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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T2072 | BET bromodomain inhibitor | Epigenetic Reader Domain | |
BET bromodomain inhibitor is a potent BET inhibitor. | |||
T10521 | ODM-207 | BET-IN-4,ODM207 | Epigenetic Reader Domain |
ODM-207 (BET-IN-4) is a potent BRD4 inhibitor. | |||
T39374 | PROTAC BET Degrader-10 | PROTACs | |
PROTAC BET Degrader-10 (WO2017007612A1, example 37) is a highly efficient and selective small molecule compound designed to degrade BET protein BRD4. PROTAC BET Degrader-10 functions by utilizing specific ligands that co... | |||
T39998 | BET bromodomain inhibitor 1 | ||
BET bromodomain inhibitor 1 is an orally active, selective inhibitor of bromodomain and extra-terminal (BET) proteins. It specifically inhibits BRD4 with an IC50 of 2.6 nM. Additionally, BET bromodomain inhibitor 1 demon... | |||
T10518 | BET-BAY 002 | Others | |
BET-BAY 002 is an effective BET inhibitor and exhibits efficacy in a multiple myeloma model. | |||
T10520 | BET-IN-2 | Epigenetic Reader Domain | |
BET-IN-2 is a BET inhibitor (IC50: 52 nM for BRD4-BD1). | |||
T10522 | BET-IN-6 | Epigenetic Reader Domain | |
BET-IN-6, a ligand with potent and high affinity for inhibiting BRD2/BRD4, plays a crucial role in the synthesis of PROTAC BRD2/BRD4 degrader-1 [1], targeting the protein BRD2/4. | |||
T13850 | PROTAC BET degrader-3 | Epigenetic Reader Domain | |
PROTAC BET Degrader-3 is a potent degrader OF BET based on PROTAC. | |||
T12559 | PROTAC BET degrader-2 | Others , PROTACs | |
PROTAC BET degrader-2 is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins (IC50 of 9.6 nM ). | |||
T13849 | PROTAC BET Degrader-1 | Epigenetic Reader Domain , PROTACs | |
PROTAC BET Degrader-1 is a potent degrader of BET based on PROTAC. | |||
T1906 | Molibresib | GSK 525762A,GSK525762,I-BET 762 | Epigenetic Reader Domain |
Molibresib (GSK525762) is an inhibitor of BET proteins (IC50: about 35 nM). | |||
T10517 | BET-BAY 002 (S enantiomer) | Others | |
The S-enantiomer of BET-BAY 002, referred to as BET-BAY 002 S enantiomer, is a potent inhibitor of BET (Bromodomain and Extra-Terminal motif proteins). | |||
T12557 | PROTAC BET-binding moiety 1 | Others | |
PROTAC BET-binding moiety 1 is a key intermediate in the synthesis of high affinity BET inhibitors | |||
T12558 | PROTAC BET-binding moiety 2 | Others | |
PROTAC BET-binding moiety 2 is an BET bromodomain inhibitor. | |||
T9619 | I-BET567 | ||
I-BET567, a potent pan-BET inhibitor with oral activity, demonstrates pIC50 values of 6.9 and 7.2 for BRD4 BD1 and BD2, respectively. This compound has exhibited efficacy in mouse models of oncology and inflammation [1]. | |||
T79610 | BET-IN-17 | Epigenetic Reader Domain | |
BET-IN-17, also known as compound 16, serves as a pan-inhibitor for BET, exhibiting inhibitory potencies (pIC50) of 7.8 for BET BD1 and 7.6 for BET BD2 [1]. | |||
T79167 | BET-IN-15 | Epigenetic Reader Domain | |
BET-IN-15 (compound 1) is a potent, orally active inhibitor of BET, demonstrating inhibitory IC50 values of 0.64 nM for BRD4-BD1 and 0.25 nM for BRD4-BD2. It exhibits antiproliferative activity [1]. | |||
T61795 | BET-IN-9 | ||
BET-IN-9 is a BET inhibitor[1]. | |||
T62055 | NVS-BET-1 | ||
NVS-BET-1 is a BET bromodomain inhibitor. NVS-BET-1 can regulate keratinocyte plasticity. | |||
T62275 | BET-IN-8 | ||
BET-IN-8 (Compound 27) is a potent inhibitor of BET (Ki: 0.83 μM, Kd: 0.571 μM), which ameliorates LPS-induced sepsis in vivo.BET-IN-8 has shown potential in sepsis. | |||
T2120 | I-BET151 | GSK1210151A | Epigenetic Reader Domain |
I-BET151 (GSK1210151A) (GSK1210151A) is a specific BET inhibitor for BRD2/3/4 (IC50: 0.5/0.25/0.79 μM, in cell-free assays). | |||
T63299 | BET-IN-1 | ||
BET-IN-1 is a potent inhibitor of BET, exhibiting good brain permeability and a reasonable metabolic stability. | |||
T79016 | BET-IN-14 | Epigenetic Reader Domain | |
BET-IN-14 is a pan BET inhibitor with an IC50 of 5.35 nM, demonstrating oral activity and anticancer properties [1]. | |||
T61253 | BET-IN-7 | ||
BET-IN-7 (Compound 1) is a highly effective BET inhibitor, possessing a K i of 12.27 μM and a K d of 89.3 μM. It exhibits promising properties for sepsis-related research [1]. | |||
T78989 | BET-IN-16 | Epigenetic Reader Domain | |
BET-IN-16 (Comp I), a bromodomain and extra-terminal (BET) inhibitor, demonstrates anticancer activity by impeding the growth of prostate cancer cells. It exhibits potent inhibitory effects with half-maximal inhibitory c... | |||
T62655 | BET bromodomain inhibitor 2 | ||
BET bromodomain inhibitor 2 is a potent inhibitor of the BET-type bromodomain (IC50: 14.1 μM). | |||
T79527 | BET BD2-IN-1 | Epigenetic Reader Domain | |
BET BD2-IN-1 (compound 45) is a potent, selective inhibitor of BET BD2, exhibiting an IC50 value of 1.6 nM. It suppresses Th17 cell differentiation through the reduced activation of STAT3 and NF-κB, making it relevant in... | |||
T72872 | HDAC/BET-IN-1 | HDAC | |
HDAC/BET-IN-1 is a chemical compound exhibiting submicromolar inhibitory activity against HDAC1 and HDAC6, with IC50 values of 0.163 μM and 0.067 μM, respectively, and against BRD4, with a Ki of 0.076 μM. Additionally, i... | |||
T22845 | I-BET151 dihydrochloride | I-BET 151 hydrochloride | Others |
I-BET 151 dihydrochloride is a BET bromodomain inhibitor that prevents BET from recruiting to chromatin. | |||
T79084 | BET bromodomain inhibitor 3 | Epigenetic Reader Domain | |
BET Bromodomain Inhibitor 3 is a BET bromodomain inhibitor with an inhibitory Ki value of >40 µM against BrdT. It is utilized in research related to contraception, cancer, and heart disease [1]. | |||
T6021 | GSK1324726A | I-BET726 | Apoptosis , Epigenetic Reader Domain |
GSK1324726A (I-BET726) is a greatly specific inhibitor of BET family proteins for BRD2(IC50=41 nM), BRD3(IC50=31 nM), and BRD4 (IC50=22 nM). | |||
T11472L | Molibresib besylate | I-BET 762 besylate,GSK 525762C | CCR |
Molibresib besylate is an inhibitor of BET bromodomain (IC50: 32.5-42.5 nM). | |||
T6828 | ZL0420 | Epigenetic Reader Domain | |
ZL0420 is a potent and selective bromodomain-containing protein 4 ( BRD4 ) inhibitor with nanomolar binding affinities to bromodomains (BDs) of BRD4. ZL0420 has IC 50 values of 27 nM against BRD4 BD1 and 32 nM against B... | |||
T70003 | I-BET469 | ||
I-BET469 is a Bromodomain and Extraterminal Inhibitor with a Low Predicted Human Dose. | |||
T17881 | (S,R,S)-AHPC-C10-NH2 | VH032-C10-NH2 | Others , Ligand for E3 Ligase |
(S,R,S)-AHPC-C10-NH2 (VH032-C10-NH2) is a synthesized E3 ligase ligand-linker conjugate, comprising the (S,R,S)-AHPC-based VHL ligand and a linker, designed for BET-targeted PROTAC applications. | |||
T6859 | I-BRD9 | GSK602 | Epigenetic Reader Domain |
I-BRD9 (GSK602) is the first selective cellular inhibitor for BRD9 with pIC50 of 7.3. | |||
T40031 | Thalidomide-O-C6-NH2 hydrochloride | 4-((6-aminohexyl)oxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride | E3 Ligase Ligand-Linker Conjugate |
Thalidomide-O-C6-NH2 hydrochloride (4-((6-aminohexyl)oxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride) is a synthesized E3 ligase ligand-linker conjugate. | |||
T13086 | I-BET762 carboxylic acid | Molibresib carboxylic acid,PROTAC BRD4-binding moiety 2,GSK525762A carboxylic acid | Epigenetic Reader Domain |
I-BET762 carboxylic acid is an inhibitor of BRD4(pIC50 of 5.1). | |||
T18661 | (S,R,S)-AHPC-C10-NH2 dihydrochloride | VH032-C10-NH2 dihydrochloride,VH032-linker 10,VH032 amide-alkylC10-amine | Others , Ligand for E3 Ligase |
(S,R,S)-AHPC-C10-NH2 dihydrochloride (VH032-linker 10) is a synthesized E3 ligase ligand-linker conjugate incorporating the (S,R,S)-AHPC based VHL ligand and a linker[1]. | |||
T5130 | DBET6 | Apoptosis , Epigenetic Reader Domain , PROTACs | |
dBET6 is a selective and cell-permeable degrader of BET based on PROTAC (IC50: 14 nM). It has antitumor activity. | |||
T4495 | DBET1 | Epigenetic Reader Domain , PROTACs | |
dBET1 is a hybrid molecule that combines (+)-JQ1 and thalidomide. It induces cereblon-dependent BET protein degradation in vitro (EC50: 430 nM) and induces apoptosis. | |||
T14550 | BETd-260 | ZBC 260 | Epigenetic Reader Domain , PROTACs |
BETd-260, a PROTAC linked by a Cereblon ligand and a BET ligand, has an inhibitory effect on BRD4 protein in leukemic cell lines. | |||
T2480 | Apabetalone | RVX-208,RVX000222 | Epigenetic Reader Domain , HIV Protease |
Apabetalone (RVX000222) , an effective BET bromodomain inhibitor, has been investigated for the treatment of diabetes, atherosclerosis, and coronary artery disease. | |||
T4195 | Betahistine | PT 9 base,Vasomotal,Serc base | Histamine Receptor |
Betahistine (Vasomotal) is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but may exacerbate bronchial asthma and peptic ulcers. Betahisti... | |||
T0464 | Carbetapentane citrate | Pentoxyverine citrate | AChR |
Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold. | |||
T76743 | Emibetuzumab | LY2875358 | c-Met/HGFR |
Emibetuzumab is a potent humanized bivalent MET antibody (IgG4 type). Emibetuzumab has antitumor activity, inhibition of HGF-dependent and independent MET pathway activation and tumor growth, and can be used to study adv... | |||
TNU0168 | 2'-Deoxy-2'-fluoro-beta-D-arabinoguanosine | Apoptosis | |
2'-Deoxy-2'-fluoro-beta-D-arabinoguanosine is a purine nucleoside analog with a broad spectrum of antitumor activity, targeting malignant tumors of the inert lymphatic system and inducing apoptosis. The anticancer mechan... | |||
T5440 | Dbet57 | Epigenetic Reader Domain , PROTACs | |
dBET57 is heterobifunctional degrader of BRD4 based on the PROTAC technology, exhibits significant degradation of BRD4BD1 with a DC50/5h of 500 nM ,and inactive on BRD4BD2 | |||
T9435 | 1-(4-Carbethoxyphenyl)-piperazin | Others | |
1-(4-Carbethoxyphenyl)-piperazin is used as a reagent for enzymes and chemical synthesis, as a model substrate for enzyme studies, and as a ligand for receptor binding assays. | |||
T12468 | PI4KIIIbeta-IN-10 | PI3K , PI4K | |
PI4KIIIbeta-IN-10 is a potent inhibitor of PI4KIIIβ (IC50 of 3.6 nM). |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
TN2539 | 1beta-Hydroxyalantolactone | IL Receptor , TNF | |
1beta-Hydroxyalantolactone is a small molecular compound isolated from the flower head of the medicinal plant giant British flower, which can inhibit the expression of TNF-α, IL-17 and IFN-γ in cells, promote the secreti... | |||
T2S0765 | Epibetulinic acid | NO Synthase , Prostaglandin Receptor | |
Epibetulinic acid has anti-inflammatory activity, it exhibits potent inhibitory effects on NO and prostaglandin E(2) production in mouse macrophages (RAW 264.7) stimulated with bacterial endotoxin. | |||
T2S2018 | 7beta-Hydroxylathyrol | 7β-Hydroxylathyrol,7-Hydroxylathyrol,7-beta-Hydroxylathyrol | P-gp |
7β-Hydroxylathyrol is a diterpenoid extract from the seed oil of Caper Spurge and displays P-gp inhibition resulting in cytotoxic properties. | |||
T3S2152 | 23-Hydroxybetulinic acid | Anemosapogenin | Others |
23-Hydroxybetulinic acid (Anemosapogenin) shows potent anti-tumor effect in vivo, but it has some toxicity, structure modification should be needed. | |||
T3121 | Betulin | Trochol,betulinic alcohol,betuline,betulinol,Betulol | Apoptosis , Endogenous Metabolite , Lipid , Fatty Acid Synthase |
Betulin (betulinol) (lup-20(29)-ene-3β, 28-diol) is an abundant, naturally occurring triterpene. It is commonly isolated from the bark of birch trees where it forms up to 30% of the dry weight of the extractive and is fo... | |||
T4S2128 | Bilobetin | PKA , PPAR | |
Bilobetin ameliorates insulin resistance by PKA-mediated phosphorylation of PPARα in rats fed a high-fat diet. | |||
T3825 | Lobetyolin | Praeruptorin D | Others |
Lobetyolin (Praeruptorin D) is compound derived from Codonopsis pilosula with antioxidative effect. | |||
TN1441 | Beta-Tocopherol | ERK , MAPK | |
Beta-Tocopherol shows effect on human erythroleukemia cell (HEL) adhesion induced by phorbol 12-myristate 13-acetate (PMA). | |||
T8166 | Pennogenin 3-O-beta-chacotrioside | Autophagy | |
Pennogenin 3-O-beta-chacotrioside is an active component isolated from Paris polyphylla with anti-colorectal cancer activity. It modulates autophagy via increasing the expressions of autophagy-related proteins LC3 and Be... | |||
T14001 | 11-Beta-hydroxyandrostenedione | NSC-17102,4-Androsten-11β-ol-3,17-dione | Endogenous Metabolite |
11-Beta-hydroxyandrostenedione (NSC-17102) is a steroid mainly found in the adrenal origin (11β-hydroxylase is present in adrenal tissue, but absent in ovarian tissue), which is a 11β-hydroxysteroid dehydrogenase isozyme... | |||
T5S0018 | Betulonic acid | (+)-Betulonic acid,Betunolic acid,Liquidambaric acid | Parasite , HSV |
1. Betulonic acid (Liquidambaric acid) amide stimulated the regenerative response in hepatocytes under conditions of combined toxic exposure and promoted recovery of their qualitative and quantitative characteristics, wh... | |||
T13092 | Tauro-Obeticholic acid | FXR | |
Tauro-Obeticholic acid is an active Obeticholic acid metabolite. Obeticholic acid is an orally bioavailable agonist of farnesoid-X receptor (FXR). | |||
T2830 | Betulinic acid | ALS-357,Lupatic acid,Betulic acid | Apoptosis , Mitophagy , NF-κB , HIV Protease , Topoisomerase , Endogenous Metabolite , Aminopeptidase , Autophagy |
Betulinic acid (ALS-357) is a pentacyclic lupane-type triterpene derivative of betulin (isolated from the bark of Betula alba, the common white birch) which has antiretroviral, antimalarial, and anti-inflammatory propert... | |||
T1373 | AC-Beta-ALA-OH | Amino Acids and Derivatives | |
It is an organic compounds with molecular fomula C5H9NO3. | |||
TN7212 | Acacetin-7-O-beta-D-galactopyranoside | Others | |
Acacetin-7-O-beta-D-galactopyranoside is a natural product found in Chrysanthemum indicum. | |||
TN4674 | Nortrachelogenin-8'-O-beta-glucoside | Others | |
Nortrachelogenin-8'-O-beta-glucoside is a lignan with a diarylhydroxybutyrolactone skeleton which isolated from the leaves and stems of Trachelospermum jasminoides (Lindl.) Lem. | |||
TN1255 | 3-O-Acetyl-11-hydroxy-beta-boswellic acid | Lipoxygenase | |
3-O-Acetyl-11-hydroxy-beta-boswellic acid is the precursor of 3-O-acetyl-9, 11-dehydro-beta-boswellic acid(a 5-lipoxygenase inhibitor ). | |||
TN1260 | 3-O-beta-D-Glucopyranosylplatycodigenin | Others | |
3-O-beta-D-Glucopyranosylplatycodigenin is isolated from the roots of Platycodon grandiflorum. | |||
T3243 | Betaine | Abromine,glycine betaine,oxyneurine,trimethylglycine,lycine | Others , Endogenous Metabolite |
Betaine (trimethylglycine) is a methyl derivative of glycine first isolated from sugar beets. It has been shown to have potential benefits for fighting heart disease, improving body composition, and helping promote muscl... | |||
T3796 | Betulinaldehyde | Betulinic aldehyde,Betulinal,Betunal | Apoptosis , Antibacterial |
Betulinaldehyde (Betunal) has the inhibition of Saccharomyces sp and alpha-glucosidase. Betulinaldehyde induces apoptosis in mouse B16 2F2 cells. Betulinaldehyde has anti-proliferative activity against mouse +SA mammary ... | |||
TC0027 | beta-Sitosterol acetate | Others | |
Beta-sitosterol is one of several plant-based substances known as phytosterols. | |||
T2S1792 | Lycobetaine | Ungeremine | Antibacterial |
1. Lycobetaine (Ungeremine) is a potential biofungicide against Penicillium roqueforti and Aspergillus niger.2. Lycobetaine have strong antibacterial activity against Flavobacterium columnare . 3. Lycobetaine effectively... | |||
TN6600 | Kaempferol 3-O-(6''-galloyl)-beta-D-glucopyranoside | HIV Protease | |
Kaempferol 3-O-(6''-galloyl)-beta-D-glucopyranoside is a glucopyranoside that inhibits HIV-2 RNase H with an IC50 of 5.19 μM. | |||
TQ0070 | Luteolin-3-O-beta-D-glucuronide | Others | |
Luteolin-3-O-beta-D-glucuronide is active in the inhibition of nitrite production in macrophages. | |||
T5979 | 1-beta-D-Arabinofuranosyluracil | Uracil 1-β-D-arabinofuranoside | Others |
1-beta-D-Arabinofuranosyluracil (Uracil 1-β-D-arabinofuranoside) isolated from the Caribbean sponge Tectitethya crypta, is a methoxyadenosine derivative. 1-beta-D-Arabinofuranosyluracil has anti-inflammatory activity, an... | |||
T4S1962 | beta-Asarone | Cis-Isoasarone,Cis-Asarone,Cis-Isoelemicin | NF-κB , JNK |
1. beta-Asarone (Cis-Isoelemicin) may be a potential preventive drug for Alzheimer's disease. 2. Beta-Asarone prevents autophagy and synaptic loss by reducing ROCK expression in SAMP8 mice. 3. The co-administration of be... | |||
T0019 | Betaine chloride | Betaine hydrochloride | Others , Chloride channel , Endogenous Metabolite |
Betaine chloride (Betaine hydrochloride) is an acidic form of betaine, a vitamin-like substance observed in grains and other foods; gains the amplification of DNA by decreasing the formation of secondary structure in GC-... | |||
T3865 | beta-Eudesmol | Beta-Selinenol | TRP/TRPV Channel , AChR |
beta-Eudesmol (Beta-Selinenol) is a noncompetitive antagonist of nicotinic acetylcholine receptors (nAChRs). It is a sesquiterpene that has been found in a variety of plants, including Cannabis, and has diverse biologica... | |||
TN1019 | Beta-mangostin | β-Mangostin | Apoptosis , Antibacterial , Parasite |
Beta-mangostin (β-Mangostin) is a xanthone compound with antibacterial and antimalarial activities. Beta-mangostin present in Cratoxylum arborescens and exhibits antimycobacterial activity against Mycobacterium tuberculo... | |||
T8335 | Lycobetaine acetate | Oxylycorine | Others |
Lycobetaine acetate (Oxylycorine) is a potential biofungicide against Penicillium roqueforti and Aspergillus niger.2. Ungeremine have strong antibacterial activity against Flavobacterium columnare | |||
T2966 | Beta-Sitosterol | Cupreol,Beta-Sitosterol,β-Sitosterol,Azuprostat,SKF 14463,22,23-Dihydrostigmasterol,Betaprost | Apoptosis , Lipase , Endogenous Metabolite |
Beta-Sitosterol (SKF 14463) has recently been shown to induce G2/M arrest, endoreduplication, and apoptosis through the Bcl-2 and PI3K/Akt signaling pathways. Beta-Sitosterol (SKF 14463) , a main dietary phytosterol foun... | |||
T3S0208 | Hederagenin 28-O-beta-D-glucopyranosyl ester | Hederagenin-28-beta-D-glucopyranoside | Others |
Hederagenin-28-beta-D-glucopyranoside, a triterpene saponin isolated from Ilex cornuta, protects cardiac myocytes against H2O2-induced damage. | |||
T8846 | beta-Escin | B-escin,AESCINE | Immunology/Inflammation related |
beta-Escin is a natural mixture of triterpenoid saponins isolated from horse chestnut (Aesculus hippocastanum) seeds, can be used as a vasoprotective anti-inflammatory, anti-edematous and anti-nociceptive agent. | |||
TN1166 | 1,3,6-Tri-O-galloyl-beta-D-glucose | 1,3,6-Tri-O-galloyl-β-D-glucose,1,3,6-Tri-O-galloylglucose | Immunology/Inflammation related |
1,3,6-Tri-O-galloyl-beta-D-glucose (1,3,6-Tri-O-galloylglucose) is a phenolic compound in Black Walnut Kernels. It shows anti-inflammatory activity. | |||
TN3500 | beta-Amyrone | β-Amyron | COX , AChR , PPAR , Antifection |
beta-Amyrone (β-Amyron) has antifungal activity against Chikungunya virus replication with an EC50 of 86 uM. beta-Amyrone has anti-inflammatory activity through inhibiting the expression of COX-2. beta-Amyrone exhibits a... | |||
TN1440 | Beta-Hydroxyisovalerylshikonin | EGFR , Tyrosine Kinases , Prostaglandin Receptor , Src , AMPK , Fatty Acid Synthase | |
Beta-Hydroxyisovalerylshikonin is an inhibitor of protein-tyrosine kinases such as v-Src and EGFR, and has been shown to induce apoptosis in several human tumor cell lines. Beta-Hydroxyisovalerylshikonin significantly de... | |||
TN1258 | 3-Acetyl-beta-boswellic acid | 3-O-Acetyl-beta-boswellic acid | DNA/RNA Synthesis |
3-Acetyl-beta-boswellic acid has antitumor activity, it inhibits synthesis of DNA, RNA and protein in human leukemia HL-60 cells in a dose dependent manner with IC50 values ranging from 0.6 to 7.1 microM. | |||
T5S2350 | Beta-Acetoxyisovalerylshikonin | Acetoxyisovalerylalkannin | Others |
Acetoxyisovalerylshikonin, a naphthoquinone derivative extracted from Arnebia euchroma, is a chemical compound. | |||
TN1182 | 11-Keto-beta-boswellic acid | 11-Keto-beta-boswellic acid | Leukotriene Receptor , NF-κB , Lipoxygenase |
11-Keto-beta-boswellic acid, a novel Nrf2 activator, and a selective 5-lipoxygenase (5-LOX) inhibitor; it exerts dose dependent cardioprotective effect manifested by dose-dependent reduction in serum lactate dehydrogenas... | |||
TN1438 | beta-Amyrin acetate | Antioxidant , HMG-CoA Reductase , Epoxide Hydrolase , Antifungal | |
beta-Amyrin acetate inhibits HMG-CoA Reductase (HMGCR) and sEH activity with IC50 of 3.4 μM. beta-Amyrin acetate has anti-inflammatory, antifungal, antioxidant, and anti-hyperlipidemic activities. | |||
T4S1439 | 6'-O-beta-D-Glucosylgentiopicroside | 6'-O-Glucosylgentiopicroside | Antifungal |
1. 6'-O-beta-D-Glucosylgentiopicroside (6'-O-Glucosylgentiopicroside) may have antifungal activity. | |||
T5713 | 2"-O-beta-L-galactopyranosylorientin | 2''-O-β-L-Galorientin | Others |
2"-O-beta-L-galactopyranosylorientin (2''-O-β-L-Galorientin) is a natual product isaolated from Trollius chinensis Bunge. | |||
T3S2156 | Chrysin 7-O-beta-gentiobioside | Chrysin 7-O-β-gentiobioside | Others |
Chrysin 7-O-beta-gentiobioside (Chrysin 7-O-β-gentiobioside), a glycosylation product of Chrysin, is from Spartium junceum. | |||
TN2633 | 15,16-Epoxy-15-ethoxy-6beta,13-dihydroxylabd-8-en-7-one | Others | |
15,16-Epoxy-15-ethoxy-6beta,13-dihydroxylabd-8-en-7-one is a natural product for research related to life sciences. The catalog number is TN2633 and the CAS number is 1374328-47-8. | |||
TN3949 | Ent-3beta-Hydroxykaur-16-en-19-oic acid | Others | |
ent-3beta-Hydroxykaur-16-en-19-oic acid is a natural product for research related to life sciences. The catalog number is TN3949 and the CAS number is 66556-91-0. | |||
TN6472 | Columbianetin beta-D-glucopyranoside | ||
Columbianetin-beta-D-glucopyranoside exhibits anti-inflammatory and analgesic properties, it also shows strong inhibiting activity against platelet aggregation. | |||
TN3306 | 8beta-Tigloyloxyreynosin | Others | |
8beta-Tigloyloxyreynosin is a natural product for research related to life sciences. The catalog number is TN3306 and the CAS number is 80368-31-6. | |||
TN6482 | Emodin-8-O-beta-gentiobioside | ||
Emodin-8-O-beta-gentiobioside is a natural product for research related to life sciences. The catalog number is TN6482 and the CAS number is 66466-22-6. | |||
TN1442 | Betulinic acid methyl ester | Antifection | |
Betulinic acid methyl ester showed antiplasmodial activity against chloroquine-resistant Plasmodium falciparum parasites in vitro.It also inhibited B16 2F2 cell proliferation by induction of apoptosis. | |||
TN6522 | Quercetin 7-O-(6''-O-malonyl)-beta-D-glucoside | ||
Quercetin 7-O-(6''-O-malonyl)-beta-D-glucoside is a natural product of Justicia, Acanthaceae. The catalog number is TN6522 and the CAS number is 98767-37-4. Quercetin 7-O-(6''-O-malonyl)-beta-D-glucoside can be used as a... | |||
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カタログ番号 | 製品名 | Species | Expression System |
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TMPH-00198 | Bet v 3 Protein, Betula pendula, Recombinant (His & Myc & SUMO) | Betula pendula | E. coli |
Could be involved in calcium metabolism in pollen. Binds 3 calcium ions. Bet v 3 Protein, Betula pendula, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The pre... | |||
TMPH-00199 | Bet v 1-A Protein, Betula pendula, Recombinant (His & SUMO) | Betula pendula | E. coli |
May be a general steroid carrier protein. Bet v 1-A Protein, Betula pendula, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 33.4 kDa and the ac... | |||
TMPY-06330 | Bet v 2 Protein, Betula verrucosa, Recombinant | Betula verrucosa | E. coli |
Bet v 2 Protein, Betula verrucosa, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 15.21 kDa. | |||
TMPY-06099 | Bet v 4 Protein, Betula pendula, Recombinant (His) | Betula pendula | E. coli |
Bet v 4 Protein, Betula pendula, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 10.3 kDa and the accession number is Q39419-1. | |||
TMPY-05716 | Integrin alpha V beta 3 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Integrin alpha-V & beta-3 (ITGAV/ITGB3) is a receptor for cytotactin, fibronectin, laminin, matrix metalloproteinase-2, osteopontin, osteomodulin, prothrombin, thrombospondin, vitronectin and von Willebrand factor. | |||
TMPY-02638 | TGF beta 1 Protein, Human/Rhesus/Cynomolgus/Canine, Recombinant | Human,Rhesus,Cynomolgus,Canine | CHO Cells |
TGF beta 1 Protein, Human/Rhesus/Cynomolgus/Canine, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 12.8 kDa and the accession number is A0A499FJK2. | |||
TMPY-02159 | Integrin alpha 5 beta 1 Protein, Human, Recombinant (Flag & His) | Human | HEK293 Cells |
Integrin alpha 5 beta 1 Protein, Human, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 192 kDa and the accession number is P08648&P05556-1. | |||
TMPY-03878 | Integrin alpha V beta 6 Protein, Human, Recombinant (Flag & His) | Human | HEK293 Cells |
Integrin alpha V beta 6 Protein, Human, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 190.4 kDa and the accession number is P06756-1&P18564-1. | |||
TMPY-05717 | Integrin alpha V beta 8 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Integrin alpha V beta 8 is a receptor for fibronectin. It recognizes the sequence R-G-D in its ligands. ITGAVB8 does not appear to assume different activation states; and the cytoplasmic tail does not connect to the cyto... | |||
TMPY-01686 | B2M/beta 2-Microglobulin Protein, Human, Recombinant (His) | Human | HEK293 Cells |
B2M/beta 2-Microglobulin Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 13.2 kDa and the accession number is P61769. | |||
TMPY-01133 | Latent TGF beta 1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Latent TGF beta 1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.4 kDa and the accession number is A0A499FJK2. | |||
TMPY-03145 | IFN-beta Protein, Human, Recombinant | Human | CHO Cells |
IFN-beta Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 20 kDa and the accession number is P01574. | |||
TMPY-00831 | IFN-beta Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
IFN-beta Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 46.7 kDa and the accession number is A0A7R8GV38. | |||
TMPY-00500 | Latent TGF beta 1 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Latent TGF beta 1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.7 kDa and the accession number is P04202. | |||
TMPY-03102 | IL-18R beta/IL-18RAP Protein, Rhesus, Recombinant (hFc) | Rhesus | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Rhesus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65.4 kDa and the accession number is XP_001108108.1. | |||
TMPY-01999 | IL-1 beta/IL-1F2 Protein, Human, Recombinant (His) | Human | E. coli |
IL-1 beta/IL-1F2 Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 32.3 kDa and the accession number is P01584. | |||
TMPY-04211 | Latent TGF beta 1 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
Latent TGF beta 1 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.7 kDa. | |||
TMPY-04925 | CD8 beta Protein, Human, Recombinant, Biotinylated | Human | HEK293 Cells |
CD8 beta Protein, Human, Recombinant, Biotinylated is expressed in HEK293 mammalian cells. The predicted molecular weight is 17.6 kDa and the accession number is P10966-1. | |||
TMPJ-01468 | Pro-Beta NGF Protein, Human, Recombinant | Human | E. coli |
The precursor form of the nerve growth factor (proNGF) like its mature form is characterized by the cystin knot motif consisting of three cystine bridges, whereas proneurotrophins and mature neurotrophins elicit opposite... | |||
TMPY-01049 | IL-1 beta/IL-1F2 Protein, Human, Recombinant | Human | E. coli |
IL-1 beta/IL-1F2 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17 kDa and the accession number is P01584. | |||
TMPY-00413 | Latent TGF beta 2 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
TGF beta 2 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46.9 kDa and the accession number is P27090. | |||
TMPY-02445 | IL-1 beta/IL-1F2 Protein, Rhesus, Recombinant | Rhesus | E. coli |
IL-1 beta/IL-1F2 Protein, Rhesus, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.5 kDa and the accession number is P48090. | |||
TMPY-03467 | IFN-beta Protein, Mouse, Recombinant | Mouse | HEK293 Cells |
IFN-beta Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 20.3 kDa and the accession number is P01575. | |||
TMPY-02227 | IL-1 beta/IL-1F2 Protein, Rat, Recombinant (mature form) | Rat | E. coli |
IL-1 beta/IL-1F2 Protein, Rat, Recombinant (mature form) is expressed in E. coli expression system. The predicted molecular weight is 17.4 kDa and the accession number is Q63264-1. | |||
TMPY-04643 | Integrin alpha V beta 6 Protein, Mouse, Recombinant (Flag & His) | Mouse | HEK293 Cells |
Integrin alpha V beta 6 Protein, Mouse, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 190.4 kDa and the accession number is NP_032428.2&NP_067334... | |||
TMPY-02153 | TNF beta Protein, Human, Recombinant | Human | E. coli |
Lymphotoxin-alpha, also known as LT-alpha, TNF-beta, Tumor necrosis factor ligand superfamily member 1, LTA TNFSF1, and TNFB, is a secreted protein that belongs to the tumor necrosis factor family. TNF-beta/TNFSF1/Lympho... | |||
TMPY-03945 | Latent TGF beta 1 Protein, Rat, Recombinant (His) | Rat | HEK293 Cells |
Latent TGF beta 1 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.7 kDa and the accession number is P17246. | |||
TMPY-00608 | TGF beta 1 Protein, Rat/Mouse, Recombinant | Mouse,Rat | HEK293 Cells |
TGF beta 1 Protein, Rat/Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 12.8 kDa. | |||
TMPJ-00249 | TGF beta 1 Protein, Human, Recombinant (Avi), Biotinylated | Human | HEK293 Cells |
Transforming Growth Factor β-1 (TGFβ-1) is a secreted protein which belongs to the TGF-β family. TGFβ-1 is abundantly expressed in bone, articular cartilage and chondrocytes and is increased in osteoarthritis (OA). TGFβ-... | |||
TMPY-00006 | GRO beta/CXCL2 Protein, Human, Recombinant | Human | E. coli |
GRO beta/CXCL2 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 7.9 kDa and the accession number is A0A024RDD9. | |||
TMPJ-00258 | TGF beta 2 Protein, Human, Recombinant | Human | HEK293 Cells |
Transforming growth factor beta-2 (TGF-β2) is a secreted protein which belongs to the TGF-beta family. It is known as a cytokine that performs many cellular functions and has a vital role during embryonic development. T... | |||
TMPY-02134 | IL-1 beta/IL-1F2 Protein, Mouse, Recombinant | Mouse | E. coli |
IL-1 beta/IL-1F2 Protein, Mouse, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.5 kDa and the accession number is P10749. | |||
TMPY-06247 | TGF beta 3 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
TGF beta 3 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 41.2 kDa and the accession number is P10600-1. | |||
TMPY-06034 | FGFR1 Protein, Human, Recombinant (beta (IIIb), His) | Human | HEK293 Cells |
FGFR1 Protein, Human, Recombinant (beta (IIIb), His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 30.8 kDa and the accession number is H9FRD4. | |||
TMPY-01446 | IL-18R beta/IL-18RAP Protein, Human, Recombinant (His) | Human | HEK293 Cells |
IL-18R beta/IL-18RAP Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40 kDa and the accession number is O95256-1. | |||
TMPY-02568 | IL-1 beta/IL-1F2 Protein, Canine, Recombinant | Canine | E. coli |
IL-1 beta/IL-1F2 Protein, Canine, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.6 kDa and the accession number is Q28292. | |||
TMPY-02205 | Beta-Catenin Protein, Human, Recombinant (His & GST) | Human | Baculovirus Insect Cells |
Beta-Catenin Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 113 kDa and the accession number is P35222-1. | |||
TMPJ-00261 | TGF beta 2 Protein, Mouse/Rat, Recombinant | Mouse,Rat | HEK293 Cells |
Transforming growth factor beta 2 (TGF-β2) is a member of TGF-beta superfamily that shares a characteristic cysteine knot structure. Mice with TGF-β2 gene deletion show defects in development of cardiac, lung, craniofaci... | |||
TMPJ-00254 | TGF beta 3 Protein, Human/Mouse/Rat, Recombinant | Human,Mouse,Rat | HEK293 Cells |
Transforming growth factor beta 3(TGFB3) is a member of a TGF -β superfamily which is defined by theirstructural and functional similarities. TGFB3 is secreted as a complex with LAP. This latent form of TGFB3becomes acti... | |||
TMPH-00513 | Proline iminopeptidase Protein, Elizabethkingia meningoseptica, Recombinant (His & Myc) | Elizabethkingia meningoseptica | E. coli |
Releases the N-terminal proline from various substrates. Cleaves specifically Pro-betaNA and small peptides containing proline at the amino terminal. No activity against hydroxyproline-betaNA. Proline iminopeptidase Prot... | |||
TMPY-02584 | 14-3-3 beta Protein, Cynomolgus, Recombinant | Cynomolgus | E. coli |
14-3-3 beta Protein, Cynomolgus, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 27.8 kDa and the accession number is Q4R572-2. | |||
TMPY-03828 | IFN-beta Protein, Rhesus, Recombinant (mFc) | Rhesus | HEK293 Cells |
IFN-beta Protein, Rhesus, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 46.4 kDa and the accession number is G7NFX1. | |||
TMPY-02456 | IFN-beta Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
IFN-beta Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 46.7 kDa and the accession number is P01575. | |||
TMPY-02630 | B2M/beta 2-Microglobulin Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
B2M/beta 2-Microglobulin Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 13 kDa and the accession number is P01887. | |||
TMPH-03628 | Beta-toxin Tz1 Protein, Tityus zulianus, Recombinant (His & Myc) | Tityus zulianus | E. coli |
Beta toxins bind voltage-independently at site-4 of sodium channels (Nav) and shift the voltage of activation toward more negative potentials thereby affecting sodium channel activation and promoting spontaneous and repe... | |||
TMPY-02161 | Integrin alpha X beta 2 Protein, Human, Recombinant (Flag & His) | Human | HEK293 Cells |
Integrin alpha X beta 2 Protein, Human, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 205 kDa and the accession number is P20702&P05107. | |||
TMPH-02471 | 14-3-3 beta/alpha Protein, Mouse, Recombinant (E. coli, His) | Mouse | E. coli |
14-3-3 beta/alpha Protein, Mouse, Recombinant (E. coli, His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 33.6 kDa and the accession number is Q9CQV8. | |||
TMPH-01333 | Fibrinogen beta chain Protein, Human, Recombinant (His) | Human | E. coli |
Fibrinogen beta chain Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 54.8 kDa and the accession number is P02675. | |||
TMPY-05800 | IKB beta/NFKBIB Protein, Human, Recombinant (GST) | Human | E. coli |
NFKBIB (NFKB Inhibitor Beta) is a Protein Coding gene. The protein encoded by this gene belongs to the NF-kappa-B inhibitor family, which inhibits NF-kappa-B by complexing with and trapping it in the cytoplasm. Phosphory... | |||
TMPH-01305 | ER beta Protein, Human, Recombinant (His) | Human | P. pastoris (Yeast) |
Nuclear hormone receptor. Binds estrogens with an affinity similar to that of ESR1/ER-alpha, and activates expression of reporter genes containing estrogen response elements (ERE) in an estrogen-dependent manner.; Lacks ... | |||
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