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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T6143 | PI-103 | PI103,PI 103 | Apoptosis , DNA-PK , PI3K , mTOR , Autophagy |
PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK). | |||
T6941 | PI-1840 | PI 1840 | PARP , Proteasome |
PI-1840(IC50 = 27 nM)is a reversible and selective chymotrypsin-like (CT-L) inhibitor, with little proteasome proteolytic effects on trypsin-like (T-L) and postglutamyl-peptide-hydrolysis-like (PGPH-L). | |||
T12454 | PI-273 | Apoptosis , PI4K | |
PI-273, a Substrate-Competitive, Specific Small-Molecule Inhibitor of PI4KIIα, Inhibits the Growth of Breast Cancer Cells | |||
T16528 | PI-828 | LY 294002, 4gamma-NH2 | Casein Kinase , PI3K |
PI-828 is a phosphatidylinositol 3-kinase (PI3K) inhibitor, which is widely used to study the physiological function of PI3K and also promotes stem cell differentiation into mesoderm. | |||
T60390 | PI-55 | 6-(2-hydroxy-3-methylbenzylamino)purine | Others |
PI-55 (6-(2-hydroxy-3-methylbenzylamino)purine) is a cytokinin receptor inhibitor that exhibits structural similarity to 6-benzylaminopurine (BAP). It competitively inhibits BAP binding on the specific Arabidopsis recept... | |||
T2083 | PI-3065 | PI3065 | DNA-PK , PI3K , mTOR |
PI-3065 is a novel potent and selective PI3K p110δ inhibitor. | |||
T2130 | Propidium Iodide | PI | Others |
Propidium Iodide (PI) is a red fluorescent dye that can be used for cell staining and is suitable for fluorescence microscopy, confocal microscopy, flow cytometry, and fluorometer analysis. In aqueous solution, the Ex/Em... | |||
T68443 | PI-540 | ||
PI-540 is a potent and selective inhibitor of class 1A phosphatidylinositide 3-kinases (PI3K). | |||
T28412 | PI-091 | ||
PI-091 inhibits platelet aggregation. | |||
T32950 | Lumi-PI | ||
Lumi-PI is used as a chemiluminescent substrate for detecting phosphatidylinositol-specific phospholipase C. | |||
T6143L | PI-103 Hydrochloride | ||
PI-103 Hydrochloride is a potent dual inhibitor of PI3K and mTOR, demonstrating inhibitory IC50 values of 8 nM for p110α, 88 nM for p110β, 48 nM for p110δ, 150 nM for p110γ, 20 nM for mTORC1, and 83 nM for mTORC2, respec... | |||
T13819 | Pi-Methylimidazoleacetic acid hydrochloride | Others | |
Pi-Methylimidazoleacetic acid hydrochloride is a potential neurotoxin. | |||
T125867 | PI 201 | ||
PI 201 is a useful organic compound for research related to life sciences. The catalog number is T125867 and the CAS number is 143605-56-5. | |||
T63527 | RIDR-PI-103 | ||
RIDR-PI-103 is a reactive oxygen species (ROS)-induced drug release prodrug containing an autocyclized portion linked to a pan-PI3K inhibitor (PI-103). In MDA-MB-361 and MDA-MB-231 cells, Doxorubicin and RIDR-PI-103 exhi... | |||
T80723 | ZK-PI-9 | ||
ZK-PI-9 acts as an inhibitor of both trehalase and chitinase activities in female pupae and functions as an insecticide [1]. | |||
T80724 | ZK-PI-5 | ||
ZK-PI-5, a potent trehalase inhibitor, has the potential to regulate Spodoptera frugiperda reproduction and may serve as a novel insecticide with significant pest control capabilities [1]. | |||
T30425 | BePI | Be-PI,NSC 664711,NSC-664711,NSC664711,Be PI | |
BePI can be a specific intercalator of both double and triple-helical DNA. | |||
T35003 | UR-PI376 | UR-PI 376,UR-PI-376,URPI-376,URPI 376 | |
UR-PI376 is a histamine H4 receptor agonist (hH4R agonist) (pEC50 = 7.47, alpha = 0.93), with low activity for hH1R and hH2R and significant selectivity for hH3R (pKB = 6.00, alpha =- 0.28), as in stable-use a membrane p... | |||
T30874 | Chemodosimeter 1 | Pi-Probe-1,Chemodosimeter-1 | |
Chemodosimeter 1 is designed as a highly selective phosphate ion (PI) sensor capable of demonstrating exogenous and endogenous ATP-catalysed PI production and is the first probe capable of tracking PI production and enri... | |||
T12462 | PI3Kδ-IN-1 | PI3K | |
PI3Kδ-IN-1 is an efficacious PI3Kδ inhibitor (IC50 of 1.7 nM). | |||
T12365 | PARP/PI3K-IN-1 | PARP , PI3K | |
PARP/PI3K-IN-1 is a novel dual poly (ADP-ribose) polymerase (PARP) and phosphatidylinositol 3-kinase (PI3K) dual inhibitor with anticancer, antitumour and antiproliferative activities for the study of breast, pancreatic ... | |||
T10804 | CHMFL-PI3KD-317 | PI3K , PI4K | |
CHMFL-PI3KD-317 is a highly potent, selective and orally active PI3Kδ inhibitor, with an IC50 of 6 nM, and exhibits over 10-1500 fold selectivity over other class I, II and III PIKK family isoforms, such as PI3Kα (IC50, ... | |||
T5831 | Selective PI3Kδ Inhibitor 1 | PI3K | |
Selective PI3Kδ Inhibitor 1 is a PI3Kδ Inhibitor( IC50 = 0.9 nM). | |||
T12589 | PI3Kα/mTOR-IN-1 | PI3K , mTOR | |
PI3Kα/mTOR-IN-1 is a potent dual inhibitor of PI3Kα/mTOR. PI3Kα/mTOR-IN-1 shows an IC50 of 7 nM for PI3Kα in a cell assay, and Kis of 12.5 nM and 10.6 nM for mTOR and PI3Kα in a cell free assay , respectively. | |||
T35530 | IHMT-PI3Kδ-372 | IHMT-PI3Kδ-372 | PI3K |
IHMT-PI3Kδ-372 is a selective inhibitor of PI3Kδ with an IC50 of 14 nM and can be used in studies about chronic obstructive pulmonary disease. | |||
T12469 | PI4KIIIbeta-IN-9 | PI3K , PI4K | |
PI4KIIIbeta-IN-9 is a potent inhibitor of PI4KIIIβ(IC50 of 7 nM). . | |||
T29126 | VU0360172 | VU-0360172,VU 0360172 | GluR |
VU0360172 is a positive allosteric modulator of mGlu5 receptors (EC50 = 16 nM; Ki = 195 nM). | |||
T12468 | PI4KIIIbeta-IN-10 | PI3K , PI4K | |
PI4KIIIbeta-IN-10 is a potent inhibitor of PI4KIIIβ (IC50 of 3.6 nM). | |||
T12459 | PI3K/mTOR Inhibitor-2 | PI3K , mTOR | |
TMIH-0273 | Hydroxyzine dihydrochloride-d10 | (R)-2-(2-(4-((4-chlorophenyl)(phenyl)methyl)pi perazin-1-yl-2,2,3,3,5,5,6,6-d8)ethoxy)ethan-1, 1-d2-1-ol dihydrochloride | |
Hydroxyzine dihydrochloride-d10 is a deuterated compound of Hydroxyzine dihydrochloride. | |||
T12457 | PI3K-IN-6 | PI3K | |
PI3K-IN-6 is an oral active and highly selective inhibitor of phosphoinositide 3-kinase (PI3K) β/δ(IC50 values of 7.8 nM/5.3 nM , respectively). | |||
T12456 | PI3K-IN-10 | PI3K | |
PI3K-IN-10 is a potent inhibitor of pan-PI3K . | |||
T12458 | PI3K-IN-9 | PI3K | |
PI3K-IN-9 is a potent and selective inhibitor of PI3Kδ(IC50 of 8.9 nM). | |||
T12463 | PI3kδ inhibitor 1 | PI3K | |
PI3kδ inhibitor 1 is a selective inhibitor of PI3Kδ (IC50 of 3.8 nM). | |||
T12461 | PI3Kdelta inhibitor 1 | PI3K | |
PI3Kdelta inhibitor 1 is a potent, selective and orally available inhibitor of PI3Kδ with an IC50 of 1.3 nM. | |||
T1826 | PI3K-IN-1 | Voxtalisib Analogue,Voxtalisib (SAR245409, XL765) Analogue,XL765,SAR245409 | DNA-PK , PI3K |
PI3K-IN-1 (Voxtalisib Analogue) is a dual inhibitor of mTOR/PI3K, mostly for p110γ , also inhibits DNA-PK and mTOR. | |||
T12455 | PI3K/HDAC-IN-1 | PI3K | |
PI3K/HDAC-IN-1 is a potent PI3K and HDAC dual inhibitor(IC50s of 8.1 nM and 1.4 nM, respectively). | |||
T36087 | PI3K-IN-22 | CAY10626 | |
PI3K-IN-22 is a dual kinase inhibitor of PI3Kα and mTOR, with IC50s of 0.9 and 0.6 nM respectively. PI3K-IN-22 could be used in cancer. | |||
T12465 | PI3Kγ inhibitor 2 | PI3K | |
PI3Kγ inhibitor 2 is an orally bioavailable inhibitor of PI3Kγ(Ki of 4 nM). | |||
T12460 | PI3K/mTOR Inhibitor-1 | PI3K | |
PI3K/mTOR Inhibitor-1 is a potent, orally bioavailable dual inhibitor of PI3K/mTOR (PI3Kα/PI3Kβ/PI3Kδ/PI3Kγ/mTOR with IC50s of 20/376/204/46/186 nM) | |||
T40196 | PI3Kγ inhibitor 5 | ||
PI3Kγ inhibitor 5 is a potent inhibitor of phosphoinositide 3-kinase γ (PI3Kγ), exhibiting an exceptional IC50 value of 34 nM. | |||
T12464 | PI3Kγ inhibitor 1 | PI3K | |
PI3Kγ inhibitor 1 is a inhibitor of PI3Kδ and PI3Kγ. | |||
T39542 | PI3Kδ-IN-8 | PI3Kδ-IN-8 | |
PI3Kδ-IN-8 is a powerful and specific oral inhibitor of PI3Kδ, exhibiting an IC50 of 3.3 nM. It demonstrates preferential inhibition of PI3Kδ when compared to PI3Kα, PI3Kβ, and PI3Kγ, with IC50 values of 377.2 nM, 241.6 ... | |||
T36315 | NVS-PI3-4 | NVS-PI3-4 | |
NVS-PI3-4 is a highly selective inhibitor of the enzyme PI3Kγ. It is specifically designed for use in scientific investigations related to allergies, inflammatory conditions, and cancerous diseases[1][2]. | |||
T39592 | PI3Kδ-IN-9 | PI3Kδ-IN-9 | |
PI3Kδ-IN-9 is a selective PI3Kδ inhibitor with an IC 50 value of 3.8 nM. | |||
T39581 | PI3K-IN-19 hydrochloride | PI3K-IN-19 hydrochloride | |
PI3K-IN-19 hydrochloride (WO2017153220, step 5) acts as a phosphatidylinositol-3-kinase (PI3K) inhibitor. | |||
T12467 | PI4KIII beta inhibitor 3 | PI3K | |
PI4KIII beta inhibitor 3 is a novel and high effective inhibitor of PI4KIIIβ (IC50 of 5.7 nM). | |||
T35527 | PI3Kα-IN-4 | PI3Kα-IN-4 | |
PI3Kα-IN-4 is a potent, selective, and orally active PI3Kα inhibitor, demonstrating an IC50 of 1.8 nM and exhibiting antitumor activity[1]. | |||
T70619 | LY2934747 | ||
LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo. | |||
T28413 | PI3KD/V-IN-01 | PI3KD/V IN 01,PI3KD/VIN01 | |
PI3KD/V-IN-01 is a potent ATP-competitive PI3Kδ/Vps34 dual inhibitor. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T13820 | Pi-Methylimidazoleacetic acid | Others | |
Pi-Methylimidazoleacetic acid is a potential neurotoxin. | |||
T8187 | Tetrahydroepiberberine | Others , Influenza Virus , Antifungal | |
Tetrahydroepiberberine, an isoquinoline alkaloid, has antifungal and selective inhibition against the PI-3 virus activities. | |||
T1205 | Chloramphenicol | Chlornitromycin,Levomycetin,Chloromycetin | ribosome , HIF/HIF Prolyl-Hydroxylase , Antibacterial , Antibiotic |
Chloramphenicol (Chloromycetin), a broad-spectrum antibiotic, blocks bacterial protein synthesis. | |||
T5285 | 3-(Methylthio)propionic acid | 3-Methylthiopropionate,4-Thiapentanoic acid,3-Methylsulfanylpropionic acid | Others , Endogenous Metabolite , Antifungal |
3-(Methylthio)propionic acid (4-Thiapentanoic acid) is one of the metabolites of methionine (especially of D-methionine). Cultures of Streptomyces lincolnensis accumulated 3-methylthioacrylic acid in amounts directly rel... | |||
TN7041 | (-)-Epipodophyllotoxin | Apoptosis | |
(-)-Epipodophyllotoxin (2) is an antiproliferative agent against cancer cells with GI50s of 0.36 and 0.24 μM in HeLa cells and MCF-7 cells, respectively. (-)-Epipodophyllotoxin can inhibit mitotic spindle assembly in vit... | |||
T14305 | Apicidin | OSI 2040 | Apoptosis , HDAC , Autophagy |
Apicidin (OSI 2040) is a histone deacetylase (HDAC) inhibitor with antiparasitic activity and antiproliferative activity.Apicidin attenuates memory deficits, inhibits cell growth and proliferation, and induces apoptosis ... | |||
TN2967 | Pinobanksin 3-acetate | 3-O-Acetylpinobanksin | Others , Antioxidant |
Pinobanksin 3-acetate (3-O-Acetylpinobanksin), a flavonoid derivative, is a strong antioxidant found in sunflowers and honey that inhibits LDL peroxidation. | |||
TN3972 | Epimedokoreanin B | Apoptosis , Others , Antibacterial | |
Epimedokoreanin B (EKB), an isoprenylated flavonoid isolated from Korean Epimedium, exhibited anticancer activity in human non-small cell lung cancer (NSCLC) A549 and NCI-H292 cells.Epimedokoreanin B also possesses anti-... | |||
TL0002 | Liquiritin apioside | Others | |
Liquiritin Apioside is one of the main active components in Suan-Zao-Ren decoction as a treatment for insomnia. | |||
T5776 | pimpinellin | Apoptosis , Anti-infection | |
Pimpinellin is a natural product that acts as antagonist of proteins with GABA receptor activity. | |||
TN1377 | α-Spinasterol | alpha-Spinasterol | COX , Antibacterial , TRP/TRPV Channel |
α-Spinasterol is a transient receptor potential vanilloid 1 (TRPV1) antagonist, has anti-inflammatory, antidepressant, antioxidant and antinociceptive effects. α-Spinasterol inhibits COX-1 andCOX-2 activities with IC50 v... | |||
T16535 | Picrotoxinin | Chloride channel , GABA Receptor | |
Picrotoxinin is a blocker of chloride channel and a noncompetitive antagonist of GABAA with an IC50 of 1.15 μM for α1β2γ2L GABAA. Picrotoxinin shows convulsant properties. | |||
TN1082 | Apigenin 7-O-malonylglucoside | Apigenin 7-O-(6''-O-malonylglucoside) | |
Apigenin 7-O-malonylglucoside (Apigenin 7-O-(6''-O-malonylglucoside)) is found in chrysanthemums and is a flavonoid as well as a glycoside. | |||
TN2023 | 8-Oxoepiberberine | Oxyepiberberine | Others |
8-Oxoepiberberine (Oxyepiberberine) is an alkaloid metabolite in the plasma after oral administration of Zuojin formula. Zuojin formula is a traditional chinese medicine used to treat gastrointestinal disease. | |||
TN2083 | Pinostrobin chalcone | ||
Pinostrobin chalcone, a chalcone analog isolated from the leguminous plant, Mucuna pruriens, exhibits anticancer activity with an IC50 value of 20.42±2.23 μg/mL against MDA-MB-231 and 22.51±0.42 μg/mL against the HT-29 c... | |||
TN1891 | Lupiwighteone | Apoptosis , BCL , PARP , Caspase | |
Lupiwighteone has anti-angiogenesis potential, it also has anticancer and cancer preventive effects on SH-SY5Y cells. | |||
T3S0027 | Picropodophyllotoxin | AXL 1717,Picropodophyllin | IGF-1R |
Picropodophyllotoxin (AXL 1717) is a cyclolignan alkaloid found in the mayapple plant family (Podophyllum peltatum), and a small molecule inhibitor of the insulin-like growth factor 1 receptor (IGF1R) with potential anti... | |||
TN2031 | γ-Terpinene | Moslene,p-Mentha-1,4-diene,Crithmene | Antioxidant |
γ-Terpinene (p-Mentha-1,4-diene) is a monoterpene compound with high antioxidant properties suitable for oral consumption. It displays direct radical scavenging abilities and is known to be a potent antinociceptive agent... | |||
T2972 | Rutaecarpine | Rutacarpine,Rhetine,Rutecarpine | COX |
Rutaecarpine (Rhetine) is an inhibitor of COX-2 with IC50 of 0.28 μM. | |||
T8709 | Nandrolone phenylpropionate | Nandrolone phenpropionate | Androgen Receptor |
Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis | |||
TN1079 | Deoxyelephantopin | NF-κB | |
Deoxyelephantopin has anti-inflammatory, hepatoprotective, and wound healing activities; it also has antitumor activity.Deoxyelephantopin inhibits NF-κB, MAPK, PI3K/Akt, and β-catenin signaling | |||
T2828 | Spiculisporic Acid | 4,5-dicarboxy-4-pentadecanolide | Others |
Spiculisporic Acid (4,5-dicarboxy-4-pentadecanolide) is a bioactive γ-butenolide isolated from a marine Aspergillus. | |||
T5S0483 | (-)-Syringaresnol-4-O-β-D-apiofuranosyl-(1→2)-β-D-glucopyranoside | (-)-Syringaresnol-4-O-beta-D-apiofuranos | Others |
(-)-Syringaresnol-4-O-β-D-apiofuranosyl-(1→2)-β-D-glucopyranoside ((-)-Syringaresnol-4-O-beta-D-apiofuranos) is a lignan glycosides from the bark of Albizzia myriophylla. | |||
T3392 | Sinapine thiocyanate | P-gp , AChE | |
Sinapine Thiocyanate, is a derivative of Sinapine (S486605), an alkaloidal amine found in black mustard seeds. It is the choline ester of Sinapic Acid (S486800). It is also a phenolic-chloine conjugates, acting as anti-o... | |||
Fr16605 | Lupinine | AChR , AChE | |
Lupinine is an alkaloid capable of counteracting ethanol anesthesia. Lupinine is an AChE and BChE inhibitor and potential CD69 activator found in species of Loranthus, Calia, and Lupinus. It may also inhibit heparin. | |||
T12830 | Sapienic acid sodium | Antibacterial | |
Sapienic acid sodium is a fatty acid commonly. It has variable antimicrobial activities against Gram-positive and Gram-negative bacteria found on the skin and in the oral cavity. | |||
T1231 | Pilocarpine nitrate | Pilagan,Pilofrin | AChR |
Pilocarpine nitrate (Pilagan) is a slowly hydrolyzed muscarinic agonist with no nicotinic effects. Pilocarpine is used as a miotic and in the treatment of glaucoma. | |||
T8148 | Mupirocin calcium hydrate | Mupirocin calcium | Others , Antibacterial , Antibiotic |
Mupirocin calcium hydrate is an antibiotic produced by Pseudomonas fluorescens, showed a high level of activity against staphylococci and streptococci and against certain gram-negative bacteria | |||
T3768 | Epifriedelanol | Epifriedelinol | Others |
Epifriedelanol (Epifriedelinol) suppresses adriamycin-induced cellular senescence, replicative senescence in human fibroblasts (HDFs) and HUVECs. Because of Epifriedelanol can reduce cellular senescence in human primary ... | |||
Fr14115 | α-Terpineol | Terpineol | IL Receptor , Anti-infection , Antibacterial |
Terpineol possesses antifungal activity against Trichophyton mentagrophytes, it also exhibits strong antimicrobial activity against periodontopathic and cariogenic bacteria. α-Terpineol (Terpineol) shows anticonvulsant, ... | |||
TN2264 | Terpinen-4-ol | Terpinine-4-ol,4-Carvomenthenol | Others , Endogenous Metabolite |
Terpinen-4-ol (4-Carvomenthenol) is a natural product from Pimpinella yunnanensis. | |||
T0814 | Ampicillin Trihydrate | NCI-C56086 | Antibacterial , Antibiotic |
Ampicillin Trihydrate (NCI-C56086), a broad-spectrum semisynthetic derivative of aminopenicillin, is a β-lactam antibiotic. | |||
T5514 | Epibrassinolide | 24-Epibrassinolide,B1105,BP55 | Apoptosis |
Epibrassinolide (BP55) (EBR) is a biologically active compound of the brassinosteroids, is a natural brassinosteroid (BR) derivative, is a plant regulator with a similar structure to mammalian steroids. | |||
T2228 | Adipic acid | Others , Endogenous Metabolite | |
Adipic acid is a precursor for the production of nylon. | |||
T5S1989 | Apiin | Apioside | Others |
1. Apiin (Apioside) is the reducing and stabilizing agent. 2. Apiin has inhibitory activity in-vitro on iNOS expression and nitrite production when added before LPS stimulation in the medium of J774.A1 cells. | |||
T2S1200 | Sinapine | Antioxidant , P-gp , AChE | |
1. Sinapine, an alkaloid from seeds of the cruciferous species, can be used as an effective natural compound for chemo-resistance. 2. Sinapine has antioxidant and radio-protective activities. | |||
T3A2467 | Allocryptopine | Thalictrimine,Fagarine I | Potassium Channel |
Allocryptopine (Thalictrimine) induces muscle contraction and relaxation in urinary bladder and ileum, respectively. | |||
T7959 | (+)-ISOPINOCAMPHEOL | Others | |
(+)-ISOPINOCAMPHEOL is a natural product. | |||
TN2070 | Picropodophyllol | Others | |
Picropodophyllol is a natural product isolated from the roots of Dysosma versipellis | |||
TN7086 | Propiosyringone | Others | |
Propiosyringone is from the degradation of Eucalyptus globulus wood by wood-rotting fungi. | |||
TN1141 | Isodeoxyelephantopin | NF-κB , Reactive Oxygen Species , Autophagy | |
Isodeoxyelephantopin exerts antitumor effects on several cancer cells by inducing apoptosis , cell cycle arrest , and inhibiting proliferation. It enhances apoptosis and inhibit invasion and osteoclastogenesis by inhibit... | |||
T67922 | Lepidiline C | Others | |
Lepidiline C is a novel imidazoles alkaloids extracted from the root of Lepidium meenii Walpers of the brassaceae family. It has shown cytotoxic activity against HL-60 cells (IC50:27.7 μM). | |||
T3834 | 8-Epideoxyloganic acid | ROS , Immunology/Inflammation related | |
8-Epideoxyloganic acid possesses bioactivities of analgesia, homeostasis and anti-inflammatory. It has the potential to serve as anti-inflammatory agents during oxidative stress, the inhibition of ROS production, possibl... | |||
T4S1024 | Picfeltarraenin IB | Others , AChE | |
1. Picfeltarraenin IB and Picfeltarraenin IA displayes no cytotoxic activity in vitro human tumor cell line panel. | |||
T2210 | Genipin | (+)-Genipin | Others , Autophagy |
Genipin ((+)-Genipin), an active aglycone derived from an iridoid glycoside called geniposide, is found in the fruit of Gardenia jasminoides Ellis. | |||
T7936 | Benzopinacole | Others | |
Benzopinacole is an anti-amoeba drug that can be used as an intermediate to synthesize a variety of compounds. | |||
TN3967 | Epieriocalyxin A | ERK , BCL , ROS , Caspase , DNA/RNA Synthesis , JNK | |
Epieriocalyxin A can suppress Caco-2 colon cancer cell growth. It could be a potential drug for colon cancer therapy in the future. | |||
T1064 | Norepinephrine bitartrate monohydrate | Levophed,Noradrenaline bitartrate monohydrate | Endogenous Metabolite , Adrenergic Receptor , Autophagy |
Norepinephrine bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator. | |||
TN2252 | Syrosingopine | Dopamine Receptor | |
Syrosingopine has selective depleting effect on brain amines is potentiated by combined treatment with disulfiram or fusaric acid, a dopamine beta-hydroxylase inhibitor. | |||
T3821 | Deapioplatycodin D | Deapi-platycodin D,DesapioplatycodinD | Others , HCV Protease |
Deapioplatycodin D and platycodin D can regulate the production and secretion of airway mucin and, at least in part, explains the traditional use of aqueous extract of APG as expectorants in diverse inflammatory pulmonar... | |||
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カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPY-00915 | Serpin A1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Serpin A1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 45.7 kDa and the accession number is P01009-1. | |||
TMPY-00547 | PITPN Protein, Human, Recombinant (His) | Human | HEK293 Cells |
PITPN Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 33.3 kDa and the accession number is Q00169. | |||
TMPY-01398 | Alpha 2 Antiplasmin/SerpinF2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Alpha 2 Antiplasmin/SerpinF2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 53.2 kDa and the accession number is P08697-1. | |||
TMPK-00540 | Serpin F2 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
Large-pool solvent/detergent (SD) plasma for transfusion exhibits reduced alpha 2-antiplasmin (alpha2-AP; SERPINF2) functional activity. The reason for the loss of alpha2-AP has not been described and could be due to the... | |||
TMPJ-00931 | Serpin A4 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Serpin Peptidase Inhibitor, Clade A (α-1 Antiproteinase, Antitrypsin), Member 4 (Serpin A4) is a member of the Serpin family. Serpin A4 exists as a monomer and some homodimers. Serpin A4 is expressed by the liver and sec... | |||
TMPJ-00302 | Serpin F2 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
Alpha-2-antiplasmin, also called Serpin F2, is a serine protease inhibitor (serpin) responsible for inactivating plasmin, and an important enzyme participates in fibrinolysis and degradation of other proteins. In liver c... | |||
TMPY-02628 | Neuroserpin Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Neuroserpin Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46 kDa and the accession number is O35684. | |||
TMPY-02210 | Serpin B9 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
SerpinB9, also known as Cytoplasmic antiproteinase 3, CAP-3, Peptidase inhibitor 9, SERPINB9 and PI-9, is a cytoplasm protein that belongs to the serpin family and Ov-serpin subfamily. Serpin-B9 ( CAP-3 / PI-9 ) is the o... | |||
TMPJ-00243 | Serpin B6 Protein, Human, Recombinant (E. coli, His) | Human | E. coli |
Serpin B6 belongs to the serpin family. Serpin B6 localizes to the cytoplasm. Serpin B6 is expressed in many tissues, abundantly by mast cells in different tissues and mastocytoma lesions. Serpin B6 may be involved in th... | |||
TMPJ-00499 | GSTP1 Protein, Human, Recombinant | Human | E. coli |
Glutathione S-transferase P (GSTP1) is an enzyme that contains 1 GST C-terminal domain, 1 GST N-terminal domain. GSTP1 belongs to the GST superfamily, the GSTs are a family of enzymes that play an important role in deto... | |||
TMPJ-00796 | Serpin E2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Serpin E2 is a secreted protein that belongs to the serpin family. Serpin E2 is a serine protease inhibitor with activity toward thrombin, trypsin, and urokinase. Serpin E2 expression is weak or absent in all normal panc... | |||
TMPY-02128 | Serpin B1 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
SerpinB1 is an endogenous inhibitor of serine proteases recognized for its anti-inflammatory and host-protective properties. Serum SerpinB1 levels are elevated in patients with type 2 diabetes compared with that in healt... | |||
TMPY-02242 | Serpin B6 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
SerpinB6, also known as Cytoplasmic antiproteinase, Peptidase inhibitor 6, Placental thrombin inhibitor, SERPINB6 and PI-6, is a cytoplasm protein that belongs to the serpin family and Ov-serpin subfamily. SerpinB6 / PI-... | |||
TMPJ-01083 | Serpin E2 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Serpin E2 is a member of the Serpin superfamily. It is differentially expressed during neuronal differentiation and is able to transform human embryonic kidney cells into neuronlike cells. Its over-expression in mice lea... | |||
TMPH-00917 | ADH4 Protein, Human, Recombinant (GST) | Human | E. coli |
Catalyzes the NAD-dependent oxidation of either all-trans-retinol or 9-cis-retinol. Also oxidizes long chain omega-hydroxy fatty acids, such as 20-HETE, producing both the intermediate aldehyde, 20-oxoarachidonate and th... | |||
TMPJ-00505 | Serpin A1 Protein, Human, Recombinant (aa 25-418, His) | Human | HEK293 Cells |
Serpin A1 is a prototype member of the Serpin superfamily of the serine protease inhibitors. As one of the most abundant proteinase inhibitors in the circulation, it is synthesized in hepatocytes, and to a lesser extent,... | |||
TMPY-01241 | Neuroserpin Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Neuroserpin Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46 kDa and the accession number is A0A0S2Z455. | |||
TMPY-01841 | Serpin I2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Serpins are the largest and most diverse family of serine protease inhibitors which are involved in some fundamental biological processes such as blood coagulation, complement activation, fibrinolysis, angiogenesis, infl... | |||
TMPY-01792 | Serpin A1b Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
Serpin A1b Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 70.2 kDa. | |||
TMPY-00621 | Serpin A1d Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Serpin A1d Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 44.9 kDa and the accession number is XP_003945711.1. | |||
TMPY-02425 | Serpin B4, Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
Overexpression of SERPINB4 in tumor cells inhibited recombinant GrM-induced as well as NK cell-mediated cell death and this inhibition depended on the reactive center loop of the serpin. | |||
TMPY-00623 | Serpin A1d Protein, Mouse, Recombinant | Mouse | HEK293 Cells |
Serpin A1d Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 44.1 kDa and the accession number is XP_003945711.1. | |||
TMPY-00619 | Serpin A1d Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
Serpin A1d Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 70.2 kDa and the accession number is XP_003945711.1. | |||
TMPJ-00022 | LGALS7 Protein, Human, Recombinant | Human | E. coli |
The Galectin family of proteins, with specificity for Nacetyllactosamine containing glycoproteins, consists of beta-galactoside binding lectins containing homologous carbohydrate recognition domains (CRDs).They also poss... | |||
TMPY-05674 | Human coronavirus (HCoV-NL63) Spike Protein (S1+S2 ECD, His) | HCoV-NL63 | Baculovirus Insect Cells |
Human coronavirus (HCoV-NL63) Spike Protein (S1+S2 ECD, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 142.4 kDa and the accession number is A0A1L2YVI8. | |||
TMPY-03236 | Human respiratory syncytial virus (RSV) Fusion protein/RSV-F (Strain RSS-2) Protein (His) | RSV | Baculovirus Insect Cells |
Human respiratory syncytial virus (RSV) Fusion protein/RSV-F (Strain RSS-2) Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.8 kDa and the accession number is P112... | |||
TMPY-05824 | Dengue virus (DENV)(type 3, strain Philippines/H87/1956) E/Envelope Protein (aa 247-675, His) | DENV | HEK293 Cells |
Dengue virus (DENV)(type 3, strain Philippines/H87/1956) E/Envelope Protein (aa 247-675, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 48.79 kDa and the accession number is A... | |||
TMPY-05670 | Human coronavirus (HCoV-NL63) Spike S1 Protein (His) | HCoV-NL63 | HEK293 Cells |
Human coronavirus (HCoV-NL63) Spike S1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 78.8 kDa and the accession number is A0A1L2YVI8. | |||
TMPY-05675 | Human coronavirus (HCoV-229E) Spike Protein (S1+S2 ECD, His) | HCoV-229E | Baculovirus Insect Cells |
Human coronavirus (HCoV-229E) Spike Protein (S1+S2 ECD, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 122.1 kDa and the accession number is A0A1L7B942. | |||
TMPY-05750 | Human coronavirus (HCoV-OC43) Spike S1 Protein (His) | HCoV-OC43 | HEK293 Cells |
Human coronavirus (HCoV-OC43) Spike S1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 89.02 kDa and the accession number is A0A2P1ZWW8. | |||
TMPY-01082 | Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (95% Homology) (His) | RSV | HEK293 Cells |
Human respiratory syncytial virus (RSV) (A, rsb1734) glycoprotein G/RSV-G Protein (95% Homology) (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.7 kDa and the accession num... | |||
TMPY-03574 | MERS-CoV Spike/S1 Protein (aa 1-725, His) | MERS-CoV | HEK293 Cells |
MERS-CoV Spike/S1 Protein (aa 1-725, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 79.9 kDa and the accession number is K0BRG7. | |||
TMPY-00891 | Neuropilin-1 Protein, Human, Recombinant (V179A, hFc) | Human | HEK293 Cells |
Neuropilin-1 Protein, Human, Recombinant (V179A, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 96.5 kDa and the accession number is O14786-2. | |||
TMPY-02429 | Human coronavirus HKU1 (isolate N1) (HCoV-HKU1) Spike S1 Protein (His) | HCoV-HKU1 | HEK293 Cells |
Human coronavirus HKU1 (isolate N1) (HCoV-HKU1) Spike S1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 85.8 kDa and the accession number is Q5MQD0. | |||
TMPY-05676 | Human coronavirus HKU1 (isolate N5) (HCoV-HKU1) Spike Protein (S1+S2 ECD, His) | HCoV-HKU1 | Baculovirus Insect Cells |
Human coronavirus HKU1 (isolate N5) (HCoV-HKU1) Spike Protein (S1+S2 ECD, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 144.4 kDa and the accession number is Q0ZME7.1. | |||
TMPY-05671 | Human coronavirus (HCoV-229E) Spike S1 Protein (His) | HCoV-229E | HEK293 Cells |
Human coronavirus (HCoV-229E) Spike S1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 58.3 kDa and the accession number is A0A1L7B942. | |||
TMPY-00402 | MERS-CoV Spike/RBD Protein fragment (aa 367-606, His) | MERS-CoV | Baculovirus Insect Cells |
MERS-CoV Spike/RBD Protein fragment (aa 367-606, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 27.7 kDa and the accession number is K0BRG7. | |||
TMPY-00356 | Neuropilin-1 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
Neuropilin-1 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 68.1 kDa and the accession number is XP_005564993.1. | |||
TMPY-01283 | Glypican 3/GPC3 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Glypican 3/GPC3 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 62 kDa and the accession number is P51654-1. | |||
TMPY-05688 | Human respiratory syncytial virus (RSV) Fusion Protein (aa 1-525, His) | RSV | Baculovirus Insect Cells |
Human respiratory syncytial virus (RSV) Fusion Protein (aa 1-525, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.12 kDa and the accession number is K7WLI9. | |||
TMPY-05740 | Neuropilin-1 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Neuropilin-1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 95.12 kDa and the accession number is P97333. | |||
TMPY-00502 | Glypican 3/GPC3 Protein, Mouse, Recombinant (His) | Mouse | Baculovirus Insect Cells |
Glypican 3/GPC3 Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 62 kDa and the accession number is Q3TWB2. | |||
TMPY-03661 | MERS-CoV Spike Protein (S1+S2 ECD, aa 1-1297, His) | MERS-CoV | Baculovirus Insect Cells |
MERS-CoV Spike Protein (S1+S2 ECD, aa 1-1297, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 44.10 kDa and the accession number is K0BRG7. | |||
TMPY-02731 | SPINK4 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
SPINK4 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 34.5 kDa and the accession number is O35679. | |||
TMPY-03512 | MERS-CoV Spike/S2 Protein (aa 726-1296, His) | MERS-CoV | Baculovirus Insect Cells |
MERS-CoV Spike/S2 Protein (aa 726-1296, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 63.84 kDa and the accession number is K0BRG7. | |||
TMPY-05677 | Human coronavirus (HCoV-OC43) Spike Protein (S1+S2 ECD, His) | HCoV-OC43 | Baculovirus Insect Cells |
Human coronavirus (HCoV-OC43) Spike Protein (S1+S2 ECD, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 145.1 kDa and the accession number is A0A2P1ZWW8. | |||
TMPY-01030 | TFPI Protein, Human, Recombinant (His) | Human | HEK293 Cells |
TFPI Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 30.6 kDa and the accession number is P10646-1. | |||
TMPY-04903 | Dengue virus (DENV) (type 3, strain Philippines/H87/1956) NS1 Protein (His) | DENV | HEK293 Cells |
Dengue virus (DENV) (type 3, strain Philippines/H87/1956) NS1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.1 kDa and the accession number is AAA99437.1. | |||
TMPY-03763 | Neuropilin-2 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Neuropilin-2 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 120.7 kDa and the accession number is O60462-3. | |||
TMPY-06013 | Human coronavirus (HCoV-OC43) Spike S2 Protein (His) | HCoV-OC43 | Baculovirus Insect Cells |
Human coronavirus (HCoV-OC43) Spike S2 Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 60.7 kDa and the accession number is A0A2P1ZWW8. | |||
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カタログ番号 | 製品名 | ||
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L1300 | PI3K-AKT-mTOR Compound Library | 420 compounds | |
A unique collection of 420 compounds targeting PI3K/Akt/mTOR signaling for research in PI3K/Akt/mTOR signaling, and drug discovery in diseases involved with PI3K/Akt/mTOR signaling; | |||
L7000 | Bioactive Lipid Compound Library | 385 compounds | |
A unique collection of 385 bioactive lipids related compounds for high throughput screening (HTS) and high content screening (HCS), including Agonists & Antagonists, Endocannabinoids, Farnesyl/geranylgeranyl derivates, ... | |||
L1200 | Epigenetics Compound Library | 953 compounds | |
Well-chosen 953 compounds related to epigenetic regulation for research in epigenetics, high throughput screening (HTS) and high content screening (HCS) for new drugs; | |||
L9400 | PPI Inhibitor Library | 485 compounds | |
A unique collection of 485 PPI-related compounds for drug screening; | |||
L9500 | Target-Focused Phenotypic Screening Library | 1796 compounds | |
A unique collection of 1796 annotated bioactive compounds with clear targets, suitable for phenotypic screening; | |||
L2510 | Lipid Metabolism Compound Library | 492 compounds | |
A unique collection of 492 compounds targeting lipid metabolism, can be used for high-throughput screening (HTS) and high-content screening (HCS). | |||
L1610 | FDA-Approved Kinase Inhibitor Library | 263 compounds | |
A unique collection of 263 kinase inhibitors/regulators for specific targeting of kinases, ready for high-throughput screening and high-content screening. | |||
L1600 | Kinase Inhibitor Library | 2720 compounds | |
A unique collection of 2720 kinase inhibitors/regulators for high throughput screening and high content screening for drug discovery in kinase related diseases; | |||
L6210 | Tibetan medicine Compound Library | 747 compounds | |
A collection of 747 natural product molecules originated from Tibetan medicine, which can be used for high-throughput and high-content screening. |