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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T11069 | DO-264 | Others | |
DO-264 is an inhibitor of autohydrolase structural domain 12 (ABHD12) (IC50: 11 nM) and an inhibitor of cellular LysoPS degradation that enhances LPS-induced phagocytosis. | |||
T4142 | PCC0208009 | IDO inhibitor 1,DO-IN-2,IDO-IN-2 | Indoleamine 2,3-Dioxygenase (IDO) |
PCC0208009 (IDO-IN-2) is an IDO inhibitor. | |||
T31559 | DO-601 | Others | |
DO-601 is a stimulant that stimulates the central nervous system. | |||
T7857 | DO1 | Disperse Orange 1 | Others |
DO1 (Disperse Orange 1) is an anti-amyloid agent which potently delays both seeded and non-seeded Aβ42 polymerization at substoichiometric concentrations | |||
T11070 | DO34 analog | Others | |
DO34 analog is a triazole DAGL(α) inhibitor. | |||
T27821 | Lexipafant | ISV-611,GR-167089,DO-6,BB-882,DO6,BB882 | Others |
Lexipafant is a platelet-activating factor (PAF) receptor antagonist. | |||
T11070L | DO34 | Others | |
DO34 is a highly potent and centrally active inhibitor of diacylglycerol lipase (IC50: 6 nM for DAGLα conversion of SAG to 2-AG). | |||
T31558 | DO53 | Others | |
DO53 is a negative control for DO34, not inhibiting DAGL. | |||
T71808 | Tisopurine | Others | |
Tisopurine is a drug used in the treatment of gout in some countries. It reduces uric acid production through inhibiting an early stage in its production. | |||
T24156 | ICI 195739 | DO870,D0870,D 0870,D-0870 | Others |
ICI 195739 is a newer antifungal agent. It inhibits neutrophil random migration, chemotaxis, and hexose monophosphate shunt activity. | |||
T19293 | DO3A tert-Butyl ester | DO3A-t-Bu-ester,DO3A tert-butyl | Others |
DOTA tert-butyl ester is a phenyl derivative of cycloteramide; it can be directly nitrated; it is more convenient to add nitro after deprotection of lithium aluminum hydride. | |||
T40025 | Pomalidomide-PEG2-CO2H | Pomalidomide 4'-PEG2-acid,Pomalidomide-PEG2-C2-acid | E3 Ligase Ligand-Linker Conjugate |
Pomalidomide-PEG2-CO2H is a synthetic E3 ligase ligand-linker conjugate containing a Pomalidomide-based cereblon ligand and a 2-unit PEG linker. | |||
T17492 | Azido-PEG2-azide | Others , PROTAC Linker | |
Azido-PEG2-azide is a PEG-based PROTAC linker that can be used in PROTAC synthesis. | |||
T17486 | Azido-PEG12-NHS ester | Others , PROTAC Linker | |
Azido-PEG12-NHS ester is a PEG-based PROTAC linker that can be used in PROTAC synthesis. | |||
T11894 | Lusaperidone | R107474 | Adrenergic Receptor |
Lusaperidone (R107474) is a potent α2-adrenergic receptor antagonist, a potential radioligand for the α (2)-adrenergic receptor, with inhibitory effects on α2A and α2C, with Ki values of 0.13 and 0.15 nM, respectively. | |||
T11075 | Donitriptan | 5-HT Receptor | |
Donitriptan is a 5-HT receptor agonist with pKis of 9.4 and 9.3 for 5-HT1B and 5-HT1D, respectively. | |||
T19319 | Ethyl docosa-4,7,10,13,16,19-hexaenoate | Others | |
Ethyl cis-4,7,10,13,16,19-Docosahexaenoate, the ethyl ester of Docosahexaenoate (DHA), is selectively enriched in the ethyl ester fraction through the alcoholysis process involving fatty acid ethyl esters from tuna oil a... | |||
T17522 | Azido-PEG9-azide | Others , PROTAC Linker | |
Azido-PEG9-azide is a PEG-based PROTAC linker that can be used in PROTAC synthesis. | |||
T8653 | DOPEXAMINE | Dopamine Receptor | |
Dopexamine is a dopaminergic agonist | |||
T22316 | Doxazosin | UK 33274 | Adrenergic Receptor |
Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms. | |||
T7759 | Thalidomide-O-amido-C4-NH2 TFA | E3 ligase Ligand-Linker Conjugates 19 TFA,Cereblon Ligand-Linker Conjugates 6 TFA | E3 Ligase Ligand-Linker Conjugate |
Thalidomide-O-amido-C4-NH2 TFA (E3 ligase Ligand-Linker Conjugates 19 TFA) is a synthesized E3 ligase ligand-linker conjugate. | |||
T40023 | Pomalidomide-PEG3-CO2H | Thalidomide-NH-PEG3-propionic acid | E3 Ligase Ligand-Linker Conjugate |
Pomalidomide-PEG3-CO2H (Thalidomide-NH-PEG3-propionic acid) is a synthesized E3 ligase ligand-linker conjugate. Pomalidomide-PEG3-CO2H incorporates the Thalidomide based cereblon ligand and 3-unit PEG linker used in PROT... | |||
T19459 | N1-Methylpseudouridine | 1-Methylpseudouridine | Others |
N1-Methylpseudouridine (1-Methylpseudouridine) is a methylpseudouridine and enhances translation through eIF2α-dependent and independent mechanisms by increasing ribosome density in mRNA. | |||
T15159 | Dorzagliatin | HMS5552 | Glucokinase |
Dorzagliatin (HMS5552) is a dual-acting glucokinase (GK) activator. It also improves glycaemic control and pancreatic β-cell function in type 2 diabetes. | |||
T0182L2 | (±) Clopidogrel hydrogen sulfate | Plavix,Clopidogrel hydrogen sulfate,Iscover | P2Y Receptor |
(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots in various conditions such as cerebrovascular disease, periph... | |||
T2148 | Carbidopa monohydrate | Carbidopa Hydrate,S(-)-Carbidopa | Decarboxylase , Aryl Hydrocarbon Receptor |
Carbidopa monohydrate (S(-)-Carbidopa) is an inhibitor of DOPA decarboxylase, preventing the conversion of levodopa to dopamine. | |||
T14038 | 4-Azido-L-phenylalanine | p-Azidophenylalanine,p-Azido-L-phenylalanine | Others |
4-Azido-L-phenylalanine (p-Azido-L-phenylalanine) is an amino acid derivative that acts as a photoaffinity marker and can be used to detect localized protein environments. | |||
T6165 | Bardoxolone Methyl | RTA 402,CDDO Methyl ester,TP-155,NSC 713200 | Apoptosis , IκB/IKK , Ferroptosis , Nrf2 , Autophagy |
Bardoxolone Methyl (TP-155) is a synthetic triterpenoid that acts as an activator of the Nrf2 pathway and an inhibitor of the NF-κB pathway with potential anti-tumor and anti-inflammatory activities. | |||
T40016 | Thalidomide-NH-CH2-COOH | 2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetic acid,(2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)glycine | Ligand for E3 Ligase |
Thalidomide-NH-CH2-COOH ((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)glycine) is a synthesized E3 ligase ligand-linker conjugate containing a Thalidomide-based cereblon ligand and a linker. | |||
T2601 | Vidofludimus | SC12267,4sc-101 | Dehydrogenase , DNA/RNA Synthesis , Interleukin |
Vidofludimus (SC12267) (4SC-101, SC12267) is a novel small molecule inhibitor of dihydroorotate dehydrogenase (DHODH). | |||
T1977 | Dorsomorphin | Compound C,BML-275 | AMPK , Autophagy , TGF-beta/Smad |
Dorsomorphin (BML-275) is an AMPK inhibitor (Ki=109 nM) that is selective and ATP-competitive. Dorsomorphin inhibits the BMP type I receptors ALK2, ALK3, and ALK6. Dorsomorphin induces autophagy, and possesses antitumor ... | |||
T3269 | Metadoxine | pyridoxine-pyrrolidone carboxylat,Metasin,Metadoxil | 5-HT Receptor , PKA |
Metadoxine (Metadoxil) is a neurotransmitter stimulant. | |||
T7191 | Diphenyleneiodonium chloride | DPI | NOS , Reactive Oxygen Species , NADPH , TRP/TRPV Channel |
Diphenyleneiodonium chloride (DPI)(DPI) is an irreversible inhibitor of iNOS and eNOS (IC50 values of 50 nM and 0.3 μM, respectively),and displays broad-spectrum bactericidal activity. | |||
T40019 | Thalidomide-5-NH2-CH2-COOH | Others | |
Thalidomide-5-NH2-CH2-COOH (compound 114) is a selective inhibitor of the protomyosin receptor kinase. It is a ligand for E3 ligase and has potential for studying one or more diseases. | |||
T7758 | Thalidomide-O-amido-PEG3-C2-NH2 TFA | E3 ligase Ligand-Linker Conjugates 14 TFA,Cereblon Ligand-Linker Conjugates 3 (TFA) | Others , E3 Ligase Ligand-Linker Conjugate , Ligand for E3 Ligase |
Thalidomide-O-amido-PEG3-C2-NH2 TFA (Cereblon Ligand-Linker Conjugates 3 (TFA)) is a synthesized E3 ligase ligand-linker conjugate. Thalidomide-O-amido-PEG3-C2-NH2 TFA incorporates the Thalidomide based cereblon ligand a... | |||
T32535 | Ladostigil | TV-3326,Ladostigil,TV 3326,TV3326,Ladostigil free base | Antioxidant , MAO , AChE |
Ladostigil (Ladostigil free base) is an orally active dual inhibitor of cholinesterase and brain-selective monoamine oxidase (MAO) with inhibitory effects on MAO-B and AChE, with IC50 values of 37.1 and 31.8 μM, respecti... | |||
T9384 | Pomalidomide-PEG3-OH | 1H-Isoindole-1,3(2H)-dione, 2-(2,6-dioxo-3-piperidinyl)-4-[[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]amino]- | PROTACs |
Pomalidomide-PEG3-OH enables the synthesis of molecules for targeted protein degradation and PROTAC (proteolysis-targeting chimeras) technology. | |||
T11077 | Dopamine D2 receptor antagonist-1 | Others | |
Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity. | |||
T4568 | Dolasetron | MDL-73147 | 5-HT Receptor |
Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy. | |||
T0716 | Molindone hydrochloride | EN-1733A | Dopamine Receptor , 5-HT Receptor , AChR |
Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain. | |||
T25705 | Imupedone | LF1695,LF-1695,LF 1695 | Others |
Imupedone (LF 1695) is a synthetic immunomodulator that modulates T lymphocytes and macrophages, induces T-cell differentiation of bone marrow precursor cells, and increases the proliferative response of lymphocytes to m... | |||
T67751 | 1H-Indole-3-carboxylic acid, 5-[2-hydroxy-3-[[2-hydroxy-1,1-bis(hydroxymethyl)ethyl]amino]propoxy]-2-methyl-1-(4-methylphenyl)-, ethyl ester | Beta Amyloid | |
Compound 5936-0108 may has modulationg effect on β-Amyloid. | |||
T14033 | 3BDO | Apoptosis , mTOR , Autophagy | |
3BDO is an activator of mTOR. It can also inhibit autophagy.. | |||
T1576 | Iopamidol | SQ-13396,Niopam,Iopamiron,Iopamiro,B-15000,Isovue | Others |
Iopamidol (SQ-13396) is a benzenedicarboxamide compound. It has a role as a radioopaque medium, an environmental contaminant and a xenobiotic. | |||
T15034 | Roluperidone | CYR-101,MIN-101,MT-210 | Sigma receptor , 5-HT Receptor |
Roluperidone (CYR-101) is a novel cyclic amide derivative. It has high equipotent affinities for 5-HT2A and σ2 receptors (Ki of 7.53 nM and 8.19 nM for 5-HT2A and σ2). | |||
T1504 | Silodosin | KAD 3213,KMD 3213 | Adrenergic Receptor |
Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist. | |||
T3648 | Hypidone hydrochloride | YL0919 | 5-HT Receptor |
Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor. | |||
T19694 | Hydronidone | F351,F-351,F 351 | Others |
Hydronidone (F-351) is Non-Steroidal Antiinflammatory Drugs. It potentially for the treatment of hepatic fibrosis. | |||
T9387 | Pomalidomide 4'-PEG2-azide | E3 Ligase Ligand-Linker Conjugate | |
Pomalidomide 4'-PEG2-azide is a synthetic E3 ligase ligand-linker conjugate containing a Pomalidomide-based cereblon ligand and a linker. | |||
T0025 | Haloperidol | Aloperidin,Serenace,Haldol | Dopamine Receptor , 5-HT Receptor |
Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function. In addition, haloperidol has shown about 50-fold efficacy than chlorpromazine, another antipsychotic dr... |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T1121 | Podofilox | Podophyllotoxin,(+)-Shikonin | Microtubule Associated , Topoisomerase |
Podofilox ((+)-Shikonin) is a lignan (LIGNANS) found in PODOPHYLLIN resin from the roots of PODOPHYLLUM plants. It is a potent spindle poison, toxic if taken internally, and has been used as a cathartic. It is very irrit... | |||
TN4495 | Maoyerabdosin | Others | |
Maoyerabdosin is a kind of natural product derived from the herbs of Isodon. | |||
T7916 | 4-Acetamidobenzenesulfonyl azide | Others | |
4-Acetamidobenzenesulfonyl azide is used in a variety of scientific research applications, including the synthesis of drugs, peptides and other biologically active molecules. It is also used as a catalyst in polymerizati... | |||
TN3972 | Epimedokoreanin B | Apoptosis , Others , Antibacterial | |
Epimedokoreanin B (EKB), an isoprenylated flavonoid isolated from Korean Epimedium, exhibited anticancer activity in human non-small cell lung cancer (NSCLC) A549 and NCI-H292 cells.Epimedokoreanin B also possesses anti-... | |||
TN7186 | Methyl 6-bromo-1H-indole-3-carboxylate | Methyl 6-bromo-1H-indole-3-carboxylate | Others |
1H-Indole-3-Carboxylic Acid,6-Bromo-,Methyl Ester (Methyl 6-bromo-1H-indole-3-carboxylate) is a marine derived natural products found in Smenospongia sp. | |||
TN7136 | 1,7-dimethyl-1H-indole-3-carbaldehyde | 1,7-dimethylindole-3-carbaldehyde,ZINC14592128,N,7-Dimethylindole-3-carbaldehyde | Others |
1,7-dimethyl-1H-indole-3-carbaldehyde (ZINC14592128) is a marine derived natural products found in Lyngbya majuscula. | |||
T4754 | Pyridoxylamine dihydrochloride | Pyridorin,Pyridoxamine dihydrochloride | Others , Endogenous Metabolite |
Pyridoxylamine dihydrochloride (Pyridorin) is a hydrochloride salt of one form of vitamin B6. | |||
T16223 | N-Dodecyl-β-D-maltoside | Lauryl Maltoside | Others |
N-Dodecyl-β-D-maltoside (Lauryl Maltoside) has also been employed in applications such as in the purification and stabilization of RNA polymerase and the detection of protein-lipid interactions. N-Dodecyl-β-D-maltoside i... | |||
T13851 | Pseudolaric Acid C2 | Others | |
Pseudolaric Acid C2 is a diterpenoid isolated from Pseudolarix kaempferi. | |||
TN7207 | Ethyl6-bromo-1H-indole-3-carboxylate | Ethyl 6-Bromoindole-3-carboxylate,ethyl 6-bromo-3-indolecarboxylate,ZINC13379655 | Others |
Ethyl6-bromo-1H-indole-3-carboxylate (Ethyl 6-Bromoindole-3-carboxylate) is a marine derived natural products found in Pleroma menoui. | |||
TN7041 | (-)-Epipodophyllotoxin | Apoptosis | |
(-)-Epipodophyllotoxin (2) is an antiproliferative agent against cancer cells with GI50s of 0.36 and 0.24 μM in HeLa cells and MCF-7 cells, respectively. (-)-Epipodophyllotoxin can inhibit mitotic spindle assembly in vit... | |||
T2773 | Vindoline | Microtubule Associated | |
Vindoline is an indole alkaloid that exhibits antimitotic activity by inhibiting microtubule assembly. | |||
T4461 | 3,5-Diiodo-L-thyronine | Diiodothyronine | Thyroid hormone receptor(THR) , Endogenous Metabolite |
3,5-Diiodo-L-thyronine (Diiodothyronine) is an iodinated thyronine hormone that regulates gene activity affecting processes such as homeostasis, lipid metabolism and insulin resistance. | |||
T5258 | Dodecanedioic acid diammonium salt | 1,10-Decanedicarboxylic acid diammonium salt | Others |
Dodecanedioic acid diammonium salt (1,10-Decanedicarboxylic acid diammonium salt) is a dicarboxylic acid which is water-soluble and involves in a metabolic pathway intermediate to those of lipids and carbohydrates. | |||
TN7160 | 3,3'-Bi[1H-indole] | 3,3'-Biindole,3-(1H-indol-3-yl)-1H-indole,1H,1'H-3,3'-biindole | Others |
3,3'-Bi[1H-indole] (3,3'-Biindole) is a marine derived natural products found in Nocardiopsis sp. | |||
T4744 | 5-HYDROXYINDOLE-3-ACETIC ACID | 5-HIAA | Others , Endogenous Metabolite |
5-Hydroxyindole-3-acetic acid (5-HIAA) is a breakdown product of serotonin that is excreted in the urine. Serotonin and 5HIAA are produced in excess amounts by carcinoid tumors, and levels of these substances may be meas... | |||
T4107 | 4-Pyridoxic Acid | Pyridoxic Acid,4-Pyridoxinsaeure | Endogenous Metabolite |
4-Pyridoxic Acid (4-Pyridoxinsaeure), a catabolite of vitamin B6, is a water-soluble B-group vitamin that can be used as a urinary diagnostic biomarker for determining the nutritional status of these vitamins. | |||
T19295 | Docosapentaenoic acid 22n-3 | Endogenous Metabolite | |
Docosapentaenoic acid 22n-3 is present in the cell membranes of all animals and is a component of phospholipids. | |||
TN7200 | 3-chloro-1H-indole | ZINC6117681,3-chloro-1H-indole | Others |
3-chloro-1H-indole (ZINC6117681) is a marine derived natural products found in Ptychodera flava. | |||
TN7092 | Lugrandoside | Others | |
Lugrandoside is a novel phenylpropanoid glycoside, lugrandoside, has been isolated from the caulinary leaves of Digitalis Lutea L. and Difitalis Grandiflora Miller. | |||
T25114 | Ascaridole | NSC-406266,NSC 406266,NSC406266 | Parasite |
Ascaridole (NSC-406266) acts as an anthelmintic compound that repels parasitic helminths (worms) in humans and plants and has weak antimalarial activity. | |||
T2S2172 | Nerolidol | (±)-Nerolidol,Peruviol | Others , Endogenous Metabolite , Antibacterial , Parasite , Antifungal |
Nerolidol (Peruviol) shows sedative effects in animals, oxidative process plays a crucial role on neuronal pathological consequence. Nerolidol is mainly related to ROS and DNA single strand breaks generated by the presen... | |||
T13513 | 5-Methoxyindole-3-acetic acid | Methoxyindoleacetic acid,5-Methoxyindoleacetic acid | Endogenous Metabolite |
5-Methoxyindole-3-acetic acid (5-Methoxyindoleacetic acid) is a metabolite of Melatonin and is isolated from pineal tissue. | |||
TQ0065 | Pseudobufarenogin | ψ-Bufarenogin | Others |
Pseudobufarenogin (ψ-Bufarenogin), a novel anti-tumor compound, suppresses liver cancer growth by inhibiting receptor tyrosine kinase-mediated signaling. | |||
T3799 | Isorhamnetin-3-O-neohespeidoside | Isorhamnetin 3-O-neohesperidin,Isorhamnetin 3-O-neohesperoside,Calendoflavoside | Antioxidant |
Isorhamnetin-3-O-neohespeidoside (Calendoflavoside) is a flavonol glycoside extract used as an anti-oxidant. | |||
T5741 | Pseudolaric acid B β-D-glucoside | Pseudolaric acid B-glucopyranoside | Others |
Pseudolaric acid B β-D-glucoside (Pseudolaric acid B-glucopyranoside) is a natural product from Pseudolarix amabilis. | |||
T0436 | 6-Acetamidohexanoic acid | 6-Acetamidocaproic acid,Acexamic Acid | Amino Acids and Derivatives , COX |
6-Acetamidohexanoic acid (Acexamic Acid) is a kind of amino acids deriviate. | |||
T0076 | Paliperidone | 9-hydroxyrisperidone | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor |
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the primary active metabolite of the older... | |||
T3S1967 | (S)-Indoximod | N-ME-Tryptophan,Abrine,L-Abrine | Others , Indoleamine 2,3-Dioxygenase (IDO) |
(S)-Indoximod (L-Abrine) exhibits inhibition of rabbit small intestine indoleamine 2, 3-dioxygenase, competitive inhibition of IDO, reduction of Foxp3 protein expression in tumor of C57BL/6 mouse allografted with mouse L... | |||
T5558 | Chelidonic acid | Jervaic acid,Jerva acid,γ-Pyrone-2,6-dicarboxylic acid | NF-κB , Caspase |
Chelidonic acid (Jervaic acid) is a component of Chelidonium majus L., used as a mild analgesic, an antimicrobial, an acentral nervous system sedative. Chelidonic acid (Jervaic acid) also shows anti-inflammatory activity... | |||
TN1723 | Hamaudol | COX | |
Hamaudol is a chromone isolated from Saposhnikovia divaricata,has analgesic and anti-inflammary activities, it showed inhibitory activity on COX-1 and COX-2 activities with values of 0.30, 0.57 mM, respectively. | |||
T4805 | α-Pyridone | 2-Hydroxypyridine | Others , Endogenous Metabolite |
α-Pyridone (2-Hydroxypyridine)e is the catalyst for generating β-oxopropyl carbonates from cyclic carbonates and alcohols and in the aminolysis of a polyglutamate. | |||
T5984 | Indole-3-carboxylic acid | 3-Indoleformic acid | Endogenous Metabolite |
Indole-3-carboxylic acid (3-Indoleformic acid) is a normal urinary indolic tryptophan metabolite . | |||
T2S0250 | Pseudoprotogracillin | Others | |
Pseudoprotogracillin is a steroidal saponin extracted from Dioscoreae. | |||
T8105 | Indole-3-carboxaldehyde | 3-Formylindole | Endogenous Metabolite |
1H-Indole-3-carboxaldehyde (3-Formylindole), also known as 3-formylindole or 3-indolealdehyde, belongs to the class of organic compounds known as indoles. Indoles are compounds containing an indole moiety, which consists... | |||
T5S0055 | Chelidonine | Helidonine,Khelidonin,Stylophorin | Apoptosis , Others , Influenza Virus |
1. Chelidonine (Stylophorin) isolated from Chelidonium majus efficiently induced apoptosis in HeLa cells through possible alteration of p38-p53 and AKT/PI3 kinase signalling pathways. 2. Chelidonine is a promising model ... | |||
T5709 | Cyperotundone | Others | |
Cyperotundone is a natural product from Cyperus rotundus | |||
T5868 | Methyl indole-3-carboxylate | Methyl 3-indolecarboxylate | Others , Antibacterial |
Methyl indole-3-carboxylate (Methyl 3-indolecarboxylate) is a natural product isolated from Heracleum candicans. | |||
T3S0027 | Picropodophyllotoxin | AXL 1717,Picropodophyllin | IGF-1R |
Picropodophyllotoxin (AXL 1717) is a cyclolignan alkaloid found in the mayapple plant family (Podophyllum peltatum), and a small molecule inhibitor of the insulin-like growth factor 1 receptor (IGF1R) with potential anti... | |||
T0969 | Doramectin | Dectomax,Cyclohexylavermectin B1 | Others , Antibiotic , Parasite |
Doramectin (Dectomax) is an antiparasitic agent. | |||
T5S0527 | Rhodojaponin III | Others | |
1. Rhodojaponin III has antifeedant and oviposition deterrence effects against many kinds of insects, BdorCSP2 of B. dorsalis could be involved in chemoreception of Rhodojaponin III and played a critical role. 2. Rhodoja... | |||
T8188 | Podophyllotoxone | Others , Microtubule Associated | |
Podophyllotoxinone, a natural compound found in Dysosma versipellis, shows inhibitory activity against L1210 leukemia and KB cells in vitro. | |||
TN2070 | Picropodophyllol | Others | |
Picropodophyllol is a natural product isolated from the roots of Dysosma versipellis | |||
T4S1519 | Pseudoginsenoside RT5 | Others | |
1. Pseudoginsenoside RT5 has anti-epilepsy, anti-depressant activity by promoting nerve growth and improve cognitive ability. 2. Pseudoginsenoside RT5 has anti-bacterial, anti-tumor and anti-malaria activities. | |||
TN7175 | 9H-Carbazole, 3,6-diiodo- | 3,6-Diiodo-9H-carbazole,3,6-diiodocarbazole | Others |
9H-Carbazole, 3,6-diiodo- (3,6-diiodocarbazole) is a marine derived natural products found in Kyrtuthrix maculans. | |||
T5226 | 2-(2-Methylbenzamido)acetic acid | 2-Methylhippuric acid,O-Toluric acid,N-(O-Toluoyl)glycine | Others , Endogenous Metabolite |
2-(2-Methylbenzamido)acetic acid (O-Toluric acid) is an acyl glycine. Acyl glycines are normally minor metabolites of fatty acids. In certain cases, the measurement of these metabolites in body fluids can be used to diag... | |||
TN7180 | 2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)- | Meridianin C | Others |
2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)- (Meridianin C) is a marine derived natural products found in Aplidium meridianum. | |||
T3578 | Pyridoxal phosphate | PLP,PAL-P,pyridoxal 5'-phosphate,Pyridoxyl phosphate,Pyridoxal 5′-phosphate,Vitamin B6 phosphate | Reverse Transcriptase , Endogenous Metabolite |
Pyridoxal phosphate (Vitamin B6 phosphate) is the active form of vitamin B6 and a coenzyme for many pyridoxal phosphate (PLP)-dependent enzymes. PLP is involved in numerous enzymatic transamination, decarboxylation and d... | |||
TN2356 | Tetradehydropodophyllotoxin | Dehydropodophyllotoxin | Others , Antifungal |
Tetradehydropodophyllotoxin (Dehydropodophyllotoxin) has anti-tumor activity. | |||
T5217 | 2-(2-Phenylacetamido)acetic acid | Phenaceturic acid,Phenyl-ac-Gly-OH,Phenylacetyl glycine | Others , Endogenous Metabolite |
Phenyl-ac-Gly-OH is an endogenous metabolite that activates β2AR and can be used in the study of ischemia/reperfusion-induced cardiac injury. | |||
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カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPY-02822 | ART4/CD297 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
ART4/CD297 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 53.7 kDa and the accession number is Q9CRA0. | |||
TMPY-02738 | ART4/CD297 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
ART4/CD297 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 28.2 kDa and the accession number is EDL10575.1. | |||
TMPH-00708 | DegP Protein, E. coli, Recombinant (His) | E. coli | P. pastoris (Yeast) |
DegP acts as a chaperone at low temperatures but switches to a peptidase (heat shock protein) at higher temperatures. Degrades transiently denatured and unfolded or misfolded proteins which accumulate in the periplasm fo... | |||
TMPY-05823 | Influenza B (B/Colorado/06/2017) Hemagglutinin/HA Protein (His) | Influenza B | HEK293 Cells |
Influenza B (B/Colorado/06/2017) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 58.86 kDa and the accession number is A0A2Z5E1Y3. | |||
TMPY-01519 | Influenza A H1N1 (A/New Caledonia/20/1999) Hemagglutinin/HA Protein (His) | H1N1 | HEK293 Cells |
Influenza A H1N1 (A/New Caledonia/20/1999) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is Q6WG00. | |||
TMPY-05918 | Influenza A H1N1 (A/Guangdong-Maonan/SWL1536/2019)/(A/Hawaii/70/2019) Hemagglutinin/HA Protein (His) | H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Guangdong-Maonan/SWL1536/2019)/(A/Hawaii/70/2019) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59.2 kDa and the accession numbe... | |||
TMPY-00416 | Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA0 Protein | H10N8 | Baculovirus Insect Cells |
Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA0 Protein is expressed in Baculovirus insect cells. The predicted molecular weight is 60.6 kDa. | |||
TMPY-02869 | MMP-12 Protein, Human, Recombinant (catalytic domain) | Human | E. coli |
Matrix metalloproteinases (MMPs) are a family of zinc-dependent endopeptidases that degrade components of the extracellular matrix (ECM) and play essential roles in various physiological processes such as morphogenesis, ... | |||
TMPY-00382 | Thioredoxin/TRX Protein, Mouse, Recombinant | Mouse | E. coli |
Thioredoxin/TRX Protein, Mouse, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 11.7 kDa and the accession number is P10639. | |||
TMPY-01384 | Endoglin/CD105 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Endoglin/CD105 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 62.3 kDa and the accession number is A0A024R878. | |||
TMPY-02662 | Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA Protein (His) | H10N8 | Baculovirus Insect Cells |
Influenza A H10N8 (A/Jiangxi-Donghu/346/2013) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.9 kDa. | |||
TMPY-06059 | Influenza A H1N1 (A/Guangdong-Maonan/SWL1536/2019) Nucleoprotein/NP Protein (His) | H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/Guangdong-Maonan/SWL1536/2019) Nucleoprotein/NP Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.7 kDa. | |||
TMPY-05895 | Influenza A H3N2 (A/swine/Colorado/A01203748/2012) Hemagglutinin/HA Protein (His) | H3N2 | HEK293 Cells |
Influenza A H3N2 (A/swine/Colorado/A01203748/2012) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 57.7 kDa and the accession number is K0FL26. | |||
TMPY-06737 | Equ c 1 Protein, Domestic horse, Recombinant | Domestic horse | E. coli |
Equ c 1 Protein, Domestic horse, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 21.1 kDa. | |||
TMPY-06187 | Influenza B (B/Colorado/06/2017) Nucleoprotein/NP Protein (His) | Influenza B | Baculovirus Insect Cells |
Influenza B (B/Colorado/06/2017) Nucleoprotein/NP Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 63.1 kDa. | |||
TMPY-05169 | Peroxiredoxin 2 Protein, Mouse, Recombinant (His) | Mouse | Baculovirus Insect Cells |
Peroxiredoxin 2 Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 24.1 kDa and the accession number is Q61171. | |||
TMPY-00245 | Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Makona-Kissidougou-C15) GP/Glycoprotein Protein (His) | EBOV | HEK293 Cells |
Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Makona-Kissidougou-C15) GP/Glycoprotein Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 69.3 kDa and the ... | |||
TMPY-00181 | Endothelin B Receptor Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Endothelin B Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 9.5 kDa and the accession number is P24530-1. | |||
TMPY-02718 | Doublecortin/DCX Protein, Human, Recombinant (aa 45-150, GST) | Human | E. coli |
DCX (doublecortin, N-GST chimera)contains 2 doublecortin domains and belongs to the doublecortin family. It is highly expressed in neuronal cells of fetal brain, but not expressed in other fetal tissues. In the adult, it... | |||
TMPY-00323 | Hepatitis C virus (HCV-1a) NS3 protease/helicase immunodominant region Protein (aa 1356-1459, GST) | HCV | E. coli |
HCV NS3 displays three enzymatic activities: serine protease, NTPase, and RNA helicase. HCV NS3 serine protease, in association with NS4A, is responsible for the cleavages of NS3-NS4A, NS4A-NS4B, NS4B-NS5A, and NS5A-NS5B... | |||
TMPY-00102 | Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) Glycoprotein/GP-RBD Protein (His) | EBOV | HEK293 Cells |
Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) Glycoprotein/GP-RBD Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 32.3 kDa and the acc... | |||
TMPY-00279 | Dengue virus DENV-2 (strain New Guinea C) NS5 (methyltransferase domain)/Nonstructural protein 5 Protein (His) | DENV | E. coli |
Dengue virus DENV-2 (strain New Guinea C) NS5 (methyltransferase domain)/Nonstructural protein 5 Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 35.5 kDa and the ac... | |||
TMPY-02084 | Thioredoxin 2/TRX2 Protein, Human, Recombinant (His) | Human | E. coli |
Thioredoxin-2, also known as TXN2, MTRX and TRX2, is a member of the thioredoxin family. Tryparedoxins (TXN) are thioredoxin-related proteins which, as trypanothione:peroxiredoxin oxidoreductases, constitute the trypanot... | |||
TMPY-06733 | PLA A2 Protein, London plane tree, Recombinant | London plane tree | HEK293 Cells |
PLA A2 Protein, London plane tree, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 40.2 kDa. | |||
TMPY-06736 | Bos d 2 Protein, Bos domesticus, Recombinant | Bos domesticus | E. coli |
Bos d 2 Protein, Bos domesticus, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 32.4 kDa. | |||
TMPY-00255 | Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) GP2/Glycoprotein Protein (Fc) | EBOV | HEK293 Cells |
Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) GP2/Glycoprotein Protein (Fc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 43.4 kDa and the accessio... | |||
TMPY-02928 | IDO Protein, Human, Recombinant | Human | E. coli |
IDO Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 45.2 kDa and the accession number is A0A348GSI3. | |||
TMPY-01095 | Podoplanin Protein, Mouse, Recombinant (His & hFc) | Mouse | HEK293 Cells |
Podoplanin Protein, Mouse, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 40.6 kDa and the accession number is Q62011. | |||
TMPY-06887 | Influenza A H1N1 (A/Hawaii/70/2019;A/Guangdong-Maonan/SWL1536/2019) Hemagglutinin/HA Protein (His) | H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/Hawaii/70/2019;A/Guangdong-Maonan/SWL1536/2019) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.24 kDa. | |||
TMPY-02462 | Peroxiredoxin 5 Protein, Mouse, Recombinant (His) | Mouse | E. coli |
Peroxiredoxin 5 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 18.5 kDa and the accession number is P99029-1. | |||
TMPY-00061 | Rift Valley fever virus (TAN/Dod-002/07) RVFV-L Protein (His) | RVFV | E. coli |
Rift Valley fever virus (TAN/Dod-002/07) RVFV-L Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 29.4 kDa and the accession number is AEB20483.1. | |||
TMPY-00555 | Podoplanin Protein, Rat, Recombinant (hFc) | Rat | HEK293 Cells |
Podoplanin Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 38.6 kDa and the accession number is Q64294. | |||
TMPY-02250 | Thioredoxin/TRX Protein, Human, Recombinant | Human | E. coli |
Thioredoxin/TRX Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 11.7 kDa and the accession number is P10599. | |||
TMPY-01311 | Podoplanin Protein, Human, Recombinant (His & hFc) | Human | HEK293 Cells |
Podoplanin Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 38.4 kDa and the accession number is Q86YL7-1. | |||
TMPY-04653 | Influenza A H5N6 (A/duck/Guangdong/GD01/2014) Hemagglutinin/HA1 Protein (His) | H5N6 | HEK293 Cells |
Influenza A H5N6 (A/duck/Guangdong/GD01/2014) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38.9 kDa and the accession number is A0A059XIJ9. | |||
TMPY-00783 | Endoglin/CD105 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Endoglin/CD105 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 87.5 kDa and the accession number is A0A024R878. | |||
TMPY-00178 | Ebola virus EBOV (subtype Zaire, strain Mayinga 1976) Glycoprotein/GP-RBD (Receptor Binding Domain) Protein (hFc) | EBOV | HEK293 Cells |
Ebola virus EBOV (subtype Zaire, strain Mayinga 1976) Glycoprotein/GP-RBD (Receptor Binding Domain) Protein (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 57.6 kDa and the acc... | |||
TMPY-00041 | Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) Glycoprotein/GP1 Protein (His) | EBOV | Baculovirus Insect Cells |
Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) Glycoprotein/GP1 Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 52.3 kDa and the acce... | |||
TMPY-00347 | Doppel/PRND Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Doppel/PRND Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 41.2 kDa and the accession number is Q9UKY0. | |||
TMPY-00015 | Influenza A H10N8 (A/duck/Guangdong/E1/2012) Hemagglutinin/HA1 Protein (His) | H10N8 | HEK293 Cells |
Influenza A H10N8 (A/duck/Guangdong/E1/2012) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37 kDa and the accession number is I6PXD4. | |||
TMPY-00312 | Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) Nucleoprotein/NP Protein (His) | EBOV | E. coli |
Ebola virus EBOV (subtype Zaire, strain H.sapiens-wt/GIN/2014/Kissidougou-C15) Nucleoprotein/NP Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 15.6 kDa and the acc... | |||
TMPY-05801 | Podoplanin Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Podoplanin Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 11.78 kDa and the accession number is Q86YL7. | |||
TMPY-04608 | Influenza A H3N2 (A/Guangdong-Luohu/1256/2009) Hemagglutinin/HA1 Protein (His) | H3N2 | HEK293 Cells |
Influenza A H3N2 (A/Guangdong-Luohu/1256/2009) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is I6T542. | |||
TMPY-00172 | Influenza A H5N1 (A/goose/Guangdong/1/1996) Hemagglutinin/HA Protein (His) | H5N1 | Baculovirus Insect Cells |
Influenza A H5N1 (A/goose/Guangdong/1/1996) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 60.1 kDa and the accession number is Q9Q0U6. | |||
TMPY-02622 | Aldolase B Protein, Human, Recombinant (GST) | Human | E. coli |
The aldolase family members involved in metabolism and glycolysis are present in three isoforms: ALDOA, ALDOB, and ALDOC. Aldolases are differentially expressed in human tissues, and aberrant expression has been observed... | |||
TMPY-04796 | VEGFR2/KDR Protein, Human, Recombinant (Domain 2&3, His) | Human | HEK293 Cells |
VEGFR2/KDR Protein, Human, Recombinant (Domain 2&3, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 24.8 kDa and the accession number is P35968-1. | |||
TMPY-04589 | Influenza A H5N1 (A/Indonesia/5/2005) Hemagglutinin/HA-specific B cell probe Protein (His) | H5N1 | Baculovirus Insect Cells |
Influenza A H5N1 (A/Indonesia/5/2005) Hemagglutinin/HA-specific B cell probe Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 58.2 kDa and the accession number is AHJ... | |||
TMPY-00199 | Ebola virus EBOV (Subtype Sudan, strain Gulu) Glycoprotein/GP1 (mucin domain deleted) Protein (aa 1-320, His) | EBOV | Baculovirus Insect Cells |
Ebola virus EBOV (Subtype Sudan, strain Gulu) Glycoprotein/GP1 (mucin domain deleted) Protein (aa 1-320, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 33.8 kDa and the acce... | |||
TMPY-01503 | Influenza A H5N3 (A/duck/Hokkaido/167/2007) Hemagglutinin/HA1 Protein (His) | H5N3 | HEK293 Cells |
Influenza A H5N3 (A/duck/Hokkaido/167/2007) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is B1AHS0. | |||
TMPY-06948 | Influenza A H1N1 (A/New Caledonia/20/1999) Hemagglutinin/HA-specific B cell probe (Y108F, and aa 339-342 SIQS→QRET, His & Avi), Biotinylated | H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/New Caledonia/20/1999) Hemagglutinin/HA-specific B cell probe (Y108F, and aa 339-342 SIQS→QRET, His & Avi), Biotinylated is expressed in Baculovirus insect cells with His and Avi tag. The predicted mo... | |||
------------------------ More ------------------------ |
カタログ番号 | 製品名 | ||
---|---|---|---|
L2400 | Endocrinology-Hormone Compound Library | 784 compounds | |
A unique collection of 784 compounds targeting endocrine system for high throughput screening (HTS) and high content screening (HCS) for new drugs; | |||
L9700 | Endoplasmic Reticulum Stress Compound Library | 193 compounds | |
A unique collection of 193 endoplasmic reticulum stress (ER stress) related compounds used for high throughput screening (HTS) and high content screening (HCS); | |||
L2501 | Human Endogenous Metabolite Compound Library Plus | 1283 compounds | |
L2500 | Human Endogenous Metabolite Library | 499 compounds | |
A collection of 499 selected human endogenous metabolites for high throughput and high content screening. | |||
L2300 | Ion Channel Inhibitor Library | 931 compounds | |
A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery; | |||
L7700 | Neural Regeneration Compound Library | 524 compounds | |
A unique collection of 149 neuroregeneration related compounds for high throughput and high content screening; | |||
L9500 | Target-Focused Phenotypic Screening Library | 1796 compounds | |
A unique collection of 1796 annotated bioactive compounds with clear targets, suitable for phenotypic screening; | |||
L2610 | Neurotransmitter Receptor Compound Library | 1513 compounds | |
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening; | |||
L7110 | Anti-Hypertension Compound Library | 678 compounds | |
678 hypertension-related small molecules for high-throughput and high-content screening. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T16909 | Donafenib | Sorafenib (D3),Bay 43-9006 (D3),Sorafenib-d3 | Raf , VEGFR |
Donafenib (Bay 43-9006 (D3)) is a deuterium-labeled Sorafenib which is a multikinase inhibitor(IC50s: 6 nM, 20 nM, and 22 nM for Raf-1, B-Raf, and VEGFR-3, respectively). | |||
T10279 | Alfacalcidol-D6 | Others | |
Alfacalcidol-D6 is a deuterated Alfacalcidol. Alfacalcidol is a non-selective VDR activator medication. | |||
T11089 | Doxercalciferol-D3 | Others | |
Doxercalciferol-d3 is the deuterated form of Doxercalciferol and ACTS as vitamin D receptor activator (VDRA), which is a vitamin D2 analogue. | |||
T12035 | Midodrine D6 hydrochloride | Others | |
Midodrine D6 hydrochloride is a vasopressor/antihypotensive agent. | |||
T12587 | Pyridostigmine-d6 bromide | Pyridostigmine D6 bromide | Others |
Pyridostigmine D6 bromide is the deuterium labeled Pyridostigmine, which is a parasympathomimetic and a reversible inhibitor of cholinesterase. | |||
TMIH-0156 | Cis-Clopidogrel-MP-13C-d3 Derivative | ||
cis-Clopidogrel-MP-13C-d3 Derivative is the 13C and deuterated compound of cis-Clopidogrel-MP Derivative. | |||
TMIH-0210 | Eluxadoline-13C-d3 | ||
Eluxadoline-13C-d3 is the 13C and deuterated compound of Eluxadoline. Eluxadoline has a CAS number of 864825-13-8. | |||
T13300 | Vilazodone-d8 | Others | |
Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial. | |||
T19297 | Doxazosin D8 | UK 33274 D8 | Others |
Doxazosin D8 (UK 33274 D8) is a deuterium labeled Doxazosin (UK 33274).Doxazosin, a quinazoline derivative, selectively antagonizes postsynaptic AP1 adrenergic receptor. | |||
TMIH-0464 | Pyridoxal-d3 Hydrochloride | ||
Pyridoxal-d3 Hydrochloride is a deuterated compound of Pyridoxal Hydrochloride. | |||
TMIH-0039 | 3 Hydroxy Midostaurin Epimer 2-d5 | CGP52421 Epimer 2-d5 | |
3 Hydroxy Midostaurin Epimer 2-d5 is a deuterated compound of 3 Hydroxy Midostaurin Epimer 2.3 Hydroxy Midostaurin Epimer 2 has a CAS number of 155848-20-7. | |||
T11656 | Indoramin D5 | Indoramine D5,Wy-21901 D5 | CDK |
Indoramin D5 is a piperidine antiadrenergic agent. Indoramin D5 is deuterium labeled Indoramin. | |||
TMIH-0452 | Primidone-d5 | ||
Primidone-d5 is a deuterated compound of Primidone. | |||
T19119 | 3-Hydroxy Midostaurin-D5 | CGP52421-D5 | Others |
3-Hydroxy Midostaurin-D5 (CGP52421-D5) is a deuterium-labeled 3-Hydroxy Midostaurin which is a metabolite of PKC412. PKC412 effectively inhibits FMS-like tyrosine kinase-3 (FLT3) autophosphorylation (IC50s: 132 nM and 9.... | |||
TMIH-0423 | Penfluridol-d7 | ||
Penfluridol-d7 is a deuterated compound of Penfluridol. Penfluridol has a CAS number of 26864-56-2. Penfluridol is a highly potent antipsychotic. | |||
T11088 | Doxepin D3 Hydrochloride | Histamine Receptor | |
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, signi... | |||
TMIH-0315 | Lurasidone Inactive Metabolite 14283-d8 | 5α/6α-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers) | |
Lurasidone Inactive Metabolite 14283-d8 is a deuterated compound of Lurasidone Inactive Metabolite 14283.Lurasidone Inactive Metabolite 14283 has a CAS number of 186204-31-9. | |||
T71145 | Racecadotril-d5 | ||
Racecadotril-d5 is intended for use as an internal standard for the quantification of racecadotril by GC- or LC-MS. Racecadotril is a prodrug form of the neprilysin (NEP) inhibitor thiorphan. In vivo, racecadotril reduce... | |||
T11535 | Haloperidol D4 | Others | |
Haloperidol D4 is deuterium-labeled haloperidol. | |||
T70313 | Indoxyl Sulfate-d5 potassium salt | ||
Indoxyl sulfate-d5 is intended for use as an internal standard for the quantification of indoxyl sulfate by GC- or LC-MS. Indoxyl sulfate is a uremic toxin and a metabolite of tryptophan. It is formed via sulfation of in... | |||
T19407 | Lurasidone Metabolite 14326 D8 | Others | |
Lurasidone Metabolite 14326 D8 is the deuterium labeled Lurasidone Metabolite 14326. | |||
TMIH-0404 | O-Desmethyl Midostaurin-d5 | ||
O-Desmethyl Midostaurin-d5 is a deuterated compound of O-Desmethyl Midostaurin. | |||
TMIH-0488 | Reduced Haloperidol-d4 | ||
Reduced Haloperidol-d4 is a deuterated compound of Reduced Haloperidol. Reduced Haloperidol has a CAS number of 34104-67-1. | |||
TMIH-0200 | Donepezil-d7 Hydrochloride | ||
Donepezil-d7 Hydrochloride is a deuterated compound of Donepezil Hydrochloride. | |||
TMIH-0465 | Pyridoxamine-d3 dihydrochloride | ||
Pyridoxamine-d3 dihydrochloride is a deuterated compound of Pyridoxamine dihydrochloride. | |||
TMIH-0046 | 3-Indoleacrylic acid-d4 | ||
3-Indoleacrylic acid-d4 is a deuterated compound of 3-Indoleacrylic acid. 3-Indoleacrylic acid has a CAS number of 1204-06-4. 3-Indoleacrylic acid is a metabolite of tryptophan produced by Peptostreptococcus species. 3-I... | |||
T13195 | Trandolapril D5 | RU44570 D5 | Others |
Trandolapril D5 is a deuterium labeled Trandolapril. Trandolapril is an orally active inhibitor of angiotensin converting enzyme (ACE) for hypertension and congestive heart failure (CHF). | |||
T70174 | Pirlindole-d4 HCl | ||
Pirlindole-d4 is intended for use as an internal standard for the quantification of pirlindole by GC- or LC-MS. Pirlindole is a selective and reversible monoamine oxidase A (MAO-A) inhibitor. It is selective for MAO-A ov... | |||
T11072 | Dofetilide D4 | UK 68789 D4 | Others |
Dofetilide D4 (UK 68789 D4), a deuterium-labeled version of Dofetilide, is categorized as a Class III antiarrhythmic medication. | |||
TMIH-0466 | Pyridoxine-d3 | ||
Pyridoxine-d3 is a deuterated compound of Pyridoxine. | |||
TMIH-0515 | Samidorphan-d5 | ||
Samidorphan-d5 is a deuterated compound of Samidorphan. Samidorphan has a CAS number of 852626-89-2. | |||
TMIH-0463 | Pyridoxal-d3 | ||
Pyridoxal-d3 is a deuterated compound of Pyridoxal. | |||
TMIH-0467 | Pyridoxine-d3 Hydrochloride | ||
Pyridoxine-d3 Hydrochloride is a deuterated compound of Pyridoxine Hydrochloride. | |||
T13141 | Thalidomide D4 | Others | |
Thalidomide D4 is a deuterium labeled Thalidomide, has immunomodulatory, anti-inflammatory and anti-angiogenic cancer properties. | |||
TMIH-0038 | 3 Hydroxy Midostaurin Epimer 1-d5 | CGP52421 Epimer 1-d5 | |
3 Hydroxy Midostaurin Epimer 1-d5 is a deuterated compound of 3 Hydroxy Midostaurin Epimer 1. 3 Hydroxy Midostaurin Epimer 1 has a CAS number of 945260-14-0. | |||
TMIH-0551 | Tapentadol-d5 | ||
Tapentadol-d5 is a deuterated compound of Tapentadol. Tapentadol has a CAS number of 175591-23-8. | |||
T19185 | Aldosterone-d8 | Aldosterone D8 | Others |
Aldosterone D8, a deuterium-labeled variant of Aldosterone produced in the adrenal zona glomerulosa, regulates blood pressure. | |||
T12485 | Pirfenidone-d5 | AMR69 D5,Pirfenidone D5 | Others |
Pirfenidone D5 is a deuterium labeled Pirfenidone. Pirfenidone is an antifibrotic agent that attenuates CCL2 and CCL12 production in fibrocyte cells. | |||
T12036 | Midostaurin-D5 | PKC412-D5,CGP 41251-D5 | Others |
Midostaurin-D5 is a deuterium labeled Midostaurin. | |||
T11536 | Haloperidol (D4') | Haloperidol D4' | Others |
Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist. | |||
TMIH-0059 | 4-Pyridoxic Acid-d3 Hydrochloride | ||
4-Pyridoxic Acid-d3 Hydrochloride is a deuterated compound of 4-Pyridoxic Acid Hydrochloride. 4-Pyridoxic Acid Hydrochloride has a CAS number of 62511-95-9. | |||
T73715 | Risperidone-d4 | ||
Risperidone-d4, a deuterium-labeled version of Risperidone, acts as a potent antagonist of the dopamine D2 and serotonin 5-HT2 receptors, and inhibits P-Glycoprotein, displaying Ki values of 5.9 nM and 4.8 nM for the dop... | |||
TMIH-0420 | Paliperidone-d4 | ||
Paliperidone-d4 is a deuterated compound of Paliperidone. Paliperidone has a CAS number of 144598-75-4. Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schi... | |||
TMID-0034 | Haloperidol-d4 TFA | ||
Haloperidol-d4 TFA is a deuterated compound of Haloperidol TFA. | |||
TMIJ-0029 | Sulfadoxine-d4 | ||
Sulfadoxine-d4 is a deuterated compound of Sulfadoxine. Sulfadoxine has a CAS number of 2447-57-6. Sulfadoxine is a broad-spectrum sulfanilamide and a synthetic analog of para-aminobenzoic acid (PABA) with bacteriostatic... | |||
T11655 | Indomethacin-D4 | Indometacin-D4 | CDK |
Indomethacin-D4 is a deuterium labeled Indomethacin. Indomethacin is a potent and nonselective inhibitor of COX1 and COX2, with IC50s of 18 nM and 26 nM for human COX-1 and COX-2, respectively, in CHO cells. | |||
TNU1192 | N1-Methyl-d3-pseudouridine | ||
N1-Methyl-d3-pseudouridine is a useful organic compound for research related to life sciences and the catalog number is TNU1192. | |||
TMIH-0109 | Bempedoic acid-d4 | ||
Bempedoic acid-d4 is a deuterated compound of Bempedoic acid. Bempedoic acid has a CAS number of 738606-46-7. ETC-1002, also known as ESP-55016 and Bempedoic acid, is an orally available, once-daily LDL-C lowering small ... | |||
TMIH-0049 | 3-O-Methyldopa-d3 | ||
3-O-Methyldopa-d3 is a deuterated compound of 3-O-Methyldopa. 3-O-Methyldopa has a CAS number of 300-48-1. | |||
TMIH-0281 | Indobufen-d5 | ||
Indobufen-d5 is a deuterated compound of Indobufen. Indobufen has a CAS number of 63610-08-2. Indobufen is an inhibitor of platelet aggregation and is a reversible platelet cyclooxygenase (Cox) activity inhibitor. Indobu... | |||
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