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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T15546 | ICA | N-[4-(2-Pyridinyl)-2-thiazolyl]-2-pyridinamine | Potassium Channel , Parasite |
ICA (N-[4-(2-Pyridinyl)-2-thiazolyl]-2-pyridinamine) is a SK channel inhibitor and exhibits antileishmanial activity (IC50: 2.1 µM). | |||
T9009 | ICA-105574 | ICA,3-nitro-N-[4-phenoxyphenyl]-benzamide | HER |
ICA-105574 (ICA) is an activator of hERG that binds to the channel to remove inactivation, thus increasing peak current amplitude and shortening the action potential. It also modulates activation kinetics of the channel. | |||
T15545 | ICA-27243 | Potassium Channel | |
ICA-27243 is less effective at activating KCNQ4 and KCNQ3/Q5. ICA-27243 is a potent and orally active KCNQ2/Q3 potassium channel opener (EC50: 0.38 μM). ICA-27243 also has antiepileptic and anticonvulsant effects. | |||
T7612 | ICA 110381 | Potassium Channel | |
ICA 110381 is a KCNQ2/Q3 potassium channel opener for the treatment of epilepsy | |||
T7336 | ICA-121431 | 2,2-Diphenyl-N-[4-(thiazol-2-ylsulfamoyl | Sodium Channel |
ICA-121431 (2,2-Diphenyl-N-[4-(thiazol-2-ylsulfamoyl) is a nanomolar potent small molecule Nav1.7 channel inhibitor with IC50 of 19 nM for rat Nav1.7, with little or no activity against human Nav1.5 or Nav1.7 channels. | |||
T3959 | ICA-069673 | ICA069673 | Potassium Channel |
ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM). | |||
T3528 | Senicapoc | ICA-17043 | Potassium Channel |
Senicapoc (ICA-17043) is a potent inhibitor of the Gardos channel and ameliorates RBC dehydration in the SAD mouse. Senicapoc blocked Ca2+-induced rubidium flux from human RBCs with an IC50 value of 11 ± 2 nM (CLT IC50 =... | |||
T11606 | ICA-105665 | PF-04895162 | Others |
ICA-105665 (PF-04895162) is a potent and orally active neuronal Kv7.2/7.3 and Kv7.3/7.5 potassium channels opener. ICA-105665 had low cytotoxic potential in human hepatocytes but inhibited liver mitochondrial function an... | |||
T6456 | CRT0044876 | NSC 69877,7-NO2-ICA,NSC 69877,7-Nitroindole-2-Carboxylic Acid | DNA/RNA Synthesis |
CRT0044876 (7-NO2-ICA) is a potent and selective APE1 inhibitor with IC50 of ~3 μM. | |||
T4539 | Nicainoprol | RU-42924 | Sodium Channel |
Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent. | |||
T7618 | Pyributicarb | TSH-888 | P450 |
Pyributicarb (TSH-888) is a potent activator of both CYP3A4 gene and human pregnane X receptor (hPXR). | |||
T61046 | Anticancer agent 43 | Apoptosis | |
Anticancer agent 43 is a potent anticancer agent that induces apoptosis through caspase 3, PARP1, and Bax protein-dependent pathways.Anticancer agent 43 induces DNA damage and can be used in the study of glioblastoma in ... | |||
T21483 | Tricaine methanesulfonate | MS-222 | Others |
Tricaine methanesulfonate (MS-222) (TMS) is an anesthetic. Many hatcheries and research studies use TMS to immobilize fish for marking or transport and to suppress sensory systems during invasive procedures. | |||
T60852 | Anticancer agent 46 | ||
Anticancer agent 46 is a potent anti-cancer agent, showing anti-proliferative activity in cellular assays, with an IC50 of 0.986 μM against MGC803 cells. | |||
T13383 | Zamicastat | BIA 5-1058 | BCRP , Hydroxylase , P-gp |
Zamicastat (BIA 5-1058) is an inhibitor of dopamine β-hydroxylase (DBH), and is also a concentration-dependent dual inhibitor of P-gp and BCRP(IC50 values of 73.8 μM and 17.0 μM, respectively). | |||
T7811 | Pilsicainide HCl | SUN 1165 | Sodium Channel |
Pilsicainide HCl (SUN 1165) is a pure sodium channel blocker | |||
T6387 | Ampiroxicam | CP 65703,Flucam | COX |
Ampiroxicam (Flucam) is a nonselective cyclooxygenase inhibitor uesd as anti-inflammatory drug. | |||
T68115 | Nicanartine | Others | |
Nicanartine is a cholesterol inhibitor that is used to treat cardiovascular disease and can be used to study atherosclerosis. | |||
T69984 | Ticalopride | 5-HT Receptor | |
Ticalopride is a 5-HT3 receptor agonist used in the treatment of digestive disorders, orofacial disorders, otorhinolaryngologic disorders, and may be used in the study of bulimia nervosa, gastroesophageal reflux, and irr... | |||
T28537 | Ricasetron | Brl 46470,Brl46470,Brl-46470 | 5-HT Receptor |
Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysis and antiemetic properties, and is used in the study of anxiety and anxiety disorders. | |||
T1727 | 4-Cyclohexyl-1-phenylthiosemicarbazide | Others | |
4-Cyclohexyl-1-phenylthiosemicarbazide is employed as an intermediate. | |||
T1794 | Micafungin sodium | Mycamine Sodium,FK 463,FK463 Sodium | Antibiotic , Antifungal |
Micafungin sodium (FK 463) is the sodium salt form of micafungin, a semi-synthetic echinocandin derived from a natural product of the fungus Coleophoma empetri with antifungal activity. | |||
T13275 | Vabicaserin hydrochloride | SCA 136 | 5-HT Receptor |
Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM). | |||
T7640 | Aldicarb sulfone | AChE | |
Aldicarb sulfone is a cholinesterase inhibitor . | |||
T77707 | Di-tert-butyl dicarbonate | BOC anhydride | Others |
Di-tert-butyl dicarbonate(BOC anhydride) is a biochemical reagent that can be used in biochemical experiments. | |||
T0826 | Meloxicam | Movalis,Mobic,Metacam | Apoptosis , COX , Autophagy |
Meloxicam (Metacam) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of meloxicam is as a Cyclooxygenase Inhibitor. The chemical classification of meloxicam is Nonsteroidal Anti-inflammatory Compounds. | |||
T5388 | 2,5-PYRIDINEDICARBOXYLIC ACID | Others | |
2,5-Pyridinedicarboxylic Acid is used in the preparation of new derivatives as antiviral agents. | |||
T16681 | Nesolicaftor | PTI-428 | CFTR , Autophagy |
Nesolicaftor (PTI-428) specifically enhances cystic fibrosis transmembrane conductance regulator protein synthesis. | |||
T21059 | Ticagrelor metabolite M5 | Ticagrelor metabolite M5,,T437700,AR-C133913XX | P2Y Receptor |
Ticagrelor metabolite M5 (T437700) is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor. Compared to Clopidogrel, Ticagrelor has faster and more consistent inhibition on ADP-receptors. Ti... | |||
T21443 | Prednicarbate | Hoe 777,Hoe-777,Dermatop E emollient,UNII-V901LV1K7D | Others |
Prednicarbate (Hoe 777) is a Corticosteroid Hormone Receptor Agonist. Prednicarbate has antipruritic, anti-inflammatory, and vasoconstrictive properties. It also decreases the number of circulating lymphocytes by inhibit... | |||
T6604 | Nepicastat hydrochloride | Nepicastat HCl,RS-25560-197 hydrochloride,SYN-117 hydrochloride,Nepicastat (SYN-117) HCl | Hydroxylase |
Nepicastat hydrochloride (RS-25560-197 hydrochloride) is an effective and specific inhibitor, which is used for bovine and human dopamine-β-hydroxylase with IC50 of 8.5 nM and 9 nM, respectively.The affinity of Nepicasta... | |||
T60272 | Isatin-β-thiosemicarbazone | IBT | HSV |
Isatin-β-thiosemicarbazone is a potent inhibitor of herpes simplex virus (HSV). isatin-β-thiosemicarbazone exhibits antiviral activity by inhibiting both HSV-1 and HSV-2. isatin-β-thiosemicarbazone is Isatin-β-thiosemica... | |||
T3116 | Atorvastatin hemicalcium salt | Lipitor,Atorvastatin hemicalcium,Atorvastatin Calcium,CI-981,Sortis | Ferroptosis , HMG-CoA Reductase , Autophagy |
Atorvastatin hemicalcium salt (Atorvastatin Calcium), an effective HMG-CoA reductase inhibitor (IC50 = 8 nM), is utilized as a cholesterol-lowering medication. | |||
T8333 | Aurintricarboxylic acid | ATA,NSC-4056,NSC4056,NSC 4056 | Apoptosis , P2X Receptor , Influenza Virus , Topoisomerase |
Aurintricarboxylic acid (NSC-4056) is a strong inhibitor of topoisomerases and other nucleases. It is a potent inhibitor of ribonuclease and topoisomerase II by preventing the binding of the nucleic acid to the enzyme. | |||
T16950 | Sudoxicam | 4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide | COX |
Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema, and antipyretic properties. | |||
T9258 | Aficamten | Others | |
Aficamten is a Next-Generation Cardiac Myosin Inhibitor for the Treatment of Hypertrophic Cardiomyopathy. | |||
T6606 | Nicaraven | Others | |
Nicaraven, a hydroxyl radical scavenger, has neuroprotective and antivasospastic effects. | |||
T3532 | 5S rRNA modificator | FAI,Furoyl Acylimidazole | Others |
5S rRNA modificator (FAI), used in 5S rRNA RNA modification, is a suitable electrophile for 2'-hydroxyl acylation on structured RNA molecules. | |||
T21195 | AICAR monophosphate | Aica ribonucleotide,AICA riboside,Acadesine 5'-monophosphate,Z-nucleotide | Others |
AICAR monophosphate (Aica ribonucleotide) is a purine precursor with antineoplastic activity and can be used in studies about type 2 diabetes. | |||
T7806 | Licarbazepine | 10,11-hydroxy-10,11 Dihydrocarbamezer | Others |
Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial seizures and bipolar disorders. | |||
T11099 | Droxicainide | Others | |
Droxicainide is an antiarrhythmic agent. | |||
T35033 | Vamicamide | FK 176,FK-176,FK176 | AChE |
Vamicamide (FK 176) is a novel anticholinergic compound. Vamicamide increases spontaneous locomotor activity in mice at 32 mg/kg (p.o.) or higher and inhibits cataleptic convulsions in mice at 100 mg/kg. | |||
T60150 | (1S,2R)-Alicapistat | Cysteine Protease | |
(1S,2R)-Alicapistat ((1S,2R)-ABT-957) is a highly efficient, orally active compound that selectively inhibits human calpains 1 and 2, with promising implications for Alzheimer's disease (AD) therapy [1]. This compound ef... | |||
T60420 | Anticancer agent 73 | DNA/RNA Synthesis | |
Anticancer agent 73 is an anticancer agent which potently targets transactivation response(TAR) RNA-binding protein 2 (TRBP) and disrupts the TRBP-Dicer interaction. Anticancer agent 73 suppresses the growth and metasta... | |||
T64319 | 4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester | Others | |
4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester is a biologically active compound used as an intermediate in the synthesis of a variety of compounds. | |||
T21404 | Fluticasone furoate | Veramyst,Allermist,Avamys,Fluticasone furoate | Glucocorticoid Receptor |
Fluticasone furoate (Avamys) is a synthetic trifluorinated corticosteroid derived from fluticasone with a Kd of 0.3 nM. Fluticasone furoate has potent anti-inflammatory, anti-asthmatic activity, and low systemic exposure... | |||
T16398 | Opicapone | BIA 9-1067 | Transferase |
Opicapone (BIA 9-1067) reduces the ATP content of the cells (IC50: 98 μM). Opicapone is an effective third-generation catechol-O-methyltransferase inhibitor for the research of Parkinson's disease and motor fluctuations. | |||
T77705 | Diethyl 2,4-dimethylpyrrole-3,5-dicarboxylate | Diethyl 3,5-dimethyl-1H-pyrrole-2,4-dicarboxylate | Others |
Diethyl 2,4-dimethylpyrrole-3,5-dicarboxylate is a biochemical reagent that can be used in biochemical reactions. | |||
T6706 | Ticarcillin sodium | Ticarpen hydrate,Aerugipen hydrate,BRL 2288,AB 2288,Monapen | Others , Antibacterial , Antibiotic |
Ticarcillin sodium (Aerugipen hydrate) is a semisynthetic antibiotic with a broad spectrum of bactericidal activity against many gram-positive and gram-negative aerobic and anaerobic bacteria. | |||
T1063 | Ticarcillin disodium | Ticarpen,Ticarcillin disodium salt | Antibacterial , Antibiotic |
Ticarcillin disodium (Ticarpen) is the disodium salt form of ticarcillin, a broad-spectrum, semi-synthetic penicillin antibiotic with bactericidal and beta-lactamase resistant activity. Similar to carbenicillin in action... |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T4S1545 | Licarin B | (-)-Licarin B,Licarine B | transporter , Antibacterial , PPAR |
1.(-)-Licarin B (Licarine B) has anti-mycobacterial activity. | |||
T7995 | α-Angelica lactone | Alpha-Angelica Lactone | Others , GST |
α-Angelica lactone has cardiotonic activity, may exert their effects by providing an increased contraction-dependent calcium pool to be released upon systolic depolarization. | |||
T1468 | Lornoxicam | Ro 13-9297,Chlortenoxicam,TS110 | COX , Endogenous Metabolite |
Lornoxicam (Chlortenoxicam) (chlortenoxicam) is a new nonsteroidal anti-inflammatory drug (NSAID) of the oxicam class with analgesic, anti-inflammatory, and antipyretic properties. Lornoxicam differs from other oxicam co... | |||
T19278 | Dicaprylyl carbonate | Dimethyl carbonate | Others |
Dicaprylyl carbonate (Dimethyl carbonate) is a solid fat derived from plants and a dry emollient. Dimethyl carbonate has good skin compatibility and comprehensive properties, such as a sunscreen filter with the ability t... | |||
T5227 | Tricaprin | Tridecanoin,Glyceryl tridecanoate,Glycerol Tridecanoate,TG(10:0/10:0/10:0),Glycerol tricaprate | Others , Endogenous Metabolite |
Tricaprin (Glycerol Tridecanoate) is also known as triacylglycerols or triacylglycerides. The triglycerides are rebuilt in the blood from their fragments and become constituents of lipoproteins, which deliver the fatty a... | |||
T13768 | (+)-Medicarpin | Estrogen/progestogen Receptor | |
(+)-Medicarpin, a pterocarpan, is an isoflavonoid compound derived from multiple medicinal plant species such as Sophora japonica, Zollernia paraensis, Platymiscium yucatamun, Machaerium aristulatum, and Platymiscium flo... | |||
T2775 | Baicalin | Baicalein 7-O-β-D-glucuronide | NF-κB , HIV Protease , GABA Receptor , Autophagy |
Baicalin (Baicalein 7-O-β-D-glucuronide) is a prolyl endopeptidase inhibitor isolated from scutellaria baicalensis, with antioxidant, anti-tumor, anti-HIV properties. | |||
T3551 | D-Pantothenic acid hemicalcium salt | D-Pantothenic Acid Calcium,Calpanate,Calcium D-pantothenate,Vitamin B5 calcium salt,Calcium pantothenate,Calcium D-Panthotenate | Apoptosis , Endogenous Metabolite |
D-Pantothenic acid hemicalcium salt (Calcium pantothenate), a kind of water soluble vitamin, can reduce the patulin content of the apple juice. | |||
T2S2150 | Noricaritin | Others | |
Noricaritin is a flavonoid derived from Epimedium root. | |||
T2732 | (-)-Epicatechin gallate | (−)-Epicatechin 3-gallate,Epicatechin gallate,(-)-Epicatechin 3-gallate,(-)-Epicatechin 3-O-gallate,ECG | Virus Protease , COX , Autophagy |
(-)-Epicatechin gallate ((-)-Epicatechin 3-O-gallate) is one of the catechin isomers and a potent antioxidant that can modulate a wide range of membrane proteins. Its bilayer-modifying potency was tested using gramicidin... | |||
T3921 | Punicalagin | SARS-CoV , HBV | |
Punicalagin is a major ellagitannin found in pomegranates that is reported to produce antioxidant, anti-inflammatory, and anticancer effects. It has been shown to prevent high-fat diet-induced obesity-associated accumula... | |||
TN3848 | Dihydrobaicalein | PLK | |
Dihydrobaicalein is a natural product from Scutellaria baicalensis, a PLK1 inhibitor (IC50:6.3 μM).Dihydrobaicalein inhibits VRK2 and PLK2. | |||
T5S2205 | Sibiricaxanthone B | Others | |
Sibiricaxanthone B is an oxygen-containing xanthone isolated from Polygala tenuifolia. | |||
T5564 | Tricarballylic acid | β-Carboxyglutaric acid,1,2,3-Propanetricarboxylic acid,Carballylic acid,Propane-1,2,3-tricarboxylic acid | aconitase , Mitochondrial Metabolism |
Tricarballylic acid (Carballylic acid) is an inhibitor of aconitase. | |||
T4S1521 | 1,4-Dicaffeoylquinic acid | HIV Protease | |
1,4-Dicaffeoylquinic acid has antioxidant activity.1,4-Dicaffeoylquinic acid is a potent and highly selective class of HIV-1 integrase inhibitors, inhibitsHIV-1 replication in MT-2 cell culture at non-toxic concentration... | |||
T6S2140 | β-Anhydroicaritin | Anhydroicaritin,Beta-Anhydroicaritin | MMP , Others , TNF , Interleukin |
1. β-Anhydroicaritin exhibits immunosuppressive effect on the mouse macrophages stimulated by LPS. 2. β-Anhydroicaritin phytosomes can inhibit enhanced bone turnover induced by ovariectomy, improve BMD the biomechanical ... | |||
TL0005 | 3,5-O-Dicaffeoylquinic acid | Isochlorogenic Acid A,(-)-3,5-Dicaffeoyl quinic acid,3,5-Dicaffeoylquinic Acid | Others |
3,5-O-Dicaffeoylquinic acid (Isochlorogenic Acid A) is an isolated compound from Artemisia argyi; its ester derivatives exert anti-leucyl-tRNA synthetase of Giardia lamblia (GlLeuRS) and potential anti-giardial effects. ... | |||
T5246 | Trans-2-butene-1,4-dicarboxylic acid | trans-2-Butene-1,4-dicarboxylic Acid,3-Hexenedioic Acid,trans-3-Hexenedioic Acid,β-Hydromuconic Acid | Others , Endogenous Metabolite |
Trans-2-butene-1,4-dicarboxylic acid (3-Hexenedioic Acid) is a normal human unsaturated dicarboxylic acid metabolite with increased excretion in patients with Dicarboxylic aciduria caused by fatty acid metabolism disorde... | |||
T3S1892 | Crassicauline A | Crassicauline I | Others |
1. Crassicauline A (Crassicauline I) and Yunaconitine possesses feeding deterrent activity against T. castaneum adults, with EC(5) values of 1134.5 and 653.4 ppm, respectively. | |||
T3808 | Icariside I | Lcariside I,Icariin I,Icarisid I | Others |
Icariside I (Lcariside I) is isolated from Epimedium herb. It can stimulate osteogenic differentiation of BMSCs and inhibit bone resorption activity of osteoclasts. | |||
TN1384 | Angelicain | Norcimifugin | Others |
Angelicain, also known as Norcimifugin, is a component found in Cimicifuga foetida that exhibits anti-inflammatory activity. | |||
T5736 | 1,3-Dicaffeoylquinic acid | CYNARIN,Cyclohexanecarboxylic acid, 1,3-bis[[3-(3,4-dihydroxyphenyl)-1-oxo-2-propen-1-yl]oxy]-4,5-dihydroxy-, (1S,3R,4R,5R)-,1,3-O-Dicaffeoylquinic acid,1,5-Dicaffeoylquinic acid | Reactive Oxygen Species , Akt , PI3K |
1,3-Dicaffeoylquinic acid (CYNARIN) is a natural product. It shows antioxidant and choleretic properties and is a potential immunosuppressive agent. | |||
T2856 | (-)-Epicatechin | L-Epicatechin,Epicatechin,(-)-Epicatechol | Ferroptosis , COX , Endogenous Metabolite |
(-)-Epicatechin (Epicatechin) is an inhibitor of cyclooxygenase-1 (COX-1), inhibiting the IL-1β-induced expression of iNOS by blocking the nuclear localization of the p65 subunit of NF-κB. | |||
T2858 | Baicalein | 5,6,7-Trihydroxyflavone | Ferroptosis , Influenza Virus , ROS , Xanthine Oxidase |
Baicalein (5,6,7-Trihydroxyflavone) is a xanthine oxidase inhibitor. | |||
T2S1158 | 4,5-Dicaffeoylquinic acid | 3,4-Dicaffeoylquinic acid,Isochlorogenic acid C | Others , HBV , Endogenous Metabolite |
1. 4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) has antiviral activity, including anti-HIV-1 integrase activity. 2. 4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) shows anti-hepatotoxic activity. | |||
T4S1718 | Punicalin | HBV , HIV Protease | |
Punicalin exerts anti-inflammatory, antioxidative, and anti-hepatotoxic activities, it shows inhibitory activity on HIV-1 reverse transcriptase in a dose-dependent manner, with an IC50 of 0.11 microg/ml (0.14 microM). | |||
TN1427 | Baicalin methyl ester | Anti-infection | |
Baicalin methyl ester shows inhibitory effects on the Avian Myeloblastosis Virus reverse transcriptase (AMV-RT). | |||
T14149 | AICAR phosphate | AICA Riboside phosphate,Acadesine phosphate | Mitophagy , NOS , YAP , AMPK |
AICAR phosphate (Acadesine phosphate) is an AMPK activator and inhibitor of autophagy, YAP, and mitophagy, as well as an adenosine analog that regulates glucose and lipid metabolism, and inhibits the production of pro-in... | |||
T5275 | 2,5-Furandicarboxylic acid | Dehydromucic Acid,2,5-Dicarboxyfuran | Others , Endogenous Metabolite |
2,5-Furandicarboxylic acid (Dehydromucic Acid) is a normal urinary metabolite in humans. 2,5-Furandicarboxylic acid is also a microbial metabolite, a product of the oxidation of hydroxymethylfurfural (HMF) by the enzyme ... | |||
T13305 | Viridicatol | Anti-infection , Antifungal | |
Viridicatol, with potent antibacterial activity against Staphylococcus aureus(MIC: 15.6 μg/mL), is isolated from the fermentation of an endophytic fungus Penicillium sp. R22 in Nerium indicum. | |||
T8167 | Medicagenic acid | Castanogenin | Antibacterial |
Medicagenic acid (Castanogenin), isolated from the roots of Herniaria glabra L, exhibits potent fungistatic effects against several plant pathogens and human dermatophytes. | |||
T13229 | Tunicamycin | Influenza Virus , Antibacterial , Antibiotic , Antifungal | |
Tunicamycin is a mixture of antibiotics that inhibit N-linked glycosylation by blocking GlcNAc phosphotransferase (GPT). Tunicamycin has antitumor activity, as well as anti-bacterial, anti-fungal, and anti-viral activity... | |||
T6S1525 | 3,4-Dicaffeoylquinic acid | Isochlorogenic acid B | Apoptosis , Antioxidant , Influenza Virus , Endogenous Metabolite |
3,4-Dicaffeoylquinic acid (Isochlorogenic acid B) has antioxidant activity. | |||
TN1918 | Medicarpin | Apoptosis , BCL , ROS , JNK | |
Medicarpin, a legume phytoalexin, acts as an estrogen receptor (ER) agonist, can stimulate osteoblast differentiation likely via ERα², promote achievement of peak bone mass, and is devoid of uterine estrogenicity; in add... | |||
T13350 | Wushanicaritin | Others | |
Wushanicaritin is a natural product isolated from the traditional Chinese medicine Epimedium plants, with antitumor effects and anti-inflammatory property. | |||
T2855 | Icariin | Ieariline | PDE , PPAR , Autophagy |
Icariin (Ieariline) is a flavonol glycoside, inhibiting PDE5 and PDE4 activities. Icariin also is a PPARα activator. | |||
T19866 | Indican | NSC-87517,3-Indoxyl-beta-D-glucopyranoside,NSC 87517,NSC87517,Indoxyl-β-D-glucoside | OAT , MRP |
Indican (Indoxyl-β-D-glucoside) is a natural protective compound that is used to protect the liver. | |||
T3398 | Icaritin | Anhydroicaritin,Cycloicaritin | Apoptosis , JAK , STAT , Autophagy |
Icaritin (Anhydroicaritin) has hormone regulation activity and cardiovascular function improvement activity. Icaritin has anticancer activity, can induce S phase arrest and apoptosis, inhibit ENKL cell proliferation. Ica... | |||
TQ0172 | 2''-O-Rhamnosylicariside II | Others | |
2''-O-Rhamnosylicariside II might be beneficial for improving postmenopausal osteoporosis. It shows potent antioxidant activity, with IC50 values of 11.5 ug/mL and 90.5 uM. | |||
T5266 | Tricaprilin | Glycerol Tri-n-octanoate,trioctanoin,tricaprylic glyceride,Glyceryl trioctanoate | Others , Endogenous Metabolite |
Tricaprilin (Glycerol Tri-n-octanoate) is used in study for patients with mild to moderate Alzheimer's disease. Tricaprilin also has a role as an anticonvulsant and a plant metabolite. | |||
TMA1948 | Sibiricaxanthone A | Sibiricaxanthone A | Others |
Sibiricaxanthone A (Sibiricaxanthone A) is a natural product from Polygala tenuifolia | |||
TN4056 | Ficaprenol 11 | Others | |
Ficaprenol 11 is a natural product of Artocarpus, Moraceae. The catalog number is TN4056 and the CAS number is 26296-50-4. Ficaprenol 11 can be used as a reference standard. | |||
TMA1890 | Icariside F2 | NF-κB | |
Icariside F2 shows modest α-glucosidase inhibitory (4.60±1.74% to 11.97±3.30%) and antioxidant activities. It also displays potent NF-κB inhibitory effects, with the IC50 value of 16.25 ± 2.19 uM. | |||
TN2406 | Myricadenin A | Others | |
Myricadenin A is a natural product from plants | |||
TN3392 | Alpha-Toxicarol | Others | |
Alpha-Toxicarol exhibits a marked inhibitory effect on mouse skin tumor promotion in an in vivo two-stage carcinogenesis test. | |||
TN5767 | Gneafricanin F | ||
Gneafricanin F is a natural product for research related to life sciences. The catalog number is TN5767 and the CAS number is 477561-12-9. | |||
T83088 | Anticancer agent 156 | ||
Compound 156, also referred to as compound 11, is a potent miliusanes-based anticancer agent that demonstrates effective inhibition of human cancer cell growth and exhibits substantial cytotoxicity against gastric cancer... | |||
TN3811 | Dehydrotoxicarol | Others | |
Dehydrotoxicarol is a natural product of Derris, Fabaceae. The catalog number is TN3811 and the CAS number is 59086-93-0. Dehydrotoxicarol can be used as a reference standard. | |||
TN4601 | Myricadiol | Others | |
Myricadiol is a potential lead compound for synthetic anti-cancer drugs. | |||
TN4018 | Ethyl 3,4-dicaffeoylquinate | Others | |
Ethyl 3,4-dicaffeoylquinate is a natural product of Inula, Asteraceae. The catalog number is TN4018 and the CAS number is 143051-73-4. Ethyl 3,4-dicaffeoylquinate can be used as a reference standard. | |||
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カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPY-04920 | ICA Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
INHCA, official full name is inhibitor of carbonic anhydrase, which is a member of the transferrin gene family. Unlike many members of that gene family it does not play a significant role in iron homeostasis but rather i... | |||
TMPJ-01140 | IA2 Protein, Human, Recombinant (aa 607-686 & aa 795-888 , His) | Human | E. coli |
IA2 Protein, Human, Recombinant (aa 607-686 & aa 795-888 , His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 26-30 KDa and the accession number is Q16849. | |||
TMPJ-01139 | IA2 Protein, Human, Recombinant (aa 576-950, His) | Human | E. coli |
IA2 Protein, Human, Recombinant (aa 576-950, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 50 KDa and the accession number is Q16849. | |||
TMPJ-01141 | IA2 Protein, Human, Recombinant (aa 687-979, His) | Human | E. coli |
IA2 Protein, Human, Recombinant (aa 687-979, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 33 KDa and the accession number is Q16849. | |||
TMPY-01283 | Glypican 3/GPC3 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Glypican 3/GPC3 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 62 kDa and the accession number is P51654-1. | |||
TMPY-00502 | Glypican 3/GPC3 Protein, Mouse, Recombinant (His) | Mouse | Baculovirus Insect Cells |
Glypican 3/GPC3 Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 62 kDa and the accession number is Q3TWB2. | |||
TMPY-05017 | ICAM-1/CD54 Protein, Rhesus, Recombinant (His) | Rhesus | HEK293 Cells |
ICAM-1/CD54 Protein, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.9 kDa and the accession number is Q5NKV6. | |||
TMPY-01142 | ICAM-1/CD54 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
ICAM-1/CD54 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 51 kDa and the accession number is A0A384MEK5. | |||
TMPY-01349 | ICAM-1/CD54 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
ICAM-1/CD54 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 51.7 kDa and the accession number is P13597-1. | |||
TMPY-00981 | ICAM-1/CD54 Protein, Human, Recombinant (aa 1-480,DDDDK) | Human | HEK293 Cells |
ICAM-1/CD54 Protein, Human, Recombinant (aa 1-480,DDDDK) is expressed in HEK293 mammalian cells. The predicted molecular weight is 50.2 kDa and the accession number is A0A384MEK5. | |||
TMPY-05476 | MICA Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
MICA Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 34.3 kDa and the accession number is A9UJR3. | |||
TMPY-02053 | MICA Protein, Human, Recombinant (His), MICA*018 | Human | HEK293 Cells |
MICA Protein, Human, Recombinant (His), MICA*018 is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 34 kDa and the accession number is AAH16929.1. | |||
TMPK-00219 | MICA Protein, Human, Recombinant (His & Avi), Biotinylated | Human | HEK293 Cells |
TMICA (MHC class I chain-related gene A) is a transmembrane glycoprotein that functions as a ligand for human NKG2D. A closely related protein, MICB, shares 85% amino acid identity with MICA. These proteins are distantly... | |||
TMPH-00402 | Classical swine fever virus Genome polyprotein (His) | CSFV | Baculovirus Insect Cells |
Classical swine fever virus Genome polyprotein (His) is expressed in Baculovirus. | |||
TMPK-00872 | ICAM-1/CD54 Protein, Canine, Recombinant (His) | Canine | HEK293 Cells |
Intercellular adhesion molecule-1 (ICAM-1; CD54) is a 90 kDa member of the immunoglobulin (Ig) superfamily and is critical for the firm arrest and transmigration of leukocytes out of blood vessels and into tissues. ICAM-... | |||
TMPH-02450 | MALD3 Protein, Malus domestica, Recombinant (His & SUMO) | Apple | E. coli |
Plant non-specific lipid-transfer proteins transfer phospholipids as well as galactolipids across membranes. May play a role in wax or cutin deposition in the cell walls of expanding epidermal cells and certain secretory... | |||
TMPY-06751 | Glypican 3/GPC3 Protein, Canine, Recombinant (His) | Canine | HEK293 Cells |
Glypican 3/GPC3 Protein, Canine, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 62.07 kDa and the accession number is A0A8C0TMC5. | |||
TMPY-06778 | ICAM-1/CD54 Protein, Human, Recombinant (aa 1-480, LEVLFQ) | Human | HEK293 Cells |
ICAM-1/CD54 Protein, Human, Recombinant (aa 1-480, LEVLFQ) is expressed in HEK293 mammalian cells. The predicted molecular weight is 50.31 kDa and the accession number is NP_000192.2. | |||
TMPY-05830 | MICA Protein, Human, Recombinant (hFc), MICA*018 | Human | HEK293 Cells |
MICA Protein, Human, Recombinant (hFc), MICA*018 is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 59.86 kDa and the accession number is AAH16929.1. | |||
TMPH-00347 | Papain Protein, Carica papaya, Recombinant (His) | Carica papaya | E. coli |
Papain Protein, Carica papaya, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 27.4 kDa and the accession number is P00784. | |||
TMPH-03091 | Silicatein Protein, Petrosia ficiformis, Recombinant (His & Myc) | Petrosia ficiformis | E. coli |
Polymerizes silica around the axial filament during spicule formation. Silicatein Protein, Petrosia ficiformis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted... | |||
TMPH-03039 | ASP2 Protein, Necator americanus, Recombinant (His) | Necator americanus | E. coli |
ASP2 Protein, Necator americanus, Recombinant (His) is expressed in E. coli. | |||
TMPH-00034 | ASFV (isolate Tick/South Africa/Pretoriuskop Pr4/1996) p12 Protein (His) | ASFV | E. coli |
Virus attachment protein. ASFV (isolate Tick/South Africa/Pretoriuskop Pr4/1996) p12 Protein (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 12.7 kDa and the accession... | |||
TMPY-06086 | SARS-CoV-2 Helicase Protein (His) | SARS-CoV-2 | E. coli |
SARS-CoV-2 Helicase Protein (His) is expressed in E. coli expression system. The predicted molecular weight is 67.8 kDa and the accession number is YP_009725308.1. | |||
TMPH-00514 | Endo H Protein, Streptomyces plicatus, Recombinant (His) | Streptomyces plicatus | P. pastoris (Yeast) |
Cleaves asparagine-linked oligomannose and hybrid, but not complex, oligosaccharides from glycoproteins. | |||
TMPH-03716 | Invasin Protein, Yersinia enterocolitica, Recombinant (His & SUMO) | Yersinia enterocolitica | E. coli |
Invasin is a protein that allows enteric bacteria to penetrate cultured mammalian cells. The entry of invasin in the cell is mediated by binding several beta-1 chain integrins. | |||
TMPY-00825 | ICAM-1/CD54 Protein, Human, Recombinant (His & hFc) | Human | HEK293 Cells |
ICAM-1/CD54 Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 77.4 kDa and the accession number is A0A384MEK5. | |||
TMPH-02928 | Testican-2 Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
May participate in diverse steps of neurogenesis. Binds calcium. Testican-2 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is... | |||
TMPY-05189 | Bla g 1 Protein, Blattella germanica, Recombinant (His) | Blattella germanica | E. coli |
Bla g 1 Protein, Blattella germanica, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 46.8 kDa and the accession number is Q9UAM5. | |||
TMPH-02466 | Ribonuclease MC Protein, Momordica charantia, Recombinant (His & Myc) | Momordica charantia | E. coli |
Ribonuclease MC Protein, Momordica charantia, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 28.7 kDa and the accession number is P23540. | |||
TMPH-03719 | YopH Protein, Yersinia enterocolitica, Recombinant (His & Myc) | Yersinia enterocolitica | E. coli |
Essential virulence determinant. This protein is a protein tyrosine phosphatase. The essential function of YopH in Yersinia pathogenesis is host-protein dephosphorylation. It contributes to the ability of the bacteria to... | |||
TMPH-00385 | Chikungunya virus (strain S27-African prototype) Non-structural protein 4 (His) | CHIKV | E. coli |
Chikungunya virus (strain S27-African prototype) Non-structural protein 4 (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 31.1 kDa and the accession number is Q8JUX6. | |||
TMPH-00204 | Azurin Protein, Bordetella bronchiseptica, Recombinant (His & Myc) | Bordetella bronchiseptica | E. coli |
Azurin Protein, Bordetella bronchiseptica, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 20.8 kDa and the accession number is P0A321. | |||
TMPH-00444 | GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His & Myc) | Chinese hamster | E. coli |
GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-00452 | Polygalacturonase Protein, Cryptomeria japonica, Recombinant (His & SUMO) | Cryptomeria japonica | E. coli |
N/A. Polygalacturonase Protein, Cryptomeria japonica, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 58.2 kDa and the accession number is P4321... | |||
TMPY-00388 | ICAM-5 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
ICAM-5 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 87.2 kDa and the accession number is Q9UMF0. | |||
TMPH-03621 | CHRNA1 Protein, Tetronarce californica, Recombinant (His) | Tetronarce californica | HEK293 Cells |
After binding acetylcholine, the AChR responds by an extensive change in conformation that affects all subunits and leads to opening of an ion-conducting channel across the plasma membrane. CHRNA1 Protein, Tetronarce cal... | |||
TMPY-01320 | ICAM-1/CD54 Protein, Mouse, Recombinant (His & hFc) | Mouse | HEK293 Cells |
ICAM-1/CD54 Protein, Mouse, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 78.3 kDa and the accession number is P13597-1. | |||
TMPH-00346 | Limulus clotting factor C Protein, Carcinoscorpius rotundicauda, Recombinant (His) | Carcinoscorpius rotundicauda | E. coli |
This enzyme is closely associated with an endotoxin-sensitive hemolymph coagulation system which may play important roles in both hemostasis and host defense mechanisms. Its active form catalyzes the activation of factor... | |||
TMPY-00826 | ICAM-2/CD102 Protein, Human, Recombinant (His & hFc) | Human | HEK293 Cells |
ICAM-2/CD102 Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 50.3 kDa and the accession number is P13598. | |||
TMPH-03130 | Uricase Protein, Pig, Recombinant (His & SUMO) | Sus scrofa (Pig) | E. coli |
Catalyzes the oxidation of uric acid to 5-hydroxyisourate, which is further processed to form (S)-allantoin. Uricase Protein, Pig, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag.... | |||
TMPH-03307 | Glypican 3/GPC3 Protein, Rat, Recombinant (His) | Rat | P. pastoris (Yeast) |
Glypican 3/GPC3 Protein, Rat, Recombinant (His) is expressed in Yeast. | |||
TMPH-03620 | CHRNA1 Protein, Tetronarce californica, Recombinant (E. coli, His) | Torpedo californica | E. coli |
After binding acetylcholine, the AChR responds by an extensive change in conformation that affects all subunits and leads to opening of an ion-conducting channel across the plasma membrane. CHRNA1 Protein, Tetronarce cal... | |||
TMPY-00191 | ICAM-5 Protein, Human, Recombinant (aa 1-132,hFc) | Human | HEK293 Cells |
ICAM-5 Protein, Human, Recombinant (aa 1-132,hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 38.6 kDa and the accession number is Q9UMF0. | |||
TMPH-02731 | ICAM4 Protein, Mouse, Recombinant (His & SUMO) | Mouse | E. coli |
Adhesion molecule that binds to leukocyte adhesion LFA-1 protein LFA-1 (integrin alpha-L/beta-2). ICAM4 is also a ligand for alpha-4/beta-1 and alpha-V integrins. Isoform 2 may modulate binding of membrane-associated ICA... | |||
TMPY-01412 | Glypican 5 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
Glypican-5 (GPC5), is a cell membrane protein that belongs to the glypican family. The glypicans compose a family of glycosylphosphatidylinositol-anchored heparan sulfate proteoglycans that may play a role in the control... | |||
TMPY-01799 | ICAM-2/CD102 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
ICAM-2/CD102 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 50 kDa and the accession number is P35330. | |||
TMPY-01680 | Lumican Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Lumican, a prototypic leucine-rich proteoglycan with keratan sulfate side chains, is a major component of the cornea, dermal, and muscle connective tissues. In these bifunctional molecules, the protein moiety binds colla... | |||
TMPY-05142 | Blo t 1 Protein, Blomia tropicalis, Recombinant (His) | Blomia tropicalis | P. pastoris (Yeast) |
Blo t 1 Protein, Blomia tropicalis, Recombinant (His) is expressed in yeast with His tag. The predicted molecular weight is 37.7 kDa and the accession number is A1KXI0. | |||
TMPY-06877 | Glypican 3/GPC3 Protein, Human, Recombinant (His & Avi), Biotinylated | Human | HEK293 Cells |
Glypican 3/GPC3 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 64.05 kDa and the accession number is P51654-1. | |||
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