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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T14066 | 9-ING-41 | Apoptosis , GSK-3 , Autophagy | |
9-ING-41 is a glycogen synthase kinase-3 inhibitor. | |||
T6357 | (S)-crizotinib | ent-crizotinib | Apoptosis , DNA/RNA Synthesis , MTH1 |
(S)-crizotinib (ent-crizotinib) (IC50 of 72 nM), an effective MTH1 (NUDT1) inhibitor, is the (S)-enantiomer of crizotinib. | |||
T1488 | Procarbazine hydrochloride | NSC-77213 HCl,Procarbazine HCl | DNA Alkylator/Crosslinker , DNA/RNA Synthesis |
Procarbazine hydrochloride (NSC-77213 HCl) is the hydrochloride salt of a methylhydrazine derivative with antineoplastic and mutagenic activities. Although the exact mode of cytotoxicity has not been elucidated, procarba... | |||
T28503 | Ralitoline | GOE-4942,PD-117818,Ralitolina,CI-946,Ralitolinum | Others |
Ralitoline (Ralitolinum) is an anticonvulsant with anticancer activity and sodium channel blocking activity. | |||
T10721 | CD73-IN-1 | CD73 | |
CD73-IN-1 is a CD73 inhibitor with anticancer activity. | |||
T68159 | Tetrazolast | Antifungal | |
Tetrazolast has anticancer activity and may have antifungal activity. | |||
T70086 | EPZ033294 | Others | |
EPZ033294 has potential anticancer and antiproliferative activity. | |||
T84364 | (R)-Monepantel | (R)-AAD1566 | Others |
(R)-Monepantel ((R)-AAD1566) has potential anticancer activity but no nematicidal activity. | |||
T60002 | DC-S239 | Histone Methyltransferase | |
DC-S239 (DC-S239) is a selective inhibitor of histone methyltransferase SETD7 (IC50 = 4.59 μM) with anticancer activity. | |||
T12682 | Emzadirib | CYT-0851,RAD51-IN-2 | DNA/RNA Synthesis |
Emzadirib (RAD51-IN-2) is a potent RAD51 inhibitor with potential anticancer activity for the study of DNA damage repair. | |||
T13905 | Stilbamidine | Ba 2652,Stilbamidin | Antifungal |
Stilbamidine (Ba 2652) has antifungal and anticancer activity and can be used to study multiple myeloma and bladder migratory cell carcinoma. | |||
T60967 | Atg4B-IN-2 | Phospholipase , Autophagy | |
Atg4B-IN-2 is a potent and selective Atg4B inhibitor with anticancer activity that inhibits the activity of Atg4B and PLA2.Atg4B-IN-2 resists the anticancer activity of anti-desiccation-resistant prostate cancer drugs th... | |||
T20890 | Alvespimycin | 17-DMAG,KOS1022,KOS 1022,KOS-1022 | HSP |
Alvespimycin (17-DMAG) is a potent Hsp90 inhibitor with potential anticancer activity, which acts by binding to Hsp90. | |||
T35300 | Zeniplatin | Zeniplatinum | Others |
Zeniplatin (Zeniplatinum) is a new cisplatin complex with anticancer activity for the treatment of metastatic melanoma and kidney cancer. | |||
T8668 | HM03 | HSP | |
HM03 is a potent and selective inhibitor of HSPA5, and has anticancer activity. | |||
T15390 | Glufosfamide | D 19575,Glucosylifosfamide mustard | Others |
Glufosfamide is a novel oxazolophosphamide compound with anticancer activity for the study of advanced non-small cell lung cancer. | |||
T78210 | STC-15 | STC15 | Others |
STC-15 is an orally active and potent METTL3 inhibitor with anticancer activity that inhibits cancer growth and induces anticancer immunity. | |||
T36491 | POMHEX | Glucokinase | |
Pomhex, a cell-permeable potent enolase inhibitor with anticancer activity, is used in the study of cancer lethality.Pomhex, a racemic mixture, is a potent and selective ENO2 inhibitor.Pomhex is inhibitory to the glycoly... | |||
T15205 | EL-102 | EL102 | Microtubule Associated , HIF |
EL-102 is a HIF1α inhibitor with anticancer activity that inhibits microtubule protein polymerization and can be used to study prostate cancer. | |||
T10395L | ATM-3507 | Myosin | |
ATM-3507 is a protomyosin inhibitor with anticancer activity that inhibits human melanoma and can be used to study ovarian cancer. | |||
T13045 | Syk-IN-3 | Syk | |
Syk-IN-3 is a Syk inhibitor with potential anti-inflammatory and anticancer activity and can be used to study immune dysregulation. | |||
T14974 | Citenamide | Cytenamide,AY-15613 | Others |
Citenamide (AY-15613) has anticancer and anticonvulsant activity and is used in the study of neurological disorders because of its sleep-promoting properties. | |||
T4228 | Nolatrexed | DNA/RNA Synthesis | |
Nolatrexed is a thymidylate synthase inhibitor with potential anticancer activity. | |||
T70388L | (R)-Enitociclib | CDK | |
(R)-Enitociclib, an enantiomer of BAY-1251152, is a CDK9 inhibitor with anticancer activity. | |||
T13639 | Deferasirox (Fe3+ chelate) | Apoptosis | |
Deferasirox (Fe3+ chelate) is an orally available iron chelator with potential anticancer activity, inhibits the anti-apoptotic activity of MCL-1, and can be used to study iron overload. | |||
T23115 | OXF BD 02 | OXFBD02 | Epigenetic Reader Domain |
OXF BD 02 is a potent and selective BRD4(1) inhibitor (IC50: 382 nM) with anticancer and anti-inflammatory activity. | |||
T77558 | 5,7-Dimethoxy-4-methylcoumarin | Antioxidant | |
5,7-Dimethoxy-4-methylcoumarin has potential antioxidant antiproliferative and anticancer or activity. | |||
T25212 | CCCI-01 | CCCI 01,CCCI01,Centrosome Clustering Chemical Inhibitor-01 | Apoptosis |
CCCI-01(Centrosome Clustering Chemical Inhibitor-01) is a centrosome cluster inhibitor. CCCI-01 has anticancer activity, induces apoptosis, and can be used in the study of non-cross-resistant anticancer compounds that bl... | |||
T60012 | HS-243 | IRAK , MAPK , CDK | |
HS-243 is an inhibitor of IRAK-4 and IRAK-1 with IC50s of 20 and 24 nM. HS-243 shows anti-inflammatory and anticancer activity. | |||
T25829 | Mopidamol | RA233,RA 233,RA-233,Rapenton,OLX 102 | PDE |
Mopidamol (RA 233) is a phosphodiesterase inhibitor, a dipyridamole derivative, with anticancer activity that prevents retinal vascular defects in experimental diabetes. | |||
T8529 | WYC-210 | Others | |
WYC-210 is a retinoid compound,and with lower anticancer activity | |||
T21773 | SP-141 | SP 141 | Mdm2 |
SP 141 is a MDM2 inhibitor.SP-141 promotes MDM2 auto-ubiquitination and degradation, with anticancer activity. | |||
T70058 | PQR514 | PI3K | |
PQR514 is a potent PI3K inhibitor with anticancer activity and inhibits cancer cell proliferation. | |||
T15236 | Entasobulin | Microtubule Associated | |
Entasobulin is an inhibitor of β-tubulin polymerization. It has a potential anticancer activity. | |||
T27454 | GSK2008607 | Raf | |
GSK2008607 is a potent B-RafV600E inhibitor with anticancer activity and can be used to study breast, colorectal, melanoma, thyroid, and ovarian cancers. | |||
T23512 | VU 0364739 hydrochloride | VU 0364739 HCl | Apoptosis , Phospholipase |
VU 0364739 hydrochloride (VU 0364739 HCl) is a selective and potent inhibitor of phospholipase D2 (PLD2) with IC50s of 20 and 1500 nM for PLD2 and PLD1, respectively.VU 0364739 hydrochloride exhibits potential anticancer... | |||
T12577 | PTP1B-IN-3 | Phosphatase | |
PTP1B-IN-3 is a selective and potent PTP1B inhibitor with anticancer activity that inhibits PTP1B and TCPTP.PTP1B-IN-3 is used in the study of diabetes. | |||
T27257 | EMD-503982 | EMD503982,EMD 503982 | Factor Xa |
EMD-503982 is a potential Factor Xa and Factor VIIa inhibitor with potential anticancer and antitumor activity for the study of thromboembolic and neurological disorders. | |||
T15055 | DB04760 | MMP-13 Inhibitor | MMP |
DB04760 is a highly selective, non-zinc-chelating inhibitor of MMP-13 (IC50: 8 nM). DB04760 obviously decreases paclitaxel neurotoxicity and has anticancer activity. | |||
T34602 | Selatinib | EGFR | |
Selatinib is an orally active and potent dual inhibitor of EGFR and ErbB2 with anticancer activity that inhibits the growth of NCI-N87 tumor cells. | |||
T20158 | Phenformin | Debeone,N-Phenethylbiguanide,Insoral,BRN 1977317,Azucaps | Apoptosis |
Phenformin (BRN 1977317) is a biguanide compound with anticancer and anti-glycemic activity, inhibits skin tumor growth and promotes keratinocyte differentiation and apoptosis. | |||
T16777 | ROC-325 | Apoptosis , Autophagy | |
ROC-325 is an effective and orally active inhibitor of autophagy with anticancer activity. ROC-325 induces renal cell carcinoma apoptosis and exhibits favorable selectivity. | |||
T16866 | SDZ281-977 | SDZ-LAP 977 | EGFR |
SDZ281-977 (SDZ-LAP 977) is a derivative of Lavendustin A. It exhibits anticancer and antiplusative activity and inhibits the growth of human vulvar cancer cells. | |||
T60852 | Anticancer agent 46 | Others | |
Anticancer agent 46 is a potent anti-cancer agent, showing anti-proliferative activity in cellular assays, with an IC50 of 0.986 μM against MGC803 cells. | |||
T69742 | SRX3177 | Epigenetic Reader Domain , PI3K , CDK | |
SRX3177 is a novel and potent inhibitor of BRD4, PI3K and CDK.SRX3177 has potential anticancer activity. | |||
T60564 | PI3K/Akt/mTOR-IN-2 | Apoptosis , Akt , PI3K , mTOR | |
PI3K/Akt/mTOR-IN-2 is a potent PI3K/AKT/mTOR inhibitor.PI3K/Akt/mTOR-IN-2 has anticancer effects and is selective for MDA-MB-231 cells with an IC50 of 2.29 μM.PI3K/Akt/mTOR-IN-2 exhibits anticancer activity and induces c... | |||
T7208 | AMD 3465 hexahydrobromide | GENZ-644494 (hexahydrobromide) | HIV Protease , CXCR |
AMD 3465 hexahydrobromide (GENZ-644494 (hexahydrobromide)) is a CXCR4 receptor antagonist with potential anticancer and anti-HIV activity. | |||
T62620 | ZY-444 | Others | |
ZY-444 has potential anticancer activity, inhibits PCa cell proliferation and metastasis, and inhibits the growth of subcutaneous tumors. | |||
T77734 | ERK5-IN-5 | ERK | |
ERK5-IN-5 is a potent extracellular signal-regulated kinase 5 (ERK5) inhibitor with anticancer activity and potential anticonvulsant activity that inhibits A549 cell proliferation. | |||
T22830 | GYY4137 | GYY 4137 morpholine salt | Others |
GYY4137 (GYY 4137 morpholine salt) is a novel water-soluble and slow releasing H2S donor with vasodilator and antihypertensive activity. GYY4137 also exhibits anti-inflammatory and anticancer activity. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T2763 | Panaxadiol | 20(R)-Panaxadiol | Others , HIF/HIF Prolyl-Hydroxylase |
Panaxadiol (20(R)-Panaxadiol) is a novel antitumor agent extracted from the Chinese medical herb Panax ginseng. | |||
T2230 | Paeoniflorin | Peoniflorin | HSP , COX |
Paeoniflorin (Peoniflorin) is a herbal constituent extracted from the root of Paeonia albiflora Pall. | |||
T0687 | Simvastatin | MK-0733,MK 733 | Apoptosis , Mitophagy , Ferroptosis , HMG-CoA Reductase , Autophagy |
Simvastatin (MK 733) is an HMG-CoA reductase inhibitor (Ki=0.2 nM) with oral activity. Simvastatin has hypolipidemic activity, inhibits hepatic production of cholesterol, and is also used for the prevention of cardiovasc... | |||
T4952 | 9-Hydroxycamptothecin | 9-HCPT,10-Hydroxycampothecin | Topoisomerase |
9-Hydroxycampothecin is a camptothecin derivative with anticancer activity. | |||
TN7226 | 2-Hydroxy-3-methoxy chalcone | ||
2-Hydroxy-3-methoxy chalcone has anticancer activity and inhibits colon cancer. | |||
T3S1957 | 9-amino-CPT | Aminocamptothecin,9-amino-2(S)-camptothecin,9-Aminocamptothecin | Topoisomerase |
9-amino-CPT (Aminocamptothecin) is an inhibitor of topoisomerase I with potent anticancer activity. | |||
T3S1265 | Liriopesides B | Nolinospiroside F | Others |
Liriopesides B (Nolinospiroside F) exhibited potential anticancer activity against human ovarian cancer A2780 cells. | |||
T5S1252 | Prosapogenin A | Progenin III | Apoptosis , Others |
Prosapogenin A (Progenin III) has anticancer activity. | |||
T8213 | Isolinderalactone | NOS , STAT | |
Isolinderalactone shows anti-inflammatory and anticancer capacity, and it exhibits moderate iNOS inhibitory activity, with the IC50 value of 0.30 uM. | |||
T6S0141 | Corylin | Antibacterial , Antibiotic , STAT | |
Corylin is a major bioactive compound isolated from Psoralea corylifolia L; it has the activity of antibiotic or anticancer. | |||
T19154 | 5-Methyl-2-thiophenecarboxaldehyde | Others | |
5-Methyl-2-thiophenecarboxaldehyde is a candidate microscopic third-order nonlinear optical (NLO) material.5-Methyl-2-thiophenecarboxaldehyde possesses a wide range of biological activities, such as anticancer activity. | |||
T4S2012 | Dihydrosanguinarine | 13,14-Dihydrosanguinarine,Dihydro Sanguinarine | Caspase , Antifungal |
Dihydrosanguinarine is a natural compound isolated from the leaves of Macleaya microcarpa,and has antifungal and anticancer activity. | |||
T0595 | Naringin | Naringoside | Mitophagy , P450 , Endogenous Metabolite , Autophagy |
Naringin (Naringoside), a flavanone glycoside, exerts various of pharmacological effects such as blood lipid lowering, antioxidant activity, anticancer activity, and inhibition of cytochrome P450 enzymes. | |||
T3819 | Ursolic acid acetate | Acetylursolic acid,3-Acetylursolic Acid | AChE |
Ursolic acid acetate (Acetylursolic acid) has cytotoxic activity, antimalarial activity, antitumor and anticancer activities. Acetylursolic acid has NO production inhibitory activities. Acetylursolic acid has inhibition ... | |||
T10584 | Bovinic acid | (9Z,11E)-Octadecadienoic acid,Rumenic acid | Endogenous Metabolite |
Bovinic acid ((9Z,11E)-Octadecadienoic acid) is a conjugated linoleic acid with anticancer and anti-atherosclerotic activity and can be used to study coronary heart disease and obesity in the elderly. | |||
T4S0051 | Coptisine sulfate | Indoleamine 2,3-Dioxygenase (IDO) | |
1. Coptisine sulfate has growth inhibitory activity against human cancer cell line in the NCI's anticancer drug screening program. | |||
T2S0837 | Astragalus Polysacharin | 2-(Chloromethyl)-4-(4-nitrophenyl)thiazole,89250-26-0 | TAM Receptor |
2-(Chloromethyl)-4-(4-nitrophenyl)thiazole is a natural product derived from Astragalus propinquus.2-(Chloromethyl)-4-(4-nitrophenyl)thiazole exhibits anticancer activity. 2-(Chloromethyl)-4-(4-nitrophenyl)thiazole posse... | |||
T8201 | Gambogenic acid | Histone Methyltransferase | |
Gambogenic acid is a natural product,is an effective inhibitor of EZH2,with anticancer activity. | |||
T2831 | Glycocholic acid | Glycocholate,cholylglycine | Others , Endogenous Metabolite |
Glycocholic acid (Glycocholate) is a bile acid with anticancer activity. Glycocholic acid targets against pump resistance-related and non-pump resistance-related pathways. | |||
TN1894 | Luteolin-4'-O-glucoside | Luteolin-4'-glucoside,Luteolin-4-o-glucoside | IL Receptor |
TN3543 | Bruceoside A | Others | |
Bruceoside A is a bitter wood glycoside that can be isolated from opuntia and has anticancer and tumor activity and can be used with the study of leukemia. | |||
T3898 | Schaftoside | APIGENIN-6-GLUCOSIDE-8-ARABINOSIDE,Shaftoside | Dynamin , Antioxidant , TLR , MyD88 , Mitochondrial Metabolism , Autophagy |
Schaftoside (APIGENIN-6-GLUCOSIDE-8-ARABINOSIDE) has antioxidant and anticancer activity. | |||
TN1745 | Hosenkoside M | (+)-Hosenkoside M | Others |
Hosenkoside M is a bazaine glycoside extracted from the balsam seeds of Fenugreek, which has anticancer activity and is used in the study of prostate cancer. | |||
TN1464 | Camellianin A | RAAS | |
Camellianin A has anticancer activity, it can inhibit the proliferation of the human hepatocellular liver carcinoma Hep G2 and human breast adenocarcinoma MCF-7 cell lines in a dose-dependent manner and induce the signif... | |||
T36528 | Illudin M | Apoptosis , DNA Alkylator/Crosslinker | |
Illudin M is a cytotoxic sesquiterpene from the fungus O. illudens that alkylates DNA. It has a cytotoxicity of 6-100 nM against HL-60 human leukemia cells.Illudin M has anticancer activity and is a pre-drug for the synt... | |||
T7059 | α-Dihydroartemisinin | α-Artenimol,α-Dihydroqinghaosu | Parasite |
α-Dihydroartemisinin (α-Dihydroqinghaosu) is an intermediate of artemisinin-based antimalarial compounds with good antimalarial and anticancer activity, and can be used in the study of lupus erythematosus. | |||
TQ0309 | Glaucocalyxin B | Autophagy | |
T3339 | Sophoridine | 5-Epidihydrosophocarpine,Dihydro-5-episophocarpine | Apoptosis , Topoisomerase |
Sophoridine (Dihydro-5-episophocarpine), a natural anticancer drug, has been used in China for decades. A series of novel N-substituted Sophoridinic acid derivatives were synthesized and evaluated for their cytotoxicity ... | |||
T7441 | Cuminaldehyde | Cuminic aldehyde,Cuminal | Endogenous Metabolite |
Cuminaldehyde (Cuminal) is a natural aldehyde with inhibitory effect on alpha-synuclein fibrillation and cytotoxicity. Cuminaldehyde shows anticancer activity,with a pleasant smell and contributes to the aroma of essenti... | |||
T3425 | Polyphyllin G | Polyphyllin VII,Polyphyllin VII,Y-0166 | Others |
Polyphyllin G (Polyphyllin VII), the the main member of polyphyllin family, shows strong anticancer activity against several carcinomas, including lung cancer, breast cancer, colorectal cancer, cervical cancer, hepatocel... | |||
T83321 | 4-Demethyldeoxypodophyllotoxin | Chk | |
4-Demethyldeoxypodophyllotoxin, an aryl tetrahydronaphthalenyl lignan analog from the roots of Podophyllum peltatum, has anticancer activity and modulates the Chk-2 signaling pathway in MCF-7 breast cancer cells. | |||
T5S1285 | (+)-(3R,8S)-Falcarindiol | Falcarindiol | Others |
1. (+)-(3R,8S)-Falcarindiol is a potential new anticancer agent that exerts its activity through inducing ER stress and apoptosis. 2. Falcarindiol induces immunosuppressive effects in vitro and in vivo and might be a nov... | |||
TN5254 | Wighteone | Erythrinin B,6-Isopentenylgenistein | Antifungal |
Wighteone (Erythrinin B) is a small molecule compound derived from Genista ephedroides with potential antifungal and anticancer activity against EGFR L858R/T790M mutant non-small cell lung cancer. | |||
T3391 | Corosolic acid | Corsolic acid,2α-Hydroxyursolic acid,Glucosol,Colosolic acid,Colosic acid | FAK , Autophagy |
Corosolic acid (Colosic acid) contains anti-angiogenic activity that can suppress FAK signaling induced by angiopoietin-1. Corosolic acid exerts anticancer activities against HCC, colon, and colorectal Y cells, by induci... | |||
T3398 | Icaritin | Anhydroicaritin,Cycloicaritin | Apoptosis , JAK , STAT , Autophagy |
Icaritin (Anhydroicaritin) has hormone regulation activity and cardiovascular function improvement activity. Icaritin has anticancer activity, can induce S phase arrest and apoptosis, inhibit ENKL cell proliferation. Ica... | |||
T7054 | N-Benzoyl-(2R,3S)-3-phenylisoserine | taxol side chain | Antiviral |
N-Benzoyl-(2R,3S)-3-phenylisoserine (taxol side chain) is an intermediate in the preparation of potent anticancer drug Paclitaxel, used to study the location of the binding sites. It shows cytotoxic, antiviral and immuno... | |||
TN1727 | Helichrysetin | Apoptosis , HIV Protease | |
Helichrysetin has mild anti-HIV-1 PR activity. Helichrysetin has great potentials for development as an anticancer agent, it has cytotoxic effect on four selected cancer cell lines, A549, MCF-7, Ca Ski, and HT-29. | |||
TN1019 | Beta-mangostin | β-Mangostin | Apoptosis , Antibacterial , Parasite |
Beta-mangostin (β-Mangostin) is a xanthone compound with antibacterial and antimalarial activities. Beta-mangostin present in Cratoxylum arborescens and exhibits antimycobacterial activity against Mycobacterium tuberculo... | |||
TNU0052 | Nebularine | 9-(beta-D-Ribofuranosyl)-9H-purine | Apoptosis |
Nebularine (9-(beta-D-Ribofuranosyl)-9H-purine) is a purine nucleoside analog with a broad spectrum of antitumor activity, targeting inert lymphoid malignancies and inducing apoptosis.The anticancer mechanism of Nebulari... | |||
TN2083 | Pinostrobin chalcone | ||
Pinostrobin chalcone, a chalcone analog isolated from the leguminous plant, Mucuna pruriens, exhibits anticancer activity with an IC50 value of 20.42±2.23 μg/mL against MDA-MB-231 and 22.51±0.42 μg/mL against the HT-29 c... | |||
T3404 | Cucurbitacin B | Cuc B,DATISCACIN,Amarine | Apoptosis , PTEN , Integrin , Endogenous Metabolite , HIF , STAT , Autophagy |
Cucurbitacin B (Cuc B) has profound in vitro and in vivo antiproliferative effects against human pancreatic Y cells. It inhibited AKT signaling activation through up-regulation of PTEN. Cucurbitacin B is an effective inh... | |||
TN1040 | Skullcapflavone II | COX , Antibacterial , TGF-beta/Smad | |
Skullcapflavone II is a flavonoid derived from Scutellaria baicalensis, a widely used herbal medicine in anti-inflammatory and anticancer therapy. Skullcapflavone II may have therapeutic potential for the treatment of al... | |||
TN3628 | Chamaejasmenin B | Others | |
Chamaejasmenin B is a compound isolated from Stellera chamaejasme L. Chamaejasmenin B has anticancer and antitumor activity, inhibiting cancer cell migration and invasion, and inhibiting tumor metastasis.Chamaejasmenin B... | |||
T3410 | Momordin Ic | Momordin 1c | Apoptosis , MAPK , PI3K |
Momordin Ic (Momordin 1c) might represent a potential anticancer activity, by inducing apoptosis through oxidative stress-regulated mitochondrial dysfunction involving the MAPK and PI3K-mediated iNOS and HO-1 pathways. A... | |||
TN1376 | α-Solanine | alpha-Solanine | Apoptosis , NF-κB |
α-Solanine (alpha-Solanine) is an alkaloid derived from potato with anticancer and antitumor activity, attenuating chondrocyte death by inhibiting the NF-κB pathway. α-Solanine inhibits the proliferation and migration of... | |||
T5S2017 | Ingenol | (-)-Ingenol | PKC |
1. Ingenol ((-)-Ingenol) mebutate is an effective treatment for actinic keratosis. 2. Formulating novel derivatives from Ingenol esters may be an innovative approach to develop new lead compounds to reactivate latent HIV... | |||
T3824 | Jaceosidin | Apoptosis , BCL , COX , UGT | |
Jaceosidin has anti-oxidative activity. Jaceosidin has anti-inflammatory activity, also a microglial inhibitor with anti-neuroinflammation activity. aceosidin has anticancer activity, modulates the ERK/ATM/Chk1/2 pathway... | |||
TN1065 | Hirsutine | Apoptosis | |
Hirsutine induces apoptosis and is a potent Dengue virus inhibitor exhibiting low cytotoxicity.Hirsutine has anticancer, cardioprotective, anti-hypertensive and anti-arrhythmic activities, it also has vasodilatation acti... | |||
T30969 | Clitocine | Apoptosis , BCL | |
Clitocine, an adenosine analogue derived from mushrooms, is a potent transcriptional readout agent, an inhibitor of nonsense mutations, and has anticancer activity, inducing the production of p53 protein in cells carryin... | |||
TN1249 | 3-Epiursolic acid | Cysteine Protease , Immunology/Inflammation related | |
3-Epiursolic acid may have antiinflammatory activity, it shows inhibition on Cathepsins L (catL), the IC50 value of 6.5 μM, cathepsins L (catL) and B play an important role in tumor progression and have been considered p... | |||
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カタログ番号 | 製品名 | Species | Expression System |
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TMPY-01865 | BLMH Protein, Mouse, Recombinant (His) | Mouse | E. coli |
The papain superfamily member bleomycin hydrolase (BLMH) is a cytoplasmic cysteine peptidase that is highly conserved through evolution. The only known activity of the enzyme is metabolic inactivation of the glycopeptide... | |||
TMPY-02072 | HSF1 Protein, Human, Recombinant (His) | Human | E. coli |
Heat shock factor protein 1, also known as heat shock transcription factor 1, HSF1, and HSTF1, is a cytoplasm and nucleus protein that belongs to the HSF family. HSF1 is the major transcription factor of HSPs (heat shock... |
カタログ番号 | 製品名 | ||
---|---|---|---|
L6110 | Alkaloid Natural Product Library | 464 compounds | |
A unique collection of 464 natural alkaloids can be used for high throughput and high content screening; | |||
L2160 | Anti-Cancer Active Compound Library | 3188 compounds | |
A unique collection of 3188 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS); | |||
L1100 | Protease Inhibitor Library | 343 compounds | |
A unique collection of 343 protease and proteasome inhibitors for research in chemical genomics, and drug screening; | |||
L6700 | Anti-Tumor Natural Product Library | 1772 compounds | |
A unique collection of 1772 natural products with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS); |