|
T15697 |
L-NMMA acetate
|
Tilarginine acetate,Methylarginine acetate |
NOS
|
|
|
|
T21335 |
Fluorogestone acetate
|
Flurogestone Acetate Flugestone Acetate Fluorogesterone Acetate SC9880 |
Others
|
|
Fluorogestone acetate (Flurogestone Acetate Flugestone Acetate Fluorogesterone Acetate SC9880) showed a high potency with short duration of activity and performed physiologically similar to progesterone. FGA was approxim... |
|
TP1103 |
Cotadutide acetate
|
MEDI0382 acetate,Cotadutide acetate (1686108-82-6 Free base) |
Glucagon Receptor
|
|
Cotadutide acetate (MEDI0382 acetate) is a potent peptide dual agonist of glucagon-like peptide-1 (GLP-1) and glucagon receptor with EC50 of 6.9 pM and 10.2 pM, respectively. |
|
TP1022 |
Protirelin Acetate
|
TSH-RF Acetate,TRH Acetate,TRF Acetate |
Thyroid hormone receptor(THR)
,
Endogenous Metabolite
|
|
Protirelin Acetate (TRH Acetate) is a thyrotropin-releasing hormone, stimulating the release of thyrotropin and prolactin from the anterior pituitary. |
|
T8359 |
Lanreotide acetate
|
Lanreotide acetate (108736-35-2 free base),BIM 23014 (acetate),BIM 23014 acetate |
Others
|
|
Lanreotide acetate (BIM 23014 acetate) is a somatostatin analogue with antineoplastic activity, used for carcinoid syndrome |
|
T38862 |
Nandrolone acetate
|
19-Nortestosterone 17β-acetate |
Others
|
|
Nandrolone acetate (19-Nortestosterone 17β-acetate) is a competitive inhibitor of isomerase with the Ki of 7 μM for Δ5-3-ketosteroid isomerase of Pseudomonas testosreroni. |
|
T20383 |
Nopol acetate
|
Nopyl acetate,Lignyl acetate,2-Pinene-10-methyl acetate |
Others
|
|
Nopol acetate (2-Pinene-10-methyl acetate) is an agent of biochemical. |
|
T13072 |
Taltirelin acetate
|
TA-0910 acetate |
Thyroid hormone receptor(THR)
|
|
Taltirelin acetate (TA-0910 acetate) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)). |
|
T1666 |
Fludrocortisone acetate
|
9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,9α-fluorocortisol acetate |
Glucocorticoid Receptor
,
Autophagy
|
|
Fludrocortisone acetate (9α-Fludrocortisone acetate) , a glucocorticoid-receptor agonist, binds to cytoplasmic receptors, translocates to the nucleus, and subsequently initiates the transcription of glucocorticoid-respon... |
|
T24584 |
P505-15 Acetate
|
PRT 062607 Acetate,P505 15 Acetate,PRT-062607 Acetate,PRT062607 Acetate,P50515 Acetate |
Tyrosinase
|
|
P505-15 Acetate is a selective inhibitor of spleen tyrosine kinase that acts by suppressing leukocyte immune function and inflammation and leading to a reduction in arthritis score and attenuated histological damage. |
|
T19067 |
Thionin acetate
|
Thionine acetate |
Others
|
|
Thionin acetate (Thionine acetate) is a metachromatic cationic histology dye used in biological staining widely. |
|
T6881L |
LTX315 acetate
|
KKWWKKW-Dip-K-NH2 acetate,Oncopore acetate,Ruxotemitide acetate,LTX315 acetate(1345407-05-7, Free base) |
Others
|
|
LTX315 acetate (Oncopore acetate) is an oncolytic peptide with potent anticancer activity, with IC50 values of 34.3 µM for MRC-5, 8.3 µM for A20, and 11 µM for AT84, respectively. |
|
TP1814L |
CEF4 acetate
|
CEF4 acetate(199727-68-9 free base) |
Others
|
|
CEF4 acetate (CEF4 acetate (199727-68-9 free base)) is a polypeptide corresponding to amino acid sequence 342-351 of the influenza A virus nucleocapsid protein. |
|
TP2112L |
TC14012 acetate
|
TC14012 acetate(368874-34-4 free base) |
CXCR
,
Arrestin
|
|
TC14012 acetate is a serum-stable derivative of T140 which is a selective and peptidomimetic CXCR4 antagonist with an IC50 of 19.3 nM. TC14012 is also a potent CXCR7 agonist with an EC50 of 350 nM for recruiting β-arrest... |
|
TP1910L1 |
CALP1 acetate
|
CALP1 acetate(145224-99-3 free base) |
CaMK
|
|
CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site. CALP1 blocks calcium influx and apoptosis (IC50 of 44.78 µM) by inhibiting the open of calcium channel. CALP1 blo... |
|
TP2501 |
Difelikefalin acetate
|
Difelikefalin acetate(1024828-77-0 free base),CR 845 acetate,FE 202845 acetate |
Opioid Receptor
|
|
Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist. CR845 exhibit low P450 CYP inhibition and low penetration into the brain. |
|
T10549 |
Bisindolylmaleimide VIII acetate
|
Ro 31-7549 acetate,Bis VIII acetate |
Apoptosis
,
PKC
|
|
Bisindolylmaleimide VIII acetate (Ro 31-7549 acetate) is a potent and selective PKC inhibitor (IC50: 158 nM for rat brain PKC). It has IC50s of 53, 195, 163, 213, and 175 nM for PKC-α, PKC-βI, PKC-βII, PKC-γ, PKC-ε, resp... |
|
T21598L |
G3335 Acetate
|
G3335 Acetate (36099-95-3 free base) |
PPAR
|
|
G3335 Acetate was discovered to be a novel PPARgamma antagonist. |
|
T20413L |
Spantide acetate
|
Spantide acetate(91224-37-2 Free base) |
Neurokinin receptor
|
|
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2. |
|
TP2338L |
Cenupatide acetate
|
Cenupatide acetate(1006388-38-0 Free base) |
Others
|
|
Cenupatide acetate is an urokinase plasminogen activator receptor (uPAR) inhibitor for treating disorders associated altered cell migration, such as cancer. |
|
T22178L |
Spadin Acetate
|
Spadin Acetate(1270083-24-3 Free base) |
Others
|
|
Spadin Acetate is a natural peptide derived from a propeptide released in blood. Spadin Acetate is able to block the TREK-1 channel activity. Spadin Acetate binds specifically to TREK-1 with an affinity of 10 nM. |
|
T20704L |
Levitide acetate
|
Levitide acetate(114281-19-5 Free base) |
Others
|
|
Levitide acetate is an antimicrobial peptide from the skin of frogs. |
|
TP1382L |
HAEGTFTSDVS acetate
|
HAEGTFTSDVS acetate(864915-61-7 free base) |
Glucagon Receptor
|
|
HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells. |
|
T11052L |
Disitertide acetate
|
P144 acetate,Disitertide acetate(272105-42-7 Free base) |
TGF-beta/Smad
|
|
Disitertide acetate (P144 acetate) is a peptidic transforming growth factor-beta 1 (TGF-β1) inhibitor specifically designed to block the interaction with its receptor. Disitertide acetate is also a PI3K inhibitor and an ... |
|
T40508L |
TRV120056 acetate
|
TRV120056 acetate (40678-47-5 Free base) |
Others
|
|
TRV120056 acetate is a Gq-biased agonist with 10-fold greater molecular efficiency on AT1R-Gq fusion proteins than AT1R-βarr2 fusion proteins. |
|
T36420 |
IM-156 acetate
|
HL271 acetate |
|
|
IM-156 acetate, an activator of NADH dehydrogenase (IC50=2.2 μM) and AMP-activated protein kinase alpha (AMPKα), is an orally available and bioavailable inhibitor of mitochondrial oxidative phosphorylation (OxPhos).IM-15... |
|
T12992 |
SPR741 acetate
|
SPR741 acetate,NAB741 acetate,SPR741 acetate (1179330-52-9 free base) |
Antibacterial
|
|
SPR741 acetate is a cationic peptide derived from polymyxin B. It exhibits antimicrobial activity against gram-negative bacteria by inhibiting severe gram-negative bacterial sensory by increasing the permeability of the ... |
|
T11836 |
Lefamulin acetate
|
BC-3781 acetate |
ribosome
,
Antibacterial
,
Antibiotic
|
|
Lefamulin acetate (BC-3781 acetate) (formally BC-3781 acetate) is a novel pleuromutilin antibiotic and is the first to be used for the systemic treatment of bacterial infections in humans. Lefamulin acetate (BC-3781 acet... |
|
T13306L |
Vapreotide acetate
|
RC-160 acetate,BMY-41606 acetate |
Neurokinin receptor
|
|
Vapreotide acetate (BMY-41606 acetate) is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM). |
|
TP1223L |
Apamin acetate
|
Apamine acetate,Apamin acetate(24345-16-2 Free base) |
Potassium Channel
|
|
Apamin acetate (Apamine acetate) is a selective Ca2+-activated blocker of K+ (SK) channels, an 18-amino acid peptide neurotoxin found in bee toxins.Apamin acetate enhances synapse growth and regeneration following lacera... |
|
TP1299L1 |
Melittin Acetate
|
Melittin Acetate(20449-79-0 Free base),Forapin Acetate |
Phospholipase
|
|
Melittin Acetate (Forapin Acetate) is a PLA2 activator. Melittin Acetate stimulates the activity of the low molecular weight PLA2, while it does not increase the activity of the high molecular weight PLA2. |
|
T9857L |
Vasopressin acetate
|
Vasopressin acetate (11000-17-2 Free base) |
Endogenous Metabolite
|
|
Vasopressin acetate, a cyclic nonapeptide, is synthesized centrally in the hypothalamus. Vasopressin acetate acts as a neurotransmitter, exerting its action by binding to specific G protein-coupled receptors. |
|
TP1759L |
GRGDSPC acetate
|
GRGDSPC,GRGDSPC acetate(91575-26-7 free base) |
Others
|
|
GRGDSPC acetate (GRGDSPC acetate (91575-26-7 free base)) is a 7-amino acid peptide of thiolated cell adhesion. |
|
TP1018L |
Urechistachykinin II acetate
|
Urechistachykinin II acetate(149097-04-1 free base),Uru-TK II acetate |
Others
|
|
Urechistachykinin II acetate (Uru-TK II acetate) is an invertebrate rapid kinin-related peptide (TRPs) isolated from carotenoid worms, shows antimicrobial activities without a hemolytic effect |
|
T21567L |
Cyclosomatostatin Acetate
|
Cyclosomatostatin Acetate （84211-54-1 Free base） |
Somatostatin
|
|
Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell proliferation, ALDH+ cell population size, and sphere-formation in c... |
|
T23077L |
Novokinin acetate
|
Novokinin acetate (358738-77-9 free base) |
RAAS
|
|
Novokinin acetate exhibited an affinity for the AT2 receptor with Ki of 7 nM, and its antihypertensive and vasorelaxing activities were blocked by PD123319, an AT2 receptor antagonist. |
|
T11918L |
Lysipressin acetate(50-57-7(fb_acetate))
|
Lysine vasopressin acetate,[Lys8]-Vasopressin acetate |
Others
|
|
Lysipressin acetate(50-57-7(fb_acetate)) ([Lys8]-Vasopressin acetate) , Induces contraction of the rabbit urinary bladder smooth muscle, activate adenylate-cyclase. Lysipressin is Antidiuretic hormone that have been foun... |
|
T40570L |
LKKTETQ acetate
|
LKKTETQ acetate (476014-70-7 Free base) |
Others
|
|
LKKTETQ acetate is the active site in the protein thymosin β4 responsible for wound healing, actin binding and cell migration. |
|
T3407L |
Rapastinel acetate
|
Rapastinel acetate (117928-94-6 Free base) |
NMDAR
,
iGluR
|
|
Rapastinel acetate is a modulator of N-methyl-D-aspartate (NMDA) receptor and a partial agonist of glycine site long-lasting antidepressant effects. |
|
TP1448L |
Astressin acetate
|
Astressin acetate (170809-51-5 Free base) |
CRFR
|
|
|
|
T7815L |
AOD9604 acetate(221231-10-3 free base)
|
AOD-9604 acetate,AOD9604 acetate,AOD 9604 acetate |
Others
|
|
AOD9604 acetate(221231-10-3 free base) is a potential anti-obesity peptide based on the human growth hormone. |
|
T7608 |
Bremelanotide Acetate
|
bremelanotide,PT-141 Acetate |
Melanocortin Receptor
|
|
Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) . |
|
T0947 |
Dexamethasone acetate
|
Dexamethasone 21-acetate,Dexamethason acetate,NSC 39471 |
Glucocorticoid Receptor
,
Mitophagy
,
IL Receptor
,
Annexin A
,
NOS
,
Antibacterial
,
Autophagy
|
|
Dexamethasone acetate (NSC 39471) is the acetate salt form of Dexamethasone, a synthetic adrenal corticosteroid with potent anti-inflammatory properties. In addition to binding to specific nuclear steroid receptors, dexa... |
|
T0337 |
Prednisolone acetate
|
Omnipred,Prednisolone-21-acetate |
Glucocorticoid Receptor
|
|
Prednisolone acetate (Omnipred) is the acetate salt form of prednisolone, a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. |
|
T14932L |
Ceruletide Ammonium acetate
|
FI-6934 Ammonium acetate,Caerulein Ammonium acetate,Ceruletide Ammonium acetate (17650-98-5 free base) |
cholecystokinin
|
|
Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) is a cholecystokinin (CCK) receptor agonist. Ceruletide Ammonium acetate is a safe and effective cholecystokinetic agent and small bowel and exocrine pancreatic stim... |
|
T38459 |
Chromium(III) acetate
|
Chromium triacetate,Chromic acetate,Chromium acetate |
Others
|
|
Chromium(III) acetate （Chromium acetate） is a small molecule ionic crosslinker that is used as a feedstock for the synthesis of other compounds. |
|
T21470L |
Davunetide acetate
|
Davunetide acetate(211439-12-2 Free base) |
Beta Amyloid
,
Microtubule Associated
|
|
Davunetide acetate is derived from activity-dependent neuroprotective protein existing in the mammalian CNS. Davunetide acetate is a microtubule-stabilizing peptide and inhibits Aβ aggregation and Aβ-induced neurotoxicit... |
|
TP2482 |
LCKLSL acetate
|
LCKLSL acetate(533902-29-3 free base) |
Annexin A
|
|
LCKLSL acetate is a competitive annexin A2 (AnxA2) inhibitor. LCKLSL acetate potently inhibits the binding of tissue plasminogen activator (tPA) to AnxA2 and the generation of plasmin. LCKLSL acetate has anti-angiogenic ... |
|
T20692L |
Schistoflrfamide acetate
|
Schistoflrfamide acetate(121801-61-4 Free base) |
Others
|
|
Schistoflrfamide acetate is isolated from the grasshopper, Schistocerca gregaria. Schistoflrfamide acetate elicited an immediate effect on the basal membrane potential of the opalescent tubule gland cells in insects. |
|
TP1535L |
GPLGIAGQ acetate
|
GPLGIAGQ acetate(109053-09-0 Free base) |
MMP
|
|
|
