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カタログ番号	製品名	別名	ターゲット
T4989	Fosfomycin Tromethamine		Antibacterial , Antibiotic
	An antibiotic produced by Streptomyces fradiae.		Antibacterial , Antibiotic
T9014	SKI-178		Apoptosis , S1P Receptor
	SKI-178 is a sphingosine kinase 1 (SphK1) inhibitor with IC50 of 0.1-1.8 μM. It induces prolonged mitosis followed by apoptotic cell death through the intrinsic apoptotic cascade. The sustained activation of CDK1 during ...		Apoptosis , S1P Receptor
T8722	IKIX1		Antifungal
	iKIX1 is an Pdr1-dependent gene activation. It re-sensitizes drug-resistant C. glabrata to azole antifungals in vitro and in animal models for disseminated and urinary tract C. glabrata infection.		Antifungal
T3131	Fosfomycin calcium	Phosphomycin calcium salt,Fosmicin	Antibacterial , Antibiotic
	Fosfomycin calcium (Phosphomycin calcium salt) is a blood-brain barrier penetrating, broad-spectrum antibiotic by irreversibly inhibiting an early stage in cell wall synthesis.		Antibacterial , Antibiotic
T8217	Enzalutamide carboxylic acid		Androgen Receptor , Drug Metabolite
	Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .		Androgen Receptor , Drug Metabolite
T10981	DCZ0415		Apoptosis , Others , NF-κB
	DCZ0415 induces antimyeloma activity in vitro, in vivo and in primary cells of drug-resistant myeloma patients. DCZ0415 is a potent TRIP13 inhibitor that can impair the repair of non-homologous end junctions and inhibit ...		Apoptosis , Others , NF-κB
T9830	GSK2556286	GSK286	Antibacterial
	GSK2556286 (GSK286) is an orally active inhibitor of Mycobacterium tuberculosis (M. tuberculosis).GSK2556286 inhibits the growth of human macrophages with an IC50 value of 0.07 μM.GSK2556286 is effective against both mul...		Antibacterial
T10378	Artelinic acid		Others
	Artelinic acid, a derivative of Artemisinin, is an antimalarial drug for the treatment of multidrug-resistant strains of Plasmodium falciparum.		Others
T10356	AQ-13 dihydrochloride		Parasite
	AQ-13 dihydrochloride is an antimalarial drug. It is effective against drug-resistant strains of Plasmodium falciparum.		Parasite
T22269	Benzyldodecyldimethylammonium Chloride Dihydrate		Antibacterial
	Benzyldodecyldimethylammonium chloride dihydrate can be used as an insecticide reagent. It can target drug-resistant bacteria, such as methicillin-resistant Staphylococcus aureus, multidrug-resistant Pseudomonas aerugino...		Antibacterial
T5315	TCA1	TCA-1,TCA 1	Antibacterial , Antibiotic
	TCA1 (TCA 1) is a small molecule with activity against drug-resistant and persistent tuberculosis.		Antibacterial , Antibiotic
T14081	Enmetazobactam	AAI101	Antibacterial
	Enmetazobactam (AAI101) is an extended-spectrum β-lactamase inhibitor for the treatment of multi-drug resistant gram-negative bacterial infections.		Antibacterial
T64860	3-(Trifluoromethyl)cinnamic acid	3-(3-(Trifluoromethyl)phenyl)acrylic acid	Antibiotic
	3-(Trifluoromethyl)cinnamic acid (3-(3-(Trifluoromethyl)phenyl)acrylic acid) can be used to study drug-resistant bacterial infections.		Antibiotic
T73586	Anticonvulsant agent 2		Others
	Anticonvulsant agent 2 is a potent orally active anticonvulsant that has shown antiepileptic activity in a model of drug-resistant epilepsy.		Others
T6824	EAI045		EGFR
	EAI045, an allosteric inhibitor, targets towards drug-resistant EGFR mutants but avoids the wild-type receptor.		EGFR
T0391	Linezolid	PNU-100766	MAO , Antibacterial , Antibiotic
	Linezolid (PNU-100766), the first of the oxazolidinone class, is a synthetic antibiotic used for the therapy of infections resulted from multi-resistant bacteria including methicillin-resistant Staphylococcus aureus (MRS...		MAO , Antibacterial , Antibiotic
T4469	Nemorubicin	Methoxymorpholinyldoxorubicin,PNU-152243A,PNU 152243	Others
	Nemorubicin (PNU 152243) is a doxorubicin derivative that differs significantly from its parent drug in terms of spectrum of antitumor activity, metabolism and toxicity profile. The drug is active on tumors resistant to ...		Others
T14188	ALLO-2		Hedgehog/Smoothened , Smo
	ALLO-2 is a Inhibitor of Drug-Resistant Smo Mutant.It inhibits Smo agonist Hh-Ag1.5-induced luciferase expression in TM3-Gli-Luc cells with IC50 of 6 nM.		Hedgehog/Smoothened , Smo
T0331L	Moxifloxacin	Avelox,Moxeza	Others , Antibacterial , Antibiotic
	Moxifloxacin (Avelox) is a fourth-generation fluoroquinolone that has been shown to be effective against Gram-positive, Gram-negative, and atypical strains, as well as multi-drug resistant Streptococcus pneumoniae.		Others , Antibacterial , Antibiotic
T11427	Antibacterial compound 2		Antifungal
			Antifungal
T61016	EMI1		EGFR
	EMI1 can be used in the mutant EGFR-associated, drug-resistant non-small-cell lung cancer(NSCLC) research. EMI1 is an inhibitor of EGFR L858R/T790M/C797S and EGFR ex19del/T790M/C797S [1].		EGFR
T10802	CHMFL-EGFR-202		EGFR
	CHMFL-EGFR-202 is a potent, irreversible inhibitor of EGFR mutant kinase (IC50s: 5.3 nM and 8.3 nM for drug-resistant mutant EGFR T790M and WT EGFR kinases).		EGFR
T10799	CHMFL-ABL-039		Bcr-Abl
	CHMFL-ABL-039 is a type II native ABL kinase and drug-resistant V299L mutant BCR-ABL inhibitor (IC50s: 7.9 nM and 27.9 nM) used in the research of chronic myeloid leukemia.		Bcr-Abl
T22646	CFM 4	CFM-4,CFM4	Apoptosis , APC
	CFM 4 is a potent small molecule CARP-1/APC-2 antagonist that prevents CARP-1 from binding to APC-2, contributes to G2M cell cycle arrest, and induces apoptosis, with an IC50 in the range of 10-15 μM.CFM 4 inhibits the g...		Apoptosis , APC
T11125	Durlobactam sodium salt	ETX2514 sodium salt	Antibacterial
	Durlobactam sodium salt (ETX2514 sodium salt) is an inhibitor of β-lactamase with IC50 values of 4 nM, 14 nM, and 190 nM for Class A KPC-2, Class C AmpC, and Class D OXA-24, respectively. Durlobactam sodium salt can be u...		Antibacterial
T23858	WCK-5153	WCK 5153,WCK5153	Antibacterial
	WCK-5153 is an enhancer of β-Lactamase and an inhibitor of PBP2 with antimicrobial activities against Pseudomonas aeruginosa. WCK-5153 can be used in studies about the treatment of serious infections caused by highly dru...		Antibacterial
T1146	Nifedipine	BAY-a-1040,Procardia XL,Procardia,Adalat	CaMK , Potassium Channel , Calcium Channel , Autophagy
	Nifedipine (Procardia) is a dihydropyridine calcium channel blocking agent. Nifedipine inhibits the transmembrane influx of extracellular calcium ions into myocardial and vascular smooth muscle cells, causing dilatation ...		CaMK , Potassium Channel , Calcium Channel , Autophagy
T67934	MRT-2359		Others
	MRT-2359 is a potent and orally available GSPT1 reducer with antitumour activity.MRT-2359 inhibits the growth of drug-resistant non-small cell lung cancer (NSCLC) and small cell lung cancer (SCLC) cells.MRT-2359 exhibits...		Others
T12343	Benzquinamide	BZQ,P2647,Benzoquinamide	Adrenergic Receptor
	Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer drugs in multidrug-resistant cells.The Ki values of Benzqui...		Adrenergic Receptor
T8972	FIT-039		Others , DNA/RNA Synthesis , CDK , HSV
	FIT-039 is a selective and ATP-competitive, orally active inhibitor of CDK9( IC50 : 5.8 μM;CDK9/cyclin T1). FIT-039 inhibits replication of HSV-1 (IC50 of 0.69 μM), HSV-2, human adenovirus, and human CMV. FIT-039 is a pr...		Others , DNA/RNA Synthesis , CDK , HSV
T28886	Suprafenacine	N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide	Microtubule Associated
	Suprafenacine (N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide) is a cell-permeable microtubule destabilizer that induces cell cycle arrest and apoptosis in G2/M phase. Suprafenacine ...		Microtubule Associated
T63746	Vamotinib	PF-114	Apoptosis , Tyrosine Kinases , Bcr-Abl
	Vamotinib (PF-114) is an orally active and specific tyrosine kinase inhibitor with antiproliferative and antitumour activity.Vamotinib inhibits the phosphorylation of BCR/ABL and BCR/ABL-T315I, which promotes apoptosis. ...		Apoptosis , Tyrosine Kinases , Bcr-Abl
T27453	GSK1733953A	DG70	Antibacterial
	GSK1733953A can be used as a small molecule Mycobacterium tuberculosis respiration inhibitor with an inhibitory effect on MenG activity and an IC50 value of 2.6 ± 0.6 μM.GSK1733953A is a selective biphenylbenzamide with ...		Antibacterial
T1852	Rac-Belinostat	NSC726630,PXD101,PX-105684	HDAC
	Rac-Belinostat (PX-105684) is a novel hydroxamic acid-type histone deacetylase (HDAC) inhibitor with antineoplastic activity. Belinostat targets HDAC enzymes, thereby inhibiting tumor cell proliferation, inducing apoptos...		HDAC
T1190	Cefmenoxime hydrochloride	Cefmenoxime hemihydrochloride,SCE-1365 hemihydrochloride	Antibacterial , Antibiotic , Antifection
	Cefmenoxime hydrochloride (Cefmenoxime hemihydrochloride) is a cephalosporin antibiotic that is administered intravenously or intramuscularly. It is active against most common gram-positive and gram-negative microorganis...		Antibacterial , Antibiotic , Antifection
T4126	CBL0137	Curaxin 137,CBLC137	NF-κB , p53
	CBL0137 (Curaxin 137), a metabolically stable curaxin, activates p53 (EC50: 0.37 μM) and inhibits NF-κB (EC50: 0.47 μM). It functionally inactivates the facilitates chromatin transcription complex (FACT), driving the eff...		NF-κB , p53
T35610	2,5-dimethyl Celecoxib		Apoptosis , Wnt/beta-catenin , Prostaglandin Receptor
	2,5-dimethyl Celecoxib is a derivative of celecoxib that does not inhibit COX-2 (IC50 = >100 μM).1 It does inhibit microsomal prostaglandin E synthase-1 (mPGES-1) in HeLa cells (IC50 = 15.6 μM) and reduces prostaglandin ...		Apoptosis , Wnt/beta-catenin , Prostaglandin Receptor
T3024	Avitinib	AC0010	EGFR , JAK , BTK
	Avitinib (AC0010), also known as AC0010 or AC0010MA, is an orally available, irreversible, epidermal growth factor receptor (EGFR) mutant-selective inhibitor, with potential antineoplastic activity. Upon oral administrat...		EGFR , JAK , BTK
T70671	IC2418
	IC2418 is an MmpL3 inhibitor, being active against drug-resistant Mycobacterium tuberculosis.
T10902	CWHM-1008		Others
	CWHM-1008 is an effective oral antimalarial drug. The EC50 values of the drug-sensitive Plasmodium falciparum 3D7 and drug-resistant Dd2 strains are 46 and 21 nM, respectively.		Others
T33683	NITD-304	NITD304
	NITD-304 is an anti-tuberculosis drug candidate for the treatment of multidrug-resistant tuberculosis (MDR-TB), showing effective activity against both MTB drug-sensitive and multidrug-resistant clinical isolates.
T70545	HI-253
	HI-253 is a potent non-nucleoside inhibitor of drug-resistant human immunodeficiency virus (HIV).
T23625	ACT-451840	ACT451840
	ACT-451840 is a drug of antimalarial activity. It has effective activity against sensitive and resistant Plasmodium falciparum strains.
T40140	Zanamivir-Cholesterol Conjugate
	Zanamivir-cholesterol conjugate is an extended-duration neuraminidase inhibitor highly effective against drug-resistant influenza strains.
T28988	TNK-6123	TNK6123
	TNK-6123 is an emivirine analog. TNK-6123 has improved activity against drug-resistant HIV mutants.
T24103	GS-9148
	GS-9148 is a dAMP analog. It also maintains its antiviral activity against drug-resistant HIV.
T70212	U 95133
	U 95133 is a potent, broad-spectrum nonnucleoside reverse transcriptase inhibitor of drug-resistant isolates of human immunodeficiency virus type 1.
T71725	IMB-XMA0038
	IMB-XMA0038 was identified as an inhibitor of MtASADH and it is a promising lead compound against drug-resistant tuberculosis.
T24130	HCI-2184	HCI2184,HCI 2184
	HCI-2184 is an inhibitor of AXL kinase and Nek2 that acts by successfully mitigating drug resistance in bortezomib-resistant multiple myeloma.
T11116	Duocarmycin MA		Others
	Duocarmycin MA can be used against multi-drug resistant cell lines.Duocarmycin MA is an antibody drug conjugates (ADCs) toxin. Duocarmycin is a DNA alkylating agent that binds in the minor groove.		Others

Compounds

Fosfomycin Tromethamine

T4989

Synonym:

Target: Antibacterial, Antibiotic

SKI-178

T9014

Synonym:

Target: Apoptosis, S1P Receptor

Synonym: Phosphomycin calcium salt,Fosmicin

Target: Antibacterial, Antibiotic

Enzalutamide carboxylic acid

T8217

Synonym:

Target: Androgen Receptor, Drug Metabolite

DCZ0415

T10981

Synonym:

Target: Apoptosis, Others, NF-κB

GSK2556286

T9830

Synonym: GSK286

Target: Antibacterial

AQ-13 dihydrochloride

T10356

Synonym:

Target: Parasite

Benzyldodecyldimethylammonium Chloride Dihydrate

T22269

Synonym:

Target: Antibacterial

TCA1

T5315

Synonym: TCA-1,TCA 1

Target: Antibacterial, Antibiotic

Enmetazobactam

T14081

Synonym: AAI101

Target: Antibacterial

3-(Trifluoromethyl)cinnamic acid

T64860

Synonym: 3-(3-(Trifluoromethyl)phenyl)acrylic acid

Target: Antibiotic

Anticonvulsant agent 2

Target: MAO, Antibacterial, Antibiotic

Nemorubicin

T4469

Synonym: Methoxymorpholinyldoxorubicin,PNU-152243A,PNU 152243

Target: Hedgehog/Smoothened, Smo

Moxifloxacin

T0331L

Synonym: Avelox,Moxeza

Target: Others, Antibacterial, Antibiotic

Antibacterial compound 2

Target: Apoptosis, APC

Durlobactam sodium salt

T11125

Synonym: ETX2514 sodium salt

Target: Antibacterial

WCK-5153

T23858

Synonym: WCK 5153,WCK5153

Target: Antibacterial

Nifedipine

T1146

Synonym: BAY-a-1040,Procardia XL,Procardia,Adalat

Target: CaMK, Potassium Channel, Calcium Channel, Autophagy

Synonym: BZQ,P2647,Benzoquinamide

Target: Adrenergic Receptor

FIT-039

T8972

Synonym:

Target: Others, DNA/RNA Synthesis, CDK, HSV

Suprafenacine

T28886

Synonym: N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide

Target: Microtubule Associated

Vamotinib

T63746

Synonym: PF-114

Target: Apoptosis, Tyrosine Kinases, Bcr-Abl

GSK1733953A

T27453

Synonym: DG70

Target: Antibacterial

Rac-Belinostat

T1852

Synonym: NSC726630,PXD101,PX-105684

Target: HDAC

Cefmenoxime hydrochloride

T1190

Synonym: Cefmenoxime hemihydrochloride,SCE-1365 hemihydrochloride

Target: Antibacterial, Antibiotic, Antifection

CBL0137

T4126

Synonym: Curaxin 137,CBLC137

Target: NF-κB, p53

2,5-dimethyl Celecoxib

T35610

Synonym:

Target: Apoptosis, Wnt/beta-catenin, Prostaglandin Receptor

Avitinib

T3024

Synonym: AC0010

Target: EGFR, JAK, BTK

Zanamivir-Cholesterol Conjugate

Synonym: HCI2184,HCI 2184

カタログ番号	製品名	別名	ターゲット
TN4660	Niranthin		Anti-infection , HBV , PAFR , Topoisomerase
	Niranthin is a potent anti-leishmanial agent, inhibits the relaxation activity of heterodimeric type IB topoisomerase of L. donovani and acts as a non-competitive inhibitor interacting with both subunits of the enzyme. N...		Anti-infection , HBV , PAFR , Topoisomerase
TN6512	Tectol		Transferase , Parasite
	Tectol has anti-plasmodial activity, it as a moderately active growth inhibitor with an IC50 3.44±0.20μM. It exhibited significant activity against human leukemia cell lines HL60 and CEM. Tectol may cause itchy dermatiti...		Transferase , Parasite
T8262	Fosfomycin sodium	Fosfomycin Disodium	Antibacterial , Antibiotic
	Fosfomycin sodium is a bactericidal, low-molecular weight, broad-spectrum antibiotic, with putative activity against several bacteria, including multidrug-resistant Gram-negative bacteria, by irreversibly inhibiting an e...		Antibacterial , Antibiotic
TQ0152	Dalfopristin	RP54476	Antibacterial , Antibiotic
	Dalfopristin (RP54476) is a semi-synthetic streptogramin antibiotic. Quinupristin/Dalfopristin (Q/D) is used for the treatment of multi-drug resistant Enterococcus faecium infections.		Antibacterial , Antibiotic
T5132	9-dihydro-13-acetylbaccatin III	13-Acetyl-9-dihydrobaccatin III,9-DHAB III	Apoptosis
	9-dihydro-13-acetylbaccatin III (9-DHAB III)is an apoptosis inducer. It shows cytotoxicity against the MCF7 cell line and drug-resistant cell line MCF7-ADR.		Apoptosis
T1589	D-Cycloserine	RO-1-9213	Others , Antibacterial , Antibiotic , iGluR
	D-Cycloserine (RO-1-9213) is a broad spectrum antibiotic used as a second line agent for treatment of drug resistant tuberculosis, always in combination with other antituberculosis agents.		Others , Antibacterial , Antibiotic , iGluR
TN2213	Imperialine 3-β-D-glucoside	Sipeimine-3-beta-D-glucoside	Others
	Imperialine 3-β-D-glucoside (Sipeimine-3-beta-D-glucoside) is a natural product. Imperialine 3-β-D-glucoside may exhibit anti-tumor properties against multi-drug resistant tumor cells.		Others
T6S1683	Demethoxycurcumin	Curcumin II,Desmethoxycurcumin,Monodemethoxycurcumin	Apoptosis , Antioxidant , Antibacterial , Autophagy
	1. Demethoxycurcumin (Desmethoxycurcumin) has antioxidant activity. 2. Demethoxycurcumin has anti-inflammatory activity. 3. Demethoxycurcumin has anti-proliferative activity. 4. Demethoxycurcumin has anti-acanthamoebic e...		Apoptosis , Antioxidant , Antibacterial , Autophagy
T5S2347	Deoxyshikonin	Arnebin 7	Others , HIF/HIF Prolyl-Hydroxylase , Antibacterial
	1. Deoxyshikonin (Arnebin 7) may be a new drug candidate for wound healing and treatment of lymphatic diseases. 2. Deoxyshikonin enhances the ability of human dermal lymphatic microvascular endothelial cells (HMVEC-dLy) ...		Others , HIF/HIF Prolyl-Hydroxylase , Antibacterial
T6S1315	Oroxylin A	6-Methoxybaicalein,Baicalein 6-methyl ether	Virus Protease , HIF/HIF Prolyl-Hydroxylase , Autophagy
	1. Oroxylin A (Baicalein 6-methyl ether) has various anti-tumor effects including apoptosis, cell cycle arrest, drug-resistant reversion. 2. Oroxylin A possesses abilities of inhibiting the ATRA-induced IL-6 production v...		Virus Protease , HIF/HIF Prolyl-Hydroxylase , Autophagy
TN3013	4,5-Dimethoxycanthin-6-one	Methylnigakinone	P450 , Antibacterial , PDE
	4,5-Dimethoxycanthin-6-one is an alkaloid isolated from Picrasma quassioides BENNET (Simaroubaceae).4,5-Dimethoxycanthin-6-one was isolated from Picrasma quassioides BENNET (Simaroubaceae) with antimicrobial activity.4,5...		P450 , Antibacterial , PDE
TN6559	Isogambogic acid
	Isogambogic acid shows cytotoxic activiity against KB and drug-resistant KB-V1 cell lines.
TN5114	Taxinine		P-gp
	Taxinine and Taxinine B can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells.		P-gp
TN1397	Ardisiacrispin B		Others
	Ardisiacrispin B displays cytotoxic effects in multi-factorial drug resistant cancer cells via ferroptotic and apoptotic cell death.		Others
T40924	Tellimagrandin II	Eugeniin
	Tellimagrandin II (Eugeniin) is the initial intermediate in the 4 C 1 -glucose derived series of ellagitannins. Additionally, it possesses the ability to inhibit antibiotic resistance exhibited by drug-resistant Staphylo...
TN2726	Jatrophane 5		P-gp
	Jatrophane 5 demonstrates the most powerful inhibition of P-gp, higher than R(+)-verapamil and tariquidar in colorectal multi-drug resistant (MDR) cells (DLD1-TxR).		P-gp
TN5113	Taxinine B		Others
	Taxinine and taxinine B can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells. Taxinine B shows stronger inhibitory effects than acetylsalicylic acid (ASA) on platelet aggregation induced by arach...		Others
TN2311	Wulignan A1		Antifection
	Wulignan A1 exhibits activity against leukemia P-388 in vitro; it also may have anti-influenza virus H1N1 and H1N1-TR (a Tamiflu drug resistant virus strain) activities.		Antifection
T81099	Staphyloferrin A
	Staphyloferrin A, a siderophore, can be utilized in conjunction with antibiotics to investigate drug-resistant bacteria implicated in skin diseases [1].
TN4382	Kazinol A		AMPK , mTOR
	Kazinol A shows strong inhibition of arachidonic acid (AA)-induced platelet aggregation. It also exhibits potent inhibition with IC50 values ranging 0.6-164 M against XOD. Kazinol A may be a candidate for the development...		AMPK , mTOR
TN2727	Jatrophane 2		P-gp , Antifection
	2,5,7,8,9,14-Hexaacetoxy-3-benzoyloxy-15-hydroxyjatropha-6(17),11E-diene (Jatrophane 2 ) exhibits significant antifeedant activity against a generalist plant-feeding insect, the cotton bollworm (Helicoverpa armigera). Ja...		P-gp , Antifection
T38330	Collinin
	Collinin is a coumarin that has been found in Z. schinifolium and has diverse biological activities.1,2,3,4 It is active against drug-susceptible and -resistant strains of M. tuberculosis (MIC50s = 3.13-6.25 μg/ml).1 Col...
TN3438	Arborinine		HCV Protease , Antifection
	Arborinine shows mild in vitro antibacterial activity, it possesses moderate levels of anti-hepatitis C virus(HCV) activities with the IC50 values being 6.4 ± 0.7 ug/ml. Arborinine shows antifeedant activity against Spod...		HCV Protease , Antifection
TN2977	3-O-trans-p-Coumaroyltormentic acid		Caspase , Antifection
	3-O-(E)-p-coumaroyl tormentic acid may be promising lead compound for developing an effective drug for treatment of leukemia, it induces apoptotic cell death in human leukemia (HL60) via mainly mitochondrial pathway by, ...		Caspase , Antifection
T36954	Nemorosone
	Nemorosone is a polycyclic polyprenylated acylphloroglucinol (PPAP) originally isolated from C. rosea that has antiproliferative properties.1 Nemorosone inhibits growth of NB69, Kelly, SK-N-AS, and LAN-1 neuroblastoma ce...

天然物製品

Niranthin

TN4660

Synonym:

Target: Anti-infection, HBV, PAFR, Topoisomerase

Tectol

TN6512

Synonym:

Target: Transferase, Parasite

Fosfomycin sodium

T8262

Synonym: Fosfomycin Disodium

Target: Antibacterial, Antibiotic

Dalfopristin

TQ0152

Synonym: RP54476

Target: Antibacterial, Antibiotic

9-dihydro-13-acetylbaccatin III

T5132

Synonym: 13-Acetyl-9-dihydrobaccatin III,9-DHAB III

Target: Others, Antibacterial, Antibiotic, iGluR

Imperialine 3-β-D-glucoside

TN2213

Synonym: Sipeimine-3-beta-D-glucoside

Target: Others

Demethoxycurcumin

T6S1683

Synonym: Curcumin II,Desmethoxycurcumin,Monodemethoxycurcumin

Target: Apoptosis, Antioxidant, Antibacterial, Autophagy

Deoxyshikonin

T5S2347

Synonym: Arnebin 7

Target: Others, HIF/HIF Prolyl-Hydroxylase, Antibacterial

Oroxylin A

T6S1315

Synonym: 6-Methoxybaicalein,Baicalein 6-methyl ether

Target: Virus Protease, HIF/HIF Prolyl-Hydroxylase, Autophagy

4,5-Dimethoxycanthin-6-one

TN3013

Synonym: Methylnigakinone

Target: P450, Antibacterial, PDE

Target: P-gp, Antifection

Target: HCV Protease, Antifection

3-O-trans-p-Coumaroyltormentic acid

TN2977

Synonym:

Target: Caspase, Antifection

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPH-03139	MDR1 Protein, Plasmodium falciparum, Recombinant (His & SUMO)	Plasmodium falciparum	E. coli
	Energy-dependent efflux pump responsible for decreased drug accumulation in multidrug-resistant cells. MDR1 Protein, Plasmodium falciparum, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-...
TMPY-03458	Sorcin/SRI Protein, Human, Recombinant	Human	Baculovirus Insect Cells
	Sorcin was originally identified in multidrug-resistant cells. It is a calcium-binding protein. Sorcin modulates excitation-contraction coupling in the heart, contributes to calcium homeostasis in the heart sarcoplasmic ...
TMPY-03267	Sorcin/SRI Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	Sorcin was originally identified in multidrug-resistant cells. It is a calcium-binding protein. Sorcin modulates excitation-contraction coupling in the heart, contributes to calcium homeostasis in the heart sarcoplasmic ...

MDR1 Protein, Plasmodium falciparum, Recombinant (His & SUMO)

TMPH-03139

Species: Plasmodium falciparum

Expression System: E. coli

Sorcin/SRI Protein, Human, Recombinant

TMPY-03458

Species: Human

Expression System: Baculovirus Insect Cells

Sorcin/SRI Protein, Human, Recombinant (His & GST)

TMPY-03267

Species: Human

Expression System: Baculovirus Insect Cells

カタログ番号	製品名
L4520	Anti-Bacterial Compound Library	904 compounds
	A unique collection of 904 antibacterial bioactive compounds, a powerful tool for antibacterial drug development;
L4400	Antibiotics Library	692 compounds
	A unique collection of 692 compounds with antibiotic activity for new antibacterial drug screening;
L1800	Anti-Infection Compound Library	2938 compounds
	A unique collection of 2938 anti-infective compounds including anti-bacterial, anti-fungi, anti-Human Cytomegalovirus (HCMV), anti-HIV, anti-SARS, anti-influenza, etc;
L4600	Selected Plant-Sourced Compound Library	3048 compounds
	A unique collection of 3048 plant-sourced compounds that derived from 277 plant species for high throughput screening (HTS) and high content screening (HCS);
L9840	Anti-Alzheimer's Disease Compound Library	986 compounds
	A unique collection of 986 compounds with anti-AD activities or acting on main drug targets of AD can be used for HTS and HCS.
L6610	Anti-infective Natural Product Library	1060 compounds
	A unique collection of 1060 species of natural products with anti-infective activity for high throughput screening (HTS) and high content screening (HCS);
L9410	Covalent Inhibitor Library	1920 compounds
	A unique collection of 1920 covalent Inhibitors and other molecules with common warheads like chloroacetyl，2-Chloropropionyl，Acryloyl，sulfonyl fluoride, alkyne，acrylamide, ketocarbonyl，disulfide bond, etc.