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カタログ番号 製品名 別名 ターゲット
T81089 Steroid sulfatase-IN-7
Steroid sulfatase-IN-7 is an irreversible inhibitor of steroid sulfatase (STS), demonstrating potent activity with an IC50 of 0.05 nM against human placental STS, rendering it suitable for application in cancer research ...
T62237 Steroid sulfatase-IN-4
Steroid sulfatase-IN-4 (Compound 16) is an irreversible inhibitor of steroid sulfatase (STS) that acts on human STS (IC50: 25 nM). steroid sulfatase-IN-4 can be used to study endometriosis.
T61212 Steroid sulfatase-IN-2
Steroid sulfatase-IN-2 is an active inhibitor of steroid sulfatase (STS), demonstrating an IC50 value of 109.5 nM. Its potential application lies in hormone-dependent cancer research, specifically estrogen-dependent brea...
T61686 Steroid sulfatase-IN-3
Steroid sulfatase-IN-3 (compound 1q) is a highly effective Steroid sulfatase (STS) inhibitor, exhibiting an IC 50 value of 25.8 nM. This compound also demonstrates antiproliferative properties against T-47D estrogen-depe...
T81091 Steroid sulfatase-IN-5
Steroid sulfatase-IN-5 (compound 10b), an inhibitor of steroid sulfatase (STS) with an IC50 of 0.32 nM, effectively suppresses T-47D breast cancer cell proliferation, demonstrating an IC50 value of 35.7 μM. This compound...
T61687 Steroid sulfatase-IN-1
Steroid sulfatase-IN-1 is a highly potent and orally active inhibitor of the enzyme Steroid sulfatase, with an impressive IC50 value of 1.71 μM. This compound exhibits notable antitumor activity, achieving a TGI (tumor g...
T81090 Steroid sulfatase-IN-6
Steroid Sulfatase-IN-6 (Compound 10c) serves as an irreversible steroid sulfatase (STS) inhibitor, exhibiting a K i value of 0.4 nM against human placenta STS, and is applicable in tumor disease research [1].
T61979 Steroid sulfatase/17β-HSD1-IN-4
Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ). Steroid sulfatase/17β-HSD1-IN-4 irreversibly inhibits hSTS a...
T62236 Steroid sulfatase/17β-HSD1-IN-3
Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1). Steroid sulfatase/17β-HSD1-IN-3 can be used to study endometriosis and ...
T61716 Steroid sulfatase/17β-HSD1-IN-1
Steroid sulfatase/17β-HSD1-IN-1 is a highly effective inhibitor of both steroid sulfatase and 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) activities, displaying an IC50 value of 28 nM against cellular human steroi...
T81092 Steroid sulfatase/17β-HSD1-IN-5
Steroid sulfatase/17β-HSD1-IN-5 serves as an irreversible inhibitor of steroid sulfatase (STS) and a reversible, selective inhibitor of 7β-hydroxysteroid dehydrogenase type1 (17β-HSD1), exhibiting IC50 values of 43 nM fo...
T83752 Biotin-SRC-1 (676–700) TFA Biotin-Steroid Receptor Coactivator 1 (676-700)
Biotin-SRC-1 (676–700), a biotinylated and truncated variant of steroid receptor coactivator 1 (SRC-1), finds application in affinity-based reporter assays such as time-resolved FRET (TR-FRET) and amplified luminescent p...
T0181 Loteprednol etabonate Lotemax,Alrex Glucocorticoid Receptor , Antibacterial , Antibiotic
Loteprednol etabonate (Lotemax) is an ophthalmic analog of the corticosteroid prednisolone with anti-inflammatory activity.
T0166 Pancuronium dibromide Pancuronium bromide,Pavulon AChR
Pancuronium dibromide (Pavulon), a competitive AChR antagonist (IC50 = 5.5 nM), acts as a skeletal muscle relaxant. Pancuronium dibromide(Pancuronium bromide) blocking neuromuscular transmission is achieved by competing ...
T1531 Mometasone furoate Sch32088 Glucocorticoid Receptor
Mometasone furoate (Sch32088) is a pregnadienediol derivative ANTI-ALLERGIC AGENT and ANTI-INFLAMMATORY AGENT that is used in the management of ASTHMA and ALLERGIC RHINITIS. It is also used as a topical treatment for ski...
T1167 Cyproterone acetate Androcur,Cyproterone 17-O-acetate Androgen Receptor
Cyproterone acetate (Cyproterone 17-O-acetate) binds the androgen receptor (AR), thereby preventing androgen-induced receptor activation in target tissues and inhibiting the growth of testosterone-sensitive tumor cells. ...
T61444 Nonsteroidal aromatase inhibitor 1
Nonsteroidal aromatase inhibitor 1 (Compound 13h) effectively inhibits the enzyme CYP19A1 with an IC50 value of 0.09 nM. Due to its potent inhibitory activity, Nonsteroidal aromatase inhibitor 1 holds promise for researc...
T76147 3α-Hydroxysteroid dehydrogenase
3α-Hydroxysteroid dehydrogenase (3α-HSD), encoded by the AKR1C4 gene, is responsible for catalyzing the transformation of 3-ketosteroids into 3α-hydroxy compounds. This enzyme significantly contributes to the inactivatio...
T4464 Irosustat 667-Coumate,BN83495,STX64 Others
Irosustat (667-Coumate) is a potent steroid sulfatase inhibitor, with an IC50 of 8 nM, and exhibits anti-breast cancer activity.
T33414 MK 0434 MK0434,MK434,MK 434,MK-0434,MK-434
MK 0434 is a steroid 5α-reductase inhibitor and hormone antagonist associated with a significant reduction in DHT.
T0870 Altrenogest R2267,RU2267,Allyltrenbolone,A35957 Estrogen/progestogen Receptor , Progesterone Receptor
Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone.
T0293 Metyrapone NSC-25265,Su-4885 Others , P450 , Dehydrogenase , Autophagy
Metyrapone (NSC-25265) is an inhibitor of the enzyme STEROID 11-BETA-MONOOXYGENASE. It is used as a test of the feedback hypothalamic-pituitary mechanism in the diagnosis of CUSHING SYNDROME.
T19213 Boldenone Cypionate Others , Androgen Receptor
Boldenone Cypionate is an androgenic anabolic steroid.
T83615 S5A1 Others
S5A1 is a synthetic steroid used in the study of diabetes.
T6502 Fluocinonide Lidex,Metosyn,Topsyn Glucocorticoid Receptor
Fluocinonide (Topsyn) (Vanos) is an effective glucocorticoid steroid, utilized in the treatment as the skin disorders anti-inflammatory agent.
T2559 Allylestrenol Gestanon,Gestanol,Gestanin Estrogen/progestogen Receptor
Allylestrenol (Gestanin) is a synthetic steroid with progestational activity.
T60929 Brassinazole (2S,3R)-Brassinazole Others
Brassinazole is a selective inhibitor of triazole-type steroid (BR) biosynthesis.Brassinazole can be used to modulate the oleuropein steroid (BR) signaling pathway, which is used to regulate plant xylem growth and develo...
T3137 Boldenone Undecylenate Parenabol,Ba 29038,Vebonol Androgen Receptor , Endogenous Metabolite
Boldenone Undecylenate (Parenabol) is a synthetic steroid.
T21452 Anecortave Acetate Retaane,Al 3789,NSC 24345,NSC 15475,Anecortave Others
Anecortave Acetate (NSC-24345), an angiostatic steroid, is used for proteomics research.
T5326 Sugammadex sodium Org25969,Sugammadex (sodium) Others
Sugammadex sodium (Org25969) , a synthetic derivative of γ-cyclodextrin, is a steroid-based neuromuscular blocker reversing agent.
T27478 GSK3987 Liver X Receptor
GSK3987 is an LXR ligand. GSK3987 recruits the steroid receptor coactivator-1 to human LXRalpha and LXRbeta with EC50s of 40 nM.
T15000 Cort108297 Glucocorticoid Receptor
Cort108297 is a selective glucocorticoid receptor modulator and a selective GR antagonist with no affinity for other steroid receptors. Cort108297 showed a high affinity for GRs (Ki: 0.45nM).
T2199 Myclobutanil Systhane Antifungal
Myclobutanil (Systhane) is a triazole chemical used as a fungicide. It is a steroid demethylation inhibitor, specifically inhibiting ergosterol biosynthesis. Ergosterol is a critical component of fungal cell membranes.
T1594 Vecuronium bromide ORG NC 45 AChR
Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking agent, with muscle relaxant activity.
T0384 Estradiol benzoate Benzoestrofol,Benzhormovarine,Benovocylin Estrogen Receptor/ERR , Estrogen/progestogen Receptor
Estradiol benzoate (Benzhormovarine) is the synthetic benzoate ester of estradiol, a steroid sex hormone vital to the maintenance of fertility and secondary sexual characteristics in females.
T23549 YM 511 P450 , Aromatase
YM 511 is a highly specific non-steroidal aromatase inhibitor. YM 511 inhibits aromatase activities in microsomes from rat ovary and human placenta competitively (IC50s of 0.4 and 0.12 nM, respectively). YM 511 slightly ...
T13684 Equilin 7-Dehydroestrone Calcium Channel
Equilin (7-Dehydroestrone) is a neurotrophic estrogenic steroid with vasodilatory activity that increases monocyte-endothelial adhesion through NF-κB signalling.Equilin similarly relaxes mesenteric arterial resistance by...
T6503 Fluorometholone Acetate NSC 47438,Flarex,Eflone,Oxylone acetate Glucocorticoid Receptor , Carbonic Anhydrase
Fluorometholone Acetate (Oxylone acetate) is a synthetic corticosteroid, used in the treatment of steroid responsive inflammatory conditions of the eye.
T6215 Abiraterone Acetate Zytiga,CB7630 P450
Abiraterone Acetate (CB7630) is an androstene derivative that inhibits STEROID 17-ALPHA-HYDROXYLASE and is used as an ANTINEOPLASTIC AGENT in the treatment of metastatic castration-resistant PROSTATE CANCER.
T6465 Dexamethasone Sodium Phosphate Dexadreson,Dexagro,Dalalone IL Receptor , COX
Dexamethasone Sodium Phosphate (Dexadreson) , an interleukin receptor modulator, has anti-inflammatory and immunosuppressant effects. It belongs to a potent glucocorticoid class of steroid synthetic drugs.
T67901 SRD5A1-IN-1 Others
SRD5A1-IN-1 is an inhibitor of steroid 5α-reductase type 1 (SRD5A1, IC50 = 1.44 µM). SRD5A1-IN-1 lowers the production of dihydrotestosterone and shows a significant decrease in the SRD5A1 protein expression.
T3316 Fluorometholone Fluoromethalone,Cortilet,Oxylone,Delmeson Glucocorticoid Receptor
Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery. It is marketed under the brand names FML (Allergan) and Flarex (Alcon). Fluorometholone acetate ophthalmic susp...
T6886 MCB-613 MCB 613 Src
MCB-613 is an effective steroid receptor coactivator (SRC) stimulator.
T1438 Butoconazole nitrate RS 35887 Estrogen/progestogen Receptor , Antifungal
Butoconazole Nitrate is the nitrate salt form of butoconazole, a synthetic imidazole derivative with fungistatic properties. Butoconazole nitrate (RS 35887) interferes with steroid biosynthesis by inhibiting the conversi...
T0947 Dexamethasone acetate Dexamethasone 21-acetate,Dexamethason acetate,NSC 39471 Glucocorticoid Receptor , Mitophagy , IL Receptor , Annexin A , NOS , Antibacterial , Autophagy
Dexamethasone acetate (NSC 39471) is the acetate salt form of Dexamethasone, a synthetic adrenal corticosteroid with potent anti-inflammatory properties. In addition to binding to specific nuclear steroid receptors, dexa...
T60924 Verosudil AR-12286 ROCK
Verosudil (AR-12286) is a highly potent Rho kinase (ROCK) inhibitor with a Ki of 2 and 2 nM against ROCK1 and ROCK2, respectively. AR-12286 reverses steroid-induced intraocular pressure in mice by decreasing intraocular ...
T2556 Nandrolone decanoate 19-Nortestosterone decanoate Others , HIV Protease
Nandrolone decanoate (19-Nortestosterone decanoate) is the decanoate salt form of nandrolone, an anabolic steroid analog of testosterone with androgenic, anabolic, and erythropoietin stimulating effects. Nandrolone enter...
T28773 SI-2 SI2,EPH 116,EPH116,EPH-116 Others
SI-2 is an inhibitor (SMI) of steroid receptor coactivator-3 (SRC-3 or AIB1). SI-2 can selectively reduce the transcriptional activities and the protein concentrations of SRC-3 in cells, and selectively induce breast can...
T72470 Estrone O-sulfamate Estrone 3-O-sulfamate Others
Estrone O-sulfamate (Estrone 3-O-sulfamate) is a potent inhibitor of steroid sulfatase (STS). Estrone O-sulfamate is a placental microsomal inhibitor (P.M.) with IC50 values of 18 nM. Estrone O-sulfamate showed inhibitor...
T9836 (E)-SI-2 Others
(E)-SI-2 is a potent small-molecule inhibitor of steroid receptor coactivator-3 (SRC-3 or AIB1) that can selectively inhibit the intrinsic transcriptional activities of SRC-3, also inhibits SRC-1 and SRC-2. It selectivel...

Compounds

Steroid sulfatase-IN-7
T81089
Synonym:
Target:
Steroid sulfatase-IN-4
T62237
Synonym:
Target:
Steroid sulfatase-IN-2
T61212
Synonym:
Target:
Steroid sulfatase-IN-3
T61686
Synonym:
Target:
Steroid sulfatase-IN-5
T81091
Synonym:
Target:
Steroid sulfatase-IN-1
T61687
Synonym:
Target:
Steroid sulfatase-IN-6
T81090
Synonym:
Target:
Steroid sulfatase/17β-HSD1-IN-4
T61979
Synonym:
Target:
Steroid sulfatase/17β-HSD1-IN-3
T62236
Synonym:
Target:
Steroid sulfatase/17β-HSD1-IN-1
T61716
Synonym:
Target:
Steroid sulfatase/17β-HSD1-IN-5
T81092
Synonym:
Target:
Biotin-SRC-1 (676–700) TFA
T83752
Synonym: Biotin-Steroid Receptor Coactivator 1 (676-700)
Target:
Loteprednol etabonate
T0181
Synonym: Lotemax,Alrex
Target: Glucocorticoid Receptor, Antibacterial, Antibiotic
Pancuronium dibromide
T0166
Synonym: Pancuronium bromide,Pavulon
Target: AChR
Mometasone furoate
T1531
Synonym: Sch32088
Target: Glucocorticoid Receptor
Cyproterone acetate
T1167
Synonym: Androcur,Cyproterone 17-O-acetate
Target: Androgen Receptor
Nonsteroidal aromatase inhibitor 1
T61444
Synonym:
Target:
3α-Hydroxysteroid dehydrogenase
T76147
Synonym:
Target:
Irosustat
T4464
Synonym: 667-Coumate,BN83495,STX64
Target: Others
MK 0434
T33414
Synonym: MK0434,MK434,MK 434,MK-0434,MK-434
Target:
Altrenogest
T0870
Synonym: R2267,RU2267,Allyltrenbolone,A35957
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Metyrapone
T0293
Synonym: NSC-25265,Su-4885
Target: Others, P450, Dehydrogenase, Autophagy
Boldenone Cypionate
T19213
Synonym:
Target: Others, Androgen Receptor
S5A1
T83615
Synonym:
Target: Others
Fluocinonide
T6502
Synonym: Lidex,Metosyn,Topsyn
Target: Glucocorticoid Receptor
Allylestrenol
T2559
Synonym: Gestanon,Gestanol,Gestanin
Target: Estrogen/progestogen Receptor
Brassinazole
T60929
Synonym: (2S,3R)-Brassinazole
Target: Others
Boldenone Undecylenate
T3137
Synonym: Parenabol,Ba 29038,Vebonol
Target: Androgen Receptor, Endogenous Metabolite
Anecortave Acetate
T21452
Synonym: Retaane,Al 3789,NSC 24345,NSC 15475,Anecortave
Target: Others
Sugammadex sodium
T5326
Synonym: Org25969,Sugammadex (sodium)
Target: Others
GSK3987
T27478
Synonym:
Target: Liver X Receptor
Cort108297
T15000
Synonym:
Target: Glucocorticoid Receptor
Myclobutanil
T2199
Synonym: Systhane
Target: Antifungal
Vecuronium bromide
T1594
Synonym: ORG NC 45
Target: AChR
Estradiol benzoate
T0384
Synonym: Benzoestrofol,Benzhormovarine,Benovocylin
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
YM 511
T23549
Synonym:
Target: P450, Aromatase
Equilin
T13684
Synonym: 7-Dehydroestrone
Target: Calcium Channel
Fluorometholone Acetate
T6503
Synonym: NSC 47438,Flarex,Eflone,Oxylone acetate
Target: Glucocorticoid Receptor, Carbonic Anhydrase
Abiraterone Acetate
T6215
Synonym: Zytiga,CB7630
Target: P450
Dexamethasone Sodium Phosphate
T6465
Synonym: Dexadreson,Dexagro,Dalalone
Target: IL Receptor, COX
SRD5A1-IN-1
T67901
Synonym:
Target: Others
Fluorometholone
T3316
Synonym: Fluoromethalone,Cortilet,Oxylone,Delmeson
Target: Glucocorticoid Receptor
MCB-613
T6886
Synonym: MCB 613
Target: Src
Butoconazole nitrate
T1438
Synonym: RS 35887
Target: Estrogen/progestogen Receptor, Antifungal
Dexamethasone acetate
T0947
Synonym: Dexamethasone 21-acetate,Dexamethason acetate,NSC 39471
Target: Glucocorticoid Receptor, Mitophagy, IL Receptor, Annexin A, NOS, Antibacterial, Autophagy
Verosudil
T60924
Synonym: AR-12286
Target: ROCK
Nandrolone decanoate
T2556
Synonym: 19-Nortestosterone decanoate
Target: Others, HIV Protease
SI-2
T28773
Synonym: SI2,EPH 116,EPH116,EPH-116
Target: Others
Estrone O-sulfamate
T72470
Synonym: Estrone 3-O-sulfamate
Target: Others
(E)-SI-2
T9836
Synonym:
Target: Others
1 2 3
カタログ番号 製品名 別名 ターゲット
TN3270 (R)-3β-Hydroxy steroid sulfotransferase-IN-11 Others
(R)-3β-Hydroxy steroid sulfotransferase-IN-11 has a wide range of applications in life science related research.
T5S1982 Periplocin Periplocoside Apoptosis , Others
1. Periplocin (Periplocoside) has anti-cancer effects on lung cancer cells, induces apoptosis and inhibits growth of cancer cells by the beta-catenin/Tcf signaling pathway. 2. Periplocin is used for treatment of rheumato...
T19470 Nandrolone propionate Others , Androgen Receptor
Nandrolone propionate is an anabolic steroid action primarily consisting of androgenic and nitrogen-retentive properties.
T8709 Nandrolone phenylpropionate Nandrolone phenpropionate Androgen Receptor
Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis
T8117 Metenolone acetate Methenolone acetate Others , Androgen Receptor
Metenolone acetate (Methenolone acetate) is an androgen and anabolic steroid (AAS) medication which is used mainly in the treatment of anemia due to bone marrow failure.
TMA0984 Cerevisterol DNA/RNA Synthesis
Cerevisterol is a cytotoxic steroid, can inhibit the activity of DNA polymerase alpha. It can stimulate NGF-mediated neurite outgrowth on PC12 cells.
T2207 Adrenosterone 11-ketoandrostenedione,11-oxoandrostenedione,Reichstein's substance G Androgen Receptor , Endogenous Metabolite
Adrenosterone (11-ketoandrostenedione) is a steroid hormone isolated from the adrenal cortex.
T14001 11-Beta-hydroxyandrostenedione NSC-17102,4-Androsten-11β-ol-3,17-dione Endogenous Metabolite
11-Beta-hydroxyandrostenedione (NSC-17102) is a steroid mainly found in the adrenal origin (11β-hydroxylase is present in adrenal tissue, but absent in ovarian tissue), which is a 11β-hydroxysteroid dehydrogenase isozyme...
TN3910 Ecdysone Apoptosis , ATPase , Glucocorticoid Receptor , Potassium Channel , Sodium Channel , Endogenous Metabolite , Autophagy
Ecdysone is a major steroid hormone in insects and herbs. Ecdysone triggers mineralocorticoid receptor activation and induces cellular apoptosis. Ecdysone signaling through Ecdysone receptor isoform B1 is required cell a...
T1048 Estradiol E2,17β-Estradiol,17β-Oestradiol,β-Estradiol Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
Estradiol (E2) is a naturally occurring steroidal sex hormone that is essential for female fertility and maintenance of secondary sexual characteristics. Estradiol upregulates IL-6 expression through estrogen receptor be...
T36857 Estrone sulfate sodium Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate Endogenous Metabolite
Estrone sulfate sodium (17β-Estrone 3-sulfate) is an endogenous steroid and an estrogen ester that is biologically inactive. It is converted by steroid sulfatase into estrone . Estrone sulfate sodium has been investigate...
T3220 Euphorbiasteroid Euphobiasteroid,Euphorbia factor L1 Others , AMPK
Euphorbiasteroid (Euphobiasteroid) (25-50 μM) decreased differentiation of 3T3-L1 cells via reduction of intracellular triglyceride (TG) accumulation.
T8043 5α-Cholestane Endogenous Metabolite
5α-Cholestane belongs to the cholestane steroid class of compounds.
T13500 3-O-Acetyl-20-Hydroxyecdysone Others
3-O-Acetyl-20-Hydroxyecdysone, a steroid extracted from the roots of Cyanotis arachnoidea C.B.Clark, is characterized by its unique structural modifications.
TN7130 Chlorogenin Others
Chlorogenin is a natural steroid derived from the herbs of Agave americana.
T7024 Qingyangshengenin Qingyangshengenin A,Cynanchagenin Others
Qingyangshengenin (Cynanchagenin) is a steroid used in the preparation of antiepileptic agents.
TN1075 Adynerin Others
Adynerin is a steroid found in the herbs of Nerium oleander.
T10048 17a-Hydroxypregnenolone Endogenous Metabolite
17a-Hydroxypregnenolone is a pregnane steroid. It is a prohormone in the formation of dehydroepiandrosterone (DHEA).
T20302 Deoxycorticosterone Desoxycorticosterone,Desoxycorticosteronum,Desoxycortone Endogenous Metabolite
Deoxycorticosterone (Desoxycortone) is a steroid metabolite produced by the adrenal gland. Deoxycorticosterone is an aldosterone precursor and possesses mineralocorticoid activity.
T73772 Estrone sulfate potassium Endogenous Metabolite
Estrone sulfate potassium is an estrogen ester and conjugate, a natural endogenous steroid.
T2912 Ergosterol Provitamin D,Ergosterin,Provitamin D2 Others , Endogenous Metabolite
Ergosterol (Provitamin D2) is a steroid extracted from Ganoderma lucidum cystocarp.
TC0026 Testosterone benzoate Others
Testosterone benzoate is a synthetic, injected anabolic androgenic steroid (AAS) and an androgen ester specifically
T3130 Testosterone phenylpropionate Testosterone hydrocinnamate,Retandrol,Testosterone 17-phenylpropionate Others
Testosterone phenylpropionate (Testosterone 17-phenylpropionate)is a steroid indicated for testosterone replacement therapy in sterilization, missing testicle, hypopituitarism, and osteoporosis.
T2748 Cortodoxone 11-Deoxycortisol,cortexolone,17α,21-dihydroxyprogesterone,Reichstein's substance S,11-Desoxycortisol Glucocorticoid Receptor , Endogenous Metabolite
Cortodoxone (11-Desoxycortisol) is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.
T3S0895 Spirostan-3-ol Sarsaponin Others
Spirostan-3-ol (Sarsaponin) is a stereoisomer of Sarsasapogenin (S142505), a steroid glycoside isolated from plant materials. A saponin with with potential anti-tumor activity via apoptosis.
T0856 Dehydroisoandrosterone 3-acetate Dehydroepiandrosterone 3-acetate,Dehydroepiandrosterone acetate,Prasterone acetate,DHEA acetate,androstenolone acetate Androgen Receptor
Dehydroisoandrosterone 3-acetate (Prasterone acetate) is a primary C19 steroid generated by the adrenal cortex.
T12536 Pregnenolone monosulfate 3β-Hydroxy-5-pregnen-20-one monosulfate NMDAR
Pregnenolone monosulfate (3β-Hydroxy-5-pregnen-20-one monosulfate) is a potent nootropic steroid that positively regulates NMDA recordings, and can be used in studies of neuroticism and depression.
TC0019 Pregnenolone acetate 3β-Hydroxy-5-pregnen-20-one acetate Cannabinoid Receptor , Endogenous Metabolite
Pregnenolone acetate is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. It acts as a signaling-specific inhibitor of cannabinoid CB1 receptor, inhibits the effects of te...
T2822 Ginsenoside Rb1 Gypenoside Ⅲ,Gypenoside III ATPase , Mitophagy , IRAK , NF-κB , Autophagy , HSV
Ginsenoside Rb1 (Gypenoside Ⅲ) is part of a class of steroid glycosides; may have properties that inhibit or prevent the growth of tumors.
T6S1842 Tenacissoside G Tenacissimoside A Others
Tenacissoside G, a C21 steroid derived from the stems of Marsdenia tenacissima, can reverse multidrug resistance in cancer cells exhibiting overexpression of P-glycoprotein.
T3033 Deoxycorticosterone acetate DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate Glucocorticoid Receptor , Endogenous Metabolite , Adrenergic Receptor
Deoxycorticosterone acetate (Cortexone acetate) is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection for replacement therapy of the adrenocortical steroid.
T4878 Hecogenin Hocogenin Others , Antifungal
Hecogenin (Hocogenin), a steroid saponin derived from Agave sisalana, serves as a specific inhibitor for human UDP-glucuronosyltransferases. Notably, it exhibits a broad range of pharmacological activities, such as anti-...
T0851 Pregnenolone 3β-Hydroxy-5-pregnen-20-one,Arthenolone Cannabinoid Receptor , Endogenous Metabolite , TRP/TRPV Channel , AChR , Autophagy
Pregnenolone (Arthenolone) is an endogenous steroid hormone synthesized from cholesterol, used in the treatment of Alzheimer's disease.
T0478 Progesterone Pregn-4-ene-3,20-dione Estrogen/progestogen Receptor , Progesterone Receptor , Opioid Receptor , Endogenous Metabolite
Progesterone (Pregn-4-ene-3,20-dione) is the major progestational steroid that is secreted primarily by the CORPUS LUTEUM and the PLACENTA. Progesterone acts on the UTERUS, the MAMMARY GLANDS and the BRAIN. It is require...
T9171 Methenolone enanthate Others
Methenolone enanthate is an androgen and anabolic steroid (AAS) medication which is used mainly in the treatment of anemia due to bone marrow failure.
T5751 Tigogenin Others
Tigogenin is one of steroidal sapogenins which is widely used for synthesizing steroid drugs. It might have protective effect on bone and be helpful in preventing the development of osteoporosis.
TN7099 Antcin A NOD
antcin A is a steroid-like phytochemical isolated from the fruiting bodies of a precious edible mushroom Antrodia cinnamomea with strong anti-inflammatory and anti-tumor effects.
T19124 3-​Oxocholic acid 3-Ketocholic acid Endogenous Metabolite
3-Oxocholic acid(3-Ketocholic acid) is the metabolite of bile acid and the main product of bile degradation by Clostridium perfringens in the intestine.3-Oxocholic acid is a steroid acid mainly found in the bile of mamma...
T2733 Sarsasapogenin Parigenin,Sarsagenin Apoptosis , NF-κB , Endogenous Metabolite
Sarsasapogenin (Parigenin) is a steroidal sapogenin, that is the aglycosidic portion of a plant saponin. It is named after sarsaparilla (Smilax sp.), a family of climbing plants found in subtropical regions. It was one o...
T7990 9-hydroxy-4-androstene-3,17-dione Others
9-hydroxy-4-androstene-3,17-dione is a steroid hormone. It has anti-tumor activity and can inhibit the growth of many types of cancer cells, including breast, prostate and lung cancer cells.
T2881 Crustecdysone Commisterone,B-ecdysone,Commisterone,20-Hydroxyecdysone,Ecdysterone,B-ecdysone,Hydroxyecdysone Others , Caspase , Endogenous Metabolite , Autophagy
Crustecdysone (Hydroxyecdysone) is a steroid hormone that regulates the processes of molting or ecdysis in insects.
T8040 Cholesterol myristate Cholesteryl myristate,Cholesteryl tetradecanoate Others , Potassium Channel , GABA Receptor , Endogenous Metabolite , AChR
Cholesterol Myristate (Cholesteryl Myristate) is a natural steroid found in traditional Chinese medicine that interacts with various ion channels, including the GABAA receptor, nicotinic acetylcholine receptor, and the i...
T3674 Hydroxysafflor yellow A HSYA,Safflomin A TGF-beta/Smad
Hydroxysafflor yellow A (Safflomin A) inhibited adipogenesis by increasing HSL promoter activities. Hydroxysafflor yellow A can effectively protect the liver from long-term alcohol injury by enhancing antioxidant capacit...
T1009 Estrone Oestrone,Fluoroethyl,Aquacrine Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
Estrone (Aquacrine) is an aromatized C18 steroid with a 3-hydroxyl group and a 17-ketone, a major mammalian estrogen. It is converted from ANDROSTENEDIONE directly, or from TESTOSTERONE via ESTRADIOL. In humans, it is pr...
T6654 Saponins Sapogenins Glycosides,Saponin Others
Saponins (Sapogenins Glycosides) are a mixture of triterpene and steroid saponins isolated from medicinal plants such as Aesculus hippocastanum L., Hedera helix L. and Ruscus aculeatus L., which are claimed to be effecti...
T0948L Corticosterone 17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,Corticosterone (From plants) Glucocorticoid Receptor , Endogenous Metabolite
Corticosterone (Kendall's compound B) is an adrenocortical steroid with salocorticoid and glucocorticoid activity that is orally active. Corticosterone is involved in the regulation of energy, immune responses, and stres...
T2777 Ginsenoside Rg1 Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,Panaxoside A,Ginsenoside A2 Apoptosis , Beta Amyloid , NF-κB
Ginsenoside Rg1 (Panaxoside Rg1) is a class of steroid glycosides, and triterpene saponins found exclusively in the plant genus Panax (ginseng). It improves spatial learning and increase hippocampal synaptophysin level i...
T1429 17α-Hydroxyprogesterone Hydroxyprogesterone,17-OHP,17-Hydroxyprogesterone Estrogen/progestogen Receptor , Progesterone Receptor , Endogenous Metabolite
17α-Hydroxyprogesterone (17-OHP) is a physiological progestin that is produced during glucocorticoid and steroid hormone synthesis and is increased during the third trimester of pregnancy. Hydroxyprogesterone binds to th...
T5574 Guggulsterone Guggulsterone E&Z Apoptosis , FXR , Akt , Caspase , JNK , Autophagy
Guggulsterone (Guggulsterone E&Z) E&Z is a 3-hydroxy steroid. It has a role as an androgen.
T4717 25-Hydroxycholesterol Others , Endogenous Metabolite , HMG-CoA Reductase
25-Hydroxycholesterol is a steroid derivative that suppresses the cleavage of sterol regulatory element binding proteins (SREBPs). It inhibits HMG-CoA reductase and so it also plays a significant role in the in vivo regu...
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天然物製品

(R)-3β-Hydroxy steroid sulfotransferase-IN-11
TN3270
Synonym:
Target: Others
Periplocin
T5S1982
Synonym: Periplocoside
Target: Apoptosis, Others
Nandrolone propionate
T19470
Synonym:
Target: Others, Androgen Receptor
Nandrolone phenylpropionate
T8709
Synonym: Nandrolone phenpropionate
Target: Androgen Receptor
Metenolone acetate
T8117
Synonym: Methenolone acetate
Target: Others, Androgen Receptor
Cerevisterol
TMA0984
Synonym:
Target: DNA/RNA Synthesis
Adrenosterone
T2207
Synonym: 11-ketoandrostenedione,11-oxoandrostenedione,Reichstein's substance G
Target: Androgen Receptor, Endogenous Metabolite
11-Beta-hydroxyandrostenedione
T14001
Synonym: NSC-17102,4-Androsten-11β-ol-3,17-dione
Target: Endogenous Metabolite
Ecdysone
TN3910
Synonym:
Target: Apoptosis, ATPase, Glucocorticoid Receptor, Potassium Channel, Sodium Channel, Endogenous Metabolite, Autophagy
Estradiol
T1048
Synonym: E2,17β-Estradiol,17β-Oestradiol,β-Estradiol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Estrone sulfate sodium
T36857
Synonym: Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate
Target: Endogenous Metabolite
Euphorbiasteroid
T3220
Synonym: Euphobiasteroid,Euphorbia factor L1
Target: Others, AMPK
5α-Cholestane
T8043
Synonym:
Target: Endogenous Metabolite
3-O-Acetyl-20-Hydroxyecdysone
T13500
Synonym:
Target: Others
Chlorogenin
TN7130
Synonym:
Target: Others
Qingyangshengenin
T7024
Synonym: Qingyangshengenin A,Cynanchagenin
Target: Others
Adynerin
TN1075
Synonym:
Target: Others
17a-Hydroxypregnenolone
T10048
Synonym:
Target: Endogenous Metabolite
Deoxycorticosterone
T20302
Synonym: Desoxycorticosterone,Desoxycorticosteronum,Desoxycortone
Target: Endogenous Metabolite
Estrone sulfate potassium
T73772
Synonym:
Target: Endogenous Metabolite
Ergosterol
T2912
Synonym: Provitamin D,Ergosterin,Provitamin D2
Target: Others, Endogenous Metabolite
Testosterone benzoate
TC0026
Synonym:
Target: Others
Testosterone phenylpropionate
T3130
Synonym: Testosterone hydrocinnamate,Retandrol,Testosterone 17-phenylpropionate
Target: Others
Cortodoxone
T2748
Synonym: 11-Deoxycortisol,cortexolone,17α,21-dihydroxyprogesterone,Reichstein's substance S,11-Desoxycortisol
Target: Glucocorticoid Receptor, Endogenous Metabolite
Spirostan-3-ol
T3S0895
Synonym: Sarsaponin
Target: Others
Dehydroisoandrosterone 3-acetate
T0856
Synonym: Dehydroepiandrosterone 3-acetate,Dehydroepiandrosterone acetate,Prasterone acetate,DHEA acetate,androstenolone acetate
Target: Androgen Receptor
Pregnenolone monosulfate
T12536
Synonym: 3β-Hydroxy-5-pregnen-20-one monosulfate
Target: NMDAR
Pregnenolone acetate
TC0019
Synonym: 3β-Hydroxy-5-pregnen-20-one acetate
Target: Cannabinoid Receptor, Endogenous Metabolite
Ginsenoside Rb1
T2822
Synonym: Gypenoside Ⅲ,Gypenoside III
Target: ATPase, Mitophagy, IRAK, NF-κB, Autophagy, HSV
Tenacissoside G
T6S1842
Synonym: Tenacissimoside A
Target: Others
Deoxycorticosterone acetate
T3033
Synonym: DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate
Target: Glucocorticoid Receptor, Endogenous Metabolite, Adrenergic Receptor
Hecogenin
T4878
Synonym: Hocogenin
Target: Others, Antifungal
Pregnenolone
T0851
Synonym: 3β-Hydroxy-5-pregnen-20-one,Arthenolone
Target: Cannabinoid Receptor, Endogenous Metabolite, TRP/TRPV Channel, AChR, Autophagy
Progesterone
T0478
Synonym: Pregn-4-ene-3,20-dione
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Opioid Receptor, Endogenous Metabolite
Methenolone enanthate
T9171
Synonym:
Target: Others
Tigogenin
T5751
Synonym:
Target: Others
antcin A
TN7099
Synonym:
Target: NOD
3-​Oxocholic acid
T19124
Synonym: 3-Ketocholic acid
Target: Endogenous Metabolite
Sarsasapogenin
T2733
Synonym: Parigenin,Sarsagenin
Target: Apoptosis, NF-κB, Endogenous Metabolite
9-hydroxy-4-androstene-3,17-dione
T7990
Synonym:
Target: Others
Crustecdysone
T2881
Synonym: Commisterone,B-ecdysone,Commisterone,20-Hydroxyecdysone,Ecdysterone,B-ecdysone,Hydroxyecdysone
Target: Others, Caspase, Endogenous Metabolite, Autophagy
Cholesterol myristate
T8040
Synonym: Cholesteryl myristate,Cholesteryl tetradecanoate
Target: Others, Potassium Channel, GABA Receptor, Endogenous Metabolite, AChR
Hydroxysafflor yellow A
T3674
Synonym: HSYA,Safflomin A
Target: TGF-beta/Smad
Estrone
T1009
Synonym: Oestrone,Fluoroethyl,Aquacrine
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Saponins
T6654
Synonym: Sapogenins Glycosides,Saponin
Target: Others
Corticosterone
T0948L
Synonym: 17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,Corticosterone (From plants)
Target: Glucocorticoid Receptor, Endogenous Metabolite
Ginsenoside Rg1
T2777
Synonym: Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,Panaxoside A,Ginsenoside A2
Target: Apoptosis, Beta Amyloid, NF-κB
17α-Hydroxyprogesterone
T1429
Synonym: Hydroxyprogesterone,17-OHP,17-Hydroxyprogesterone
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Endogenous Metabolite
Guggulsterone
T5574
Synonym: Guggulsterone E&Z
Target: Apoptosis, FXR, Akt, Caspase, JNK, Autophagy
25-Hydroxycholesterol
T4717
Synonym:
Target: Others, Endogenous Metabolite, HMG-CoA Reductase

Recombinant Proteins

カタログ番号 製品名 Species Expression System
TMPH-02139 CYP17A1 Protein, Human, Recombinant (GST) Human E. coli
A cytochrome P450 monooxygenase involved in corticoid and androgen biosynthesis. Catalyzes 17-alpha hydroxylation of C21 steroids, which is common for both pathways. A second oxidative step, required only for androgen sy...
TMPH-02140 CYP21A2 Protein, Human, Recombinant (E. coli, His) Human E. coli
A cytochrome P450 monooxygenase that plays a major role in adrenal steroidogenesis. Catalyzes the hydroxylation at C-21 of progesterone and 17alpha-hydroxyprogesterone to respectively form 11-deoxycorticosterone and 11-d...
TMPH-02141 CYP21A2 Protein, Human, Recombinant (His) Human P. pastoris (Yeast)
A cytochrome P450 monooxygenase that plays a major role in adrenal steroidogenesis. Catalyzes the hydroxylation at C-21 of progesterone and 17alpha-hydroxyprogesterone to respectively form 11-deoxycorticosterone and 11-d...
TMPJ-00207 AKR1C2 Protein, Human, Recombinant Human E. coli
Aldo-Keto Reductase Family 1 Member C2 (AKR1C2) plays a role in concert with the 5-α/5-β-Steroid Reductases to convert Steroid hormones into the 3-α/5-α and 3-α/5-β-Tetrahydrosteroids. AKR1C2 catalyzes the inactivation o...
TMPH-00220 Adrenodoxin, mitochondrial Protein, Bovine, Recombinant (His) Bovine E. coli
Essential for the synthesis of various steroid hormones. Participates in the reduction of mitochondrial cytochrome P450 for steroidogenesis. Transfers electrons from adrenodoxin reductase to CYP11A1, a cytochrome P450 th...
TMPH-00199 Bet v 1-A Protein, Betula pendula, Recombinant (His & SUMO) Betula pendula E. coli
May be a general steroid carrier protein. Bet v 1-A Protein, Betula pendula, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 33.4 kDa and the ac...
TMPH-03654 Vaccinia virus (strain Western Reserve) 3-beta-HSD Protein (His & Myc) VACV E. coli
Catalyzes the oxidative conversion of Delta(5)-ene-3-beta-hydroxy steroid, and the oxidative conversion of ketosteroids. The 3-beta-HSD enzymatic system plays a crucial role in the biosynthesis of all classes of hormonal...
TMPH-01811 OR7D4 Protein, Human, Recombinant (His & KSI) Human E. coli
Odorant receptor. Selectively activated by androstenone and the related odorous steroid androstadienone. OR7D4 Protein, Human, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The p...
TMPJ-01076 FKBP4 Protein, Human, Recombinant (His) Human E. coli
FKBP4 act as a regulator of microtubule dynamics by inhibiting MAPT/TAU ability to promote microtubule assembly. FKBP4 may play a role in the intracellular trafficking of heterooligomeric forms of steroid hormone recepto...
TMPY-00481 AKR1C4 Protein, Human, Recombinant (His) Human E. coli
Aldo-keto reductases comprise of AKR1C1-AKR1C4, four enzymes that catalyze NADPH dependent reductions and have been implicated in biosynthesis, intermediary metabolism, and detoxification. there is a strong correlation ...
TMPH-01747 FDXR Protein, Human, Recombinant (His & SUMO) Human E. coli
Serves as the first electron transfer protein in all the mitochondrial P450 systems including cholesterol side chain cleavage in all steroidogenic tissues, steroid 11-beta hydroxylation in the adrenal cortex, 25-OH-vitam...
TMPH-00288 Adrenodoxin reductase Protein, Bovine, Recombinant (His) Bovine P. pastoris (Yeast)
Serves as the first electron transfer protein in all the mitochondrial P450 systems including cholesterol side chain cleavage in all steroidogenic tissues, steroid 11-beta hydroxylation in the adrenal cortex, 25-OH-vitam...
TMPH-00287 Adrenodoxin reductase Protein, Bovine, Recombinant (E. coli, His) Bovine E. coli
Serves as the first electron transfer protein in all the mitochondrial P450 systems including cholesterol side chain cleavage in all steroidogenic tissues, steroid 11-beta hydroxylation in the adrenal cortex, 25-OH-vitam...
TMPH-03128 TSPO Protein, Pig, Recombinant (His & Myc & SUMO) Sus scrofa (Pig) E. coli
Promotes the transport of cholesterol across mitochondrial membranes and may play a role in lipid metabolism, but its precise physiological role is controversial. It is apparently not required for steroid hormone biosynt...
TMPH-01303 HSD17B11 Protein, Human, Recombinant (His & Myc) Human E. coli
Can convert androstan-3-alpha,17-beta-diol (3-alpha-diol) to androsterone in vitro, suggesting that it may participate in androgen metabolism during steroidogenesis. May act by metabolizing compounds that stimulate stero...
TMPJ-00158 Apolipoprotein A-I/APOA1 Protein, Human, Recombinant Human E. coli
Apolipoprotein A1 (APOA1) is a secreted protein which belongs to the Apolipoprotein A1/A4/E family. APOA1 is the major protein component of high density lipoprotein (HDL) in plasma. APOA1 plays a critical role in various...
TMPY-00867 Kallikrein 13/KLK13 Protein, Human, Recombinant (His) Human HEK293 Cells
Tissue kallikrein 13 (hK13), also known as KLK-L4 (kallikrein-like gene 4), is a member of the human tissue kallikrein family of serine proteases having diverse physiological functions in many tissues. The KLK13 gene res...
TMPY-03991 DBI Protein, Human, Recombinant (His) Human E. coli
The diazepam binding inhibitor (DBI), alternatively known as the acyl-CoA binding protein (ACBP), is involved in multiple biological actions. The polypeptide binds to the peripheral, or mitochondrial, benzodiazepine rece...
CYP17A1 Protein, Human, Recombinant (GST)
TMPH-02139
Species: Human
Expression System: E. coli
CYP21A2 Protein, Human, Recombinant (E. coli, His)
TMPH-02140
Species: Human
Expression System: E. coli
CYP21A2 Protein, Human, Recombinant (His)
TMPH-02141
Species: Human
Expression System: P. pastoris (Yeast)
AKR1C2 Protein, Human, Recombinant
TMPJ-00207
Species: Human
Expression System: E. coli
Adrenodoxin, mitochondrial Protein, Bovine, Recombinant (His)
TMPH-00220
Species: Bovine
Expression System: E. coli
Bet v 1-A Protein, Betula pendula, Recombinant (His & SUMO)
TMPH-00199
Species: Betula pendula
Expression System: E. coli
Vaccinia virus (strain Western Reserve) 3-beta-HSD Protein (His & Myc)
TMPH-03654
Species: VACV
Expression System: E. coli
OR7D4 Protein, Human, Recombinant (His & KSI)
TMPH-01811
Species: Human
Expression System: E. coli
FKBP4 Protein, Human, Recombinant (His)
TMPJ-01076
Species: Human
Expression System: E. coli
AKR1C4 Protein, Human, Recombinant (His)
TMPY-00481
Species: Human
Expression System: E. coli
FDXR Protein, Human, Recombinant (His & SUMO)
TMPH-01747
Species: Human
Expression System: E. coli
Adrenodoxin reductase Protein, Bovine, Recombinant (His)
TMPH-00288
Species: Bovine
Expression System: P. pastoris (Yeast)
Adrenodoxin reductase Protein, Bovine, Recombinant (E. coli, His)
TMPH-00287
Species: Bovine
Expression System: E. coli
TSPO Protein, Pig, Recombinant (His & Myc & SUMO)
TMPH-03128
Species: Sus scrofa (Pig)
Expression System: E. coli
HSD17B11 Protein, Human, Recombinant (His & Myc)
TMPH-01303
Species: Human
Expression System: E. coli
Apolipoprotein A-I/APOA1 Protein, Human, Recombinant
TMPJ-00158
Species: Human
Expression System: E. coli
Kallikrein 13/KLK13 Protein, Human, Recombinant (His)
TMPY-00867
Species: Human
Expression System: HEK293 Cells
DBI Protein, Human, Recombinant (His)
TMPY-03991
Species: Human
Expression System: E. coli
カタログ番号 製品名
L4710 Nonsteroidal Anti-Inflammatory Compound Library

530 compounds
530 non-steroidal anti-inflammatory compounds for high-throughput and high-content screening.
L1510 Nuclear Receptor Compound Library

531 compounds
A unique collection of 531 nuclear receptor signaling targeted compounds for high throughput and high content screening;
L6810 Traditional Chinese Medicine Monomer Library

2755 compounds
A unique collection of 2755 compounds (TCM monomers) sourcing from traditional Chinese Medicines, is a powerful tool for drug discovery and research in mechanism;
L6800 Chinese Pharmacopoeia Natural Product Library

2051 compounds
A unique collection of 2051 natural products included in Chinese Pharmacopoeia (CP), a powerful tool for drug development and pharmacological study;