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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T21649L | GnRH Associated Peptide (1-13) Acetate(human) | GnRH Associated Peptide (GAP) (1-13), human Acetate (100111-07-7 Free base),GnRH Associated Peptide (1-13), Acetate(human) (100111-07-7 Free base) | Others |
GnRH Associated Peptide (GAP) (1-13), human Acetate was found to be a potent inhibitor of prolactin secretion and to stimulate the release of gonadotropins. Active immunization with peptides corresponding to GAP sequence... | |||
T80919 | Tumour-associated MUC1 epitope | ||
Tumor-associated MUC1 epitope, a biologically active peptide, is the distinctive feature of MUC1 mucin—a significantly glycosylated type I transmembrane glycoprotein. Its extracellular domain comprises variable numbers o... | |||
TP1420 | Microtubule-associated protein tau (26-44) | ||
Microtubule-associated protein tau (26-44) is a synthetic peptide with an amino group conjugated to glutamine and a carboxyl group conjugated to lysine. | |||
T76323 | GnRH Associated Peptide (25-53), human | ||
Gonadotropin-Releasing Hormone-Associated Peptide (GAP) (25-53), Human, also known as hGAP-25-53, is a fragment of the human gonadotropin-releasing hormone-associated peptide that serves as an immunogen for producing ant... | |||
T76324 | GnRH Associated Peptide (1-24), human | ||
Gonadotropin-Releasing Hormone-Associated Peptide (GAP) (1-24), human, also known as hGAP-1-24, is the 1-24 fragment of the human GAP, which is connected to the luteinizing hormone-releasing hormone (LH-RH) through a 3 a... | |||
T82346 | Galanin message associated peptide (1-41) amide | ||
Galanin message-associated peptide (1-41) amide is a peptide hormone [1]. | |||
T3080 | Pyridone 6 | Janus-Associated Kinase Inhibitor I,JAK Inhibitor,CMP 6,JAK Inhibitor I | Tyrosine Kinases , JAK |
Pyridone 6 (JAK Inhibitor)(CMP 6) is a potent and selective inhibitor of JAK1 (IC50=15 nM, murine JAK1), JAK2 (IC50=1 nM), JAK3 (Ki=5 nM), and Tyk2 (IC50=1 nM); displaying significantly weaker affinities (130 nM to 10 mM... | |||
T2155 | Thiazovivin | ROCK | |
Thiazovivin, a ROCK inhibitor (IC50: 0.5 μM), increases the survival rate of hESC. | |||
T14367 | AZ1495 | IRAK , CDK , Haspin Kinase | |
AZ1495 is an oral active inhibitor of Interleukin-1 receptor associated kinase 4 (IRAK4), with IC50 values of 5 nM and 23 nM for IRAK4 and IRAK1, respectively. Which Shows activity in treatment of mutant MYD88L265P diffu... | |||
T5110 | IRAK inhibitor 6 | IRAK | |
IRAK inhibitor 6 is an inhibitor of interleukin-1 receptor-associated kinase 4 (IRAK-4, IC50: 160 nM). | |||
T4140 | IRAK4-IN-1 | IRAK | |
IRAK4-IN-1 is an interleukin-1 receptor associated kinase 4 (IRAK4) inhibitor with an IC50 of 7 nM. | |||
T7301 | BDP5290 | ROCK | |
BDP5290 is a potent inhibitor of both ROCK and MRCK(IC50s of 5 nM, 50 nM, 10 nM and 100 nM for ROCK1, ROCK2, MRCKα and MRCKβ, respectively.) | |||
T5094 | IRAK inhibitor 1 | IRAK , JNK | |
IRAK inhibitor 1 is an effective IRAK-4 inhibitor (IC50: 216 nM), is poorly active against JNK-1 (IC50: 3.801 μM) and JNK-2 (IC50>10 μM). | |||
T7391 | SAR407899 | ROCK , Rho | |
SAR407899 is Rho kinase inhibitor potently inhibits endothelin-1-induced constriction of renal resistance arteries. | |||
T15798 | LX7101 | ROCK , LIM Kinase , PKA | |
LX7101 is an effective inhibitor of LIMK and ROCK2 (IC50: 24, 1.6, and 10 nM for LIMK1, LIMK2, and ROCK2, respectively). It also inhibits PKA (IC50 <1 nM). | |||
T1898 | RKI-1447 | RKI1447 | ROCK |
RKI-1447 is a potent inhibitor of ROCK1 and ROCK2. It has anti-invasive and antitumor activities. | |||
T3513 | GSK180736A | GSK180736 | ROCK , GRK , PKA |
GSK180736A is an effective and selective GRK2 inhibitor (IC50: 0.77 μM) and >100-fold selectivity over other GRKs. It is a weak inhibitor of PKA (IC50: 30 μM), but highly effective against ROCK1 (IC50: 100 nM). | |||
T12746 | ROCK inhibitor-2 | ROCK | |
ROCK inhibitor-2 is a selective dual inhibitor of ROCK1 and ROCK2 (IC50s of 17 nM and 2 nM, respectively). | |||
T14960 | Chroman 1 | ROCK | |
Chroman 1 is an inhibitor of ROCK2 (IC50: 1 nM). | |||
T2633 | GSK429286A | RHO-15 | ROCK |
GSK429286A (RHO-15) is a specific inhibitor of ROCK1/2 (IC50: 14/63 nM). | |||
T12747 | ROCK2-IN-2 | ROCK | |
TQ0187 | SR-3677 | ROCK , Autophagy | |
SR-3677 is an effective and specific inhibitor of ROCK2 (IC50: 3 nM). | |||
T1870 | Y-27632 | ROCK , Apoptosis | |
Y-27632 (Y-27632) is an orally potent, ATP-competitive inhibitor of ROCK-I and ROCK-II. Y-27632 also inhibits isolation-induced apoptosis in mouse prostate stem or progenitor cells. | |||
TQ0167 | Zimlovisertib | PF-06650833,PF06650833 | IRAK |
Zimlovisertib (PF-06650833) is an effective, selective and orally active inhibitor of interleukin-1 receptor-associated kinase 4 (IRAK4) (IC50s: 0.2 and 2.4 nM in the cell and PBMC assay). | |||
T4299 | AS-2444697 | IRAK | |
AS-2444697 is an inhibitor of IRAK-4 (C50 = 21 nM). AS-2444697 exhibits renoprotective effects through anti-inflammatory action. AS-2444697 potently inhibits human and rat IRAK-4 activity. | |||
T11673 | IRAK4-IN-4 | IRAK , cGAS | |
IRAK4-IN-4 (compound 15) inhibits cyclic GMP-AMP synthase (cGAS) with an IC50 of 2.1 nM.IRAK4-IN-4 is an interleukin-1 receptor–associated kinase 4 (IRAK4) inhibitor, has an IC50 of 2.8 nM. | |||
T4095 | ZINC00881524 | ROCK inhibitor | ROCK |
ZINC00881524 (ROCK inhibitor) is an effective and specific ROCK inhibitor. | |||
T9203 | JH-X-119-01 | IRAK | |
JH-X-119-01 is a highly potent and selective covalent inhibitor of IRAK-1. | |||
T2011 | RKI1313 | RKI 1313,RKI-1313 | ROCK |
RKI1313 (RKI-1313) was a selective inhibitor for ROCK-dependent signaling, cytoskeletal changes, anchorage-independent colony formation, migration, and invasion. | |||
T14989 | CMPD101 | ROCK , GRK , PKC | |
CMPD101 is a membrane-permeable small-molecule inhibitor of GRK2/3 (IC50: 18 nM and 5.4 nM). Which can be used for the study of heart failure. CMPD101 exhibits less selectively against GRK1, GRK5, ROCK-2 and PKCα with I... | |||
T7885 | Afuresertib hydrochloride | ROCK , Akt , PKC | |
Afuresertib hydrochloride is an inhibitor of Akt kinase (Kis of 0.08/2/2.6 nM for Akt1/Akt2/Akt3 respectively) | |||
T15781 | LP-935509 | Serine/threonin kinase , AAK1 (AP2 associated kinase 1) | |
LP-935509 is highly brain-penetrant and reverses fully established pain behavior following the SNL procedure. LP-935509 is also an effective inhibitor of BIKE (IC50=14 nM) and a modest inhibitor of GAK (IC50=320 nM). LP-... | |||
T9053 | Lats-IN-1 | Others , YAP | |
Lats-IN-1 is a potent and ATP-competitive Lats1 and Lats2 kinases inhibitor. It promotes Yap-dependent proliferation in postmitotic mammalian tissues. | |||
T13384L | Y-33075 dihydrochloride | CaMK , ROCK , PKC | |
Y-33075 dihydrochloride is a selective inhibitor of ROCK(IC50 of 3.6 nM). | |||
T7648 | HA-100 | Myosin , PKA , PKC | |
HA-100 is an inhibitor of protein kinase | |||
T2482 | AT13148 | ROCK , SGK , Akt , PKA , S6 Kinase | |
AT13148 is an oral-active and ATP-competitive, multi-AGC kinase inhibitor for Akt1/2/3, p70S6K, PKA, and ROCKI/II. | |||
T1911 | Afuresertib | GSK2110183C,GSK2110183 | ROCK , Akt , PKC |
Afuresertib (GSK2110183) is an orally bioavailable inhibitor of the serine/threonine protein kinase Akt (protein kinase B) with potential antineoplastic activity. | |||
T4276L | Hydroxyfasudil | Hydroxy-Fasudil,HA-1100 | ROCK , PKA |
Hydroxyfasudil (Hydroxy-Fasudil) is a ROCK inhibitor(IC50s of 0.73 and 0.72 μM for ROCK1 and ROCK2, respectively). | |||
T4488 | GSK-25 | GSK25 | ROCK , S6 Kinase , mTOR |
GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and p70S6K (RSK1 IC50 of 398 nM, p70S6K IC50 of 1000nM), and a dramatically improved P450 profile (>2.2 uM at all isozymes tested). | |||
T7764 | CCG-222740 | ROCK , Rho , Ras | |
CCG-222740 is an inhibitor of Rho/MRTF pathway | |||
TQ0110 | ROCK-IN-2 | TC-S 7001,Azaindole 1 | ROCK |
ROCK-IN-2 (Azaindole 1) is a selective and ATP-competitive ROCK inhibitor with IC50 of 0.6 and 1.1 nM for human ROCK-1 and ROCK-2. | |||
T5354 | IRAK4-IN-7 | CA-4948 | IRAK |
IRAK4-IN-7 (CA-4948) is a selective and potent IRAK4 kinase inhibitor with in vivo activity in a TLR4-induced cytokine release model. | |||
T9027 | CA-4948 | Emavusertib | IRAK , FLT |
CA-4948 (Emavusertib) is a potent IRAK4/FLT3 inhibtor. CA-4948 with anti-tumor activity. | |||
T9631 | IRAK-4 protein kinase inhibitor 2 | IRAK | |
IRAK-4 protein kinase inhibitor 2 is a potent interleukin-1 receptor-associated kinase-4 (IRAK-4) inhibitor(IC50 = 4 μM). | |||
T12885 | SGC-AAK1-1 | AAK1 (AP2 associated kinase 1) | |
SGC-AAK1-1 is a potent and selective inhibitor of AAK1 (AP2 associated kinase 1) (IC50 of 270 nM and a Ki of 9 nM),and is a chemical probe. | |||
T3518 | GSK269962A | GSK269962B,GSK 269962,GSK269962A HCl | ROCK , S6 Kinase |
GSK269962A (GSK269962A HCl) is a selective ROCK(Rho-associated protein kinase) inhibitor with IC50 values of 1.6 and 4 nM for ROCK1 and ROCK2, respectively. | |||
T23308 | SAR407899 hydrochloride | ROCK | |
ATP-competitive ROCK inhibitor | |||
T6867 | Belumosudil | KD025,Rezurock,ROCK inhibitor,SLx-2119 | ROCK |
Belumosudil (Rezurock) is an orally available, and specific ROCK2 inhibitor (IC50/Ki: 60/41 nM). | |||
T60012 | HS-243 | IRAK , MAPK , CDK | |
HS-243 is an inhibitor of IRAK-4 and IRAK-1 with IC50s of 20 and 24 nM. HS-243 shows anti-inflammatory and anticancer activity. | |||
T2457 | IRAK-1-4 Inhibitor I | IRAK-1/4 Inhibitor I,IRAK-1/4 Inhibitor | IRAK |
IRAK-1-4 Inhibitor I is a dual inhibitor of IRAK4 and IRAK1. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
TQ0183 | Narciclasine | Lycoricidinol | ROCK |
Narciclasine (Lycoricidinol), a natural product, modulates the Rho/Rho-kinase/LIM kinase/cofilin signaling pathway, greatly increasing GTPase RhoA activity. | |||
T2822 | Ginsenoside Rb1 | Gypenoside Ⅲ,Gypenoside III | ATPase , Mitophagy , IRAK , NF-κB , Autophagy , HSV |
Ginsenoside Rb1 (Gypenoside Ⅲ) is part of a class of steroid glycosides; may have properties that inhibit or prevent the growth of tumors. | |||
T6389 | Anacardic Acid | 6-pentadecylsalicylic Acid,Hydroginkgolic acid | Others , Epigenetic Reader Domain , Histone Acetyltransferase , Antibacterial |
Anacardic Acid (6-pentadecylsalicylic Acid) is an effective inhibitor of p300 and p300/CBP-associated factor histone acetyltranferases. It also has antimicrobial activity, antibacterial activity, and inhibits prostagland... | |||
T19581 | Tiglyl carnitine | Endogenous Metabolite | |
Tiglyl carnitine is associated with lung cancer and carnitine and glycine to 3-ketothiolase deficiency . | |||
T5883 | 4-Ethylphenol | Others , Endogenous Metabolite | |
4-Ethylphenol is the volatile phenol associated with the aroma in wine. | |||
TN3594 | Cardanol (C15:1) | Apoptosis , Others | |
Cardanol (C15:1), found in cashew nut shell liquid, induces mitochondria-associated apoptosis in human melanoma cells. | |||
T22974 | Methyl 2,5-dihydroxycinnamate | EGFR | |
EGF receptor-associated tyrosine kinases inhibitor | |||
T19391 | L-Hexanoylcarnitine | Others | |
L-Hexanoylcarnitine is found to be associated with celiac disease, is an acylcarnitine. | |||
T15157 | Dodecanoylcarnitine | Lauroylcarnitine | Endogenous Metabolite |
Dodecanoylcarnitine ((-)-Lauroylcarnitine) has been associated with disturbances in fatty acid oxidation, and the use of Dodecanoylcarnitine resulted in an increase in the permeability of salmon calcitonin. | |||
T22218 | 2'-Deoxyguanosine | Deoxyguanosine,Guanine deoxyriboside | Endogenous Metabolite |
2'-Deoxyguanosine (Guanine deoxyriboside) is a purine nucleoside that is recognized by members of the 2'-dG-II family.2'-Deoxyguanosine has been associated with aging, mutation, and carcinogenesis, and is oxidized by mol... | |||
TN1219 | 20-Hydroxyganoderic acid G | ||
20-Hydroxyganoderic acid G is a lanosterane triterpenoid obtained from the ethanolic extract of Ganoderma curtisii (Ganoderma curtisii) cotyledons. 20-Hydroxyganoderic Acid G inhibited LPS-activated BV-2 microglia, with ... | |||
T5S2076 | Senkyunolide I | Others , Caspase | |
1. Senkyunolide I has neuroprotective effect, associated with its anti-oxidation and anti-apoptosis properties. | |||
TN1296 | 5-Feruloylquinic acid | 5-O-Feruloylquinic acid,5-FQA | Tyrosinase , Sirtuin |
5-Feruloylquinic acid (5-FQA) is a potent Sirt1 agonist, it is a potential lead compound that can be further tested in drug development process for diseases associated with aging. | |||
TN1295 | 5-O-Caffeoylshikimic acid | IL Receptor , TNF , NO Synthase | |
5-O-Caffeoylshikimic acid shows anti-oxidative activity; it also shows anti-inflammatory activity, the underlying mechanism was associated with downregulation of nuclear factor-κB. | |||
T2862 | Desaminotyrosine | Phloretate,3-(4-Hydroxyphenyl)propanoic acid,Hydro-p-coumaric acid,3-(4-Hydroxyphenyl)propionic acid,Phloretic acid | Others , Influenza Virus , Endogenous Metabolite |
Desaminotyrosine (3-(4-Hydroxyphenyl)propionic acid) is a microbially associated metabolite. Desaminotyrosine protects from influenza through augmentation of type I interferon signaling. | |||
T3S0507 | Homovanillic acid | Homovaniuic acid,Vanilacetic acid,Vanillacetic acid | Others , Endogenous Metabolite |
Homovanillic acid (Vanillacetic acid) is a dopamine metabolite found to be associated with aromatic L-amino acid decarboxylase deficiency, growth hormone deficiency, celiac disease, and sepiapterin reductase deficiency. | |||
TQ0118 | Britannilactone | Desacetylinulicin | Others |
Britannilactone (Desacetylinulicin) is a sesquiterpene from Inula britannica with anti-inflammatory and anti-tumor activity.Britannilactone has been associated with this antimelanotic activity and can be used in studies ... | |||
T4S1796 | Heterophyllin B | PI3K | |
Heterophyllin B effectively suppresses the adhesion and invasion of the human esophageal carcinoma cells by mediating the PI3K/AKT/β-catenin pathways and regulating the expression levels of adhesion- and invasion-associa... | |||
T3343 | 5-methoxyflavone | 5-methoxy-2-phenylchromen-4-one | DNA/RNA Synthesis |
5-methoxyflavone (5-methoxy-2-phenylchromen-4-one) is a naturally occurring, low molecular weight flavonoids compound that associated with a wide wariety of biological activities. | |||
T3369 | Nuciferine | (-)-Nuciferine,VLT 049,Sanjoinine E | Dopamine Receptor , 5-HT Receptor |
Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera. It has a profile of action associated with dopamine receptor blockade. | |||
TN1507 | Clematichinenoside AR | TNF , Autophagy | |
Clematichinenoside AR exerts anti-inflammatory and immunosuppressive properties, it has anti-arthritic effects on PI3K/Akt signaling pathway and TNF-α± associated with collagen-induced arthritis. | |||
T4894 | L-Arabinitol | L-(-)-Arabitol | Endogenous Metabolite |
L-Arabinitol (L-(-)-Arabitol) is a potential biomarker for the comsuption of the food products such as sweet potato, deerberry, moth bean. L-Arabinitol is associated with Alzheimer's disease and ribose-5-phosphate isomer... | |||
T19315 | Ethyl nonanoate | Ethyl pelargonate | Others , Endogenous Metabolite |
Ethyl nonanoate (Ethyl pelargonate) is an abundant ester in spirits, and its presence is usually associated with the aroma of alcoholic beverages. | |||
T4872 | Palmitoleic acid | (Z)-Hexadec-9-enoic acid,(Z)-9-hexadecenoic acid | Endogenous Metabolite |
Palmitoleic acid ((Z)-Hexadec-9-enoic acid) is found to be associated with isovaleric acidemia, which is an inborn error of metabolism. | |||
T1709 | 2'-Deoxyinosine | Guanine deoxyriboside,Deoxyinosine | Others , Endogenous Metabolite |
2'-Deoxyinosine (Guanine deoxyriboside) inhibits the growth of human colon-carcinoma cell lines and is associated with purine nucleoside phosphorylase (PNP) deficiency. | |||
T5279 | Ethylmalonic acid | alpha-Carboxybutyrate,2-Ethylmalonic acid | Others , Endogenous Metabolite |
Ethylmalonic acid (alpha-Carboxybutyrate) can be found in blood, cerebrospinal fluid (CSF), and urine, as well as in human fibroblasts, prostate, and skeletal muscle tissues. Moreover, ethylmalonic acid is found to be as... | |||
TN6952 | Hexadecane | n-Hexadecane | |
Hexadecane (n-Hexadecane) acts as a carbon source for fungi and is associated with biodegradation by anaerobic organisms.Hexadecane inhibited skin hyperkeratinization in guinea pig skin experiments. | |||
T6S1587 | Notoginsenoside R2 | 20(S)-Notoginsenoside R2,Ginsenoside Ng-R2 | Others , Nrf2 |
Notoginsenoside R2 (20(S)-Notoginsenoside R2) has neuroprotection against 6-OHDA-induced neurotoxicity, is associated with Notoginsenoside R2-mediated P90RSK and Nrf2 activation through MEK1/2-ERK1/2 pathways. | |||
T3840 | Dihydroresveratrol | 3,4',5-Trihydroxybibenzyl | Estrogen Receptor/ERR , Others |
Dihydroresveratrol (3,4',5-Trihydroxybibenzyl) is a major metabolite of resveratrol that is produced by animal-associated bacteria, including the gut microbiota. Dihydroresveratrol and dihydroresveratrol monosulfate are ... | |||
T4S1983 | Periplogenin | 5-beta-Hydroxydigitoxigenin,Desoxostrophanthidin | Others |
1. Periplogenin (Desoxostrophanthidin) plays protective roles against thyrotoxicosis and associated cardiovascular problems, are mediated through its direct antithyroidal and/or LPO inhibiting properties. | |||
T7036 | 2,4'-Dihydroxybenzophenone | Antioxidant | |
2,4'-Dihydroxybenzophenone can effectively protect C57BL/6J mice from APAP-induced hepatotoxicity. Its mechanisms might be associated with its Antioxidant activity. | |||
T0507 | L-Pyroglutamic acid | pidolic acid,L-pyroglutamate,5-Oxoproline | Others , Endogenous Metabolite |
L-Pyroglutamic acid (pidolic acid), a cyclized derivative of the L-GLUTAMIC ACID, can elevate blood levels. This function may be associated with problems of GLUTATHIONE or GLUTAMINE metabolism. | |||
TN6779 | Clausine E | Others | |
Clausine E is an inhibitor of fat mass and obesity-associated protein (FTO) demethylase activity. The binding of Clausine E to FTO was driven by positive entropy and negative enthalpy changes. | |||
T3768 | Epifriedelanol | Epifriedelinol | Others |
Epifriedelanol (Epifriedelinol) suppresses adriamycin-induced cellular senescence, replicative senescence in human fibroblasts (HDFs) and HUVECs. Because of Epifriedelanol can reduce cellular senescence in human primary ... | |||
T5565 | Undecanedioic acid | Others , Endogenous Metabolite | |
Undecanedioic acid has been found in parts of human aortas with advanced atherosclerotic lesions associated with intercellular matrix macromolecules and specifically with elastin. | |||
T10017 | 1-Linoleoyl Glycerol | Glycerol 1-monolinolate,Monolinolein,Glyceryl monolinoleate,1-Linoleoyl-rac-glycerol | Phospholipase |
1-Linoleoyl Glycerol (Monolinolein) is fatty acid glycerol that has been isolated from Saururus Chinensis roots. The (R)-1-Linoleoyl Glycerol and (S)-1-Linoleoyl Glycerol exhibit Lipoprotein-associated phospholipase A2 (... | |||
T3911 | Pulchinenoside A | Anemoside A3 | Others |
Pulchinenoside A (Anemoside A3) is an attractive candidate for further development as a cognitive enhancer capable of alleviating memory dysfunctions associated with aging and neurodegenerative diseases. | |||
T4766 | 3-Methylglutaric acid | Endogenous Metabolite | |
Methylglutaric acid is a leucine metabolite. A large amount of methylglutaric acid is identified in urine of patients with deficiency of 3-methylglutaconyl coenzyme A hydratase (PMID 6181239 ). Methylglutaric acid is als... | |||
T5692 | Pyrroloquinoline quinone | Others , Endogenous Metabolite | |
Pyrroloquinoline quinone (PQQ), as a well-known redox enzyme cofactor, PQQ can protect NS/PCs against glutamate toxicity associated with ROS-mediated mitochondrial pathway, | |||
T3861 | Isobavachalcone | Corylifolinin,Isobacachalcone | Apoptosis , Others , Reactive Oxygen Species , Akt , Autophagy |
Isobavachalcone (Corylifolinin) is a chalcone constituent of Angelica keiskei, has potent anti-inflammatory activity, possible can ameliorate neuronal injury in brain diseases associated with inflammation. | |||
T3823 | D-Pinitol | Pinitol,Inzitol,D-(+)-Pinitol,Methylinositol,3-O-Methyl-D-chiro-inositol | Others , Influenza Virus |
D-Pinitol (Methylinositol) has anti-inflammatory activity. D-Pinitol(Methylinositol) exerts insulin-like activity, used for many diabetic associated conditions. D-Pinitol(Methylinositol) is a safe nutrient to reduce calo... | |||
TN1711 | Gossypetin | Antioxidant , p38 MAPK , MAPK , Antibacterial | |
Gossypetin, a hexahydroxylated flavonoid extractable from Rhodiola rosea Linn. is a potent MKK3 and MKK6 inhibitor that strongly attenuates the MKK3/6-p38 signaling pathway.Gossypetin exhibits antimutagenic, antiatherosc... | |||
T5S1285 | (+)-(3R,8S)-Falcarindiol | Falcarindiol | Others |
1. (+)-(3R,8S)-Falcarindiol is a potential new anticancer agent that exerts its activity through inducing ER stress and apoptosis. 2. Falcarindiol induces immunosuppressive effects in vitro and in vivo and might be a nov... | |||
T5226 | 2-(2-Methylbenzamido)acetic acid | 2-Methylhippuric acid,O-Toluric acid,N-(O-Toluoyl)glycine | Others , Endogenous Metabolite |
2-(2-Methylbenzamido)acetic acid (O-Toluric acid) is an acyl glycine. Acyl glycines are normally minor metabolites of fatty acids. In certain cases, the measurement of these metabolites in body fluids can be used to diag... | |||
T2P2919 | (2S,3R,4S)-4-Hydroxyisoleucine | (4S)-4-Hydroxy-L-isoleucine,Hydroxyisoleucine | PI3K |
(2S,3R,4S)-4-Hydroxyisoleucine (Hydroxyisoleucine) from fenugreek (Trigonella foenum-graecum) seeds is a potential insulinotropic (anti-diabetic) and anti-obesity amino acid. HIL stimulates glucose-dependent insulin secr... | |||
T3921 | Punicalagin | SARS-CoV , HBV | |
Punicalagin is a major ellagitannin found in pomegranates that is reported to produce antioxidant, anti-inflammatory, and anticancer effects. It has been shown to prevent high-fat diet-induced obesity-associated accumula... | |||
T3771 | Methyl protodioscin | Smilax saponin B,NSC-698790 | Apoptosis |
Methyl protodioscin (Smilax saponin B) potentially increase HDL cholesterol while reducing LDL cholesterol and triglycerides. Methyl protodioscin has antitumor property. Methyl protodioscin induced apoptotic process in h... | |||
T3S0137 | Bavachalcone | Antibacterial , Antibiotic | |
Bavachalcone is a major bioactive compounds isolated from Psoralea corylifolia L. it may be useful as a therapeutic drug for bone resorption-associated diseases.Bavachalcone can protect the endothelial function by increa... | |||
T3787 | Didymin | Isosakuranetin-7-O-rutinoside,Neoponcirin | Apoptosis , Others |
Didymin (Neoponcirin) has antioxidant property. Didymin induces apoptosis by inhibiting N-Myc and upregulating RKIP in neuroblastoma, may used for neuroblastoma therapy. Didymin may be a potential therapeutic molecule fo... | |||
T6194 | Fidaxomicin | Tiacumicin B,OPT-80,Clostomicin B1,PAR-101 | Apoptosis , DNA/RNA Synthesis , Antibacterial , Antibiotic |
Fidaxomicin (Tiacumicin B) is a semisynthetic macrolide antibiotic used to treat Clostridium difficile-associated diarrhea in adults. Fidaxomicin has minimal systemic absorption and has not been linked to serum enzyme el... | |||
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カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPY-05200 | CD79B Protein, Cynomolgus, Rhesus, Recombinant (His) | Cynomolgus,Rhesus | HEK293 Cells |
CD79B Protein, Cynomolgus, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.7 kDa and the accession number is H9ZFT8. | |||
TMPY-05153 | TROP-2 Protein, Cynomolgus, Rhesus, Recombinant (His) | Cynomolgus,Rhesus | HEK293 Cells |
TROP-2 Protein, Cynomolgus, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 28.7 kDa and the accession number is XP_001114599.1. | |||
TMPY-05302 | CD79 Protein, Human, Recombinant (Flag & His) | Human | HEK293 Cells |
CD79 Protein, Human, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 37.5 kDa and the accession number is NP_001774.1&NP_000617.1. | |||
TMPY-05275 | CD79B Protein, Human, Recombinant (His) | Human | HEK293 Cells |
CD79B Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.7 kDa and the accession number is P40259-1. | |||
TMPY-01253 | LAMP1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
LAMP1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 39.8 kDa and the accession number is A0A024RDY3. | |||
TMPJ-00113 | CD79B Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
CD79B Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-Fc tag. The predicted molecular weight is 45-65 KDa and the accession number is P40259. | |||
TMPY-01604 | CTLA-4 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
CTLA-4 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 15.46 kDa and the accession number is Q6GTR6. | |||
TMPY-00590 | CD79A Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
CD79A Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 39 kDa and the accession number is P11911. | |||
TMPY-03432 | KEAP1 Protein, Human, Recombinant | Human | Baculovirus Insect Cells |
KEAP1 Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 69.7 kDa and the accession number is Q14145. | |||
TMPY-03888 | KEAP1 Protein, Human, Recombinant (His & GST) | Human | Baculovirus Insect Cells |
KEAP1 Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 97.37 kDa and the accession number is A0A024R7C0. | |||
TMPY-02101 | KEAP1 Protein, Human, Recombinant (His & GST & Avi) | Human | Baculovirus Insect Cells |
KEAP1 Protein, Human, Recombinant (His & GST & Avi) is expressed in Baculovirus insect cells with His, GST and Avi tag. The predicted molecular weight is 99.2 kDa and the accession number is Q14145. | |||
TMPY-01030 | TFPI Protein, Human, Recombinant (His) | Human | HEK293 Cells |
TFPI Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 30.6 kDa and the accession number is P10646-1. | |||
TMPH-00296 | Pregnancy-associated protein bPAP Protein, Bovine, Recombinant (His & Myc) | Bovine | E. coli |
Pregnancy-associated protein bPAP Protein, Bovine, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 17.3 kDa and the accession number is P84... | |||
TMPH-00043 | Fanconi-associated nuclease 1 Protein, Ailuropoda melanoleuca, Recombinant (His & Myc) | Ailuropoda melanoleuca | E. coli |
Fanconi-associated nuclease 1 Protein, Ailuropoda melanoleuca, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 21.5 kDa and the accession n... | |||
TMPY-02667 | TROP-2 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
TROP-2 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 29.4 kDa and the accession number is Q8BGV3. | |||
TMPY-02245 | SNAP-25 Protein, Human, Recombinant (His) | Human | E. coli |
Synaptosomal-associated protein 25, also known as Super protein, Synaptosomal-associated 25 kDa protein, SNAP25 and SNAP, is a cytoplasm and cell membrane protein that belongs to the SNAP-25 family. SNAP25 / SUP contains... | |||
TMPY-04483 | IRAK4 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
Interleukin-1 receptor-associated kinase 4, also known as Renal carcinoma antigen NY-REN-64, IRAK-4, and IRAK4, is a member of the protein kinase superfamily, TKL Ser/Thr protein kinase family, and Pelle subfamily. IRAK4... | |||
TMPY-05159 | Granzyme A/GZMA Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Granzyme A/GZMA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.5 kDa and the accession number is P12544-1. | |||
TMPY-03425 | Tau Protein, Human, Recombinant (His) | Human | E. coli |
MAPT (microtubule-associated protein tau) can produce tau proteins. Tau proteins are proteins that stabilize microtubules. They are abundant in neurons of the central nervous system and are less common elsewhere, but are... | |||
TMPJ-00211 | CD47 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
CD47 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 30-45 KDa and the accession number is Q08722. | |||
TMPY-04348 | CTLA-4 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
CTLA-4 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 15 kDa and the accession number is P16410-1. | |||
TMPY-04824 | CTLA-4 Protein, Human, Recombinant | Human | HEK293 Cells |
CTLA-4 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 13.5 kDa and the accession number is P16410-1. | |||
TMPJ-01172 | IL-17 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Interleukin-17 is a potent pro-inflammatory cytokine produced by activated memory T cells. There are at least six members of the IL-17 family in humans and in mice. Mature mouse IL-17A shares 61% and 89% amino acid seque... | |||
TMPH-00028 | Adeno-associated virus 2 (isolate Srivastava/1982) Rep78 Protein (His & MBP) | AAV-2 | E. coli |
Plays an essential role in the initiation of viral DNA synthesis. Binds specifically to an inverted terminal repeat element (ITR) on the 3' and 5' ends of the viral DNA, where it cleaves a site specifically to generate a... | |||
TMPY-01262 | TROP-2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
TROP-2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 29.4 kDa and the accession number is P09758. | |||
TMPJ-00254 | TGF beta 3 Protein, Human/Mouse/Rat, Recombinant | Human,Mouse,Rat | HEK293 Cells |
Transforming growth factor beta 3(TGFB3) is a member of a TGF -β superfamily which is defined by theirstructural and functional similarities. TGFB3 is secreted as a complex with LAP. This latent form of TGFB3becomes acti... | |||
TMPY-04171 | MFAP3 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
MFAP3 (Microfibril Associated Protein 3) is a Protein Coding gene. The human gene encoding MFAP3 has a very simple structure, containing only two translated exons encoding a protein of 362 amino acids. The gene was found... | |||
TMPY-00047 | Dengue virus DENV-2 (Strain New Guinea C) Capsid protein/DENV-C Protein (His) | DENV | E. coli |
Dengue virus DENV-2 (Strain New Guinea C) Capsid protein/DENV-C Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 14 kDa and the accession number is W0GCK5. | |||
TMPY-03135 | Contactin 3 Protein, Rat, Recombinant (His) | Rat | HEK293 Cells |
Contactin 3 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 109.2 kDa and the accession number is Q62682. | |||
TMPY-03163 | Contactin 3 Protein, Rat, Recombinant (hFc) | Rat | HEK293 Cells |
Contactin 3 Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 134.8 kDa and the accession number is Q62682. | |||
TMPJ-00249 | TGF beta 1 Protein, Human, Recombinant (Avi), Biotinylated | Human | HEK293 Cells |
Transforming Growth Factor β-1 (TGFβ-1) is a secreted protein which belongs to the TGF-β family. TGFβ-1 is abundantly expressed in bone, articular cartilage and chondrocytes and is increased in osteoarthritis (OA). TGFβ-... | |||
TMPJ-00566 | MFAP4 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Microfibril-associated glycoprotein 4(MFAP4) is a secreted protein and contains 1 fibrinogen C-terminal domain, similarity to a bovine microfibril-associated protein. The protein has binding specificities for both collag... | |||
TMPY-03137 | CD79B Protein, Rat, Recombinant (His) | Rat | HEK293 Cells |
CD79B Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.8 kDa and the accession number is O70153. | |||
TMPY-03035 | CD79B Protein, Rat, Recombinant (hFc) | Rat | HEK293 Cells |
CD79B Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.2 kDa and the accession number is O70153. | |||
TMPJ-00147 | FOLR1 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
FOLR1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-Fc tag. The predicted molecular weight is 55-75 kDa and the accession number is P15328. | |||
TMPY-02888 | MAX Protein, Human, Recombinant (His & GST) | Human | Baculovirus Insect Cells |
MYC associated factor X contains 1 basic helix-loop-helix (bHLH) domain and belongs to the MAX family. It is highly expressed in the brain, heart, and lung while lower levels are seen in the liver, kidney, and skeletal m... | |||
TMPK-00900 | MFAP4 Protein, Human, Recombinant (His & Flag) | Human | HEK293 Cells |
MFAP4 Protein, Human, Recombinant (His & Flag) is expressed in HEK293 mammalian cells with N-His-Flag tag. The predicted molecular weight is 28.6 kDa and the accession number is P55083-1. | |||
TMPY-02916 | LAMP1 Protein, Rat, Recombinant (hFc) | Rat | HEK293 Cells |
LAMP1 Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65.1 kDa and the accession number is P14562. | |||
TMPY-03685 | LAMP2 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
LAMP2 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.4 kDa and the accession number is G7Q3L7. | |||
TMPY-00461 | BTLA Protein, Rat, Recombinant (mFc) | Rat | HEK293 Cells |
BTLA Protein, Rat, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 43.4 kDa and the accession number is Q6PNM1-1. | |||
TMPY-04047 | BTLA Protein, Rhesus, Recombinant (hFc) | Rhesus | HEK293 Cells |
BTLA Protein, Rhesus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 41.4 kDa and the accession number is A0A8J8XCU2. | |||
TMPY-02753 | Contactin 3 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Contactin 3 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 110 kDa and the accession number is Q07409. | |||
TMPK-01159 | MFAP4 Protein, Mouse, Recombinant (His & Flag) | Mouse | HEK293 Cells |
MFAP4 Protein, Mouse, Recombinant (His & Flag) is expressed in HEK293 mammalian cells with N-His-Flag tag. The predicted molecular weight is 28.7 kDa and the accession number is Q9D1H9-1. | |||
TMPY-05101 | BTLA Protein, Rhesus, Recombinant (His) | Rhesus | HEK293 Cells |
BTLA Protein, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 19.3 kDa and the accession number is A0A8J8XCU2. | |||
TMPK-00477 | MFAP4 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
MFAP4 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 27.60 kDa and the accession number is A0A2K5TQS8. | |||
TMPY-06815 | SYAP1 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
Synapse-associated protein 1 (SYAP1), also known as PRO3113 and BSTA, belongs to the synapse-associated BSD domain family, featuring three α-helices and two conserved tryptophan and phenylalanine residues located at the ... | |||
TMPJ-01362 | UBAP1 Protein, Human, Recombinant (His) | Human | E. coli |
Ubiquitin-Associated Protein 1 (UBAP1) belongs to the UBA domain family. Members of this family are related to ubiquitin and the ubiquitination pathway. Because of their cytogenetic location, this UBA domain family membe... | |||
TMPH-02267 | AGTRAP Protein, Human, Recombinant (His & Myc & SUMO) | Human | E. coli |
Appears to be a negative regulator of type-1 angiotensin II receptor-mediated signaling by regulating receptor internalization as well as mechanism of receptor desensitization such as phosphorylation. Induces also a decr... | |||
TMPJ-01179 | SWSAP1 Protein, Human, Recombinant (His) | Human | E. coli |
SWSAP1 is a nucleus ATPase protein, interacts with ZSWIM7 and forms a functional complex. The complexs involved in homologous recombination repair and stabilizes each other. SWS1AP1 also interacts with RAD51, RAD51B, RAD... | |||
TMPY-02402 | WTAP Protein, Human, Recombinant (GST) | Human | E. coli |
Wilms' tumor 1-associating protein (WTAP) was previously identified as a protein associated with Wilms' tumor-1 (WT-1) protein that is essential for the development of the genitourinary system. WT1 was originally identif... | |||
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