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天然化合物

リコンビナントタンパク質

同位体標識化合物

カタログ番号	製品名	別名	ターゲット
T23745	APA-APA-MPO	APA APA MPO,APAAPAMPO	Others
	APA-APA-MPO is a PCAF bromodomain/Tat-AcK50 association inhibitor.		Others
T40191	17-GMB-APA-GA		Others
	17-GMB-APA-GA, a potent HSP90 inhibitor, is an ADC cytotoxin commonly employed for studying latent T. gondii infection.		Others
T23746	APA-H-MPO	APAHMPO	Others
	APA-H-MPO is a PCAF bromodomain/Tat-AcK50 association inhibitor.		Others
T3407	Rapastinel	GLYX-13,Thr-Pro-Pro-Thr-NH2,TPPT-amide	NMDAR , iGluR
	Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.		NMDAR , iGluR
T67849	O-Desethyl Dapagliflozin	Empagliflozin-4	SGLT
	O-Desethyl Dapagliflozin (Empagliflozin-4) is a SGLT2 inhibitor, IC50=33nM.		SGLT
T5819	Rapastinel Trifluoroacetate	Thr-Pro-Pro-Thr-NH2 Trifluoroacetate,GLYX-13 Trifluoroacetate	NMDAR , iGluR
	Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.		NMDAR , iGluR
T6638	Retapamulin	SB-275833	ribosome , Antibacterial , Antibiotic
	Retapamulin (SB-275833), a Pleuromutilin Antibacterial, binds to both E. coli and S. aureus ribosomes with similar potencies (Kd: 3 nM).		ribosome , Antibacterial , Antibiotic
T6127	Rucaparib Phosphate	AG-014699 phosphate,PF-01367338,AG-014699,PF-01367338 phosphate	PARP
	Rucaparib Phosphate (PF-01367338 phosphate) is an inhibitor of PARP (Ki: 1.4 nM for PARP1) that is used in clinical therapy to sensitize cancer cells to chemotherapy.		PARP
T10820L1	Ciraparantag acetate	Ciraparantag acetate(1438492-26-2 Free base)	Others
	Ciraparantag acetate, an anticoagulant reversal agent, is a small molecule specifically designed to bind noncovalently by charge-charge interaction to unfractionated heparin and low-molecular-weight heparin. It shows bin...		Others
T2480	Apabetalone	RVX-208,RVX000222	Epigenetic Reader Domain , HIV Protease
	Apabetalone (RVX000222) , an effective BET bromodomain inhibitor, has been investigated for the treatment of diabetes, atherosclerosis, and coronary artery disease.		Epigenetic Reader Domain , HIV Protease
T1010	Verapamil hydrochloride	Manidon,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride	P450 , Calcium Channel , P-gp
	Verapamil hydrochloride (Verapamil HCl) is a calcium channel blocker that is a class IV anti-arrhythmia agent.		P450 , Calcium Channel , P-gp
T9430	Venadaparib	NOV140101,IDX-1197	PARP
	Venadaparib (NOV140101) (IDX-1197) is a potent, selective and orally active PARP inhibitor with IC50s of 1.4 nM and 1.0 nM for PARP1 and PARP2, respectively. Venadaparib is insensitive to PARP-5. Venadaparib prevents the...		PARP
T4463	Rucaparib	AG-14447,PF-01367338,AG014699	PARP
	Rucaparib (PF-01367338) is an inhibitor of PARP with Ki of 1.4 nM for PARP1 in a cell-free assay, and also shows binding affinity to eight other PARP.		PARP
T16339	Norverapamil hydrochloride	(±)-Norverapamil hydrochloride,D591 hydrochloride	Calcium Channel , P-gp , Drug Metabolite
	Norverapamil hydrochloride (D591 hydrochloride) ((±)-Norverapamil hydrochloride) is an N-demethylated metabolite of Verapamil and it is an L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor.		Calcium Channel , P-gp , Drug Metabolite
TQ0245	Sapacitabine	CS682,CYC682	Nucleoside Antimetabolite/Analog
	Sapacitabine (CS682) is an orally available nucleoside analog precursor compound with potential anti-tumor activity for the study of acute myeloid leukemia.		Nucleoside Antimetabolite/Analog
T7587	Tenapanor	RDX-5791,RDX 5791,AZD 1722,Tenapanor free base,RDX5791,AZD-1722,AZD1722	Sodium Channel
	Tenapanor (RDX 5791) is an inhibitor of the sodium-proton (Na(+)/H(+)) exchanger NHE3, which plays a prominent role in sodium handling in the gastrointestinal tract and kidney. Tenapanor possesses an excellent preclinica...		Sodium Channel
T11506	Guaiapate	Mg 5454,Klamar	Others
	Guaiapate has an antitussive and sedative effect.		Others
T9497	Niraparib tosylate monohyrate		PARP
	Niraparib, also know as MK-4827, is an inhibitor of poly (ADP-ribose) polymerase (PARP) with potential antineoplastic activity. MK4827 inhibits PARP activity, enhancing the accumulation of DNA strand breaks and promoting...		PARP
T6763	Xevinapant	ARRY-334543,SM-406,AT406,Debio-1143	IAP
	Xevinapant (Debio-1143) is a potent Smac mimetic and an antagonist of IAP (inhibitor of apoptosis protein via E3 ubiquitin ligase), binding to XIAP-BIR3, cIAP1-BIR3 and cIAP2-BIR3 with Ki of 66.4 nM, 1.9 nM, and 5.1 nM, ...		IAP
T76742	Emapalumab	NI-0501	COX
	Emapalumab (NI-0501) is an IgG1 monoclonal antibody that humanizes human monoclonal antibodies against interferon gamma, blocking its binding to cell surface receptors and activating inflammatory signaling. Emapalumab ha...		COX
T12146	N-Desmethyl-Apalutamide	N-Desmethyl Apalutamide	P450 , Androgen Receptor
	N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.		P450 , Androgen Receptor
T3353	Niraparib hydrochloride	MK-4827 hydrochloride,MK-4827 (hydrochloride)	Apoptosis , Others , PARP
	Niraparib hydrochloride (MK-4827 hydrochloride) is an inhibitor of poly (ADP-ribose) polymerase (PARP) with potential antineoplastic activity. Niraparib hydrochloride inhibits PARP activity, enhancing the accumulation of...		Apoptosis , Others , PARP
T3098	Vorapaxar sulfate	SCH 530348 sulfate,Zontivity,vorapaxar monosulfate	Protease-activated Receptor
	Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.		Protease-activated Receptor
T9593	Senaparib	IMP4297	PARP
	Senaparib (IMP4297) is a novel highly potent and selective oral PARP1/2 inhibitor with strong antitumor activity.		PARP
T26641L	Apadenoson TFA	BAY 68-4986 TFA,Apadenoson TFA(250386-15-3 Free base),Discontinued TFA	Adenosine Receptor
	Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.		Adenosine Receptor
T63971	Canocapavir	ZM-H1505R	HBV
	Canocapavir (ZM-H1505R) is a novel orally available HBV coat protein modulator with antiviral activity that induces conformational changes in the linker region of the HBV core protein, and can be used for the treatment o...		HBV
T16999	Tavapadon	PF-6649751,CVL-751	Dopamine Receptor
	Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.		Dopamine Receptor
T0078L	Lapatinib ditosylate monohydrate	Lapatinib ditosylate monohydrate,Lapatinib ditoluenesulfonate monohydrate,Lapatinib tosilate hydrate,Lapatinib tosilate,Tykerb,Tyverb	EGFR , Ferroptosis , Autophagy
	Lapatinib ditosylate (Lapatinib tosilate) monohydrate is a tyrosine kinase receptor inhibitor used in the therapy of advanced breast cancer and other solid tumors. Lapatinib ditosylate monohydrate therapy is associated w...		EGFR , Ferroptosis , Autophagy
T4460	Dapagliflozin ((2S)-1,2-propanediol, hydrate)	BMS-512148 (2S)-1,2-propanediol, hydrate,Dapagliflozin propanediol monohydrate	SGLT
	Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-transporter type 2 (SGLT2). It is in development for the tre...		SGLT
T6235	Lapatinib Ditosylate	Lapatinib (GW-572016) Ditosylate,GW-572016 ditosylate,Tykerb ditosylate	EGFR , Ferroptosis , Autophagy
	Lapatinib Ditosylate (Tykerb ditosylate) is an effective EGFR and ErbB2 inhibitor (IC50: 10.8/9.2 nM for EGFR/ErbB2).		EGFR , Ferroptosis , Autophagy
T14301	Apararenone	MT-3995	Glucocorticoid Receptor
	Apararenone (MT-3995) is a receptor antagonist of mineralocorticoid receptor which can be used to treat non-alcoholic steatohepatitis and diabetic nephropathy.		Glucocorticoid Receptor
T3218	Napabucasin	BBI608	STAT
	Napabucasin (BBI608) is an orally available Stat3 and Y cell stemness inhibitor.		STAT
T16807	Rucaparib monocamsylate	Rucaparib Camsylate	PARP
	Rucaparib monocamsylate (Rucaparib Camsylate) is a PARP inhibitor (PARP1,Ki of 1.4 nM). Rucaparib Camsylate also displays binding affinity to eight other PARP domains.		PARP
T0113	Mebhydrolin napadisylate	Incidal,Diazolin,Mebhydroline 1,5-naphthalenedisulfonate salt,Omeril,Diazoline	5-HT Receptor , AChR , Histamine Receptor
	Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic dermatosis.		5-HT Receptor , AChR , Histamine Receptor
T6892	Niraparib tosylate	MK-4827 (tosylate),MK 4827 tosylate,Niraparib (MK-4827) tosylate	Apoptosis , PARP
	Niraparib tosylate (MK-4827 (tosylate))(with IC50 of 3.8 nM/2.1 nM) is a selective PARP1/PARP2 inhibitor.		Apoptosis , PARP
T68055	Devapamil	Devapamilo,Devapamilum	Calcium Channel
	Devapamil (Devapamilo) is a phenylalkylamine that blocks L-type calcium currents from the inner side of membrane cells in a use-dependent manner.		Calcium Channel
T4434	Tirapazamine	Tirazone,Win59075,SR4233,SR259075	Others
	Tirapazamine (Win59075) is a potent cytotoxic agent under hypoxic conditions, can induce apoptosis by inducing breaks in single and double-stranded DNA, as well as chromosomal breaks. The compound sensitizes cells to oth...		Others
T2389	Dapagliflozin	BMS-512148	SGLT , HIF
	Dapagliflozin (BMS-512148) is a selective sodium-glucose co-transporter subtype 2 (SGLT2) inhibitor with antihyperglycemic activity.		SGLT , HIF
T16802	Lonapalene	RS4317	Lipoxygenase
	Lonapalene (RS4317) is a 5-lipoxygenase (5-LO) inhibitor with anti-psoriasis efficacy.Lonapalene topically blocks skin inflammation.		Lipoxygenase
T15273	Fedovapagon	VA483,A106483	Vasopressin Receptor
	Fedovapagon (VA106483) is a selective and potent agonist of the vasopressin V2 receptor (V2R) that inhibits the growth of intersegmental vessels in zebrafish. Fedovapagon can be used to study overactive bladder, nocturia...		Vasopressin Receptor
T74048	PAPA NONOate		Endogenous Metabolite , NO Synthase
	PAPA NONOate is a pH-regulated NO donor.PAPA NONOate has potential antitumor activity and can be used to study diabetic wound healing disorders.		Endogenous Metabolite , NO Synthase
T15052	Dapansutrile		NOD-like Receptor (NLR) , NOD
	Dapansutrile is a potent, selective and orally active NLRP3 inflammasome inhibitor, with Anti-inflammatory and analgesic activity.		NOD-like Receptor (NLR) , NOD
TP1223L	Apamin acetate	Apamine acetate,Apamin acetate(24345-16-2 Free base)	Potassium Channel
	Apamin acetate (Apamine acetate) is a selective Ca2+-activated blocker of K+ (SK) channels, an 18-amino acid peptide neurotoxin found in bee toxins.Apamin acetate enhances synapse growth and regeneration following lacera...		Potassium Channel
T7013	Vorapaxar	SCH 530348,MK-5348	Protease-activated Receptor
	Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).		Protease-activated Receptor
T0078	Lapatinib	GSK572016,GW572016	EGFR , Ferroptosis , Autophagy
	Lapatinib (GW572016) is an inhibitor of ErbB2 and EGFR (IC50=9.2/10.8 nM) with oral activity. Lapatinib has antitumor activity and can be used to treat advanced or metastatic breast cancer with HER2 overexpression.		EGFR , Ferroptosis , Autophagy
TQ0125	Capadenoson	BAY 68-4986	Adenosine Receptor
	Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.		Adenosine Receptor
T60097	Methyl (E)-sinapate		Others
	Methyl (E)-sinapate is isolated from the Polygala sibirica L.var. megalopha Fr.		Others
T3231	Niraparib	MK-4827	Apoptosis , Others , PARP
	Niraparib (MK-4827) is a PARP inhibitor that selectively inhibits PARP1 and PARP2 (IC50=3.8/2.1 nM). Niraparib has antitumor activity, inhibits DNA damage repair, and induces apoptosis.		Apoptosis , Others , PARP
T2339	Apalutamide	ARN-509	Androgen Receptor , GABA Receptor
	Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.		Androgen Receptor , GABA Receptor
T22323	Enoxaparin sodium		Thrombin
	Enoxaparin sodium is a low-molecular-weight heparin (LMWH) that has recently been approved by the US FDA for use in patients with medically managed ST-segment myocardial infarction (STEMI), or STEMI with subsequent percu...		Thrombin

Compounds

APA-APA-MPO

T23745

Synonym: APA APA MPO,APAAPAMPO

Synonym: GLYX-13,Thr-Pro-Pro-Thr-NH2,TPPT-amide

Target: NMDAR, iGluR

O-Desethyl Dapagliflozin

T67849

Synonym: Empagliflozin-4

Target: SGLT

Rapastinel Trifluoroacetate

T5819

Synonym: Thr-Pro-Pro-Thr-NH2 Trifluoroacetate,GLYX-13 Trifluoroacetate

Target: ribosome, Antibacterial, Antibiotic

Rucaparib Phosphate

T6127

Synonym: AG-014699 phosphate,PF-01367338,AG-014699,PF-01367338 phosphate

Target: PARP

Ciraparantag acetate

T10820L1

Synonym: Ciraparantag acetate(1438492-26-2 Free base)

Target: Others

Apabetalone

T2480

Synonym: RVX-208,RVX000222

Target: Epigenetic Reader Domain, HIV Protease

Verapamil hydrochloride

T1010

Synonym: Manidon,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride

Target: P450, Calcium Channel, P-gp

Venadaparib

T9430

Synonym: NOV140101,IDX-1197

Target: PARP

Rucaparib

T4463

Synonym: AG-14447,PF-01367338,AG014699

Target: PARP

Norverapamil hydrochloride

T16339

Synonym: (±)-Norverapamil hydrochloride,D591 hydrochloride

Target: Calcium Channel, P-gp, Drug Metabolite

Sapacitabine

TQ0245

Synonym: CS682,CYC682

Target: Nucleoside Antimetabolite/Analog

Tenapanor

T7587

Synonym: RDX-5791,RDX 5791,AZD 1722,Tenapanor free base,RDX5791,AZD-1722,AZD1722

Target: Sodium Channel

Guaiapate

T11506

Synonym: Mg 5454,Klamar

Target: Others

Niraparib tosylate monohyrate

Synonym: ARRY-334543,SM-406,AT406,Debio-1143

N-Desmethyl-Apalutamide

T12146

Synonym: N-Desmethyl Apalutamide

Target: P450, Androgen Receptor

Niraparib hydrochloride

T3353

Synonym: MK-4827 hydrochloride,MK-4827 (hydrochloride)

Target: Apoptosis, Others, PARP

Vorapaxar sulfate

T3098

Synonym: SCH 530348 sulfate,Zontivity,vorapaxar monosulfate

Target: Protease-activated Receptor

Synonym: BAY 68-4986 TFA,Apadenoson TFA(250386-15-3 Free base),Discontinued TFA

Target: Adenosine Receptor

Synonym: PF-6649751,CVL-751

Target: Dopamine Receptor

Lapatinib ditosylate monohydrate

T0078L

Synonym: Lapatinib ditosylate monohydrate,Lapatinib ditoluenesulfonate monohydrate,Lapatinib tosilate hydrate,Lapatinib tosilate,Tykerb,Tyverb

Target: EGFR, Ferroptosis, Autophagy

Dapagliflozin ((2S)-1,2-propanediol, hydrate)

T4460

Synonym: BMS-512148 (2S)-1,2-propanediol, hydrate,Dapagliflozin propanediol monohydrate

Target: SGLT

Lapatinib Ditosylate

T6235

Synonym: Lapatinib (GW-572016) Ditosylate,GW-572016 ditosylate,Tykerb ditosylate

Target: EGFR, Ferroptosis, Autophagy

Apararenone

T14301

Synonym: MT-3995

Target: Glucocorticoid Receptor

Rucaparib monocamsylate

T16807

Synonym: Rucaparib Camsylate

Target: PARP

Mebhydrolin napadisylate

T0113

Synonym: Incidal,Diazolin,Mebhydroline 1,5-naphthalenedisulfonate salt,Omeril,Diazoline

Target: 5-HT Receptor, AChR, Histamine Receptor

Niraparib tosylate

T6892

Synonym: MK-4827 (tosylate),MK 4827 tosylate,Niraparib (MK-4827) tosylate

Target: Apoptosis, PARP

Devapamil

T68055

Synonym: Devapamilo,Devapamilum

Target: Calcium Channel

Tirapazamine

T4434

Synonym: Tirazone,Win59075,SR4233,SR259075

Synonym: VA483,A106483

Target: Vasopressin Receptor

PAPA NONOate

T74048

Synonym:

Target: Endogenous Metabolite, NO Synthase

Dapansutrile

T15052

Synonym:

Target: NOD-like Receptor (NLR), NOD

Apamin acetate

TP1223L

Synonym: Apamine acetate,Apamin acetate(24345-16-2 Free base)

Target: Potassium Channel

Vorapaxar

T7013

Synonym: SCH 530348,MK-5348

Target: Protease-activated Receptor

Lapatinib

T0078

Synonym: GSK572016,GW572016

Target: EGFR, Ferroptosis, Autophagy

Capadenoson

TQ0125

Synonym: BAY 68-4986

Target: Adenosine Receptor

Target: Apoptosis, Others, PARP

Apalutamide

T2339

Synonym: ARN-509

Target: Androgen Receptor, GABA Receptor

カタログ番号	製品名	別名	ターゲット
TN1569	Deoxylapachol		Antifection , Antifungal
	Deoxylapachol has anti-wood rot activity, it can inhibit the brown rot fungi Gloeophyllum sepiarium CBS 353.74 and Gloeophyllum trabeum CBS 318.50 and the white rot fungi Merulius tremellosus CBS 280.73 and Phlebia brevi...		Antifection , Antifungal
TN4893	Rapanone	2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione	Apoptosis , Phospholipase , Antibacterial , Parasite
	Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) is a natural benzoquinone that is a potent and selective inhibitor of human synovial PLA2.		Apoptosis , Phospholipase , Antibacterial , Parasite
T19503	Papain		Others , Cysteine Protease
	Papain is a cysteine protease of the peptidase C1 family. Papain is used in food, pharmaceutical, textile, and cosmetic industries.		Others , Cysteine Protease
T9218	Andrograpanin	19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE	p38 MAPK
	Andrograpanin (19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE) is a bioactive compound from Andrographis paniculata. Andrograpanin has anti-inflammatory and anti-infectious properties.		p38 MAPK
TN2281	Sinapaldehyde	trans-3,5-Dimethoxy-4-hydroxy cinnamaldehyde	Antibacterial
	Sinapaldehyde (trans-3,5-Dimethoxy-4-hydroxy cinnamaldehyde) is a natural product. Sinapaldehyde exhibits moderate antibacterial against Methicillin resistant S. aureus (MRSA) and E. coli with MIC values of 128 and 128 μ...		Antibacterial
T4136	Lapachol	Bethabarra wood,CI75490,Greenhartin,Tecomin	Others , Influenza Virus , Antibacterial , Parasite , Antifungal
	Lapachol (CI75490) has antimicrobial properties against many pathogens. It has anti-inflammatory, analgesic and antibiotic properties. It is an inhibitor of epithelial tumors in Drosophila melanogaster heterozygote.
TN7058	Dihydrolapachenole	6-methoxy-2,2-dimethyl-3,4-dihydro-2H-benzo[h]chromene	Others
	Dihydrolapachenole (6-methoxy-2,2-dimethyl-3,4-dihydro-2H-benzo[h]chromene) can be isolated from T. chrysantha.		Others
TN1375	α-Lapachone	alpha-Lapachone	Topoisomerase , Antifection
	α-Lapachone has antineoplastic activity, it shows an approximately trypanocidal activity against Trypanosoma cruzi.		Topoisomerase , Antifection
T6004	Tetrahydropapaverine hydrochloride	Tetrahydropapaverine HCl,Norlaudanosine HCl,Tetrahydroalkali hydrochloride	Hydroxylase
	Tetrahydropapaverine hydrochloride (Norlaudanosine HCl) , an analogue of salsolinol and tetrahydropapaveroline, has neurotoxicity on dopamine neurons.		Hydroxylase
T6407	β-Lapachone	Beta-Lapachone,NSC-26326,SL-11001,ARQ-501	IDO , Apoptosis , Topoisomerase , Autophagy
	β-Lapachone (ARQ-501) is a specific DNA topoisomerase I inhibitor, and no inhibitory activities against DNA topoisomerase II or ligase.		IDO , Apoptosis , Topoisomerase , Autophagy
T1537	Rapamycin	Sirolimus,AY 22989,NSC-2260804	Others , Endogenous Metabolite , Antibiotic , mTOR , Autophagy , Antifungal
	Rapamycin (AY 22989) is a natural product of macrolides, an mTOR inhibitor with specificity (HEK293 cells: IC50=0.1 nM). Rapamycin has immunosuppressive activity and induces autophagy.
TN7466	Isosecotanapartholide		Others
			Others
TN1929	Methyl sinapate		Others
	Methyl sinapate can increase the frequency of cells with chromosome aberrations in the CHO K-1 cells treated with MMC, 4NQO or UV.		Others
TN3318	9-Hydroxy-alpha-lapachone		Antifection
	9-Hydroxy-alpha-lapachone can highly inhibit the growth of H. pylori, it exhibits potent inhibitory activity against H. pylori Cystathionine gamma-synthase, with IC(50) values of 4.64 microM. It may have anti-inflammator...		Antifection
TN3019	4,9-Dihydroxy-alpha-lapachone		Others
	4,9-Dihydroxy-alpha-lapachone has antitumor-promoting effects, it exhibits significant inhibitory activity against 12-O-tetradecanoylphorbol 13-acetate (TPA)-induced Epstein-Barr virus early antigen (EBV-EA) activation i...		Others
TN3321	9-Methoxy-alpha-lapachone		Others
	9-Methoxy-alpha-lapachone has antitumor-promoting effect, it exhibits significant inhibitory activity against 12-O-tetradecanoylphorbol 13-acetate (TPA)-induced Epstein- Barr virus early antigen (EBV-EA) activation in Ra...		Others
T65249	Hydroxylapatite		Others
	Hydroxylapatite is a natural product for research related to life sciences and the catalog number is T65249.		Others
T25305	Demethoxyrapamycin	AY 24668,AY24668,AY-24668	Others
	Demethoxyrapamycin is a new antifungal antibiotic agent which is co-produced with rapamycin by Streptomyces hygroscopicus.		Others
T79984	Chaparrinone		Antiviral , Parasite
	Chaparrinone, a bittersweet analog from Ailanthus altissima (Mill.), has antimalarial, antitumor, and antiviral activities and has been used in the study of tobacco mosaic virus infections and SARS virus infections.		Antiviral , Parasite
TN5027	Sinapaldehyde glucoside		Others
	Sinapaldehyde glucoside is a natural product of Phellodendron, Rutaceae. The catalog number is TN5027 and the CAS number is 154461-65-1. Sinapaldehyde glucoside can be used as a reference standard.		Others
TN6365	3-Deoxy-11,13-dihydroisosecotanapartholide
	3-Deoxy-11,13-dihydroisosecotanapartholide is a natural product for research related to life sciences. The catalog number is TN6365 and the CAS number is 572924-43-7.
TN4269	Isocarapanaubine		Others
	Isocarapanaubine and reserpiline are cytotoxic constituents from the barks of Ochrosia elliptica.		Others

天然物製品

Deoxylapachol

TN1569

Synonym:

Target: Antifection, Antifungal

Rapanone

TN4893

Synonym: 2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione

Target: Apoptosis, Phospholipase, Antibacterial, Parasite

Papain

T19503

Synonym:

Target: Others, Cysteine Protease

Andrograpanin

T9218

Synonym: 19-HYDROXY-8(17),13-LABDADIEN-16,15-OLIDE

Target: p38 MAPK

Sinapaldehyde

TN2281

Synonym: trans-3,5-Dimethoxy-4-hydroxy cinnamaldehyde

Target: Antibacterial

Lapachol

T4136

Synonym: Bethabarra wood,CI75490,Greenhartin,Tecomin

Target: Others, Influenza Virus, Antibacterial, Parasite, Antifungal

Dihydrolapachenole

TN7058

Synonym: 6-methoxy-2,2-dimethyl-3,4-dihydro-2H-benzo[h]chromene

Target: Others

α-Lapachone

TN1375

Synonym: alpha-Lapachone

Target: Topoisomerase, Antifection

Tetrahydropapaverine hydrochloride

T6004

Synonym: Tetrahydropapaverine HCl,Norlaudanosine HCl,Tetrahydroalkali hydrochloride

Target: Hydroxylase

β-Lapachone

T6407

Synonym: Beta-Lapachone,NSC-26326,SL-11001,ARQ-501

Target: IDO, Apoptosis, Topoisomerase, Autophagy

Rapamycin

T1537

Synonym: Sirolimus,AY 22989,NSC-2260804

Target: Others, Endogenous Metabolite, Antibiotic, mTOR, Autophagy, Antifungal

Isosecotanapartholide

9-Hydroxy-alpha-lapachone

TN3318

Synonym:

Target: Antifection

4,9-Dihydroxy-alpha-lapachone

TN3019

Synonym:

Target: Others

9-Methoxy-alpha-lapachone

Synonym: AY 24668,AY24668,AY-24668

Target: Antiviral, Parasite

Sinapaldehyde glucoside

TN5027

Synonym:

Target: Others

3-Deoxy-11,13-dihydroisosecotanapartholide

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-00644	Aminopeptidase A Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	Aminopeptidase A Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 107.2 kDa and the accession number is Q07075.
TMPY-02896	Aminopeptidase A Protein, Mouse, Recombinant (His)	Mouse	Baculovirus Insect Cells
	Aminopeptidase A Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 106 kDa and the accession number is P16406.
TMPY-04894	SARS-CoV (strain WH20) Plpro/papain-like protease (His)	SARS	E. coli
	SARS-CoV (strain WH20) Plpro/papain-like protease (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 36.65 kDa and the accession number is AAX16193.1.
TMPY-01500	Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA1 Protein (His)	H5N1	HEK293 Cells
	Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is A0FFY3...
TMPH-03650	Turnip mosaic virus (TuMV) (strain Japanese) Genome polyprotein (His & Myc)	TuMV	E. coli
	N/A. Turnip mosaic virus (TuMV) (strain Japanese) Genome polyprotein (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 66.6 kDa and the accession number ...
TMPH-00573	DAPA aminotransferase Protein, E. coli, Recombinant (His & Myc)	E. coli	E. coli
	Catalyzes the transfer of the alpha-amino group from S-adenosyl-L-methionine (SAM) to 7-keto-8-aminopelargonic acid (KAPA) to form 7,8-diaminopelargonic acid (DAPA). It is the only animotransferase known to utilize SAM a...
TMPH-00808	HBV-D subtype ayw (isolate Japan/JYW796/1988) Protein X (His)	HBV-D	E. coli
	HBV-D subtype ayw (isolate Japan/JYW796/1988) Protein X (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 22.6 kDa and the accession number is Q9QMI3.
TMPY-01622	Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA Protein (His)	H5N1	HEK293 Cells
	Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60 kDa and the accession number is A0FFY3.
TMPY-06031	Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA1 Protein (His), Biotinylated	H5N1	HEK293 Cells
	Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA1 Protein (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession nu...
TMPJ-01431	SARS-CoV-2 Papain-Like Protease Protein	SARS-CoV-2	E. coli
	Replication of severe acute respiratory syndrome (SARS) coronavirus (SARS-CoV) requires proteolytic processing of the replicase polyprotein by two viral cysteine proteases, a chymotrypsin-like protease (3CLpro) and a pap...
TMPK-01384	SARS PLpro/papain-like protease Protein (His)	SARS	E. coli
	The coronaviral proteases, papain-like protease (PLpro) and 3C-like protease (3CLpro), are attractive antiviral drug targets because they are essential for coronaviral replication. Although the primary function of PLpro ...
TMPH-00347	Papain Protein, Carica papaya, Recombinant (His)	Carica papaya	E. coli
	Papain Protein, Carica papaya, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 27.4 kDa and the accession number is P00784.
TMPH-00714	SapA Protein, E. coli, Recombinant (His & Myc)	E. coli	E. coli
	Not part of a putrescine export system. Very similar to a S.typhimurium protein implicated in antimicrobial peptide resistance, but the SapBCDF operon in E.coli is implicated in putrescine export. SapA Protein, E. coli, ...
TMPY-06038	Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA Protein (His), Biotinylated	H5N1	HEK293 Cells
	Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA Protein (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60 kDa and the accession num...
TMPY-00254	Tapasin Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Tapasin Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 43.5 kDa and the accession number is AAH80574.1.
TMPY-00567	Influenza A H2N2 (A/Japan/305/1957) Hemagglutinin/HA1 Protein (His)	H2N2	HEK293 Cells
	Influenza A H2N2 (A/Japan/305/1957) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.5 kDa and the accession number is Q6XU87.
TMPY-05682	SARS-CoV-2 Plpro/papain-like protease Protein (aa 1564-1880, His)	SARS-CoV-2	E. coli
	SARS-CoV-2 Plpro/papain-like protease Protein (aa 1564-1880, His) is expressed in E. coli expression system. The predicted molecular weight is 36.79 kDa and the accession number is QVD65746.1.
TMPY-01135	Influenza A H2N2 (A/Japan/305/1957) Hemagglutinin/HA Protein (His)	H2N2	HEK293 Cells
	Influenza A H2N2 (A/Japan/305/1957) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is P03451.
TMPK-01352	SARS-CoV-2 PLpro/papain-like protease Protein (His & Avi)	SARS	E. coli
	The coronaviral proteases, papain-like protease (PLpro) and 3C-like protease (3CLpro), are attractive antiviral drug targets because they are essential for coronaviral replication. Although the primary function of PLpro ...
TMPH-02364	Japanese encephalitis virus Genome polyprotein (His & SUMO)	JEV	E. coli
	Japanese encephalitis virus Genome polyprotein (His & SUMO) is expressed in E. coli.
TMPH-02177	Tapasin Protein, Human, Recombinant (His & Myc)	Human	E. coli
	Involved in the association of MHC class I with transporter associated with antigen processing (TAP) and in the assembly of MHC class I with peptide (peptide loading). Tapasin Protein, Human, Recombinant (His & Myc) is e...

Aminopeptidase A Protein, Human, Recombinant (His)

TMPY-00644

Species: Human

Expression System: Baculovirus Insect Cells

Aminopeptidase A Protein, Mouse, Recombinant (His)

TMPY-02896

Species: Mouse

Expression System: Baculovirus Insect Cells

SARS-CoV (strain WH20) Plpro/papain-like protease (His)

TMPY-04894

Species: SARS

Expression System: E. coli

Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA1 Protein (His)

TMPY-01500

Species: H5N1

Expression System: HEK293 Cells

Turnip mosaic virus (TuMV) (strain Japanese) Genome polyprotein (His & Myc)

TMPH-03650

Species: TuMV

Expression System: E. coli

DAPA aminotransferase Protein, E. coli, Recombinant (His & Myc)

TMPH-00573

Species: E. coli

Expression System: E. coli

HBV-D subtype ayw (isolate Japan/JYW796/1988) Protein X (His)

TMPH-00808

Species: HBV-D

Expression System: E. coli

Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA Protein (His)

TMPY-01622

Species: H5N1

Expression System: HEK293 Cells

Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA1 Protein (His), Biotinylated

TMPY-06031

Species: H5N1

Expression System: HEK293 Cells

SARS-CoV-2 Papain-Like Protease Protein

TMPJ-01431

Species: SARS-CoV-2

Expression System: E. coli

SARS PLpro/papain-like protease Protein (His)

TMPK-01384

Species: SARS

Expression System: E. coli

Papain Protein, Carica papaya, Recombinant (His)

TMPH-00347

Species: Carica papaya

Expression System: E. coli

SapA Protein, E. coli, Recombinant (His & Myc)

TMPH-00714

Species: E. coli

Expression System: E. coli

Influenza A H5N1 (A/Japanese white-eye/Hong Kong/1038/2006) Hemagglutinin/HA Protein (His), Biotinylated

TMPY-06038

Species: H5N1

Expression System: HEK293 Cells

Tapasin Protein, Human, Recombinant (His)

TMPY-00254

Species: Human

Expression System: HEK293 Cells

Influenza A H2N2 (A/Japan/305/1957) Hemagglutinin/HA1 Protein (His)

TMPY-00567

Species: H2N2

Expression System: HEK293 Cells

SARS-CoV-2 Plpro/papain-like protease Protein (aa 1564-1880, His)

TMPY-05682

Species: SARS-CoV-2

Expression System: E. coli

Influenza A H2N2 (A/Japan/305/1957) Hemagglutinin/HA Protein (His)

TMPY-01135

Species: H2N2

Expression System: HEK293 Cells

SARS-CoV-2 PLpro/papain-like protease Protein (His & Avi)

TMPK-01352

Species: SARS

Expression System: E. coli

Japanese encephalitis virus Genome polyprotein (His & SUMO)

TMPH-02364

Species: JEV

Expression System: E. coli

Tapasin Protein, Human, Recombinant (His & Myc)

TMPH-02177

Species: Human

Expression System: E. coli

Isotope Products

カタログ番号	製品名	別名	ターゲット
TMIH-0093	Apalutamide-d4
	Apalutamide-d4 is a deuterated compound of Apalutamide.
T12243	Norverapamil-d7	D591 D7,(±)-Norverapamil D7	Others
	Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .		Others
TMIH-0547	S-Verapamil-d7 HCL
	S-Verapamil-d7 HCL is a deuterated compound of S-Verapamil HCL. S-Verapamil HCL has a CAS number of 1188265-55-5.
TMIH-0002	(+/-)-Verapamil hydrochloride-d7
	(+/-)-Verapamil hydrochloride-d7 is a deuterated compound of (+/-)-Verapamil hydrochloride. (+/-)-Verapamil hydrochloride has a CAS number of 152-11-4. Verapamil hydrochloride is a calcium channel blocker that is a class...
TMIH-0399	Norverapamil-d7 HCl
	Norverapamil-d7 HCl is a deuterated compound of Norverapamil HCl. Norverapamil HCl has a CAS number of 67812-42-4. Norverapamil hydrochloride ((±)-Norverapamil hydrochloride) is an N-demethylated metabolite of Verapamil ...
TMIH-0092	Apalutamide-13C-d3
	Apalutamide-13C-d3 is the 13C and deuterated compound of Apalutamide. Apalutamide has a CAS number of 956104-40-8. Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activ...
T12292	Olaparib-d5	KU0059436 D5,AZD2281 D5,Olaparib D5	Others
	Olaparib D5 is a deuterium labeled Olaparib. Olaparib is a potent and oral inhibitor of PARP.		Others
T10958	Dapagliflozin-d5	BMS-512148 D5	Others
	Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.		Others
TMIH-0294	Lapatinib-d4
	Lapatinib-d4 is a deuterated compound of Lapatinib. Lapatinib has a CAS number of 231277-92-2. Lapatinib is a dual inhibitor of Lapatinib is a dual ErbB2/EGFR (IC50: 9.2/10.8 nM) inhibitor
TMIH-0094	Apalutamide-d7
	Apalutamide-d7 is a deuterated compound of Apalutamide. Apalutamide has a CAS number of 956104-40-8. Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
T12691	Rapamycin-d3	AY-22989-d3,Sirolimus-d3	Others
	Rapamycin-d3 is the deuterium labeled Rapamycin. Rapamycin is a potent and specific inhibitor of mTOR(IC50 of 0.1 nM in HEK293 cells).		Others
TMIH-0508	R-Verapamil-d7 HCL
	R-Verapamil-d7 HCL is a deuterated compound of R-Verapamil HCL. R-Verapamil HCL has a CAS number of 1188265-55-5.
TMIH-0372	N-desmethyl Apalutamide-d4
	N-desmethyl Apalutamide-d4 is a deuterated compound of N-desmethyl Apalutamide. N-desmethyl Apalutamide has a CAS number of 1332391-11-3. N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is a...