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Search Results for " iNOS "

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281

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174

天然化合物

25

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1

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カタログ番号 製品名 別名 ターゲット
T83625 iNOS-IN-14 3-bromo-1H-indazole-7-carbonitrile NOS
iNOS-IN-14 (3-bromo-1H-indazole-7-carbonitrile) is a potent nitric oxide synthase (NOS) inhibitor that inhibits the NADPH oxidase activity of nNOS.
T72638 iNOS inhibitor-10 NO Synthase
iNOS Inhibitor-10, with an IC50 of 65 nM, exhibits antiproliferative effects on triple-negative breast cancer cells [1].
T62849 iNOS-IN-2
iNOS-IN-2 (Compound 53) is a potent inducible nitric oxide synthase (iNOS) protein down-regulator. iNOS-IN-2 effectively inhibits NO production (IC50: 6.4 μM). iNOS-IN-2 can be used in studies of chronic inflammation.
T62987 iNOs-IN-1
iNOs-IN-1 (YPW) is a potent inhibitor of inducible nitric oxide synthase (iNOS) with anti-inflammatory effects. iNOs-IN-1 significantly inhibits IL-6 and iNOS expression in a dose-dependent manner in murine macrophages, ...
T63261 iNOs-IN-3
iNOs-IN-3 is an orally active nitric oxide synthase (iNOS) inhibitor with an IC50 value of 3.342 μM that exhibits anti-inflammatory effects and can be used to study LPS-induced acute lung injury (ALI).
T63104 iNOS/PGE2-IN-1
iNOS/PGE2-IN-1 is an iNOS/PGE2 inhibitor and a potent anti-inflammatory agent. iNOS/PGE2-IN-1 exhibits an inhibitory effect on LPS-induced NO production and has a low ulcerogenic potential.
T21700 NOS-IN-1  2-Imino-4-methylpiperidine (acetate) NOS
NOS-IN-1 (2-Imino-4-methylpiperidine acetate) is a potent and orally active inhibitor of NO synthase (NOS) isoforms. NOS-IN-1 exhibits IC50s of 0.1 μM, 0.2 μM, and 1.1μM for human iNOS (hiNOS), hnNOS and heNOS, respectiv...
T19916 TRIM 1-(2-Trifluoromethylphenyl)imidazole NOS
TRIM (1-(2-Trifluoromethylphenyl)imidazole) is an inhibitor of nNOS.
T1127 Beclometasone dipropionate Beclovent,Beclomethasone dipropionate,Beconase,Vancenase Glucocorticoid Receptor
Beclometasone dipropionate (Vancenase) is the dipropionate ester of a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. After cell surface receptor attachment and cell entry, beclomethasone...
T22419 S-Methylisothiourea sulfate (S)-Methylisothiourea sulfate NOS , NO Synthase , HSV
S-Methylisothiourea sulfate ((S)-Methylisothiourea sulfate) is a potent and selective inhibitor of iNOS and exerts beneficial effects in rodent models of septic shock[1].
T23046 N-tert-butyl-α-Phenylnitrone (Z)-N-benzylidene-2-Methylpropan-2-aMine oxide ROS , COX
N-tert-butyl-α-Phenylnitrone ((Z)-N-benzylidene-2-Methylpropan-2-aMine oxide) inhibits COX2 catalytic activity. N-tert-butyl-α-Phenylnitrone((Z)-N-benzylidene-2-Methylpropan-2-aMine oxide) possesses potent reactive oxyge...
T4509 Inositol nicotinate Inositol niacinate,Hexanicotol,Myo-Inositol hexanicotinate,Mesotal,Dilexpal,Inositol hexanicotinate Others
Inositol nicotinate (Mesotal) has the effect of lowering cholesterol and expanding peripheral blood vessels for hypercholesterolemia and atherosclerosis.
T7621 6-​Thioinosine 6-Mercaptopurine riboside,6TI Nucleoside Antimetabolite/Analog
6-Thioinosine (6TI) is a purine antimetabolite, acts as an anti-adipogenesis agent.
T27083 Crebinostat Epigenetic Reader Domain , Histone Acetyltransferase , HDAC
Crebinostat is a potent histone deacetylase (HDAC) inhibitor, inhibiting HDAC1, HDAC2, HDAC3, and HDAC6 with IC50s of 0.7 nM, 1.0 nM, 2.0 nM, and 9.3 nM, respectively.Crebinostat increases the density of synapsin-1 punct...
T12516 Polyinosinic-polycytidylic acid sodium Poly(I:C) sodium Apoptosis , Others , TLR
Polyinosinic-polycytidylic acid sodium (Poly(I:C) sodium) is a synthetic analog of double-stranded RNA and an agonist of toll-like receptor 3 (TLR3) and retinoic acid inducible gene I (RIG-I)-like receptors (RIG-I and MD...
T3661 Citarinostat ACY241,HDAC-IN-2 HDAC
ACY-241, also known as Citarinostat (ACY241), is a potent, selective and orally available histone deacetylase (HDAC) inhibitor, with potential antineoplastic activity. Upon oral administration, ACY-241 inhibits the activ...
T6233 Entinostat SNDX-275,MS-275 Apoptosis , HDAC , Autophagy
Entinostat (MS-275) (MS-275) is an inhibitor of HDACs that inhibits HDAC1 and HDAC3 (IC50s: 0.18/0.74 μM).
T16729 Remetinostat SHP-141 HDAC
Remetinostat (SHP-141), a hydroxamic acid-based inhibitor of histone deacetylase enzymes, is currently being developed for the treatment of cutaneous T-cell lymphoma.
T4477 Domatinostat tosylate 4SC-202 tosylate,4SC-202 Apoptosis , HDAC
Domatinostat tosylate (4SC-202) is a selective inhibitor of class I HDAC for HDAC1/2/3 (IC50: 1.20/1.12/0.57 μM). It also displays inhibitory activity against Lysine-specific demethylase 1 (LSD1).
T6055 Quisinostat JNJ-26481585 Apoptosis , HDAC , Autophagy
Quisinostat (JNJ-26481585) (JNJ-26481585) is a novel second-generation HDAC inhibitor with highest potency for HDAC1 with IC50 of 0.11 nM, modest potent to HDACs 2, 4, 10, and 11; greater than 30-fold selectivity against...
T4481 Tucidinostat HBI-8000,Chidamide,CS 055 HDAC
Tucidinostat (Chidamide) is an effective and orally bioavailable HDAC enzymes class I (HDAC1/2/3) and class IIb (HDAC10) inhibitor, with IC50s of 95, 160, 67 and 78 nM, less active on HDAC8/11 (IC50: 733/432 nM), and sho...
T6279L Givinostat hydrochloride ITF2357 hydrochloride,Givinostat HCl,ITF2357,ITF 2357,ITF-2357,ITF2357 HCl HDAC
Givinostat hydrochloride (ITF2357 hydrochloride) is an inhibitor of HDAC with IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively. Givinostat hydrochloride exhibits anti-inflammatory, anti-angiogenic, and antineopla...
T2454 Dacinostat NVP-LAQ824,LAQ824 HDAC , Autophagy
LAQ824 (Dacinostat (NVP-LAQ824)) is a novel HDAC inhibitor with IC50 of 32 nM and is an activator of the p21 promoter.
T6481 Droxinostat NS 41080 Apoptosis , HDAC
Droxinostat (NS 41080) is a selective inhibitor of HDAC, mostly for HDACs 6 and 8 with IC50 of 2.47 μM and 1.46 μM, greater than 8-fold selective against HDAC3 and no inhibition to HDAC1, 2, 4, 5, 7, 9, and 10.
T1852 Rac-Belinostat NSC726630,PXD101,PX-105684 HDAC
Rac-Belinostat (PX-105684) is a novel hydroxamic acid-type histone deacetylase (HDAC) inhibitor with antineoplastic activity. Belinostat targets HDAC enzymes, thereby inhibiting tumor cell proliferation, inducing apoptos...
T2383 Panobinostat NVP-LBH589,LBH589 Apoptosis , HIV Protease , HDAC , Autophagy
Panobinostat (NVP-LBH589) is a broad-spectrum HDAC inhibitor (IC50=5 nM) with oral activity and non-selectivity. Panobinostat has antitumor activity and induces apoptosis and autophagy.
T2078 Fimepinostat CUDC-907,PI3K/HDAC Inhibitor,CUDC 907 Apoptosis , PI3K , HDAC
Fimepinostat (CUDC 907) is an orally bioavailable inhibitor of both phosphoinositide 3-kinase (PI3K) class I and pan-histone deacetylase (HDAC) enzymes, with potential antineoplastic activity. Upon oral administration, C...
T2512 Mocetinostat MGCD0103,MG0103 Apoptosis , HDAC , Autophagy
Mocetinostat (MG0103) is an orally available HDAC inhibitor with most potency for HDAC1 (IC50: 0.15 μM), 2- to 10- fold selectivity against HDAC2/3/11.
T4370 Resminostat hydrochloride 4SC-201 hydrochloride,RAS2410 hydrochloride HDAC
Resminostat hydrochloride (RAS2410 hydrochloride) is an effective inhibitor of HDAC1/HDAC3/HDAC6 (IC50: 42.5/50.1/71.8 nM), respectively, and shows less potent activities against HDAC8 (IC50: 877 nM).
TNU0810 2′-C-Methyl-6-O-methylinosine 2′-C-Methyl-6-O-methylinosine Nucleoside Antimetabolite/Analog
2′-C-Methyl-6-O-methylinosine (2′-C-Methyl-6-O-methylinosine) is a hypoxanthine analog with a wide range of physical activities for the study of a variety of tumor diseases.
TNU0187 2',5-Difluoro-2'-deoxy-1-arabinosyluracil 2'-Deoxy-2'-fluoro-5-fluoro-arabinouridine Nucleoside Antimetabolite/Analog
2',5-Difluoro-2'-deoxy-1-arabinosyluracil (2'-Deoxy-2'-fluoro-5-fluoro-arabinouridine) is a urinary pyrimidine nucleoside analogue with potential antiepileptic and antihypertensive activity, which can be used to study an...
T1583 Vorinostat MK0683,suberoylanilide hydroxamic acid,SAHA Apoptosis , Mitophagy , Virus Protease , HDAC , Autophagy
Vorinostat (SAHA) is a pan-histone deacetylase (HDAC) inhibitor (IC50=10 nM) with inhibitory activity against HDAC1/2/3/6/7/11. Vorinostat has antitumor activity, induces cell differentiation, blocks the cell cycle and i...
T0020 Sodium 4-aminosalicylate dihydrate Sodium 4-Aminosalicylate,4-Amino-salicylic acid sodium salt Free radical scavengers , NF-κB , Antibacterial , Antibiotic
Sodium 4-aminosalicylate dihydrate (4-Amino-salicylic acid sodium salt) is the sodium salt form of aminosalicylic acid, an analog of para-aminobenzoic acid (PABA) with antitubercular activity. Sodium 4-aminosalicylate di...
T0598 Iminostilbene Dibenzazepine Others
Iminostilbene (Dibenzazepine) (Dibenzazepine) is a chemical precursor of carbamazepine which is used primarily in the treatment of epilepsy and neuropathic pain.
T0431 Abexinostat CRA 24781,PCI24781,PCI-24781,PCI 24781,CRA 024781 HDAC
PCI-24781 (Abexinostat (PCI24781)) is a new pan-HDAC inhibitor mainly targeting HDAC1 (Ki: 7 nM), also have moderate inhibitory for HDACs 2, 3, 6, and 10 and greater than 40-fold selectivity against HDAC8. Phase 1/2.
T17028 Tefinostat CHR-2845 HDAC
Tefinostat (CHR-2845) is a potent monocyte/macrophage-targeted histone deacetylase (HDAC) inhibitor. Tefinostat is cleaved to the active acid CHR-2847 by the intracellular esterase human carboxylesterase-1 (hCE-1).Tefino...
T3614 Inosine pranobex Groprinosin,Isoprinosine,Immunovir,Delimmun IL Receptor , HIV Protease
Inosine pranobex (Delimmun) has a number of immunomodulatory effects, including inducing T-lymphocyte differentiation, augmenting macrophage and NK cell functions, and stimulating IL-2 production. Through these effects a...
T6362 Domatinostat 4SC202,4SC 202,4SC-202 (free base),4SC-202 Apoptosis , HDAC
Domatinostat (4SC202) is a selective class I HDAC inhibitor with IC50 of 1.20 μM, 1.12 μM, and 0.57 μM for HDAC1, HDAC2, and HDAC3, respectively. Also displays inhibitory activity against Lysine specific demethylase 1 (L...
T6865 Quisinostat dihydrochloride Quisinostat 2HCl,Quisinostat (JNJ-26481585) 2HCl,JNJ26854165(Quisinostat) 2HCl,JNJ-26481585 2HCl Apoptosis , HDAC , Autophagy
Quisinostat dihydrochloride (JNJ26854165(Quisinostat) 2HCl) is a novel second-generation HDAC inhibitor with highest potency for HDAC1 with IC50 of 0.11 nM in a cell-free assay, modest potent to HDACs 2, 4, 10, and 11; g...
T1890 Pracinostat SB939 Apoptosis , HDAC
Pracinostat (SB939) is a novel HDAC inhibitor with improved in vivo properties compared to other HDAC inhibitors currently in Clinicalal trials, allowing oral dosing. Data demonstrate that Pracinostat is a potent and eff...
T6279 Givinostat hydrochloride monohydrate ITF2357,ITF-2357 hydrochloride monohydrate,Givinostat,Gavinostat hydrochloride monohydrate HDAC
Givinostat hydrochloride monohydrate (ITF2357) is an HDAC inhibitor.
T8551 Nitrobenzylthioinosine NBMPR AChR , Adenosine Receptor
Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
T71138L Binospirone MDL 73005EF 5-HT Receptor
Binospirone (MDL 73005EF) is a 5-HT1A receptor agonist with anxiolytic activity used in the study of glaucoma and movement disorders associated with neurologic dysfunction.
TNU0442 2’-beta-C-Methyl inosine 2'-C-Methylinosine Antiviral , DNA/RNA Synthesis
2’-beta-C-Methyl inosine (2’-C-Methylinosine) is an HCV RNA polymerase inhibitor with antiviral activity and is being studied for the treatment of hepatitis C virus infection.
T23171 Polyinosinic-polycytidylic acid Poly(I:C) TLR
Polyinosinic-polycytidylic acid (Poly(I:C)) is a double-stranded RNA (dsRNA) and a TLR3 agonist. Polyinosinic-polycytidylic acid induces natural immunity in mammals.
T9835 4-QUinolinecarboxamide, N-[3-[[[2-[4-(aminosulfonyl)phenyl]ethyl]amino]carbonyl]phenyl]-1,2-dihydro-2-oxo- Others
4-QUinolinecarboxamide, N-[3-[[[2-[4-(aminosulfonyl)phenyl]ethyl]amino]carbonyl]phenyl]-1,2-dihydro-2-oxo- is an amine.
T2489 Ricolinostat ACY-1215,Rocilinostat Apoptosis , HDAC
Ricolinostat (Rocilinostat) is an orally bioavailable, specific inhibitor of histone deacetylase 6 (HDAC6) with potential antineoplastic activity.
T8517 Belinostat PX105684,PXD101,PXD-101 HDAC , Autophagy
Belinostat (PXD101) is an inhibitor of hydroxamic acid-type histone deacetylase (HDAC, IC50 of 27 nM in HeLa cell extracts),and with antineoplastic activity.
T1296 4-Aminosalicylic acid Aminosalicylic acid,4-aminosalicylate,para-aminosalicylic acid,Aminopar NF-κB , Lipoxygenase , COX , Glutathione Peroxidase , Antibacterial , Antibiotic
4-Aminosalicylic acid (para-aminosalicylic acid) is an analog of para-aminobenzoic acid (PABA) with antitubercular activity.
T125614 Clematiunicinoside D
Clematiunicinoside D is a useful organic compound for research related to life sciences. The catalog number is T125614 and the CAS number is 1699748-21-4.

Compounds

iNOS-IN-14
T83625
Synonym: 3-bromo-1H-indazole-7-carbonitrile
Target: NOS
iNOS inhibitor-10
T72638
Synonym:
Target: NO Synthase
iNOS-IN-2
T62849
Synonym:
Target:
iNOs-IN-1
T62987
Synonym:
Target:
iNOs-IN-3
T63261
Synonym:
Target:
iNOS/PGE2-IN-1
T63104
Synonym:
Target:
NOS-IN-1 
T21700
Synonym: 2-Imino-4-methylpiperidine (acetate)
Target: NOS
TRIM
T19916
Synonym: 1-(2-Trifluoromethylphenyl)imidazole
Target: NOS
Beclometasone dipropionate
T1127
Synonym: Beclovent,Beclomethasone dipropionate,Beconase,Vancenase
Target: Glucocorticoid Receptor
S-Methylisothiourea sulfate
T22419
Synonym: (S)-Methylisothiourea sulfate
Target: NOS, NO Synthase, HSV
N-tert-butyl-α-Phenylnitrone
T23046
Synonym: (Z)-N-benzylidene-2-Methylpropan-2-aMine oxide
Target: ROS, COX
Inositol nicotinate
T4509
Synonym: Inositol niacinate,Hexanicotol,Myo-Inositol hexanicotinate,Mesotal,Dilexpal,Inositol hexanicotinate
Target: Others
6-​Thioinosine
T7621
Synonym: 6-Mercaptopurine riboside,6TI
Target: Nucleoside Antimetabolite/Analog
Crebinostat
T27083
Synonym:
Target: Epigenetic Reader Domain, Histone Acetyltransferase, HDAC
Polyinosinic-polycytidylic acid sodium
T12516
Synonym: Poly(I:C) sodium
Target: Apoptosis, Others, TLR
Citarinostat
T3661
Synonym: ACY241,HDAC-IN-2
Target: HDAC
Entinostat
T6233
Synonym: SNDX-275,MS-275
Target: Apoptosis, HDAC, Autophagy
Remetinostat
T16729
Synonym: SHP-141
Target: HDAC
Domatinostat tosylate
T4477
Synonym: 4SC-202 tosylate,4SC-202
Target: Apoptosis, HDAC
Quisinostat
T6055
Synonym: JNJ-26481585
Target: Apoptosis, HDAC, Autophagy
Tucidinostat
T4481
Synonym: HBI-8000,Chidamide,CS 055
Target: HDAC
Givinostat hydrochloride
T6279L
Synonym: ITF2357 hydrochloride,Givinostat HCl,ITF2357,ITF 2357,ITF-2357,ITF2357 HCl
Target: HDAC
Dacinostat
T2454
Synonym: NVP-LAQ824,LAQ824
Target: HDAC, Autophagy
Droxinostat
T6481
Synonym: NS 41080
Target: Apoptosis, HDAC
Rac-Belinostat
T1852
Synonym: NSC726630,PXD101,PX-105684
Target: HDAC
Panobinostat
T2383
Synonym: NVP-LBH589,LBH589
Target: Apoptosis, HIV Protease, HDAC, Autophagy
Fimepinostat
T2078
Synonym: CUDC-907,PI3K/HDAC Inhibitor,CUDC 907
Target: Apoptosis, PI3K, HDAC
Mocetinostat
T2512
Synonym: MGCD0103,MG0103
Target: Apoptosis, HDAC, Autophagy
Resminostat hydrochloride
T4370
Synonym: 4SC-201 hydrochloride,RAS2410 hydrochloride
Target: HDAC
2′-C-Methyl-6-O-methylinosine
TNU0810
Synonym: 2′-C-Methyl-6-O-methylinosine
Target: Nucleoside Antimetabolite/Analog
2',5-Difluoro-2'-deoxy-1-arabinosyluracil
TNU0187
Synonym: 2'-Deoxy-2'-fluoro-5-fluoro-arabinouridine
Target: Nucleoside Antimetabolite/Analog
Vorinostat
T1583
Synonym: MK0683,suberoylanilide hydroxamic acid,SAHA
Target: Apoptosis, Mitophagy, Virus Protease, HDAC, Autophagy
Sodium 4-aminosalicylate dihydrate
T0020
Synonym: Sodium 4-Aminosalicylate,4-Amino-salicylic acid sodium salt
Target: Free radical scavengers, NF-κB, Antibacterial, Antibiotic
Iminostilbene
T0598
Synonym: Dibenzazepine
Target: Others
Abexinostat
T0431
Synonym: CRA 24781,PCI24781,PCI-24781,PCI 24781,CRA 024781
Target: HDAC
Tefinostat
T17028
Synonym: CHR-2845
Target: HDAC
Inosine pranobex
T3614
Synonym: Groprinosin,Isoprinosine,Immunovir,Delimmun
Target: IL Receptor, HIV Protease
Domatinostat
T6362
Synonym: 4SC202,4SC 202,4SC-202 (free base),4SC-202
Target: Apoptosis, HDAC
Quisinostat dihydrochloride
T6865
Synonym: Quisinostat 2HCl,Quisinostat (JNJ-26481585) 2HCl,JNJ26854165(Quisinostat) 2HCl,JNJ-26481585 2HCl
Target: Apoptosis, HDAC, Autophagy
Pracinostat
T1890
Synonym: SB939
Target: Apoptosis, HDAC
Givinostat hydrochloride monohydrate
T6279
Synonym: ITF2357,ITF-2357 hydrochloride monohydrate,Givinostat,Gavinostat hydrochloride monohydrate
Target: HDAC
Nitrobenzylthioinosine
T8551
Synonym: NBMPR
Target: AChR, Adenosine Receptor
Binospirone
T71138L
Synonym: MDL 73005EF
Target: 5-HT Receptor
2’-beta-C-Methyl inosine
TNU0442
Synonym: 2'-C-Methylinosine
Target: Antiviral, DNA/RNA Synthesis
Polyinosinic-polycytidylic acid
T23171
Synonym: Poly(I:C)
Target: TLR
4-QUinolinecarboxamide, N-[3-[[[2-[4-(aminosulfonyl)phenyl]ethyl]amino]carbonyl]phenyl]-1,2-dihydro-2-oxo-
T9835
Synonym:
Target: Others
Ricolinostat
T2489
Synonym: ACY-1215,Rocilinostat
Target: Apoptosis, HDAC
Belinostat
T8517
Synonym: PX105684,PXD101,PXD-101
Target: HDAC, Autophagy
4-Aminosalicylic acid
T1296
Synonym: Aminosalicylic acid,4-aminosalicylate,para-aminosalicylic acid,Aminopar
Target: NF-κB, Lipoxygenase, COX, Glutathione Peroxidase, Antibacterial, Antibiotic
Clematiunicinoside D
T125614
Synonym:
Target:
1 2 3 4 5 6
カタログ番号 製品名 別名 ターゲット
T6S1665 Irisflorentin Others , NO Synthase
1. Irisflorentin blocks apoptosis pathways, by exerting its effects by promoting rpn-3 expression to enhance the activity of proteasomes and down-regulating egl-1 expression. 2. Irisflorentin has anti-inflammatory mechan...
T2738 Dehydroandrographolide NOS , Influenza Virus
Dehydroandrographolide is a natural compound extracted from herbal medicine Andrographis paniculata (Burm f) Nees.
TN6951 Ethyl linoleate Others
Ethyl linoleate is a natural product.
T6S1572 Sauchinone ERK , p38 MAPK , NF-κB
1. Sauchinone is a useful adjunctive treatment for bacterial infection. 2. Sauchinone, an active lignan found in Saururus chinensis, to regulate the activation of HSCs, to prevent liver fibrosis, and to inhibit oxidative...
TN2139 Regaloside B NOS , COX , NO Synthase
Regaloside B, a phenylpropanoid isolated from Lilium longiflorum, exhibits anti-inflammatory activity by inhibiting the expression of iNOS (inducible nitric oxide synthase) and COX-2 (cyclooxygenase-2).
T0610 Piceatannol trans-Piceatannol,Astringenin Apoptosis , Serine/threonin kinase , PKA , Syk , PKC , Autophagy
Piceatannol (Astringenin) is an anti-inflammatory, immunomodulatory and antiproliferative agent. It inhibits p56lck and syk protein tyrosine kinases and inhibits NF-κB activation and gene expression of TNF-induced. It is...
T5S0045 Isofraxidin 6,8-Dimethoxyumbelliferone,Phytodolor MMP , ERK , p38 MAPK , TLR , COX
1. Isofraxidin (Phytodolor) protects leukemia cells from radiation-induced apoptosis via ROS/mitochondria pathway in a p53-independent manner. 2. Isofraxidin has a protective effect against LPS-induced ALI, and the prote...
T1079 Metronidazole Flagyl,Metronidazol,Anagiardil Apoptosis , NADPH , Hydrogenase , Antibacterial , Antibiotic , Parasite , Antifection
Metronidazole (Metronidazol) is a synthetic nitroimidazole derivative with antiprotozoal and antibacterial activities.
TCS2170 2,5-Dihydroxyacetophenone Quinacetophenone,2-Acetylhydroquinone,2-5-dihydroxyacetophenone,Acetylhydroquinone,DHAP ERK , NF-κB , Tyrosinase
1. 2,5-Dihydroxyacetophenone (Quinacetophenone) possess anti-anxiety, and neuroprotective qualities. 2. 2,5-Dihydroxyacetophenone (Quinacetophenone) reatment can induce a sustained activation of JNK, ERK1/2, and p38 MAPK...
TN1109 3-O-Acetyl-16α-hydroxydehydrotrametenolic acid 3-O-Acetyl-16 alpha-hydroxydehydrotrametenolic acid NOS , NO Synthase , Prostaglandin Receptor
3-O-Acetyl-16α-hydroxydehydrotrametenolic acid (3-O-Acetyl-16 alpha-hydroxydehydrotrametenolic acid) shows anti-inflammatory activity, it can inhibit NO production and iNOS expression in LPS-stimulated Raw264.7 cells.
T4897 Inosine-5'-triphosphate trisodium salt ITP,Inosine 5'-triphosphate trisodium salt Others , Endogenous Metabolite
Inosine-5'-triphosphate trisodium salt (ITP) is used in studies on the impact of deamination of ATP and GTP by various enzymes and chemical processes. Inosine-5'-triphosphate trisodium salt (ITP) may be used as a substra...
TN3861 Dihydropinosylvin Anti-infection
Dihydropinosylvinin is an phytoalexin, it shows antifungal activity against Cladosporium cladosporioides, Botryodiplodia theobromae, Aspergillus niger and Penicillium schlerotgenum, it also exhibits strong antibacterial ...
T3755 Pinostilbene Others
Pinostilbene obviously attenuates the phosphorylation of c-Jun and JNK triggered by 6-OHDA.
TN1808 Isovitexin 2''-O-arabinoside Others
Isovitexin 2''-O-arabinoside is a flavonoid found in the alfalfa plant.
T5S2228 6‴-Feruloylspinosin 6'''-Feruloylspinosin NF-κB
6‴-Feruloylspinosin (6'''-Feruloylspinosin) may possess anti-inflammatory activity.
T4685 INOSINIC ACID Inosine 5′-monophosphate,IMP,I-5'-P Endogenous Metabolite
Inosinic acid (IMP) is a purine nucleotide which has hypoxanthine as the base and one phosphate group esterified to the sugar moiety. Inosinic acid is a nucleotide present in muscle and other tissues. It is formed by the...
T4818 Thyminose 2-Deoxy-D-ribose,2-Deoxy-D-arabinose,2-Deoxy-D-erythropentose Others , Endogenous Metabolite
Thyminose (2-Deoxy-D-arabinose) induces Apoptosis by inhibiting the synthesis and increasing the efflux of glutathione.
T5S1679 Acetylshengmanol Arabinoside Acetylcimigenol 3-O-alpha-L-arabinopyran Others
Acetylcimigenol 3-O-alpha-L-arabinopyranoside is an extract derived from Cimicifuga.
TN6910 Aloinoside B 11-o-Rhamnosylaloin B
Aloinoside B (11-o-Rhamnosylaloin B) is a glycoside from aloe vera.
T5796 Plantainoside D Isoplantamajoside RAAS , PKC
Plantainoside D (Isoplantamajoside) shows potent antioxidative effects as those of ascorbic acid, it shows angiotensin-converting enzyme (ACE) inhibitory inhibitory activity in vitro with the IC(50) value of 2.17 mM, it ...
T0437 Inosine INO 495,NSC 20262 ROS , Endogenous Metabolite , Adenosine Receptor
Inosine (NSC-20262) is a purine nucleoside that has hypoxanthine linked by the N9 nitrogen to the C1 carbon of ribose. It has immunomodulatory, neuroprotective, and analgesic properties.
T1709 2'-Deoxyinosine Guanine deoxyriboside,Deoxyinosine Others , Endogenous Metabolite
2'-Deoxyinosine (Guanine deoxyriboside) inhibits the growth of human colon-carcinoma cell lines and is associated with purine nucleoside phosphorylase (PNP) deficiency.
T2S0112 Yibeinoside A Sinpeinine-3-O-β-glucoside Others
Yibeinoside A (Sinpeinine-3-O-β-glucoside) is an alkaloid from Fritillaria pallidiflora.
TN1487 Chrysin 6-C-arabinoside 8-C-glucoside Others
Chrysin 6-C-arabinoside 8-C-glucoside and chrysin-6-C-glucosyl-8-C-arabinoside are α±-glucosidase inhibitors, α±-glucosidase inhibitors are widely used in the treatment of type 2 diabetes.
T8144 Raffinose Melitose,Melitriose Others , Endogenous Metabolite
Raffinose (Melitriose) is an indigestible short-chain oligosaccharide, a trisaccharide composed of galactose, glucose and fructose, found in many plants. It can be hydrolyzed by α-galactosidase (α-GAL) to D-galactose and...
T8012 Scyllo-Inositol Scyllitol Beta Amyloid , Endogenous Metabolite
Scyllo-Inositol (Scyllitol) is one of the inositol stereoisomers, rare in the nature, and expected as a promising disease-modifying therapeutic agent for Alzheimer's disease.
TN1488 Chrysin 6-C-glucoside 8-C-arabinoside Others
Chrysin 6-C-glucoside 8-C-arabinoside and Chrysin-6-C-arabinosyl-8-C-glucoside are α±-glucosidase inhibitors, α±-glucosidase inhibitors are widely used in the treatment of type 2 diabetes.
TN2083 Pinostrobin chalcone
Pinostrobin chalcone, a chalcone analog isolated from the leguminous plant, Mucuna pruriens, exhibits anticancer activity with an IC50 value of 20.42±2.23 μg/mL against MDA-MB-231 and 22.51±0.42 μg/mL against the HT-29 c...
T13752 L-(+)-Arabinose Endogenous Metabolite
L-(+)-Arabinose selectively inhibits intestinal sucrase activity in a non-competitive manner, inhibiting glucose elevation caused by sucrose intake.
T0421 I-Inositol Inositol,myo-Inositol,meso-Inositol Endogenous Metabolite
i-Inositol (myo-Inositol) is a intracellular phosphate compound, involved in cell signaling and may stimulate tumor cell differentiation.
T4875 Palatinose hydrate 6-O-α-D-Glucopyranosyl-D-fructose, Isoma Others , Endogenous Metabolite
Palatinose hydrate (6-O-α-D-Glucopyranosyl-D-fructose, Isoma) is a disaccharide having an α(1→6) linkage between D-glucose and D-fructose and is similar to sucrose in its physicochemical properties. It is produced from s...
T5073 Inosine 5'-monophosphate disodium salt hydrate Inosine 5'-monophosphate disodium salt,5'-IMP-Na2,Disodium 5'-inosinate monohydrate Others , Endogenous Metabolite
Inosine 5'-monophosphate disodium salt hydrate (Inosine 5'-monophosphate disodium salt), or inosinic acid, is the ribonucleotide of hypoxanthine and the first nucleotide formed during purine synthesis.
T5915 D-chiro-Inositol D-(+)-CHIRO-INOSITOL Endogenous Metabolite
D-chiro-Inositol (D-(+)-CHIRO-INOSITOL) is an epimer of myo-inositol that is found in certain mammalian glycosylphosphatidylinositol protein anchors and inositol phosphoglycans possessing insulin-like bioactivity.
T9076 Spinosad Others
Spinosad is a naturally-occurring insecticide found in the the soil bacterium S. spinosa. It is a mixture of the macrocyclic lactones spinosyn A and spinosyn D, which act as agonists of insect nicotinic acetylcholinester...
T67867 Mycaminosyltylonolide Antibacterial
Mycaminosyltylonolide is a macrolide antibiotic that is tylonolide having a beta-D-mycaminosyl residue attached at position 5. Mycaminosyltylonolide is a potent antibiotic with antibacterial activity and inhibits lucifer...
T21495 Spinosyn A Others
Spinosyn A is a polyketide-derived macrolide produced by Saccharopolyspora spinosa and is an active ingredient in several commercial insecticides.
T19083 1-Methylinosine N1-Methylinosine,Inosine, 1-methyl Nucleoside Antimetabolite/Analog , Endogenous Metabolite
1-Methylinosine (N1-Methylinosine) is a modified nucleotide found at position 37 in tRNA 3' to the anticodon of eukaryotic tRNA and has a role as a metabolite.
TN1836 Kudinoside D LDL , AMPK , PPAR
Kudinoside D exerts anti-adipogenic effects through modulation of adipogenic transcription factors via AMPK signaling pathway.
TN6745 PALATINOSE TNP-470,Isomaltulose Others
PALATINOSE (TNP-470) is a natural occurring disaccharide composed of alpha-1,6-linked glucose and fructose。 PALATINOSE has a beneficial effect on liver metabolic functions and might therefore be a good substitute for suc...
TMS1830 Disodium 5'-inosinate Disodium Inosinate,Sodium Inosinate,5'-IMP disodium salt Others
Disodium 5'-inosinate (5'-IMP disodium salt) is a flavor agent.
T3843 Pinosylvin 3,5-stilbenediol,5-Styrylresorcinol Apoptosis , Others , Antibacterial , Autophagy
Pinosylvin (5-Styrylresorcinol) induces autophagy via AMPK activation. Pinosylvin is likely to act as a pro-angiogenic factor.
T0588 D-(-)-Arabinose D(-)-Arabinose,D-arabinose Others
D-(-)-Arabinose is a reducing sugar useful as a substrate in analysis of arabinose isomerases and synthesis of D-erythroascorbic acid in yeast. It shows strong growth inhibition against the Caenorhabditis elegans with an...
T3S0309 D(+)-Raffinose pentahydrate D-Raffinose pentahydrate,Raffinose Others , Endogenous Metabolite
D(+)-Raffinose pentahydrate (D-Raffinose pentahydrate) is a trisugar composed of fructose, galactose and glucose that occurs naturally in a variety of vegetables and grains. D(+)-Raffinose pentahydrate is a functional ol...
T6S2227 Spinosin Flavoayamenin Others
1. Spinosin (Flavoayamenin) ameliorated memory impairment induced through AβO, the serotonergic neurotransmitter system, and these effects were regulated, in part, through neuroprotective activity via the anti-inflammato...
TN2082 Pinostrobin Beta Amyloid , IL Receptor , Serine/threonin kinase , TNF
Pinostrobin, a potent flavonoid inducer, exerts a neuroprotective effect against Aα²(25-35)-induced neurotoxicity in PC12 cells, at least in part, via inhibiting oxidative damage and calcium overload, as well as suppress...
T7523 Guanidinosuccinic acid Others , Endogenous Metabolite
Guanidinosuccinic acid (GSA) has been identified as a uremic toxin, is a nitrogenous metabolite isolated in excess from serum and urine.
T4882 Arabinose DL-Arabinose Others , Endogenous Metabolite
Arabinose (DL-Arabinose), also known as (+/-)-arabinose or aloe sugar. Arabinose has been primarily detected in feces. Within the cell, Arabinose is primarily located in the cytoplasm. Arabinose exists in all eukaryotes,...
T2S0461 D-Arabinose Others , Endogenous Metabolite
Inexpensive starting material for chiral synthesis.
T0646 5-Aminosalicylic Acid Mesalazine,5-ASA,Mesalamine NF-κB , Lipoxygenase , COX , Glutathione Peroxidase , Endogenous Metabolite , PAK , PPAR
5-Aminosalicylic Acid (5-ASA) is an anti-inflammatory agent, structurally related to the SALICYLATES, which is active in INFLAMMATORY BOWEL DISEASE. It is considered to be the active moiety of SULPHASALAZINE.
TN5594 Tinosporol B
Tinosporol B is a natural product for research related to life sciences. The catalog number is TN5594 and the CAS number is 2244777-13-5.
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天然物製品

Irisflorentin
T6S1665
Synonym:
Target: Others, NO Synthase
Dehydroandrographolide
T2738
Synonym:
Target: NOS, Influenza Virus
Ethyl linoleate
TN6951
Synonym:
Target: Others
Sauchinone
T6S1572
Synonym:
Target: ERK, p38 MAPK, NF-κB
Regaloside B
TN2139
Synonym:
Target: NOS, COX, NO Synthase
Piceatannol
T0610
Synonym: trans-Piceatannol,Astringenin
Target: Apoptosis, Serine/threonin kinase, PKA, Syk, PKC, Autophagy
Isofraxidin
T5S0045
Synonym: 6,8-Dimethoxyumbelliferone,Phytodolor
Target: MMP, ERK, p38 MAPK, TLR, COX
Metronidazole
T1079
Synonym: Flagyl,Metronidazol,Anagiardil
Target: Apoptosis, NADPH, Hydrogenase, Antibacterial, Antibiotic, Parasite, Antifection
2,5-Dihydroxyacetophenone
TCS2170
Synonym: Quinacetophenone,2-Acetylhydroquinone,2-5-dihydroxyacetophenone,Acetylhydroquinone,DHAP
Target: ERK, NF-κB, Tyrosinase
3-O-Acetyl-16α-hydroxydehydrotrametenolic acid
TN1109
Synonym: 3-O-Acetyl-16 alpha-hydroxydehydrotrametenolic acid
Target: NOS, NO Synthase, Prostaglandin Receptor
Inosine-5'-triphosphate trisodium salt
T4897
Synonym: ITP,Inosine 5'-triphosphate trisodium salt
Target: Others, Endogenous Metabolite
Dihydropinosylvin
TN3861
Synonym:
Target: Anti-infection
Pinostilbene
T3755
Synonym:
Target: Others
Isovitexin 2''-O-arabinoside
TN1808
Synonym:
Target: Others
6‴-Feruloylspinosin
T5S2228
Synonym: 6'''-Feruloylspinosin
Target: NF-κB
INOSINIC ACID
T4685
Synonym: Inosine 5′-monophosphate,IMP,I-5'-P
Target: Endogenous Metabolite
Thyminose
T4818
Synonym: 2-Deoxy-D-ribose,2-Deoxy-D-arabinose,2-Deoxy-D-erythropentose
Target: Others, Endogenous Metabolite
Acetylshengmanol Arabinoside
T5S1679
Synonym: Acetylcimigenol 3-O-alpha-L-arabinopyran
Target: Others
Aloinoside B
TN6910
Synonym: 11-o-Rhamnosylaloin B
Target:
Plantainoside D
T5796
Synonym: Isoplantamajoside
Target: RAAS, PKC
Inosine
T0437
Synonym: INO 495,NSC 20262
Target: ROS, Endogenous Metabolite, Adenosine Receptor
2'-Deoxyinosine
T1709
Synonym: Guanine deoxyriboside,Deoxyinosine
Target: Others, Endogenous Metabolite
yibeinoside A
T2S0112
Synonym: Sinpeinine-3-O-β-glucoside
Target: Others
Chrysin 6-C-arabinoside 8-C-glucoside
TN1487
Synonym:
Target: Others
Raffinose
T8144
Synonym: Melitose,Melitriose
Target: Others, Endogenous Metabolite
Scyllo-Inositol
T8012
Synonym: Scyllitol
Target: Beta Amyloid, Endogenous Metabolite
Chrysin 6-C-glucoside 8-C-arabinoside
TN1488
Synonym:
Target: Others
Pinostrobin chalcone
TN2083
Synonym:
Target:
L-(+)-Arabinose
T13752
Synonym:
Target: Endogenous Metabolite
i-Inositol
T0421
Synonym: Inositol,myo-Inositol,meso-Inositol
Target: Endogenous Metabolite
Palatinose hydrate
T4875
Synonym: 6-O-α-D-Glucopyranosyl-D-fructose, Isoma
Target: Others, Endogenous Metabolite
Inosine 5'-monophosphate disodium salt hydrate
T5073
Synonym: Inosine 5'-monophosphate disodium salt,5'-IMP-Na2,Disodium 5'-inosinate monohydrate
Target: Others, Endogenous Metabolite
D-chiro-Inositol
T5915
Synonym: D-(+)-CHIRO-INOSITOL
Target: Endogenous Metabolite
Spinosad
T9076
Synonym:
Target: Others
Mycaminosyltylonolide
T67867
Synonym:
Target: Antibacterial
Spinosyn A
T21495
Synonym:
Target: Others
1-Methylinosine
T19083
Synonym: N1-Methylinosine,Inosine, 1-methyl
Target: Nucleoside Antimetabolite/Analog, Endogenous Metabolite
Kudinoside D
TN1836
Synonym:
Target: LDL, AMPK, PPAR
PALATINOSE
TN6745
Synonym: TNP-470,Isomaltulose
Target: Others
Disodium 5'-inosinate
TMS1830
Synonym: Disodium Inosinate,Sodium Inosinate,5'-IMP disodium salt
Target: Others
Pinosylvin
T3843
Synonym: 3,5-stilbenediol,5-Styrylresorcinol
Target: Apoptosis, Others, Antibacterial, Autophagy
D-(-)-Arabinose
T0588
Synonym: D(-)-Arabinose,D-arabinose
Target: Others
D(+)-Raffinose pentahydrate
T3S0309
Synonym: D-Raffinose pentahydrate,Raffinose
Target: Others, Endogenous Metabolite
Spinosin
T6S2227
Synonym: Flavoayamenin
Target: Others
Pinostrobin
TN2082
Synonym:
Target: Beta Amyloid, IL Receptor, Serine/threonin kinase, TNF
Guanidinosuccinic acid
T7523
Synonym:
Target: Others, Endogenous Metabolite
Arabinose
T4882
Synonym: DL-Arabinose
Target: Others, Endogenous Metabolite
D-Arabinose
T2S0461
Synonym:
Target: Others, Endogenous Metabolite
5-Aminosalicylic Acid
T0646
Synonym: Mesalazine,5-ASA,Mesalamine
Target: NF-κB, Lipoxygenase, COX, Glutathione Peroxidase, Endogenous Metabolite, PAK, PPAR
Tinosporol B
TN5594
Synonym:
Target:

Recombinant Proteins

カタログ番号 製品名 Species Expression System
TMPH-03169 PLC-H Protein, Pseudomonas aeruginosa, Recombinant (His & Myc & SUMO) Pseudomonas aeruginosa E. coli
Hydrolyzes sphingomyelin in addition to phosphatidylcholine. PLC-H Protein, Pseudomonas aeruginosa, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted...
TMPH-00167 L-arabinose isomerase Protein, Bacillus subtilis, Recombinant (His & Myc) Bacillus subtilis E. coli
Catalyzes the conversion of L-arabinose to L-ribulose. L-arabinose isomerase Protein, Bacillus subtilis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecu...
TMPH-02034 Retinoschisin Protein, Human, Recombinant (His) Human E. coli
Retinoschisin Protein, Human, Recombinant (His) is expressed in E. coli.
TMPH-03407 NIFH Protein, Rhizobium leguminosarum, Recombinant (GST & His & Myc) Rhizobium leguminosarum E. coli
The key enzymatic reactions in nitrogen fixation are catalyzed by the nitrogenase complex, which has 2 components: the iron protein and the molybdenum-iron protein. NIFH Protein, Rhizobium leguminosarum, Recombinant (GST...
TMPH-00045 Aln g I Protein, Alnus glutinosa, Recombinant (E. coli, His) Alnus glutinosa E. coli
Aln g I Protein, Alnus glutinosa, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 21.2 kDa and the accession number is P38948.
TMPY-03172 Argininosuccinate lyase Protein, Human, Recombinant (His & GST) Human Baculovirus Insect Cells
The recycling of citrulline by argininosuccinate synthase 1 (ASS1) and argininosuccinate lyase (ASL) is crucial to maintain arginine availability and nitric oxide (NO) production. Nitric oxide (NO) plays an established r...
TMPH-03177 RhlR Protein, Pseudomonas aeruginosa, Recombinant (His & Myc & SUMO) Pseudomonas aeruginosa E. coli
Necessary for transcriptional activation of the rhlAB genes encoding the rhamnosyltransferase. It also functions as a transcriptional activator of elastase structural gene (lasB). Binds to autoinducer molecules BHL (N-bu...
TMPH-03173 OprF Protein, Pseudomonas aeruginosa, Recombinant (His) Pseudomonas aeruginosa E. coli
Has porin activity, forming small water-filled channels. Also has a structural role in determining cell shape and ability to grow in low-osmolarity medium. OprF Protein, Pseudomonas aeruginosa, Recombinant (His) is expre...
TMPH-03171 Lysyl endopeptidase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
Lysine-specific endoprotease. Involved in corneal virulence. Lysyl endopeptidase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted mo...
TMPH-03179 LpxC Protein, Pseudomonas aeruginosa, Recombinant (His & Myc & SUMO) Pseudomonas aeruginosa E. coli
Catalyzes the hydrolysis of UDP-3-O-myristoyl-N-acetylglucosamine to form UDP-3-O-myristoylglucosamine and acetate, the committed step in lipid A biosynthesis. LpxC Protein, Pseudomonas aeruginosa, Recombinant (His & Myc...
TMPH-03178 TusA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
Sulfur carrier protein which probably makes part of a sulfur-relay system. TusA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted mol...
TMPH-03172 OprI Protein, Pseudomonas aeruginosa, Recombinant (His) Pseudomonas aeruginosa E. coli
OprI Protein, Pseudomonas aeruginosa, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 12.9 kDa and the accession number is P11221.
TMPH-03164 Beta-lactamase OXA-10 Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
Hydrolyzes both carbenicillin and oxacillin. Beta-lactamase OXA-10 Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight...
TMPH-03167 ToxR Protein, Pseudomonas aeruginosa, Recombinant (His) Pseudomonas aeruginosa E. coli
Positive regulation of toxA gene transcription. toxR Protein, Pseudomonas aeruginosa, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 32.9 kDa and the acces...
TMPH-03174 LecA Protein, Pseudomonas aeruginosa, Recombinant (His) Pseudomonas aeruginosa E. coli
D-galactose specific lectin. Binds in decreasing order of affinity: melibiose, methyl-alpha-D-galactoside, D-galactose, methyl-beta-D-galactoside, N-acetyl-D-galactosamine. Similar to plant lectins in its selective (carb...
TMPH-03176 LasA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
LasA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 36.0 kDa and the accession number is P14789.
TMPH-03165 Beta-lactamase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
Beta-lactamase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 56.7 kDa and the accession number is P24735.
TMPH-03166 Elastase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
Cleaves host elastin, collagen, IgG, and several complement components as well as endogenous pro-aminopeptidase. Autocatalyses processing of its pro-peptide. Processes the pro-peptide of pro-chitin-binding protein (cbpD)...
TMPH-03180 LpxC Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
Catalyzes the hydrolysis of UDP-3-O-myristoyl-N-acetylglucosamine to form UDP-3-O-myristoylglucosamine and acetate, the committed step in lipid A biosynthesis. LpxC Protein, Pseudomonas aeruginosa, Recombinant (His & SUM...
TMPH-03168 Exotoxin A Protein, Pseudomonas aeruginosa, Recombinant (His & KSI) Pseudomonas aeruginosa E. coli
An NAD-dependent ADP-ribosyltransferase (ADPRT). Catalyzes the transfer of the ADP ribosyl moiety of oxidized NAD (NAD(+)) onto eukaryotic elongation factor 2 (eEF-2) thus arresting protein synthesis. Has an LD(50) of 65...
TMPH-03175 Porin P Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
Anion specific, the binding site has higher affinity for phosphate than chloride ions. Porin O has a higher affinity for polyphosphates (tripolyphosphate and pyrophosphate) while porin P has a higher affinity for orthoph...
TMPH-00046 Aln g I Protein, Alnus glutinosa, Recombinant (Yeast, His) European alder P. pastoris (Yeast)
Aln g I Protein, Alnus glutinosa, Recombinant (Yeast, His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 19.2 kDa and the accession number is P38948.
TMPH-00346 Limulus clotting factor C Protein, Carcinoscorpius rotundicauda, Recombinant (His) Carcinoscorpius rotundicauda E. coli
This enzyme is closely associated with an endotoxin-sensitive hemolymph coagulation system which may play important roles in both hemostasis and host defense mechanisms. Its active form catalyzes the activation of factor...
TMPH-03170 PvdA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) Pseudomonas aeruginosa E. coli
PvdA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 65.5 kDa and the accession number is Q51548.
TMPH-01552 IRF1 Protein, Human, Recombinant (GST & His) Human Baculovirus Insect Cells
Transcriptional regulator which displays a remarkable functional diversity in the regulation of cellular responses. Regulates transcription of IFN and IFN-inducible genes, host response to viral and bacterial infections,...
PLC-H Protein, Pseudomonas aeruginosa, Recombinant (His & Myc & SUMO)
TMPH-03169
Species: Pseudomonas aeruginosa
Expression System: E. coli
L-arabinose isomerase Protein, Bacillus subtilis, Recombinant (His & Myc)
TMPH-00167
Species: Bacillus subtilis
Expression System: E. coli
Retinoschisin Protein, Human, Recombinant (His)
TMPH-02034
Species: Human
Expression System: E. coli
NIFH Protein, Rhizobium leguminosarum, Recombinant (GST & His & Myc)
TMPH-03407
Species: Rhizobium leguminosarum
Expression System: E. coli
Aln g I Protein, Alnus glutinosa, Recombinant (E. coli, His)
TMPH-00045
Species: Alnus glutinosa
Expression System: E. coli
Argininosuccinate lyase Protein, Human, Recombinant (His & GST)
TMPY-03172
Species: Human
Expression System: Baculovirus Insect Cells
RhlR Protein, Pseudomonas aeruginosa, Recombinant (His & Myc & SUMO)
TMPH-03177
Species: Pseudomonas aeruginosa
Expression System: E. coli
OprF Protein, Pseudomonas aeruginosa, Recombinant (His)
TMPH-03173
Species: Pseudomonas aeruginosa
Expression System: E. coli
Lysyl endopeptidase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03171
Species: Pseudomonas aeruginosa
Expression System: E. coli
LpxC Protein, Pseudomonas aeruginosa, Recombinant (His & Myc & SUMO)
TMPH-03179
Species: Pseudomonas aeruginosa
Expression System: E. coli
TusA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03178
Species: Pseudomonas aeruginosa
Expression System: E. coli
OprI Protein, Pseudomonas aeruginosa, Recombinant (His)
TMPH-03172
Species: Pseudomonas aeruginosa
Expression System: E. coli
Beta-lactamase OXA-10 Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03164
Species: Pseudomonas aeruginosa
Expression System: E. coli
toxR Protein, Pseudomonas aeruginosa, Recombinant (His)
TMPH-03167
Species: Pseudomonas aeruginosa
Expression System: E. coli
LecA Protein, Pseudomonas aeruginosa, Recombinant (His)
TMPH-03174
Species: Pseudomonas aeruginosa
Expression System: E. coli
LasA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03176
Species: Pseudomonas aeruginosa
Expression System: E. coli
Beta-lactamase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03165
Species: Pseudomonas aeruginosa
Expression System: E. coli
Elastase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03166
Species: Pseudomonas aeruginosa
Expression System: E. coli
LpxC Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03180
Species: Pseudomonas aeruginosa
Expression System: E. coli
Exotoxin A Protein, Pseudomonas aeruginosa, Recombinant (His & KSI)
TMPH-03168
Species: Pseudomonas aeruginosa
Expression System: E. coli
Porin P Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03175
Species: Pseudomonas aeruginosa
Expression System: E. coli
Aln g I Protein, Alnus glutinosa, Recombinant (Yeast, His)
TMPH-00046
Species: European alder
Expression System: P. pastoris (Yeast)
Limulus clotting factor C Protein, Carcinoscorpius rotundicauda, Recombinant (His)
TMPH-00346
Species: Carcinoscorpius rotundicauda
Expression System: E. coli
PvdA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
TMPH-03170
Species: Pseudomonas aeruginosa
Expression System: E. coli
IRF1 Protein, Human, Recombinant (GST & His)
TMPH-01552
Species: Human
Expression System: Baculovirus Insect Cells
カタログ番号 製品名
L2900 Oxidation-Reduction Compound Library

1264 compounds
1264 small molecule compounds with pro-oxidant or anti-oxidant activity for high-throughput and high-content screening.