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カタログ番号	製品名	別名	ターゲット
T37426	FIIN-1	FGFR irreversible inhibitor-1	FGFR
	FIIN-1 (FGFR irreversible inhibitor-1) is an irreversible and selective FGFR inhibitor with Kd of 2.8, 6.9, 5.4, 120, 32 and 120 nM for FGFR1, FGFR2, FGFR3, FGFR4, Flt1, Flt14, respectively.FIIN-1 inhibited FGFR1, FGFR2,...		FGFR
T16143	MRTX-1257		Ras
	MRTX-1257 is a selective, irreversible, and covalent inhibitor of KRAS G12C. It has an IC50 of 900 pM for KRAS dependent ERK phosphorylation in H358 cells. MRTX1257 demonstrated 31% bioavailability in the mouse, with fre...		Ras
T10140	4-Diethylaminobenzaldehyde		Dehydrogenase
	4-Diethylaminobenzaldehyde is a reversible aldehyde dehydrogenase (ALDH) inhibitor (Ki: 4 nM for ALDH1). It displays a potent anti-androgenic effect (IC50: 1.71μM).		Dehydrogenase
T2164	Wiskostatin		Others
	Wiskostatin is a selective inhibitor of N-WASP, a ubiquitously expressed member of the Wiskott-Aldrich Syndrome protein (WASp) family that regulates actin polymerization.		Others
T22461	YKL-5-124		CDK
	YKL-5-124, a potent, selective and covalent CDK7 inhibitor with an IC50 of 9.7 nM, 1300 nM and 3020 nM for CDK7/Mat1/CycH, CDK2 and CDK9 respectively, displays biochemical and cellular selectivity for CDK7 over CDK12/13...		CDK
T9399	Menin-MLL inhibitor 20		Epigenetic Reader Domain , Histone Methyltransferase
	Menin-MLL inhibitor 20 is an irreversible inhibitor of menin-MLL interaction with antitumor activities.		Epigenetic Reader Domain , Histone Methyltransferase
T6685	Sulbactam sodium	CP-45899-2	Antibacterial , Antibiotic
	Sulbactam sodium (CP-45899-2) (Unasyn) is an irreversible β-lactamase inhibitor.		Antibacterial , Antibiotic
T9865	Almonertinib mesylate		EGFR
	Almonertinib mesylate is an irreversible inhibitor of EGFR tyrosine kinase with high selectivity for EGFR-sensitizing and T790M resistance mutations. Almonertinib mesylate can be used in the non-small cell lung cancer st...		EGFR
T1631	Sulbactam	CP45899	Antibacterial , Antibiotic
	Sulbactam (CP45899) is a semi-synthetic beta-lactamase inhibitor. The beta-lactam ring of sulbactam irreversibly binds to beta-lactamase at or near its active site, thereby blocking enzyme activity and preventing metabol...		Antibacterial , Antibiotic
T36841	IPI-9119		Fatty Acid Synthase
	IPI-9119 is an orally active, selective and irreversible FASN inhibitor (IC50 = 0.3 nM).		Fatty Acid Synthase
T21652	RN-1 dihydrochloride		Histone Demethylase , MAO
	RN-1 dihydrochloride is an effective and selective irreversible inhibitor of lysine-specific demethylase 1 (LSD1, IC50 = 70 nM).		Histone Demethylase , MAO
T8421	TED-347		YAP
	TED-347 is an irreversible and covalent inhibitor of TEAD4-Yap1 protein-protein interaction(EC50 of 5.9 μM), and inhibits glioblastoma cell viability.		YAP
T60076	Oritinib	SH-1028	EGFR
	Oritinib (SH-1028) is an inhibitor of EGFR with IC50s of 18, 0.7, 4, 0.1, 1.4 and 0.89 nM for EGFR (wt), EGFR (L858R), EGFR (L861Q), EGFR (L858R/T790M), EGFR (d746-750), EGFR (d746-750/T790M), respectively. Oritinib can ...		EGFR
T14336	Allitinib	AST-1306,ALS 1306	EGFR
	Allitinib (AST-1306) (AST-1306) has anti-cancer activity，and it is an irreversible EGFR and ErbB2 inhibitor with IC50s of 0.5 and 3 nM, respectively. [1]		EGFR
T3626	Acalabrutinib	ACP-196	BTK
	Acalabrutinib (ACP-196), also known as ACP-196, is an orally available inhibitor of Bruton's tyrosine kinase (BTK) with potential antineoplastic activity. Upon administration, ACP-196 inhibits the activity of BTK and pre...		BTK
T4535	Etomoxir sodium salt	(R)-Etomoxir sodium salt,Na salt,Etomoxir	Apoptosis , Others
	Etomoxir sodium salt ((R)-Etomoxir sodium salt) is a carnitine palmitoyltransferase 1a (CPT-1a) inhibitor that blocks fatty acid synthesis. Etomoxir sodium salt has antitumor activity.		Apoptosis , Others
T1447	Fenclonine	Fenchlonine,PCPA,CP-10188,4-Chloro-DL-phenylalanine,DL-4-Chlorophenylalanine	Hydroxylase
	Fenclonine (CP-10188) is a selective and irreversible inhibitor of tryptophan hydroxylase, a rate-limiting enzyme in the biosynthesis of serotonin (5-HYDROXYTRYPTAMINE). Fenclonine(CP-10188) acts pharmacologically to dep...		Hydroxylase
T6331	Allitinib tosylate	AST-1306 TsOH,AST-6,Allitinib,AST-1306,AST-1306 (TsOH)	EGFR , FLT
	Allitinib tosylate (AST-1306) is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of 0.5 nM and 3 nM, respectively.		EGFR , FLT
T16492	PF-06459988		EGFR
	PF-06459988 is a novel, effective, orally active, irreversible, and selective epidermal growth factor receptor (EGFR) mutant inhibitor. PF-06459988 has high efficiency and high affinity for EGFRs double mutants containin...		EGFR
T4217	INF39		NOD-like Receptor (NLR) , NOD
	INF39 is a noncytotoxic and irreversible NLRP3 inhibitor.		NOD-like Receptor (NLR) , NOD
TQ0310	FMK		S6 Kinase
	FMK is an irreversible inhibitor of RSK2 kinase.		S6 Kinase
T15948	MAFP	Methyl Arachidonyl Fluorophosphonate	Phospholipase
	MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase. MAFP is an active-site directed and irreversible inhibitor of cPLA2 and iPLA2.		Phospholipase
T5340	MPO-IN-28		Glutathione Peroxidase
	MPO-IN-28 is a novel potent, irreversible Myeloperoxidase (MPO) inhibitor with IC50 of 44 nM.		Glutathione Peroxidase
T2630	Poziotinib	HM781-36B,NOV120101	Apoptosis , EGFR , HER
	Poziotinib (NOV120101)(NOV120101; HM781-36B) is an irreversible HER1/2/4 inhibitor (IC50s: 3/5/23 nM).		Apoptosis , EGFR , HER
T12584	PXS-5120A		Others , Monoamine Oxidase
	PXS-5120A is an irreversible fluoroallylamine Lysyl Oxidase-like 2/3 (LOXL2/3) inhibitor with anti-fibrotic activity.		Others , Monoamine Oxidase
T13088	Tarloxotinib bromide	TH-4000	EGFR , HER
			EGFR , HER
T13378	Z-Asp-CH2-DCB		Others
	Z-Asp-CH2-DCB is an irreversible inhibitor of broad spectrum caspase.		Others
TQ0300	Conduritol B epoxide		Glucosidase
	Conduritol B epoxide is an irreversible inhibitor of β-glucosidase (GCase).		Glucosidase
T3466	FIIN-3		EGFR , FGFR
	FIIN-3 is an irreversible inhibitor of FGFR.		EGFR , FGFR
T23602	ABC99	ABC 99,ABC-99	Wnt/beta-catenin
	ABC99 is a selective irreversible inhibitor of the wnt-deacylating enzyme. ABC99 inhibited NOTUM (IC50: 13 nM). It also showed excellent selectivity across the serine hydrolase family.		Wnt/beta-catenin
T1578	Pargyline hydrochloride	Pargylamine hydrochloride	MAO , Monoamine Oxidase
	Pargyline hydrochloride (Pargylamine hydrochloride) is an irreversible monoamine oxidase(MAO) inhibitor with antihypertensive properties.		MAO , Monoamine Oxidase
T9004	TM2-115		Parasite
	TM2-115 is a inhibitor of malaria parasite histone methyltransferases that results in rapid and irreversible parasite death [1].		Parasite
T5492	JAK3-IN-6		JAK
	JAK3-IN-6 is irreversible Janus Associated Kinase 3 (JAK3) inhibitor, with an IC50 of 0.15 nM		JAK
T1941	GSK3787		PPAR
	GSK3787 is a specific and irreversible PPARδ inhibitor（pIC50= 6.6）.		PPAR
T10864	Corin		Histone Demethylase , HDAC
	Corin is an irreversible inhibitor of HDAC1(IC50 = 147 nM) and LSD1(Ki = 110 nM).		Histone Demethylase , HDAC
T0821	Iproniazid Phosphate	Isoproniazid phosphate	MAO , Monoamine Oxidase
	Iproniazid Phosphate is a non-selective, irreversible monoamine oxidase inhibitor (MAOI).		MAO , Monoamine Oxidase
T6008	CNX-2006	CNX 2006,CNX2006	EGFR
	CNX-2006 is a novel irreversible mutant-selective EGFR inhibitor with IC50 of < 20 nM, with very weak inhibition at wild-type EGFR.		EGFR
T3677	GSK2879552	GSK2879552 2HCl	Histone Demethylase
	GSK2879552 is a selective, orally bioavailable, irreversible, mechanism-based inactivator of lysine-specific demethylase 1 (LSD1)/corepressor, with potential antineoplastic activity.		Histone Demethylase
T6370	AEBSF hydrochloride	AEBSF HCl,Pefabloc SC	Thrombin , Serine Protease , Influenza Virus
	AEBSF hydrochloride (Pefabloc SC) is an irreversible inhibitor of serine proteases, such as chymotrypsin, kallikrein, thrombin, plasmin, and trypsin.		Thrombin , Serine Protease , Influenza Virus
T41277	PACMA 31		Others
	PACMA 31 is an irreversible and covalent inhibitor of protein disulfide isomerase (PDI) with an IC50 of 10 μM. PACMA 31 significantly suppresses ovarian tumor growth and exhibits tumor targeting ability.		Others
T15303	FMK 9a		Cysteine Protease , Autophagy
	FMK 9a is an irreversible inhibitor of ATG4B with IC50 values of 80 and 73 nM in the TR-FRET and cellular-based LRA assays.		Cysteine Protease , Autophagy
T37906	Dibenamine hydrochloride		Adrenergic Receptor
	Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.		Adrenergic Receptor
T5199	COH000		E1/E2/E3 Enzyme
	COH000 is a covalent and irreversible inhibitor of small ubiquitin-like modifier (SUMO)-activating enzyme and inhibited SUMOylation (IC50: ~ 0.2 μM in vitro).		E1/E2/E3 Enzyme
T9706	BTK inhibitor 17		BTK
	BTK inhibitor 17 is a potent irreversible BTK inhibitor (IC50 = 2.1 nM). BTK inhibitor 17 can be used in rheumatoid arthritis studies.		BTK
T6836	FIIN-2		FGFR
	FIIN-2, an irreversible, pan-FGFR inhibitor, inhibits FGFR1/2/3/4 with IC50 of 3.09 nM, 4.3 nM, 27 nM and 45.3 nM, respectively.		FGFR
T3634	Osimertinib mesylate	Mereletinib mesylate,AZD-9291 mesylate	EGFR
	Osimertinib mesylate (Mereletinib mesylate) is an irreversible and mutant selective EGFR inhibitor (IC50s: 12/1 nM for EGFR(L858R) and EGFR(L858R/T790M)).		EGFR
T26389	4-POBN	NSC-640,NSC640,4-Aminobenzohydrazide,NSC 640,Myeloperoxidase Inhibitor 1,4-ABAH	Glutathione Peroxidase
	4-POBN (Myeloperoxidase Inhibitor 1) is a potent and irreversible inhibitor of myeloperoxidase (IC50 = 0.3 µM). 4-POBN can be used in studies about subacute stroke.		Glutathione Peroxidase
TP1466	Z-YVAD-FMK		Caspase
	AA-Z-YVAD-FMK is a Irreversible caspase-1 inhibitor,with anti-inflammatory and anti-tumor activities.		Caspase
T4006	Pentostatin	Nipent,CI-825,Covidarabine,Deoxycoformycin	Adenosine deaminase , Adenosine Receptor
	Pentostatin (CI-825) is an extremely effective and irreversible inhibitor of adenosine deaminase (Ki: 2.5 pM).		Adenosine deaminase , Adenosine Receptor
T3721	Avitinib maleate		EGFR
	Avitinib maleate is a pyrrolopyrimidine-based irreversible epidermal growth factor receptor (EGFR) inhibitor.		EGFR

Compounds

FIIN-1

T37426

Synonym: FGFR irreversible inhibitor-1

4-Diethylaminobenzaldehyde

T10140

Synonym:

Target: Dehydrogenase

Menin-MLL inhibitor 20

T9399

Synonym:

Target: Epigenetic Reader Domain, Histone Methyltransferase

Sulbactam sodium

T6685

Synonym: CP-45899-2

Target: Antibacterial, Antibiotic

Almonertinib mesylate

Target: Antibacterial, Antibiotic

IPI-9119

T36841

Synonym:

Target: Fatty Acid Synthase

RN-1 dihydrochloride

T21652

Synonym:

Target: Histone Demethylase, MAO

Synonym: AST-1306,ALS 1306

Synonym: (R)-Etomoxir sodium salt,Na salt,Etomoxir

Target: Apoptosis, Others

Fenclonine

T1447

Synonym: Fenchlonine,PCPA,CP-10188,4-Chloro-DL-phenylalanine,DL-4-Chlorophenylalanine

Target: Hydroxylase

Allitinib tosylate

T6331

Synonym: AST-1306 TsOH,AST-6,Allitinib,AST-1306,AST-1306 (TsOH)

Target: NOD-like Receptor (NLR), NOD

Synonym: Methyl Arachidonyl Fluorophosphonate

Target: Phospholipase

MPO-IN-28

T5340

Synonym:

Target: Glutathione Peroxidase

Poziotinib

T2630

Synonym: HM781-36B,NOV120101

Target: Apoptosis, EGFR, HER

PXS-5120A

T12584

Synonym:

Target: Others, Monoamine Oxidase

Synonym: ABC 99,ABC-99

Target: Wnt/beta-catenin

Pargyline hydrochloride

T1578

Synonym: Pargylamine hydrochloride

Target: MAO, Monoamine Oxidase

Target: Histone Demethylase, HDAC

Iproniazid Phosphate

T0821

Synonym: Isoproniazid phosphate

Target: MAO, Monoamine Oxidase

CNX-2006

T6008

Synonym: CNX 2006,CNX2006

Target: EGFR

GSK2879552

T3677

Synonym: GSK2879552 2HCl

Target: Histone Demethylase

AEBSF hydrochloride

T6370

Synonym: AEBSF HCl,Pefabloc SC

Target: Thrombin, Serine Protease, Influenza Virus

Target: Cysteine Protease, Autophagy

Dibenamine hydrochloride

T37906

Synonym:

Target: Adrenergic Receptor

COH000

T5199

Synonym:

Target: E1/E2/E3 Enzyme

Synonym: Mereletinib mesylate,AZD-9291 mesylate

Target: EGFR

4-POBN

T26389

Synonym: NSC-640,NSC640,4-Aminobenzohydrazide,NSC 640,Myeloperoxidase Inhibitor 1,4-ABAH

Target: Glutathione Peroxidase

Synonym: Nipent,CI-825,Covidarabine,Deoxycoformycin

Target: Adenosine deaminase, Adenosine Receptor

カタログ番号	製品名	別名	ターゲット
TN6848	Piperonylic acid	2H-1,3-benzodioxole-5-carboxylic acid	P450
	Piperonylic acid (2H-1,3-benzodioxole-5-carboxylic acid) is a natural molecule bearing a methylenedioxy function that closely mimics the structure of trans-cinnamic acid. Piperonylic acid selectively inactivate the CYP73...		P450
T3009	3-Nitropropanoic acid	3-NP acid,Bovinocidin,3-NP,β-Nitropropionic acid	Apoptosis , Dehydrogenase , Antibacterial
	3-Nitropropanoic acid (Bovinocidin) is an irreversible inhibitor of succinate dehydrogenase.		Apoptosis , Dehydrogenase , Antibacterial
T2898	Andrographolide	Andrographis	SARS-CoV , Influenza Virus , NF-κB , Autophagy
	Andrographolide (Andrographis)(Andrographis), an irreversible antagonist of NF-κB, has anti-inflammatory and anti-platelet aggregation activities and potential antineoplastic.		SARS-CoV , Influenza Virus , NF-κB , Autophagy
T6841	Fumagillin	NSC9168,Amebacilin	Others , HIV Protease , Antibiotic , Parasite
	Fumagillin (Amebacilin) is a selective and potent irreversible inhibitor of Methionine aminopeptidase 2 (MetAP2), used as an antibiotic to treat microsporidiosis.		Others , HIV Protease , Antibiotic , Parasite
T16012	Marizomib	NPI-0052,Salinosporamide A,ML858	Proteasome
	Marizomib (ML858) is a novel irreversible brain-permeable proteasome inhibitor that inhibits CT-L (β5), CT-T-laspase-like (C-L, β1), and trypsin-like (T-L, β2) 20S proteasomes with IC50s of 3.5, 28, and 430 nM, respectiv...		Proteasome
T11802	L-Canaline		Others
	L-Canaline, a nonprotein amino acid found in many leguminous plants, exhibits potent anticancer and antiproliferative effects. It effectively inhibits the growth of the malaria parasite Plasmodium falciparum with an IC50...		Others
T14055	5Z-7-Oxozeaenol	FR148083,L783279,LL-Z 1640-2	VEGFR , FLT , MEK , MAPK , PDGFR , Antibiotic , Src
	5Z-7-Oxozeaenol (FR148083) is a potent, irreversible and selective inhibitor of transforming growth factor (TGF)-β-activated kinase 1 with IC50 of 8.1 nM for TAK1 and low activity against MEK1 with IC50 of 411 nM, it is ...		VEGFR , FLT , MEK , MAPK , PDGFR , Antibiotic , Src
T75541	Tanshinone IIA anhydride
	Tanshinone IIA anhydride is a potent, irreversible inhibitor of human carboxylesterase (CE), exhibiting inhibitory constants (K i values) of 1.9 nM for human CE1 and 1.4 nM for human intestinal CE (hiCE), respectively [1...
T72508	Palmatine hydroxide
	Palmatine hydroxide is an orally active, irreversible inhibitor of indoleamine 2,3-dioxygenase 1 (IDO-1), demonstrating IC50 values of 3 μM for HEK 293-hIDO-1 and 157μM for rhIDO-1. Additionally, it uncompetitively inhib...

天然物製品

Piperonylic acid

TN6848

Synonym: 2H-1,3-benzodioxole-5-carboxylic acid

Target: P450

3-Nitropropanoic acid

T3009

Synonym: 3-NP acid,Bovinocidin,3-NP,β-Nitropropionic acid

Target: Apoptosis, Dehydrogenase, Antibacterial

Andrographolide

T2898

Synonym: Andrographis

Target: SARS-CoV, Influenza Virus, NF-κB, Autophagy

Fumagillin

T6841

Synonym: NSC9168,Amebacilin

Target: Others, HIV Protease, Antibiotic, Parasite

Marizomib

T16012

Synonym: NPI-0052,Salinosporamide A,ML858

Synonym: FR148083,L783279,LL-Z 1640-2

Target: VEGFR, FLT, MEK, MAPK, PDGFR, Antibiotic, Src

Tanshinone IIA anhydride

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPH-00722	PykF Protein, E. coli, Recombinant (His)	E. coli	E. coli
	Catalyzes the formation of pyruvate in the last step of glycolysis, it is irreversible under physiological conditions. The reaction is critical for the control of metabolic flux in the second part of glycolysis.
TMPH-03721	IbpA Protein, Yersinia pestis bv. Antiqua, Recombinant (His)	Yersinia pestis	E. coli
	Associates with aggregated proteins, together with IbpB, to stabilize and protect them from irreversible denaturation and extensive proteolysis during heat shock and oxidative stress. Aggregated proteins bound to the Ibp...
TMPH-03702	MTA/SAH nucleosidase Protein, Vibrio cholerae serotype O1, Recombinant (His & Myc)	Vibrio cholerae	E. coli
	Catalyzes the irreversible cleavage of the glycosidic bond in both 5'-methylthioadenosine (MTA) and S-adenosylhomocysteine (SAH/AdoHcy) to adenine and the corresponding thioribose, 5'-methylthioribose and S-ribosylhomocy...
TMPY-03617	GMPR Protein, Human, Recombinant (His)	Human	E. coli
	GMPR, also known as GMPR1, belongs to the IMPDH/GMPR family.This familyofenzymesincludesIMP dehydrogenaseandGMP reductase. These enzymes are involved inpurine metabolism and adopt aTIM barrelstructure. GMPR is an enzyme ...
TMPH-00567	MTA/SAH nucleosidase Protein, E. coli, Recombinant (His & Myc)	E. coli	E. coli
	Catalyzes the irreversible cleavage of the glycosidic bond in both 5'-methylthioadenosine (MTA) and S-adenosylhomocysteine (SAH/AdoHcy) to adenine and the corresponding thioribose, 5'-methylthioribose and S-ribosylhomocy...
TMPH-00692	MTA/SAH nucleosidase Protein, E. coli O9:H4, Recombinant (His & Myc)	E. coli	E. coli
	Catalyzes the irreversible cleavage of the glycosidic bond in both 5'-methylthioadenosine (MTA) and S-adenosylhomocysteine (SAH/AdoHcy) to adenine and the corresponding thioribose, 5'-methylthioribose and S-ribosylhomocy...
TMPH-01597	KYAT1 Protein, Human, Recombinant (His & SUMO)	Human	E. coli
	Catalyzes the irreversible transamination of the L-tryptophan metabolite L-kynurenine to form kynurenic acid (KA), an intermediate in the tryptophan catabolic pathway which is also a broad spectrum antagonist of the thre...
TMPH-02395	Lassa virus (strain GA391) GPC Protein (His)	LASV	in vitro E. coli expression system
	class I viral fusion protein that directs fusion of viral and host endosomal membranes, leading to delivery of the nucleocapsid into the cytoplasm. Membrane fusion is mediated by irreversible conformational changes induc...
TMPH-01598	CCBL2 Protein, Human, Recombinant (His & SUMO)	Human	E. coli
	Catalyzes the irreversible transamination of the L-tryptophan metabolite L-kynurenine to form kynurenic acid (KA), an intermediate in the tryptophan catabolic pathway which is also a broad spectrum antagonist of the thre...
TMPH-02393	Lassa virus (strain Mouse/Sierra Leone/Josiah/1976) GPC Protein (His & Myc)	LASV	E. coli
	interacts with the host receptor. Mediates virus attachment to host receptor alpha-dystroglycan DAG1. This attachment induces virion internalization predominantly through clathrin- and caveolin-independent endocytosis.; ...
TMPY-03501	Optineurin Protein, Human, Recombinant (His & GST)	Human	Baculovirus-Insect Cells
	OPTN (Optineurin) is a Protein Coding gene. The Optineurin gene encodes the coiled-coil containing protein optineurin. Optineurin is a multifunctional adaptor protein intimately involved in various vesicular trafficking ...
TMPH-02412	Lymphocytic choriomeningitis virus (LCMV) (strain WE) GPC Protein (His & Myc)	LCMV	E. coli
	class I viral fusion protein that directs fusion of viral and host endosomal membranes, leading to delivery of the nucleocapsid into the cytoplasm. Membrane fusion is mediated by irreversible conformational changes induc...
TMPH-02345	Influenza A H1N1 (train A/Hickox/1940) Hemagglutinin/HA Protein (His & SUMO)	H1N1	E. coli
	Binds to sialic acid-containing receptors on the cell surface, bringing about the attachment of the virus particle to the cell. This attachment induces virion internalization either through clathrin-dependent endocytosis...
TMPH-02394	Lassa virus (strain GA391) GPC Protein (His & Myc)	LASV	E. coli
	class I viral fusion protein that directs fusion of viral and host endosomal membranes, leading to delivery of the nucleocapsid into the cytoplasm. Membrane fusion is mediated by irreversible conformational changes induc...
TMPJ-00819	Trp A Protein, E. coli, Recombinant	E.coli	E. coli
	Tryptophan synthase is an enzyme that catalyzes the final two steps in the biosynthesis of tryptophan. It is commonly found in Eubacteria, Archaebacteria, Protista, Fungi, and Plantae, but is absent from animals such as ...
TMPJ-00820	Trp B Protein, E. coli, Recombinant (His)	E.coli	E. coli
	Tryptophan synthase is an enzyme that catalyzes the final two steps in the biosynthesis of tryptophan. It is commonly found in Eubacteria, Archaebacteria, Protista, Fungi, and Plantae, but is absent from animals such as ...
TMPH-02413	Lymphocytic choriomeningitis virus (LCMV) (strain Armstrong) GPC Protein (His & SUMO)	LCMV	E. coli
	class I viral fusion protein that directs fusion of viral and host endosomal membranes, leading to delivery of the nucleocapsid into the cytoplasm. Membrane fusion is mediated by irreversible conformational changes induc...
TMPY-03452	PTS Protein, Human, Recombinant (His)	Human	E. coli
	PTS(6-pyruvoyltetrahydropterin synthase) belongs to the PTPS family. It catalyzes the elimination of inorganic triphosphate from dihydroneopterin triphosphate, which is the second and irreversible step in the biosynthesi...
TMPY-01284	METTL11A Protein, Human, Recombinant (GST)	Human	E. coli
	Methyltransferase-like protein 11A, also known as METTL11A, is a member of the methyltransferase superfamily and METTL11 family. Methyltransferase is a type of transferase enzyme which transfers a methyl group from a don...
TMPY-01285	METTL11A Protein, Human, Recombinant	Human	E. coli
	Methyltransferase-like protein 11A, also known as METTL11A, is a member of the methyltransferase superfamily and METTL11 family. Methyltransferase is a type of transferase enzyme which transfers a methyl group from a don...
TMPJ-00990	S100B Protein, Mouse, Recombinant (His)	Mouse	E. coli
	S100-B, is an acidic protein with a molecular weight of 21 kDa belonging to the S100 family. S100-B contains two EF-hand-type calcium-binding motifs separated by a hinge region with a hydrophobic cleft. S100-B plays an i...
TMPY-02063	Alpha-2-macroglobulin Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	alpha-2-macroglobulin, also known as α2-macroglobulin (α2M and A2M), is an abundant protein of the plasma of vertebrates and members of several invertebrate phyla and functions as a broad-spectrum protease-binding protei...
TMPH-01262	PRKN Protein, Human, Recombinant (His & Myc)	Human	Baculovirus
	Functions within a multiprotein E3 ubiquitin ligase complex, catalyzing the covalent attachment of ubiquitin moieties onto substrate proteins. Substrates include SYT11 and VDAC1. Other substrates are BCL2, CCNE1, GPR37, ...
TMPH-01263	PRKN Protein, Human, Recombinant (His & SUMO)	Human	E. coli
	Functions within a multiprotein E3 ubiquitin ligase complex, catalyzing the covalent attachment of ubiquitin moieties onto substrate proteins. Substrates include SYT11 and VDAC1. Other substrates are BCL2, CCNE1, GPR37, ...
TMPH-02631	PRKN Protein, Mouse, Recombinant (GST)	Mouse	E. coli
	Functions within a multiprotein E3 ubiquitin ligase complex, catalyzing the covalent attachment of ubiquitin moieties onto substrate proteins. Substrates include SYT11 and VDAC1. Other substrates are BCL2, CCNE1, GPR37, ...
TMPH-03281	PRKN Protein, Rat, Recombinant (His & Myc)	Rat	Baculovirus
	Functions within a multiprotein E3 ubiquitin ligase complex, catalyzing the covalent attachment of ubiquitin moieties onto substrate proteins. Substrates include SYT11 and VDAC1. Other substrates are BCL2, CCNE1, GPR37, ...

PykF Protein, E. coli, Recombinant (His)

TMPH-00722

Species: E. coli

Expression System: E. coli

IbpA Protein, Yersinia pestis bv. Antiqua, Recombinant (His)

TMPH-03721

Species: Yersinia pestis

Expression System: E. coli

MTA/SAH nucleosidase Protein, Vibrio cholerae serotype O1, Recombinant (His & Myc)

TMPH-03702

Species: Vibrio cholerae

Expression System: E. coli

GMPR Protein, Human, Recombinant (His)

TMPY-03617

Species: Human

Expression System: E. coli

MTA/SAH nucleosidase Protein, E. coli, Recombinant (His & Myc)

TMPH-00567

Species: E. coli

Expression System: E. coli

MTA/SAH nucleosidase Protein, E. coli O9:H4, Recombinant (His & Myc)

TMPH-00692

Species: E. coli

Expression System: E. coli

KYAT1 Protein, Human, Recombinant (His & SUMO)

TMPH-01597

Species: Human

Expression System: E. coli

Lassa virus (strain GA391) GPC Protein (His)

TMPH-02395

Species: LASV

Expression System: in vitro E. coli expression system

CCBL2 Protein, Human, Recombinant (His & SUMO)

TMPH-01598

Species: Human

Expression System: E. coli

Lassa virus (strain Mouse/Sierra Leone/Josiah/1976) GPC Protein (His & Myc)

TMPH-02393

Species: LASV

Expression System: E. coli

Optineurin Protein, Human, Recombinant (His & GST)

TMPY-03501

Species: Human

Expression System: Baculovirus-Insect Cells

Lymphocytic choriomeningitis virus (LCMV) (strain WE) GPC Protein (His & Myc)

TMPH-02412

Species: LCMV

Expression System: E. coli

Influenza A H1N1 (train A/Hickox/1940) Hemagglutinin/HA Protein (His & SUMO)

TMPH-02345

Species: H1N1

Expression System: E. coli

Lassa virus (strain GA391) GPC Protein (His & Myc)

TMPH-02394

Species: LASV

Expression System: E. coli

Trp A Protein, E. coli, Recombinant

TMPJ-00819

Species: E.coli

Expression System: E. coli

Trp B Protein, E. coli, Recombinant (His)

TMPJ-00820

Species: E.coli

Expression System: E. coli

Lymphocytic choriomeningitis virus (LCMV) (strain Armstrong) GPC Protein (His & SUMO)

TMPH-02413

Species: LCMV

Expression System: E. coli

PTS Protein, Human, Recombinant (His)

TMPY-03452

Species: Human

Expression System: E. coli

METTL11A Protein, Human, Recombinant (GST)

TMPY-01284

Species: Human

Expression System: E. coli

METTL11A Protein, Human, Recombinant

TMPY-01285

Species: Human

Expression System: E. coli

S100B Protein, Mouse, Recombinant (His)

TMPJ-00990

Species: Mouse

Expression System: E. coli

Alpha-2-macroglobulin Protein, Human, Recombinant (His)

TMPY-02063

Species: Human

Expression System: Baculovirus-Insect Cells

PRKN Protein, Human, Recombinant (His & Myc)

TMPH-01262

Species: Human

Expression System: Baculovirus

PRKN Protein, Human, Recombinant (His & SUMO)

TMPH-01263

Species: Human

Expression System: E. coli

PRKN Protein, Mouse, Recombinant (GST)

TMPH-02631

Species: Mouse

Expression System: E. coli

PRKN Protein, Rat, Recombinant (His & Myc)

TMPH-03281

Species: Rat

Expression System: Baculovirus

カタログ番号	製品名
L9410	Covalent Inhibitor Library	1920 compounds
	A unique collection of 1920 covalent Inhibitors and other molecules with common warheads like chloroacetyl，2-Chloropropionyl，Acryloyl，sulfonyl fluoride, alkyne，acrylamide, ketocarbonyl，disulfide bond, etc.
L6150	Covalent Natural Product Library	583 compounds
	Detialed biological information and pharmacological information of the products, providing theoretical direction and research basis for screening.

ライブラリー

Covalent Inhibitor Library

L9410

Compounds: 1920

Covalent Natural Product Library

L6150

Compounds: 583