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Dopamine Receptor 5-HT Receptor Adrenergic Receptor

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カタログ番号	製品名	別名	ターゲット
T1539	Iloperidone	HP 873	Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
	Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.		Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
T0082	Domperidone	R33812	Dopamine Receptor
	Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent. It blocks the action of. It has strong affinities for the D2 and D3 dopamine receptors, which are found in the chemoreceptor trigger z...		Dopamine Receptor
T1536	Promestriene	3-propyl ethyl,17B-methyl estradiol,Promestriano	Estrogen/progestogen Receptor
	Promestriene (3-propyl ethyl) (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation. It is described as a tropic agent and antiseborrheic.		Estrogen/progestogen Receptor
T9317	TAK-041	NBI-1065846	GPR
	TAK-041 (NBI-1065846) is a potent and selective GPR139 agonist.		GPR
T1504	Silodosin	KAD 3213,KMD 3213	Adrenergic Receptor
	Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.		Adrenergic Receptor
T27287	Estredox	E 2CDS,E-2-CDS,IDR 90104,E-2CDS,IDR-90104,E 2 CDS
	Estredox, an estrogen receptor agonist, is used potentially for the treatment of vasomotor symptoms.
T4549	Tibolone	tibolonum,tibolona	Estrogen/progestogen Receptor
	Tibolone is an estrogen-like compound used for the treatment of the symptoms associated with menopausal transition (i.e., climacteric symptoms) and also for the treatment of osteoporosis.		Estrogen/progestogen Receptor
T21281	Zolamide	CL 5343,Tio-urasin,5-Amino-TDSNH2	Others
	Zolamide (CL 5343) may be used to prevent altitude sickness and reduce the symptoms.		Others
T6653	Salmeterol Xinafoate	Salmetedur,GR 33343X xinafoate,Arial	HIV Protease , Adrenergic Receptor
	Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptom...		HIV Protease , Adrenergic Receptor
T7160	Lofexidine		Adrenergic Receptor
	Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.		Adrenergic Receptor
T0317	Buflomedil hydrochloride	Buflomedil HCl,Fonzylane,Loftyl	Adrenergic Receptor
	Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.		Adrenergic Receptor
T16114	Pavinetant	MLE-4901,AZD4901,AZD2624	Neurokinin receptor
	Pavinetant (MLE-4901) is an orally available neurokinin-3 receptor (NK3R) antagonist used to improve menopausal symptoms.		Neurokinin receptor
T5023	Propiverine hydrochloride		Others , Calcium Channel , AChR
	Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).		Others , Calcium Channel , AChR
T22316	Doxazosin	UK 33274	Adrenergic Receptor
	Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.		Adrenergic Receptor
T0113	Mebhydrolin napadisylate	Incidal,Diazolin,Mebhydroline 1,5-naphthalenedisulfonate salt,Omeril,Diazoline	5-HT Receptor , AChR , Histamine Receptor
	Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic dermatosis.		5-HT Receptor , AChR , Histamine Receptor
T11986L	Mebeverine acid hydrochloride
	Mebeverine acid hydrochloride is an effective, oral compound to act directly on the smooth muscle of the gastrointestinal tract to relieve spasticity symptoms.
T19399	L-Ornithine L-aspartate	Ornithine Aspartate	Others
	L-Ornithine L-aspartate (Ornithine Aspartate) lowers blood ammonia concentration and to eliminate symptoms of hepatic encephalopathy associated with liver cirrhosis.		Others
T1303	Auranofin	SKF-39162	Others , SARS-CoV , Antibacterial
	Auranofin (SKF-39162) is an antirheumatic agent, is used to treat rheumatoid arthritis, improves arthritis symptoms including painful or tender and swollen joints and morning stiffness.		Others , SARS-CoV , Antibacterial
T21419	Diphenhydramine	Debendrin,PM 255,PM255,Dabylen,Syntedril,PM-255	Histamine Receptor
	Diphenhydramine (Syntedril), a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the treatment of allergies. Diphenhydramine is also used in th...		Histamine Receptor
T50055	Milacemide		MAO
	Milacemide is a glycine prodrug and MAO-B inhibitor. Milacemide has been studied for its effects on human memory and as a potential treatment for the symptoms of Alzheimer's disease.		MAO
T15239	Epristeride	SKF105657,ONO-9302	Apoptosis , Reductase
	Epristeride (ONO-9302) is an orally active, selective and non-competitive steroidal 5-α-reductase isoform 2 inhibitor that inhibits SR isoform 2.Episteride reduces prostate size and improves symptoms in men with BPH.Epis...		Apoptosis , Reductase
T1180	Blonanserin	AD-5423	Dopamine Receptor , Sigma receptor , 5-HT Receptor , Adrenergic Receptor
	Blonanserin (AD-5423) is an atypical antipsychotic approved in Japan in January, 2008. Relative to many other antipsychotics, blonanserin has an improved tolerability profile, lacking side effects such as extrapyramidal ...
T0784	Tolfenamic Acid	GEA 6414,Tolfedine	COX
	Tolfenamic Acid (GEA 6414) is one of the class of non-steroidal anti-inflammatory drugs (NSAIDs). It is used to treat the symptoms of migraine.		COX
T6701	Terazosin hydrochloride dihydrate	Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate	Adrenergic Receptor
	Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).		Adrenergic Receptor
T4563	Thonzylamine	neohetramine	Histamine Receptor
	Thonzylamine (neohetramine) is an antihistamine and anticholinergic drug. It is available as combination products with Clofedanol or Phenylephrine for temporary relief of symptoms of common cold, hay fever (allergic rhin...		Histamine Receptor
T8634	8-Bromotheophylline	Bromotheophylline	Others
	8-Bromotheophylline (Bromotheophylline) is the active moiety of pamabrom, a mixture of 2-amino-2-methyl-propanol and bromotheophylline. From this mixture, 8-Bromotheophylline acts as a weak diuretic that has been used al...		Others
T0477	Zileuton	Abbott 64077,A 64077	Ferroptosis , Lipoxygenase , COX
	Zileuton (A 64077) is a synthetic derivative of hydroxyurea with antiasthmatic properties. The leukotriene inhibitor zileuton blocks 5-lipoxygenase, which catalyzes the formation of leukotrienes from arachidonic acid; ca...		Ferroptosis , Lipoxygenase , COX
T39252	TAK-418		Histone Demethylase
	TAK-418 is a selective and orally active inhibitor of LSD1/KDM1A enzyme with an IC50 of 2.9 nM. TAK-418 unlocks abnormal epigenetic mechanisms and improves autism symptoms in models of neurodevelopmental disorders.		Histone Demethylase
T21390	Fexofenadine	Carboxyterfenadine,Telfast,MDL 16.455,Allegra	Histamine Receptor
	Fexofenadine (Carboxyterfenadine), an antihistamine pharmaceutical drug, is used to treat allergy symptoms, such as nasal congestion, hay fever, and urticaria. Compared to first-generation antihistamines, Fexofenadine is...		Histamine Receptor
T39024	PrNMI		Cannabinoid Receptor
	PrNMI is a highly effective and orally active agonist targeting the peripherally restricted cannabinoid 1 receptor (CB1R). It exhibits pronounced analgesic properties, efficiently suppressing both chemotherapy-induced pe...		Cannabinoid Receptor
T79600	Zharp2-1		RIP kinase
	Zharp2-1, a RIPK2 inhibitor, inhibits the transcription of inflammatory cytokines induced by MDP-induced or Listeria monocytogenes infection and alleviates MDP-induced peritonitis symptoms in mice, which can be used for ...		RIP kinase
T1458	Epalrestat	ONO2235	Reductase
	Epalrestat (ONO2235), an aldose reductase inhibitor, is well tolerated in Long-term therapy. It can effectually ameliorate the associated symptoms of diabetic neuropathy and delay the progression of the disease, particul...		Reductase
T1292	Tiapride hydrochloride		Dopamine Receptor
	Tiapride is a selective blocker of D2/3 dopamine receptors in the brain. It is used in the therapy of various psychiatric and neurological disorders containing dyskinesia, negative symptoms of psychosis, alcohol withdraw...		Dopamine Receptor
T39229	YNT-185		OX Receptor
	YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R, respectively. Furthermore, YNT-185 effectively alleviates symptoms of ...		OX Receptor
T0219	Valdecoxib	SC 65872	COX
	Valdecoxib (SC 65872) is a prescription drug used in the treatment of osteoarthritis, rheumatoid arthritis, and painful menstruation and menstrual symptoms. It is classified as a nonsteroidal anti-inflammatory drug, or N...		COX
T4195	Betahistine	PT 9 base,Vasomotal,Serc base	Histamine Receptor
	Betahistine (Vasomotal) is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may exacerbate bronchial asthma and peptic ulcers. Betahisti...		Histamine Receptor
T0331	Moxifloxacin hydrochloride	BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl	Topoisomerase , Antibacterial , Antibiotic
	Moxifloxacin hydrochloride (BAY12-8039 HCl) is a fourth generation fluoroquinolone with expanded activity against gram-positive bacteria as well as atypical pathogens. Moxifloxacin has been linked to mild ALT elevations ...		Topoisomerase , Antibacterial , Antibiotic
T22277L	BMS-P5 free base		PAD
	BMS-P5 free base is a specific and orally active peptidylarginine deiminase 4 (PAD4) inhibitor. BMS-P5 Blocks Formation of Neutrophil Extracellular Traps and Delays Progression of Multiple Myeloma. Administration of BMS-...		PAD
T60522	Letosteine	Viscotiol	Others
	Letosteine (Viscotiol) is an orally active, effective, and safe expectorant that can be used in the study of acute or chronic respiratory diseases, for example, bronchopulmonary disease. Letosteine dissolves bronchial mu...		Others
T21385	Cinitapride	Paxapride,Cidine,cinitapride tartrate,Blaston,Cintapro,Cinmove	5-HT Receptor
	Cinitapride (Blaston) is a gastroprokinetic agent. It slows the actions of the muscles to reduce the symptoms of conditions such as acid reflux, delayed gastric emptying, and ulcer dyspepsia. Cinitapride acts as an antag...		5-HT Receptor
T67729	UCM-1306		Dopamine Receptor
	UCM-1306 is a potent and orally active allosteric modulator (PAM) of human dopamine D1 receptor. UCM-1306 could increase the maximal effect of endogenous dopamine (DA) both in human and mouse D1 receptors. UCM-1306 could...		Dopamine Receptor
T28165	NF-1819	NF 1819,NF1819	Lipase
	NF-1819 is a potent and selective irreversible MGL (β-lactam-based monoacylglycerol lipase) inhibitor. NF-1819 alleviates symptoms in a MS model in vivo and exhibits analgesic effects in an acute inflammatory pain model ...		Lipase
T6426	Buclizine dihydrochloride	Longifene,Buclina,Buclizine HCl,UCB-4445	5-HT Receptor , AChR , Histamine Receptor
	Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and antivertigo activities. Buclizine dihydrochloride binds to and ...		5-HT Receptor , AChR , Histamine Receptor
T26684	Auten-99 HBr	Auten-99,Auten-99 hydrochloride. Auten-99 HBr,Auten99,Auten 99	Phosphatase
	Auten-99 HBr (Auten-99) is a myotubularin phosphatase Jumpy inhibitor exerting potent neuroprotective effects. AUTEN-99 activates autophagy in cell cultures and animal models. AUTEN-99 appears to effectively penetrate th...		Phosphatase
TP1904L	FSLLRY-NH2 TFA(245329-02-6 free base)		Protease-activated Receptor
	FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK activation and collagen production in iso...		Protease-activated Receptor
T1568	Amoxapine	CL-67772	GlyT
	Amoxapine (CL-67772) exerts its antidepressant effect by inhibiting the re-uptake of norepinephrine and, to a lesser degree, of serotonin, at adrenergic nerve endings and blocks the response of dopamine receptors to dopa...		GlyT
T11326	Frovatriptan succinate hydrate	Frovelan,Frova	5-HT Receptor
	Frovatriptan succinate hydrate (Frova) is effective in treating the full spectrum of migraine including the associated symptoms of nausea, vomiting, photophobia, and phonophobia. Frovatriptan succinate hydrate can also b...		5-HT Receptor
T2319	Acotiamide monohydrochloride trihydrate	Acotiamide hydrochloride,YM-443 HCl,Z-338 HCl	AChE
	Acotiamide monohydrochloride trihydrate (Z-338 HCl) is the hydrochloride salt form of acotiamide, a prokinetic agent with gastrointestinal (GI) motility-enhancing activity. Although the exact mechanism by which acotiamid...		AChE
T4616	Metoclopramide	5-Chloro-2-methoxyprocainamide	Dopamine Receptor , 5-HT Receptor
	Metoclopramide (5-Chloro-2-methoxyprocainamide) is a dopamine D2 antagonist which has been used for treatment of a variety of gastrointestinal symptoms over the last thirty years. In various countries, metoclopramide is ...		Dopamine Receptor , 5-HT Receptor
T0976	Propoxur	Aprocarb,Propoxure,Baygon	AChR , Antifungal
	Propoxur (Propoxure) is an insecticide used to control cockroaches, flies, mosquitoes, and lawn and turf insects. Acute (short-term) exposure of humans to propoxur by ingestion leads to cholinesterase inhibition of red b...		AChR , Antifungal

Compounds

Iloperidone

T1539

Synonym: HP 873

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

Domperidone

T0082

Synonym: R33812

Target: Dopamine Receptor

Promestriene

T1536

Synonym: 3-propyl ethyl,17B-methyl estradiol,Promestriano

Target: Estrogen/progestogen Receptor

Synonym: KAD 3213,KMD 3213

Target: Adrenergic Receptor

Estredox

T27287

Synonym: E 2CDS,E-2-CDS,IDR 90104,E-2CDS,IDR-90104,E 2 CDS

Target:

Tibolone

T4549

Synonym: tibolonum,tibolona

Target: Estrogen/progestogen Receptor

Zolamide

T21281

Synonym: CL 5343,Tio-urasin,5-Amino-TDSNH2

Target: Others

Salmeterol Xinafoate

T6653

Synonym: Salmetedur,GR 33343X xinafoate,Arial

Target: HIV Protease, Adrenergic Receptor

Lofexidine

T7160

Synonym:

Target: Adrenergic Receptor

Buflomedil hydrochloride

T0317

Synonym: Buflomedil HCl,Fonzylane,Loftyl

Target: Adrenergic Receptor

Pavinetant

T16114

Synonym: MLE-4901,AZD4901,AZD2624

Target: Neurokinin receptor

Propiverine hydrochloride

T5023

Synonym:

Target: Others, Calcium Channel, AChR

Doxazosin

T22316

Synonym: UK 33274

Target: Adrenergic Receptor

Mebhydrolin napadisylate

T0113

Synonym: Incidal,Diazolin,Mebhydroline 1,5-naphthalenedisulfonate salt,Omeril,Diazoline

Target: 5-HT Receptor, AChR, Histamine Receptor

Mebeverine acid hydrochloride

T11986L

Synonym:

Target:

L-Ornithine L-aspartate

T19399

Synonym: Ornithine Aspartate

Target: Others, SARS-CoV, Antibacterial

Diphenhydramine

T21419

Synonym: Debendrin,PM 255,PM255,Dabylen,Syntedril,PM-255

Target: Histamine Receptor

Synonym: SKF105657,ONO-9302

Target: Apoptosis, Reductase

Blonanserin

T1180

Synonym: AD-5423

Target: Dopamine Receptor, Sigma receptor, 5-HT Receptor, Adrenergic Receptor

Tolfenamic Acid

T0784

Synonym: GEA 6414,Tolfedine

Target: COX

Terazosin hydrochloride dihydrate

T6701

Synonym: Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate

Target: Adrenergic Receptor

Thonzylamine

T4563

Synonym: neohetramine

Target: Histamine Receptor

8-Bromotheophylline

T8634

Synonym: Bromotheophylline

Target: Others

Zileuton

T0477

Synonym: Abbott 64077,A 64077

Target: Ferroptosis, Lipoxygenase, COX

TAK-418

T39252

Synonym:

Target: Histone Demethylase

Fexofenadine

T21390

Synonym: Carboxyterfenadine,Telfast,MDL 16.455,Allegra

Target: Histamine Receptor

PrNMI

T39024

Synonym:

Target: Cannabinoid Receptor

Tiapride hydrochloride

T1292

Synonym:

Target: Dopamine Receptor

Synonym: PT 9 base,Vasomotal,Serc base

Target: Histamine Receptor

Moxifloxacin hydrochloride

T0331

Synonym: BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl

Target: Topoisomerase, Antibacterial, Antibiotic

Synonym: Paxapride,Cidine,cinitapride tartrate,Blaston,Cintapro,Cinmove

Target: 5-HT Receptor

UCM-1306

T67729

Synonym:

Target: Dopamine Receptor

NF-1819

T28165

Synonym: NF 1819,NF1819

Target: Lipase

Buclizine dihydrochloride

T6426

Synonym: Longifene,Buclina,Buclizine HCl,UCB-4445

Target: 5-HT Receptor, AChR, Histamine Receptor

Auten-99 HBr

T26684

Synonym: Auten-99,Auten-99 hydrochloride. Auten-99 HBr,Auten99,Auten 99

Target: Phosphatase

FSLLRY-NH2 TFA(245329-02-6 free base)

TP1904L

Synonym:

Target: Protease-activated Receptor

Frovatriptan succinate hydrate

T11326

Synonym: Frovelan,Frova

Target: 5-HT Receptor

Acotiamide monohydrochloride trihydrate

T2319

Synonym: Acotiamide hydrochloride,YM-443 HCl,Z-338 HCl

Target: AChE

Metoclopramide

T4616

Synonym: 5-Chloro-2-methoxyprocainamide

Target: Dopamine Receptor, 5-HT Receptor

Propoxur

T0976

Synonym: Aprocarb,Propoxure,Baygon

Target: AChR, Antifungal

カタログ番号	製品名	別名	ターゲット
TMS0418	Dihydroergotoxine mesylate	Ergoloid mesylates	GABA Receptor
	Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.		GABA Receptor
T4S0290	Araloside A	Chikusetsusaponin IV	RAAS , Fas/FasL
	Araloside A (Chikusetsusaponin IV) might relieve cutaneous symptoms caused by excessive apoptotic cell death in the skin through the Fas/FasL pathway.		RAAS , Fas/FasL
T20754	Deltamethrin	Butoss,RU-22974,Esbecythrin,K-Othrin,Decamethrin,RU 22974	Others
	Deltamethrin (RU 22974), a neurotoxic pyrethroid insecticide, produces a reversible sequence of motor symptoms in rats involving hind limb rigidity and choreoathetosis.Deltamethrin is globally used in crop protection, co...		Others
T3888	Scopolin	Murrayin,Scopoloside	Sirtuin
	Scopolin (Scopoloside) formation is increased by the enhanced activity of PAL. Scopolin can reduce the clinical symptoms of rat AIA by inhibiting inflammation and angiogenesis, and this compound may be a potent agent for...		Sirtuin
T8194L	Soy Isoflavone		Others
	Soy Isoflavone is extracted from the seeds of leguminous plants. The isoflavones in soybeans are natural phytoestrogens, which have good medicinal value and can reduce the incidence of breast cancer in women, relieve men...		Others
T4S1999	Valepotriate	Valtrate	Apoptosis , HIV Protease
	Valepotriate (Valtrate) fraction can have sedative effects and affect behavioral parameters related to recognition memory. Valepotriates, a new class of cytotoxic and antitumor agents, they are very potent cytotoxic agen...		Apoptosis , HIV Protease
T2S2173	(E)-Naringenin chalcone	Isosalipurpol,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone	Others
	Naringenin chalcone (Isosalipurpol) has antiallergic activity Naringenin chalcone suppresses asthmatic symptoms by inhibiting Th2 cytokine production from CD4 T cells. Naringenin chalcone is a potent tomato flavonoid tha...		Others
T15248	Estetrol	Donesta	Estrogen Receptor/ERR , Endogenous Metabolite
	Estetrol(Donesta) is an orally available, selective modulator of the estrogen receptor, a naturally occurring estrogen synthesized by the human fetal liver during pregnancy.Estetrol has effects on the endometrium or cent...		Estrogen Receptor/ERR , Endogenous Metabolite
T2520	Desloratadine	Sch34117,NSC 675447	Endogenous Metabolite , Histamine Receptor
	Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties. Desloratadine diminishes the typical histaminergic effects on H1-receptors in bronchial smoot...		Endogenous Metabolite , Histamine Receptor
T4776	Glycerol	Glycerin	Endogenous Metabolite
	Glycerol or glycerin is a colourless, odourless, viscous liquid that is sweet-tasting and mostly non-toxic. It is widely used in the food industry as a sweetener and humectant and in pharmaceutical formulations. Glycerol...		Endogenous Metabolite
T0729	Benzyl benzoate	Ascabiol,Novoscabin,Scabitox,Benzoic acid benzyl ester	Parasite
	Benzyl benzoate (Benzoic acid benzyl ester) is one of the older preparations used for the therapy of scabies. Scabies is a skin infection caused by the Sarcoptes scabiei. Its symptoms are red spots, severe itching (parti...		Parasite
T3011	2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid	Kynurenine,Dl-Kynurenine,Kynurenin,3-Anthraniloylalanine	Others , Endogenous Metabolite
	2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid (3-Anthraniloylalanine) is a ketone and an amino acid derivative with diverse biological functions, including vasodilatory, immunoregulatory and neuromodulatory activities. 2-...		Others , Endogenous Metabolite
T6491	(-)-(S)-Equol	(−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	(-)-(S)-Equol (4',7-Dihydroxyisoflavan) is an orally bioavailable, non-steroidal estrogen naturally produced by the metabolism of the isoflavonoid daidzein by human intestinal microflora, with potential chemoprotective a...
T4723	D-Tagatose	D-(-)-Tagatose,d-tagatos	Others , Endogenous Metabolite
	D-Tagatose (D-(-)-Tagatose), a rare natural hexoketose, is an isomer of d-galactose. D-Tagatose occurs naturally in Sterculia setigera gum, and it is also found in small quantities in various foods such as sterilized and...		Others , Endogenous Metabolite
TN2299	Vindesine		Others
	Vindesine is a microtubule inhibitor and widely used to treat malignancies. Vindesine neuropathy seems to be the cause of the patient's neurological symptoms.		Others
TN1741	Homomangiferin	芒果	Others
	Homomangiferin has important medicinal properties and is widely used to relieve many symptoms, for example coughing and asthma.Homomangiferin shows antitumoural effects against MDA-MB-231 cells.		Others
T37177	Norcholic Acid
	Norcholic acid is a bile acid and 23-carbon derivative of cholic acid .1Levels of norcholic acid are increased in the urine of patients with liver cirrhosis or cerebrotendinous xanthomatosis (CTX), an inborn error of met...
TN4383	Kazinol U		IL Receptor , IκB/IKK , NOS , NF-κB
	Kazinol U may have therapeutic value in delaying pancreatic β-cell destruction in type 1 diabetes by blocking the NF-ÎºB pathway in pancreatic β-cells reduces cell damage. Kazinol U shows estrogenic activity with ligand-...		IL Receptor , IκB/IKK , NOS , NF-κB
T73844	Nortriptyline
	Nortriptyline (Desmethylamitriptyline), the primary active metabolite of Amitriptyline, functions as a tricyclic antidepressant, effectively alleviating symptoms of depression. It is also recognized as a potent autophagy...
T36845	Isogarcinol
	Isogarcinol is a natural polyisoprenylated benzophenone first isolated from plant species in the genus Garcinia. It has immunosuppressant actions, inhibiting the protein phosphatase calcineurin (IC50 = 36 μM) and suppres...
TN3351	Aflatrem		GABA Receptor
	Aflatrem is a tremorgenic mycotoxin with acute neurotoxic effects, a single low dose of aflatrem is able to induce degeneration of neuronal processes in hippocampal neurotransmitter systems. Aflatrem potentiates the gamm...		GABA Receptor
T75600	Coronatine
	Coronatine is a plant growth regulator synthesized by Pseudomonas syringae, mimicking bioactive jasmonic acid conjugates or octadecanoid signal molecules in higher plants, which induces pathogenic symptoms. It enhances t...

天然物製品

Dihydroergotoxine mesylate

TMS0418

Synonym: Ergoloid mesylates

Target: GABA Receptor

Araloside A

T4S0290

Synonym: Chikusetsusaponin IV

Target: RAAS, Fas/FasL

Deltamethrin

T20754

Synonym: Butoss,RU-22974,Esbecythrin,K-Othrin,Decamethrin,RU 22974

Target: Others

Scopolin

T3888

Synonym: Murrayin,Scopoloside

Target: Apoptosis, HIV Protease

(E)-Naringenin chalcone

T2S2173

Synonym: Isosalipurpol,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone

Target: Estrogen Receptor/ERR, Endogenous Metabolite

Desloratadine

T2520

Synonym: Sch34117,NSC 675447

Target: Endogenous Metabolite, Histamine Receptor

Glycerol

T4776

Synonym: Glycerin

Target: Endogenous Metabolite

Benzyl benzoate

T0729

Synonym: Ascabiol,Novoscabin,Scabitox,Benzoic acid benzyl ester

Target: Parasite

2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid

T3011

Synonym: Kynurenine,Dl-Kynurenine,Kynurenin,3-Anthraniloylalanine

Target: Others, Endogenous Metabolite

(-)-(S)-Equol

T6491

Synonym: (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite

D-Tagatose

T4723

Synonym: D-(-)-Tagatose,d-tagatos

Target: Others, Endogenous Metabolite

Target: IL Receptor, IκB/IKK, NOS, NF-κB

Target: GABA Receptor

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-04826	LILRB5/CD85c Protein, Human, Recombinant (His)	Human	HEK293 Cells
	A genetic variant in LILRB5 (leukocyte immunoglobulin-like receptor subfamily-B) (rs12975366: T > C: Asp247Gly) has been reported to be associated with lower creatine phosphokinase (CK) and lactate dehydrogenase (LDH) le...
TMPY-03855	DNase I Protein, Human, Recombinant (His)	Human	HEK293 Cells
	DNase1, also known as deoxyribonuclease I and DNL1, is a member of the DNase family. DNaseI is a nuclease that cleaves DNA preferentially at phosphodiester linkages adjacent to a pyrimidine nucleotide, yielding 5'-phos...
TMPY-00117	FGF-16 Protein, Human, Cynomolgus, Recombinant	Human,Cynomolgus	Baculovirus Insect Cells
	Fibroblast growth factor 16 (FGF16) is preferentially expressed in the heart after birth, suggesting its regulation is associated with tissue-specific chromatin remodeling and DNA-protein interactions. Mutation of the ME...
TMPH-03579	TSST-1 Protein, S. aureus, Recombinant (His & SUMO)	Staphylococcus aureus	E. coli
	Responsible for the symptoms of toxic shock syndrome. TSST-1 Protein, S. aureus, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 37.9 kDa and th...
TMPH-03594	Exotoxin type A Protein, S. pyogenes, Recombinant (His & SUMO)	Streptococcus pyogenes	E. coli
	Causative agent of the symptoms associated with scarlet fever, have been associated with streptococcal toxic shock-like disease and may play a role in the early events of rheumatic fever. Exotoxin type A Protein, S. pyog...
TMPY-05186	LILRB5/CD85c Protein, Human, Recombinant (His), Biotinylated	Human	HEK293 Cells
	A genetic variant in LILRB5 (leukocyte immunoglobulin-like receptor subfamily-B) (rs12975366: T > C: Asp247Gly) has been reported to be associated with lower creatine phosphokinase (CK) and lactate dehydrogenase (LDH) le...
TMPY-06273	LILRB5/CD85c Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	A genetic variant in LILRB5 (leukocyte immunoglobulin-like receptor subfamily-B) (rs12975366: T > C: Asp247Gly) has been reported to be associated with lower creatine phosphokinase (CK) and lactate dehydrogenase (LDH) le...
TMPJ-01277	CRT2 Protein, Human, Recombinant	Human	E. coli
	Calreticulin-3 belongs to the calreticulin family, members of which are calcium binding chaperones localized mainly in the endoplasmic reticulum. It can be divided into a N-terminal globular domain, a proline-rich P-doma...
TMPY-04476	MVK Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	Mevalonate kinase belongs to the GHMP kinase family, Mevalonate kinase subfamily. It can be found in a wide variety of organisms from bacteria to mammals. Mevalonate kinase may be a regulatory site in the cholesterol bio...
TMPJ-00869	GLB1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	β Galactosidase is a lysosomal β Galactosidase that hydrolyzes the terminal β Galactose from Ganglioside and Keratan sulfate. In lysosome, the mature β Galactosidase protein associates with Cathepsin A and Neuraminidase ...
TMPY-02961	PANP/C12orf53 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	C12orf53 is mainly expressed in adult brain and cerebellum. It also can be detected in fetal brain and virtually no expression in spleen, heart, kidney, liver and dorsal ganglion relative to brain. C12orf53 acts as a lig...
TMPY-03452	PTS Protein, Human, Recombinant (His)	Human	E. coli
	PTS(6-pyruvoyltetrahydropterin synthase) belongs to the PTPS family. It catalyzes the elimination of inorganic triphosphate from dihydroneopterin triphosphate, which is the second and irreversible step in the biosynthesi...
TMPY-02516	Interferon alpha 10/IFNA10 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Interferon alpha-10 (IFNA10) is a member of the interferon family. Interferons belong to the group of the regulatory glycoproteins, of low molecular mass. They are the products of infected cell-genome, but not virus, as ...

LILRB5/CD85c Protein, Human, Recombinant (His)

TMPY-04826

Species: Human

Expression System: HEK293 Cells

DNase I Protein, Human, Recombinant (His)

TMPY-03855

Species: Human

Expression System: HEK293 Cells

FGF-16 Protein, Human, Cynomolgus, Recombinant

TMPY-00117

Species: Human,Cynomolgus

Expression System: Baculovirus Insect Cells

TSST-1 Protein, S. aureus, Recombinant (His & SUMO)

TMPH-03579

Species: Staphylococcus aureus

Expression System: E. coli

Exotoxin type A Protein, S. pyogenes, Recombinant (His & SUMO)

TMPH-03594

Species: Streptococcus pyogenes

Expression System: E. coli

LILRB5/CD85c Protein, Human, Recombinant (His), Biotinylated

TMPY-05186

Species: Human

Expression System: HEK293 Cells

LILRB5/CD85c Protein, Human, Recombinant (hFc)

TMPY-06273

Species: Human

Expression System: HEK293 Cells

CRT2 Protein, Human, Recombinant

TMPJ-01277

Species: Human

Expression System: E. coli

MVK Protein, Human, Recombinant (His & GST)

TMPY-04476

Species: Human

Expression System: Baculovirus Insect Cells

GLB1 Protein, Human, Recombinant (His)

TMPJ-00869

Species: Human

Expression System: HEK293 Cells

PANP/C12orf53 Protein, Human, Recombinant (hFc)

TMPY-02961

Species: Human

Expression System: HEK293 Cells

PTS Protein, Human, Recombinant (His)

TMPY-03452

Species: Human

Expression System: E. coli

Interferon alpha 10/IFNA10 Protein, Human, Recombinant (hFc)

TMPY-02516

Species: Human

Expression System: HEK293 Cells

カタログ番号	製品名
L9830	Anti-Parkinson's Disease Compound Library	857 compounds
	A unique collection of 857 compounds with anti-PD activities or acting on main drug targets of PD can be used for HTS and HCS.
L9840	Anti-Alzheimer's Disease Compound Library	986 compounds
	A unique collection of 986 compounds with anti-AD activities or acting on main drug targets of AD can be used for HTS and HCS.
L2196	Anti-Ovarian Cancer Compound Library	1867 compounds

L6720	Anti-COVID-19 Traditional Chinese Medicine Compound Library	1147 compounds
	A unique collection of 1147 monomers from 60 TCM plants, a powerful tool for anti-COVID-19 drug discovery, can be used for HTS and HCS screening；

ライブラリー

Anti-Parkinson's Disease Compound Library

L9830

Compounds: 857

Anti-Alzheimer's Disease Compound Library

L9840

Compounds: 986

Anti-Ovarian Cancer Compound Library

L2196

Compounds: 1867

Anti-COVID-19 Traditional Chinese Medicine Compound Library

L6720

Compounds: 1147