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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
TP1254 | [Met5]-Enkephalin, amide TFA | 5-Methionine-enkephalin amide (TFA) | Opioid Receptor |
[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors. | |||
TP1113L | [Leu5]-Enkephalin, amide acetate | [Leu5]-Enkephalin, amide acetate(60117-24-0 free base) | Opioid Receptor |
[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist. | |||
TP2446L | Angiotensin amide acetate | Angiotensin amide acetate(53-73-6 Free base) | Others |
Angiotensin amide acetate is a derivative of Angiotensin amide, an octapeptide amide that increases blood pressure through vasoconstriction. | |||
T3984 | GLP-1(7-36), amide | MKC 253,Human GLP-1-(7-36)-amide,Glucagon-like Peptide 1 (7-36) amide,Glucagon-Like Peptide (GLP) I (7-36), amide, human,GLP-1(7-36),GLP-1-(7-36)-amide | Glucagon Receptor |
GLP-1(7-36), amide (MKC 253) is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays various antidiabetic effects by potentiating glucose-... | |||
TP1858L | Phe-Met-Arg-Phe, amide acetate | Phe-Met-Arg-Phe, amide acetate(64190-70-1 freebase) | Potassium Channel |
Phe-Met-Arg-Phe, amide acetate dose dependently (ED50=23 nM) activates a K+ current in the peptidergic caudodorsal neurons. This peptide appears to localize with neuropeptide Y in some regions of the brain. | |||
T7623 | PAR-4 Agonist Peptide, amide | AY-NH2,PAR-4 Agonist Peptide, amide(2TFA),PAR-4-AP | Protease-activated Receptor |
PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4). | |||
TP1378 | 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) | 2-Furoyl-LIGRLO-amide | Protease-activated Receptor |
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist. | |||
TP1002L | γ-1-MSH, amide acetate (72629-65-3 free base) | γ-1-MSH, amide acetate | Others |
γ-1-MSH, amide acetate (72629-65-3 free base), a putative hormone in the N-terminal region of the ACTH/beta- endorphin (beta-EP) precursor protein, was studied by RIA with an antiserum against gamma 3-MSH in ACTH-produci... | |||
T0643 | Diclofenac Amide | Others | |
Diclofenac Amide is used as a intermediates of Diclofenac. | |||
T21983L | PKI 14-22 amide, myristoylated Acetate | PKI 14-22 amide, myristoylated Acetate(201422-03-9 Free base) | PKA |
PKI 14-22 amide, myristoylated Acetate inhibit cAMP-dependent protein kinase (PKA) and blocks hyperalgesia produced by spinal administration of 8-bromo-cAMP. | |||
T37891L | GLP-1(32-36)amide acetate | GLP-1(32-36)amide acetate(1417302-71-6 Free base) | Others |
GLP-1(32-36)amide acetate is a pentapeptide and derived from the C terminus of the glucoregulatory hormone GLP-1. GLP-1(32-36)amide acetate could inhibit weight gain and modulate whole body glucose metabolism in diabetic... | |||
T75888 | PKA Inhibitor Fragment (6-22) amide TFA | PKI-(6-22)-amide TFA,PKA Inhibitor Fragment (6-22) amide TFA(121932-06-7 Free base) | PKA |
PKA Inhibitor Fragment (6-22) amide TFA (PKA Inhibitor Fragment (6-22) amide TFA) is an inhibitor of the highly potent cAMP-dependent protein kinase A (PKA) inhibitor (Ki: 2.8 nM).PKA Inhibitor Fragment (6-22) amide TFA ... | |||
T37890L | GLP-1(28-36)amide acetate | GLP-1(28-36)amide acetate(1225021-13-5 Free base) | Antioxidant , Glucagon Receptor |
GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities. | |||
T38852L | TRAP-6 amide acetate | Protease-activated Receptor | |
TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1]. | |||
T5518 | N-acetylcysteine amide | Reactive Oxygen Species , ROS | |
N-Acetylcysteine amide is a thiol antioxidant and neuroprotective agent that can permeate cell membranes and the blood-brain barrier. | |||
TP1793L | Nociceptin (1-13) amide TFA | Opioid Receptor | |
Nociceptin (1-13), amide is a potent agonist Opioid receptor-like1 (ORL1) receptor with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain membranes. | |||
T9417L | Gamma-preprotachykinin amide (72-92) acetate | gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base) | Others |
gamma-preprotachykinin amide (72-92) acetate is a 21 amino acid peptide belonging to the tachykinin (TK) family and including neurokinin A (NKA) in its C-terminal sequence. gamma-preprotachykinin amide (72-92) acetate po... | |||
TP2252 | GLP-1 (9-36) amide | Glucagon Receptor | |
antagonist at the human GLP-1 receptor | |||
T38063 | N-Acetyl lysyltyrosylcysteine amide | Glutathione Peroxidase | |
N-Acetyl lysyltyrosylcysteine amide is a non-toxic myeloperoxidase (MPO) tripeptide inhibitor that is potent, reversible, and specific.N-Acetyl lysyltyrosylcysteine amide effectively inhibits MPO production in vivo. N-Ac... | |||
T37588L | GIP (1-30) amide, porcine acetate | IGF-1R | |
GIP (1-30) amide, porcine acetate is an agonist of fully glucose-dependent insulinotropic polypeptide (GIP) receptor. GIP (1-30) amide, porcine acetate can weakly inhibit gastric acid secretion and strongly stimulate ins... | |||
T21674L | PKA inhibitor fragment (6-22) amide Acetate | PKA inhibitor fragment (6-22) amide Acetate(121932-06-7 Free base) | PKA |
PKA inhibitor fragment (6-22) amide Acetate is a synthetic peptide which selectively inhibits PKA activity by binding to its substrate site (IC50 < 2 nM). | |||
TP1140L | Neuropeptide Y (29-64), amide, human acetate | Neuropeptide Y Receptor | |
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity. | |||
TP1250L | Acetyl-PHF6 amide acetate(878663-43-5 freebase) | AcPHF6 acetate,Ac-VQIVYK-NH2 acetate | Others |
Acetyl-PHF6 amide acetate(878663-43-5 freebase) (AcPHF6 acetate) is a tau derived hexapeptide. | |||
TP2212L | A-MSH, amide Acetate(581-05-5 free base) | Melanocortin Receptor | |
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities. α-MSH is a post-translational derivative of pro-opiomelano... | |||
TP1065 | PAR-4 Agonist Peptide, amide TFA | PAR-4-AP (TFA),AY-NH2 (TFA) | Protease-activated Receptor |
PAR-4 Agonist Peptide, amide TFA (PAR-4-AP (TFA)), is a selective activator of the proteinase-activated receptor-4 (PAR-4), demonstrating specificity by not influencing PAR-1 or PAR-2, and its activity can be inhibited b... | |||
T17580 | Biotin-PEG4-Amide-C6-Azide | Others , PROTAC Linker | |
Biotin-PEG4-Amide-C6-Azide is a PEG-based PROTAC linker that can be used in PROTAC synthesis. | |||
T7513 | Protease-Activated Receptor-2, amide | SLIGKV-NH2 | Protease-activated Receptor |
Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M) | |||
T9691L | (D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate | Thyroid hormone receptor(THR) | |
(D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate is a highly potent antagonist of parathyroid hormone (PTH) The Ki value is 69 nM in bovine renal cortical membrane. | |||
T37618 | Leukotriene B4 dimethyl amide | Leukotriene B4 dimethyl amide | |
LTB4 dimethyl amide is a moderate inhibitor of LTB4-induced degranulation of human neutrophils (Ki = 130 nM) and lysozyme release from rat PMNL. LTB4 dimethyl amide appears to be an antagonist of the LTB4 receptor on gui... | |||
T38756 | Thiol-C10-amide-PEG8 | Thiol-C10-amide-PEG8 | |
Thiol-C10-amide-PEG8 is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome sys... | |||
T25474 | GW-Amide | Glycyl-tryptophanamide,GW Amide | |
GW-Amide is a molluscan neuropeptide that exhibits potent modulatory effects on molluscan muscles. | |||
TP1183 | Amylin, amide, human | DAP amide, human | |
Amylin, a 37-amino acid polypeptide that is structurally related to calcitonin, is secreted from the B cells of the pancreas. Amylin has anoretic effects in rats. Amylin may be responsible for the etiology of insulin res... | |||
T39900 | Thalidomide-O-amide-C5-NH2 | Thalidomide-O-amide-C5-NH2 | |
Thalidomide-O-amide-C5-NH2 is a chemically synthesized conjugate, serving as an E3 ligase ligand-linker, which combines a cereblon ligand derived from Thalidomide with a linker that is commonly employed in PROTAC technol... | |||
T39791 | Mal-amide-PEG2-oxyamine-Boc | Mal-amide-PEG2-oxyamine-Boc | |
Mal-amide-PEG2-oxyamineBoc is a polyethylene glycol (PEG)-based linker molecule that possesses a Boc-protected oxyamine functionality. This compound serves as a valuable tool in the efficient synthesis of PROTACs (proteo... | |||
T35471 | A 410099.1 amide-PEG3-amine | A 410099.1 amide-PEG3-amine | |
Functionalized IAP ligand for PROTAC research and development; incorporates an IAP ligand plus a short amide-PEG linker with terminal amine ready for conjugation to a target protein ligand. Part of a range of functional... | |||
T36285 | VH 032 amide-PEG1-acid | VH 032 amide-PEG1-acid | |
Functionalized von-Hippel-Lindau (VHL) protein ligand for PROTAC research and development; incorporates an E3 ligase ligand plus a PEG1 linker with terminal carboxylic acid ready for conjugation to a target protein lig... | |||
T36279 | VH 032 amide-alkylC3-amine | VH 032 amide-alkylC3-amine | |
Functionalized von-Hippel-Lindau (VHL) protein ligand for PROTAC research and development; incorporates an E3 ligase ligand plus an alkyl C3 linker and terminal amine ready for conjugation to a target protein ligand. Pa... | |||
T36278 | VH 032 amide-alkylC3-acid | VH 032 amide-alkylC3-acid | |
Functionalized von-Hippel-Lindau protein ligand (VHL) for research and development; incorporates an E3 ligase ligand plus alkylC3 linker with terminal carboxylic acid ready for conjugation to a target protein ligand. Par... | |||
TP1255 | [Met5]-Enkephalin, amide | 5-Methionine-enkephalin amide | |
[Met5]-Enkephalin, amide is an agonist for δ opioid receptors as well as putative ζ (zeta) opioid receptors.Met-enkephalin circulates in several forms, some of which may be derived from proteins other than proenkephalin ... | |||
T38784 | Histone H3 (1-25), amide | Histone H3 (1-25), amide | |
Histone H3 (1-25), amide is a N-terminal peptide fragment of histone H3 that serves as a substrate for histone methyltransferases (HMTs). It can be utilized to identify the substrate for HMTs. Compared to histone H3 (15-... | |||
T35469 | A 410099.1 amide-alkylC4-amine | A 410099.1 amide-alkylC4-amine | |
Functionalized IAP ligand for PROTAC research and development; incorporates an IAP ligand plus an amide-alkylC4 linker with terminal amine ready for conjugation to a target protein ligand. Part of a range of functionali... | |||
T35470 | A 410099.1 amide-PEG2-amine | A 410099.1 amide-PEG2-amine | |
Functionalized IAP ligand for PROTAC research and development; incorporates an IAP ligand plus a short amide-PEG linker with terminal amine ready for conjugation to a target protein ligand. Part of a range of functional... | |||
T35472 | A 410099.1 amide-PEG4-amine | A 410099.1 amide-PEG4-amine | |
Functionalized IAP ligand for PROTAC research and development; incorporates an IAP ligand plus an amide-PEG4 linker with terminal amine ready for conjugation to a target protein ligand. Part of a range of functionalized... | |||
T36281 | VH 032 amide-alkylC5-amine | VH 032 amide-alkylC5-amine | |
Functionalized von-Hippel-Lindau protein ligand (VHL) for PROTAC research and development; incorporates an E3 ligase ligand plus an alkyl linker with terminal amine ready for conjugation to a target protein ligand. Part ... | |||
T36277 | VH 032 amide-alkylC2-acid | VH 032 amide-alkylC2-acid | |
Functionalized von-Hippel-Lindau protein ligand (VHL) for PROTAC research and development; incorporates an E3 ligase ligand plus alkylC2 linker with terminal carboxylic acid ready for conjugation to a target protein lig... | |||
T36267 | VH 032 amide-PEG4-amine | VH 032 amide-PEG4-amine | |
Functionalized von-Hippel-Lindau protein ligand (VHL) for PROTAC research and development; incorporates an E3 ligase ligand plus a PEG linker ready for conjugation to a target protein ligand. Part of a range of function... | |||
T36283 | VH 032 amide-alkylC8-acid | VH 032 amide-alkylC8-acid | |
Functionalized von-Hippel-Lindau protein ligand (VHL) for PROTAC research and development; incorporates an E3 ligase ligand plus alkylC8 linker with terminal carboxylic acid ready for conjugation to a target protein lig... | |||
T36280 | VH 032 amide-alkylC4-acid | VH 032 amide-alkylC4-acid | |
Functionalized von-Hippel-Lindau protein ligand (VHL) for PROTAC research and development; incorporates an E3 ligase ligand plus alkylC4 linker with terminal carboxylic acid ready for conjugation to a target protein lig... | |||
T38999 | Biotin-C4-amide-C5-NH2 | Biotin-C4-amide-C5-NH2 | |
Biotin-C4-amide-C5-NH2 is a cleavable linker employed for the synthesis of antibody-drug conjugates (ADCs). | |||
T0823 | Thioctamide | Lipoamide,Thioctic acid amide | Others |
Thioctamide (Thioctic acid amide) is a trivial name for 6, 8-dithiooctanoic amide. It is 6, 8-dithiooctanoic acid's functional form where the carboxyl group is attached to protein (or any other amine) by an amide linkage... |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
TP1232L | Amylin, amide, rat acetate(124447-81-0,free base) | Amylin Receptor | |
Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors. | |||
T13802 | Oleamide | Oleic acid amide | Others , Endogenous Metabolite |
Oleamide (Oleic acid amide) is an endogenous fatty acid amide and can be used in the synthesis of de novo in the mammalian nervous system. | |||
T22455 | Vindesine sulfate | DVA,Desacetylvinblastine amide,DAVA,Desacetyl Vinblastine amide,VDS | Others |
Vindesine sulfate (Desacetyl Vinblastine amide) is a vinca alkaloid which is a synthetic derivative of vinblastine, binds to the microtubular proteins of the mitotic spindle, leading to crystallization of the microtubule... | |||
T7445 | Acetamide | ethanamide,Acetic acid amide | Endogenous Metabolite |
Acetamide (ethanamide) is found in red beetroot,is used primarily as a solvent and a plasticizer. | |||
T20091 | Stearamide | Stearic acid amide,NSC 66462,NSC66462,NSC-66462 | |
Stearamide(Stearic acid amide) is a primary fatty acid amide that is cytotoxic and fish toxic and can be used to increase the properties of nanoparticles. | |||
T1426 | Pyrazinamide | Pyrazinoic acid amide,Pyrazinecarboxamide | Antibacterial , Antibiotic , Autophagy , Fatty Acid Synthase |
Pyrazinamide (Pyrazinecarboxamide), an antimycobacterial, is utilized therapeutically as an antitubercular agent, which is a synthetic pyrazinoic acid amide derivative. | |||
T0326L | L-Glutamine | L-Glutamic acid 5-amide | Ferroptosis , Endogenous Metabolite , GluR |
L-Glutamine (L-Glutamic acid 5-amide) , a non-essential amino acid, is synthesized from glutamic acid and ammonia. | |||
T39007 | 3,4-Dimethoxybenzamide | Others | |
3,4-Dimethoxybenzamide, amide, is found in the solid culture of Streptoverticillium morookaense . 3,4-Dimethoxybenzamide can be used as the starting material to preparation Itopride hydrochloride. | |||
TN2085 | Piperlonguminine | Anti-infection , Antibacterial , Antifungal | |
Piperlonguminine is an alkaloid amide isolated from the Piper species. Piperlonguminine shows anti-inflammatory, antitumor, neuroprotective, anti-platelet, anti-melanogenic, antifungal and antibacterial activities.Piperl... | |||
T2859 | Biochanin A | 4-Methylgenistein,Olmelin | EGFR , FAAH , Autophagy |
Biochanin A (4-Methylgenistein) is an isoflavone derivative isolated from red clover Trifolium pratense with anticarcinogenic properties. Biochanin A is a naturally occurring fatty acid amide hydrolase (FAAH) inhibitor. | |||
TN1965 | N-Benzyllinolenamide | N-Benzyllinolenamide | FAAH , Autophagy |
N-Benzyllinolenamide is a natural product. It is an inhibitor of fatty acid amide hydrolase (FAAH, IC50 of 41.8 μM). | |||
T12139 | N-(3-Methoxybenzyl)Palmitamide | FAAH | |
N-(3-Methoxybenzyl)Palmitamide is a promising FAAH inhibitor, treatment of pain, inflammation and CNS degenerative disorders. | |||
T3S2105 | N-Benzylpalmitamide | Macamide 1,N-Benzylhexadecanamide | Others , FAAH , Autophagy |
N-Benzylpalmitamide (Macamide 1) inhibits fatty acid amide hydrolase (FAAH) in a time-dependent manner and could potentially offer a good alternative for the treatment of pain, inflammation and CNS degenerative disorders... | |||
T4859 | 1-Monomyristin | rac-Glycerol 1-myristate,Glyceryl myristate,Monomyristin,2,3-Dihydroxypropyl tetradecanoate | Others , FAAH , Endogenous Metabolite , Antibacterial , Autophagy , Antifungal |
1-Monomyristin (2,3-Dihydroxypropyl tetradecanoate) , a 1-monoglyceride of myristic acid, has antibacterial activity against several Gram-positive bacterial strains. 1-Myristoyl-rac-glycerol is used in colloidal chemistr... | |||
T1321 | Nonivamide | Nonanoic acid vanillylamide,Pelargonic acid vanillylamide,Vanillyl-N-nonylamide,Pseudocapsaicin | TRP/TRPV Channel |
Nonivamide (Nonanoic acid vanillylamide) is found in herbs and spices. Nonivamide is an alkaloid from Capsicum species Nonivamide is a flavoring ingredient. Nonivamide is an organic compound and a capsaicinoid. It is an ... | |||
T6926 | Palmitoylethanolamide | Mackpeart DR 14V,N-palmitoylethanolamine,Loramine P 256,Impulsin,AM 3112,Palmidrol | Influenza Virus , Endogenous Metabolite , PPAR |
Palmitoylethanolamide (Impulsin) is an endogenously fatty acid amide. It has a role as an anti-inflammatory drug, an antihypertensive agent, a neuroprotective agent and an anticonvulsant.Upon administration, palmitoyleth... | |||
TN4171 | Grossamide | NO Synthase | |
Grossamide (GSE) Grossamide is a lignan amide derived from thioguanosine.6-Thioguanosine (GSE) is a selective and potent miR-210 (miRNA-210) inhibitor.6-Thioguanosine (GSE) is a selective and potent miR-210 (miRNA-210) i... | |||
T4834 | Indole-3-acetamide | 3-Indoleacetamide,3-Indolylacetamide | Others , Endogenous Metabolite |
1H-Indole-3-acetamide (3-Indolylacetamide), also known as auxin amide or 2-(3-indolyl)acetamide, belongs to the class of organic compounds known as 3-alkylindoles. Within the cell, 1H-indole-3-acetamide is primarily loca... | |||
TN7035 | N-benzylpentadecanamide | N-(Phenylmethyl)pentadecanamide | Others |
N-benzylpentadecanamide (N-(Phenylmethyl)pentadecanamide) is a natural product. | |||
TN1966 | N-(3-Methoxybenzyl)Oleamide | N-Benzyloleamide,MAC 18:1 | Antioxidant |
N-(3-Methoxybenzyl)Oleamide (MAC 18:1), an agmatine isolated from Lepidium meyenii, has pharmacological effects on exercise-induced fatigue, which may be related to the modulation of energy metabolism and improvement of ... | |||
T5704 | Entadamide-A-β-D-glucopyranoside | (E)-N-[2-(β-D-Glucopyranosyloxy)ethyl]- | Others |
Entadamide-A-β-D-glucopyranoside ((E)-N-[2-(β-D-Glucopyranosyloxy)ethyl]-) has Anti-inflammatory, analgesic function. | |||
TN7141 | Indole-3-glyoxylamide | 2-(1H-indol-3-yl)-2-oxoacetamide,3-(alpha-Oxoglycyl)-1H-indole,3-Indoleglyoxamide | Others |
Indole-3-glyoxylamide (3-Indoleglyoxamide) is a marine derived natural products found in Spongosorites sp. | |||
TN1558 | N-Vanillyldecanamide | Decylic acid vanillylamide | Others |
N-Vanillyldecanamide (Decylic acid vanillylamide), isolated from fruits of Capsicum annuum, significantly reduced free radical length in alfalfa seedlings in a dose-dependent manner. | |||
TN1457 | Bryonamide B | ||
Bryonamide B is a cucurbitane triterpene that can be extracted from Bryonia aspera. | |||
TN7034 | N-benzyl-heptadecanamide | N-Benzylheptadecanamide | Others |
N-benzyl-heptadecanamide (N-Benzylheptadecanamide) is a macamide in maca. | |||
T5814 | Aurantiamide | TMC-58B | p38 MAPK , NF-κB |
Aurantiamide has anti-cancer, anti-inflammatory and antinociceptive activities, it may suppress the growth of malignant gliomas by blocking autophagic flux.Aurantiamide has an anti-neuroinflammatory effect on LPS stimula... | |||
T4767 | Formamide | Carbamaldehyde,Methanamide,NSC 748,Formimidic acid | Others , Endogenous Metabolite |
Formamide (NSC-748) is a metabolite used for biological monitoring of workers exposed to N-N-dimethylformamide (DMF). There is a case of significant association between ever having been exposed to DMF and subsequent deve... | |||
T12296 | Oleoylethanolamide | N-Oleoylethanolamide,Oleamide MEA,Oleic acid monoethanolamide | Endogenous Metabolite , PPAR |
Oleoylethanolamide (N-Oleoylethanolamide) is a high affinity endogenous agonist of PPAR-α. | |||
T1165 | Ethionamide | Bayer 5312,2-ethylthioisonicotinamide,Ethinamide | Dehydrogenase , CAT , Antibacterial , Antibiotic |
Ethionamide (2-ethylthioisonicotinamide) is a nicotinamide derivative, with antibacterial activity, used to treat tuberculosis. Although the exact mechanism of action of ethionamide is unknown, it may inhibit the synthes... | |||
T8150 | Nudifloramide | 1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide | PARP , Endogenous Metabolite |
Nudifloramide (1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide) is one of the end degradation products of nicotinamide-adenine dinucleotide (NAD). | |||
T0617 | Nicotinamide N-oxide | Nicotinamide-N-oxide,Nicotinamide 1-oxide,1-oxynicotinamide | c-Myc , Endogenous Metabolite , CXCR , Drug Metabolite |
Nicotinamide N-oxide (Nicotinamide 1-oxide) is recognized as an in vivo metabolite of nicotinamide which is a precurser of nicotinamide-adenine dinucleotide (NAD+) in animals. The enzyme that catalyzes the reduction of n... | |||
T0769 | Aceglutamide | N2-Acetylglutamine,α-N-Acetyl-L-glutamine | Amino Acids and Derivatives , Endogenous Metabolite , Autophagy |
Aceglutamide (N2-Acetylglutamine) is an acetyl derivative of the amino acid L-glutamine, used to improve memory. | |||
TN1643 | Ferulamide | 4-Hydroxy-3-methoxycinnamide | PAFR , AChR |
Ferulamide (4-Hydroxy-3-methoxycinnamide), a Ferulic acid derivative, shows potent inhibitory activity against arachidonic acid-induced platelet aggregation. | |||
T13795 | Nicotinamide riboside | Sirtuin | |
Nicotinamide riboside increases NAD[+] levels and activates SIRT1 and SIRT3, culminating in enhanced oxidative metabolism and protection against high fat diet-induced metabolic abnormalities. | |||
T6780 | Benzamide | Amid kyseliny benzoove,Phenylcarboxyamide,Benzoylamide | PARP , Endogenous Metabolite |
Benzamide (Amid kyseliny benzoove), an inhibitor of poly(ADP-ribose) polymerase, is a derivative of benzoic acid. | |||
T26288 | Clovamide | trans-Clovamide,N-trans-Caffeoy-L-dopa | Apoptosis , Influenza Virus , ROS , Antibacterial |
Trans-Clovamide (trans-Clovamide) is a naturally occurring caffeoyl conjugate identified in the antioxidant polyphenolic fraction of cocoa (T. cacao L.) Trans-Clovamide is a potent antioxidantand that has shown neuroprot... | |||
TN2239 | Strictosamide | ATPase , Potassium Channel , Sodium Channel , Parasite , Antifungal | |
Strictosamide possesses antibacterial and antiviral activities, it also may have important effects on inflammation and inflammatory pain. | |||
T5222 | N-(5-Aminopentyl)acetamide | Monoacetylcadaverine,N-Acetylcadaverine,N-Acetyl-1,5-pentanediamine | Others , Endogenous Metabolite |
N-(5-Aminopentyl)acetamide (N-Acetylcadaverine) is the acetylated form of the polyamine cadaverine. Cadaverine is produced by the breakdown of amino acids in living and dead organisms and is toxic in large doses. N-(5-Am... | |||
T14193 | α-Galactosylceramide | KRN7000,α-GalCer | Others |
α-Galactosylceramide (KRN7000) is a synthetic glycolipid with antitumorial and immunostimulatory and is a very potent NKT cell agonist and binds effectively to CD1d. The complex of α-Galactosylceramide and CD1d can bind ... | |||
TN7045 | N-phenethylbenzamide | N-(2-Phenylethyl)benzamide,Solina New Impurity 21,4-(DICHLOROMETHYL)PYRIDINE HCL | Others |
N-phenethylbenzamide (Solina New Impurity 21) is a natural product. | |||
TN7126 | N-Vanillyloctanamide | Others | |
N-Vanillyloctanamide is a capsaicinoid from the fruits of Capsicum annuum L. var. annuum. N-Vanillyloctanamide reduces the radical length of Lactuca sativa seedling, this inhibition being dose-dependent. | |||
T8120 | N-Benzyloctadecanamide | N-Benzylstearamide | Others |
N-Benzyloctadecanamide is a distinct class of secondary metabolites in Lepidium meyenii Walp. (Maca). | |||
TN7036 | N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide | (9Z,12Z,15Z)-N-[(3-Methoxyphenyl)methyl]-9,12,15-octadecatrienamide,Macamide Impurity 14 | Wnt/beta-catenin |
N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide (Macamide Impurity 14) induces osteogenic differentiation and subsequent bone formation of mesenchymal stem cells by activating the canonical Wnt/β-catenin signaling pa... | |||
T66582 | 6-Methylnicotinamide | Endogenous Metabolite | |
6-Methylnicotinamide is a derivative of nicotinamide, an endogenous metabolite. 6-Methylnicotinamide is used to make co-crystals/salts. In the acute phase of cerebral hemorrhage (ICH), a sudden increase in 6-Methylnicoti... | |||
T5233 | N-Methylnicotinamide | N'-Methylnicotinamide,Nicotinic Acid Methylamide,N-Methylpyridine-3-carboxamide | Others , Endogenous Metabolite |
N-Methylnicotinamide (Nicotinic Acid Methylamide) is a metabolite of niacin (or nicotinamide) and is commonly found in human urine. However low levels of urinary excretion of N-Methylnicotinamide (Nicotinic Acid Methylam... | |||
TN1352 | N-(3-Methoxybenzyl-(9z,12z)-octadecadienamide | (9Z,12Z)-N-(3-Methoxybenzyl)octadeca-9,12-dienamide,n-3-methoxybenzyl-9z-12z-octadecadienamide | Drug Metabolite |
N-(3-Methoxybenzyl-(9z,12z)-octadecadienamide ((9Z,12Z)-N-(3-Methoxybenzyl)octadeca-9,12-dienamide) is a Macamide impurity that may be used in the study of metabolic diseases. | |||
T6942 | Picolinamide | 2-Pyridinecarboxamide,2-Carbamoylpyridine,2-Picolinamide,Picolinoylamide | PARP |
Picolinamide (Picolinoylamide) is found to be a strong inhibitor of poly (ADP-ribose) synthetase of nuclei from rat pancreatic islet cells. | |||
T32614 | L-Clausenamide | (-)-Clausenamide | Microtubule Associated |
L-Clausenamide is an alkaloid extracted from the leaves of the yellow bark (Clausena lansium (Lour) skeels) and can be used to improve cognitive function. L-Clausenamide inhibits beta-amyloid (Aβ) toxicity and prevents t... | |||
TN7061 | Yuanamide | Others | |
Yuanamide is a natural compound that belongs to the class of alkaloids. | |||
TN7142 | N-methyl-1H-indole-2-carboxamide | 1H-indole-2-carboxylic acid methylamide,ZINC35137534 | Others |
N-methyl-1H-indole-2-carboxamide (ZINC35137534) is a marine derived natural products found in Neosartorya pseudofischeri. | |||
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カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPH-02561 | CES1C Protein, Mouse, Recombinant (GST) | Mouse | E. coli |
Involved in the detoxification of xenobiotics and in the activation of ester and amide prodrugs. Involved in the extracellular metabolism of lung surfactant. | |||
TMPH-02562 | CES1C Protein, Mouse, Recombinant (His & Myc) | Mouse | HEK293 Cells |
Involved in the detoxification of xenobiotics and in the activation of ester and amide prodrugs. Involved in the extracellular metabolism of lung surfactant. | |||
TMPH-02563 | CES1C Protein, Mouse, Recombinant | Mouse | E. coli |
Involved in the detoxification of xenobiotics and in the activation of ester and amide prodrugs. Involved in the extracellular metabolism of lung surfactant. CES1C Protein, Mouse, Recombinant is expressed in E. coli expr... | |||
TMPH-03260 | Carboxypeptidase A1 Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
Carboxypeptidase that catalyzes the release of a C-terminal amino acid, but has little or no action with -Asp, -Glu, -Arg, -Lys or -Pro. Catalyzes the conversion of leukotriene C4 to leukotriene F4 via the hydrolysis of ... | |||
TMPY-01189 | GFPT1 Protein, Human, Recombinant | Human | E. coli |
Glutamine:fructose-6-phosphate amidotransferase 1 (GFAT), also known as GFPT1, is a member of the N-terminal nucleophile aminotransferases and the first rate-limiting enzyme for the entry of glucose into the hexosami... | |||
TMPH-02778 | Mcpt4 Protein, Mouse, Recombinant (E. coli, His) | Mouse | E. coli |
Has chymotrypsin-like activity. Hydrolyzes the amide bonds of synthetic substrates having Tyr and Phe residues at the P1 position. Preferentially hydrolyzes the 'Tyr-4-|-Ile-5' bond of angiotensin I and the 'Phe-20-|-Ala... | |||
TMPJ-00474 | CPA1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Carboxypeptidase A1 (CPA1) is secreted as a pancreatic peptidase that comes from the precursor form of inactive procarboxypeptidase. CPA1 comprises a signal peptide, a pro region and a mature chain, and can be activated ... | |||
TMPJ-00602 | CPA2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Carboxypeptidase A2 (CPA) is a secreted pancreatic procarboxy-peptidase that cleaves the C-terminal amide or ester bond of peptides that have a free C-terminal carboxyl group. The hydrolytic action of CPA2 was identified... |
カタログ番号 | 製品名 | ||
---|---|---|---|
L7810 | High Solubility Polyfunctional Group Fragment Library | 1159 compounds | |
Highly soluble multifunctional fragment library contains 1159 kinds of fragment molecules. |