.2 kDa and the accession number is P07333-1.
TMPY-00881	CSF1R Protein, Human, Recombinant	Human	HEK293 Cells
	CSF1R Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 55.1 kDa and the accession number is P07333-1.
TMPY-00127	M-CSF/CSF1 Protein, Human, Recombinant	Human	HEK293 Cells
	M-CSF/CSF1 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 18.4 kDa and the accession number is P09603-2.
TMPJ-00327	M-CSF/CSF1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Macrophage Colony-Stimulating Factors (m-csf) are cytokines that act in hematopoiesis by controlling the production, differentiation, and function of 2 related white cell populations of the blood, the granulocytes and th...
TMPY-01280	FOLR2 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Folate receptor beta, also known as Folate receptor 2, FBP, and FOLR2, is a member of the folate receptor family. FOLR2 is expressed in placenta and hematopoietic cells. The expression of FOLR2 is increased in malignant ...
TMPY-05181	M-CSF/CSF1 Protein, Human, Recombinant, Biotinylated	Human	HEK293 Cells
	M-CSF/CSF1 Protein, Human, Recombinant, Biotinylated is expressed in HEK293 mammalian cells. The predicted molecular weight is 18.4 kDa and the accession number is P09603-2.
TMPY-04229	M-CSF/CSF1 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	M-CSF/CSF1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 51.9 kDa and the accession number is P09603-2.
TMPK-01395	TENM2 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Teneurin-2 is a member of a novel family of transmembrane proteins characterized to date in fish, birds, mammals, and Drosophila (e.g., the pair-rule gene product Ten-m). Teneurin-2, a vertebrate homologue of the Drosoph...
TMPH-02246	TGS1 Protein, Human, Recombinant (His & SUMO)	Human	E. coli
	Catalyzes the 2 serial methylation steps for the conversion of the 7-monomethylguanosine (m(7)G) caps of snRNAs and snoRNAs to a 2,2,7-trimethylguanosine (m(2,2,7)G) cap structure. The enzyme is specific for guanine, and...
TMPY-00005	FGF-8a Protein, Human, Recombinant	Human	E. coli
	In mammalian embryos, transient Fgf8 expression defines the developing isthmic region, lying between the midbrain and the first rhombomere, but there has been uncertainty about the existence of a distinct isthmic segment...
TMPY-00891	Neuropilin-1 Protein, Human, Recombinant (V179A, hFc)	Human	HEK293 Cells
	Neuropilin-1 Protein, Human, Recombinant (V179A, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 96.5 kDa and the accession number is O14786-2.
TMPY-00748	Nectin-2 Protein, Human, Recombinant	Human	HEK293 Cells
	Nectin-2 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 36.2 kDa and the accession number is Q92692-2.
TMPY-00850	ST2/IL-1 RL1 Protein, Human, Recombinant	Human	HEK293 Cells
	ST2/IL-1 RL1 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 35.6 kDa and the accession number is Q01638-2.
TMPY-00871	LAYN Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	LAYN Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 49.5 kDa and the accession number is Q6UX15-2.
TMPY-04116	KRAS Protein,Human,Recombinant(G12C & Q61H, His)	Human	E. coli
	KRAS Protein,Human,Recombinant(G12C & Q61H, His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 23.3 kDa and the accession number is P01116-2.
TMPY-05288	PLGF/PGF Protein, Human, Recombinant (aa 19-149)	Human	E. coli
	PLGF/PGF Protein, Human, Recombinant (aa 19-149) is expressed in E. coli expression system. The predicted molecular weight is 14.9 kDa and the accession number is P49763-2.
TMPY-00341	FGFR3 Protein, Human, Recombinant (alpha IIIb, His)	Human	HEK293 Cells
	FGFR3 Protein, Human, Recombinant (alpha IIIb, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40 kDa and the accession number is P22607-2.
TMPY-02792	GDNF Protein, Human, Recombinant (HEK293)	Human	HEK293 Cells
	GDNF Protein, Human, Recombinant (HEK293) is expressed in HEK293 mammalian cells. The predicted molecular weight is 15.1 kDa and the accession number is P39905-2.
TMPY-02011	CD96 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	CD96 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 55 kDa and the accession number is P40200-2.
TMPY-00849	ST2/IL-1 RL1 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	ST2/IL-1 RL1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 61.72 kDa and the accession number is Q01638-2.
TMPY-01691	Clusterin Protein, Human, Recombinant (CLU34, His)	Human	HEK293 Cells
	Clusterin Protein, Human, Recombinant (CLU34, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 51.5 kDa and the accession number is P10909-2.
TMPY-02358	CD98 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	CD98 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 49.2 kDa and the accession number is P10852-2.
TMPJ-01449	3CLpro/3C-like Protease Protein, SARS-CoV-2, Recombinant	SARS-CoV-2	E. coli
	The viral main proteinase (M pro , also called 3CL pro ), which controls the activities of the coronavirus replication complex. It functions as a cysteine protease engaging in the proteolytic cleavage of the viral precur...
TMPH-02884	CTDP1 Protein, Mouse, Recombinant (His & Myc)	Mouse	E. coli
	Processively dephosphorylates 'Ser-2' and 'Ser-5' of the heptad repeats YSPTSPS in the C-terminal domain of the largest RNA polymerase II subunit. This promotes the activity of RNA polymerase II. Plays a role in the exit...
TMPJ-01448	3CLpro/3C-like Protease Protein, SARS-CoV-2, Recombinant (His)	2019-nCoV	E. coli
	The viral main proteinase (M pro , also called 3CL pro ), which controls the activities of the coronavirus replication complex. It functions as a cysteine protease engaging in the proteolytic cleavage of the viral precur...
TMPY-04113	KRAS Protein,Human,Recombinant(G12D & Q61H, His)	Human	E. coli
	KRAS Protein,Human,Recombinant(G12D & Q61H, His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 23.3 kDa and the accession number is P01116-2.
TMPY-01985	CD32B/Fcgr2b Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	CD32B/Fcgr2b Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 24 kDa and the accession number is P31994-2.
TMPY-04844	BTN3A1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	BTN3A1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.6 kDa and the accession number is O00481-2.
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