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カタログ番号	製品名	別名	ターゲット
T4316	ML365		Potassium Channel
	ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).		Potassium Channel
T0280	Spiperone	Spiroperidol,Spiropitan	Dopamine Receptor
	Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds. It has been recommended in the treatment of SCHIZOPHRENIA.		Dopamine Receptor
TP1088	N-Acetylcarnosine	N-Acetyl-L-carnosine	Others
	N-Acetylcarnosine (N-Acetyl-L-carnosine) is thought to be able to combat some of the effects of oxidative stress as it has anti-oxidant properties.		Others
T12146	N-Desmethyl-Apalutamide	N-Desmethyl Apalutamide	P450 , Androgen Receptor
	N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.		P450 , Androgen Receptor
T22416	RO495	CS-2667	Tyrosine Kinases , JAK
	RO495 (CS-2667), a potent inhibitor of TYK2, inhibits TYK2 with IC50 of 1.5nM as tested in cell-based pharmacological assays		Tyrosine Kinases , JAK
T15233	Endovion	NS3728	Chloride channel
	Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.		Chloride channel
TN6963	Hentriacontane		NF-κB
	Hentriacontane is a natural product.		NF-κB
T24932	Vatanidipine	AE-0047,AE 0047,AE0047	Calcium Channel
	Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lasting hypotensive action was observed in various experimental hypertensi...		Calcium Channel
T14978	CL-82198		MMP
	CL-82198, a selective MMP-13 inhibitor, serves as a pharmacological intervention to halt the progression of osteoarthritis (OA). Its mechanism of action involves binding to the S1’ pocket of MMP-13, ensuring its selectiv...		MMP
T4688	Pipequaline hydrochloride	PK-8165 hydrochloride	GABA Receptor
	Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely re...		GABA Receptor
T21720	GP-82996	Cdk4/6 Inhibitor IV,CINK4	CDK
	GP-82996 (CINK4) is a pharmacological inhibitor specifically targeting CDK4/6, exhibiting IC50 values of 1.5 μM for CDK4/cyclin D1, 5.6 μM for CDK6/cyclin D1, and 25 μM for Cdk5/p35. It effectively induces apoptosis in U...		CDK
T21777	VU0359595	VU0359595-1,CID-53361951,ML-270	Phospholipase
	VU0359595 (ML-270) is a potent and selective pharmacological phospholipase D1 (PLD1) inhibitor with an IC50 of 3.7 nM. VU0359595 is >1700-fold selective for PLD1 over PLD2 (IC50 of 6.4 μM). VU0359595 can be used for the ...		Phospholipase
T5159	Olodaterol hydrochloride	BI-1744 HCl,BI 1744 hydrochloride	Adrenergic Receptor
	Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and activating β2-adrenergic receptors...		Adrenergic Receptor
T0797	Cimetidine	SKF-92334	Histamine Receptor
	Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological actions. It inhibits GASTRIC ACID secretion, as well as PEP...		Histamine Receptor
T1540	Doxepin hydrochloride	Toruan,Doxepin HCl,Aponal,Novoxapin	P450 , Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , AChR , Norepinephrine , Histamine Receptor
	Doxepin hydrochloride (Aponal) is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation. Its mechanism of action is not fully understood, but it ap...
T35028	Valiglurax	VU2957,VU 0652957,VU 2957,VU-0652957,VU0652957,VU-2957	GluR
	Valiglurax (VU2957), also known as VU0652957 and VU2957, is a potent, selective, CNS penetrant, and orally bioavailable mGlu4 PAM. VU2957 possessed attractive in vitro and in vivo pharmacological and DMPK properties acro...		GluR
T11016	DGAT-1 inhibitor 2		Transferase
	DGAT-1 inhibitor 2 is an effective DGAT-1 inhibitor; anti-obesity drug. Objective: DGAT-1 acyl-CoA: diacylglycerol acyltransferase 1 (DGAT1) is one of two known DGAT enzymes that catalyze the final step of triglyceride s...		Transferase
T12654	(Rac)-Acolbifene	(Rac)-EM-652,EM-343	Estrogen Receptor/ERR
			Estrogen Receptor/ERR
T67917	ML353	VU0478006	Potassium Channel
	ML353 (VU0478006) is a selective activator of TREK-1 and TREK-2 and a selective ligand (Ki =18.2 nM) for the mGlu5 Silencing Allosteric Modulator (SAM). ML353 has potential as a solution to the intrinsic activity or phar...		Potassium Channel
T0005	Aspirin	Acetylsalicylate,Acetylsalicylic Acid,ASA	Mitophagy , Virus Protease , COX , Autophagy
	Aspirin (Acetylsalicylic Acid) is a potent and selective inhibitor of COX with various pharmacological activities, such as anti-inflammation and pain relief. Aspirin is a histone deacetylase inhibitors to up-regulate cel...		Mitophagy , Virus Protease , COX , Autophagy
T1787	Levobupivacaine		Sodium Channel
	Levobupivacaine is an amino-amide local anaesthetic drug belonging to the family of n-alkylsubstituted pipecoloxylidide. It is the S-enantiomer of bupivacaine. Levobupivacaine hydrochloride is commonly marketed by AstraZ...		Sodium Channel
Fr13587	7-Chloro-4-(piperazin-1-yl)quinoline
	7-Chloro-4-(piperazin-1-yl)quinolone is an important scaffold in medicinal chemistry. It exhibited either alone or as hybrid with other active pharmacophores diverse pharmacological profiles. 7-Chloro-4-(piperazin-1-yl)q...
T0455	Clozapine	HF 1854,LX 100-129	Dopamine Receptor , Adrenergic Receptor , AChR
	Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and displays a unique pharmacological profile. Clozapine is a...		Dopamine Receptor , Adrenergic Receptor , AChR
T36520	COR659		Cannabinoid Receptor , GABA Receptor
	COR659 is a GABAB positive allosteric modulator (PAM) . COR659 suppresses alcohol and chocolate self-administration in rats[1]. COR659 apparently exerts its effects via a composite mechanism, including positive allosteri...		Cannabinoid Receptor , GABA Receptor
T29533	ABT-866	ABT 866,A 286666
	ABT-866 is a novel alpha-adrenoceptor agent with mixed pharmacological properties.
T31178	Dabequin	dabechin,G 800
	Dabequin is a derivative of aminoquinoline. It is said to have pharmacological activity against Plasmodium fukiparum.
T68749	EBOV-IN-C31
	EBOV-IN-C31 is a novel PP1-targeting Ebola Virus (EBOV) inhibitor with improved pharmacological properties.
T11893L	Lurasidone metabolite 14326 hydrochloride	Lurasidone metabolite 14326 hydrochloride (186204-33-1 free base)	Others
	Lurasidone metabolite 14326 hydrochloride, an active metabolite of the atypical antipsychotic Lurasidone, maintains its significant function in pharmacological efficacy.		Others
T28822	SNAP 398299	SNAP-398299,SNAP398299
	SNAP 398299, a galanin receptor antagonist, is a potential novel pharmacological treatment for mood disorders.
T33607	NBI-34041	NBI34041,SB 723620,SB-723620,SB723620
	NBI-34041 is an effective and high-affinity CRF1 receptor antagonist that effectively reduces endocrine responses to CRF(1) receptor-mediated pharmacological and behavioral challenges.
T23628	AD-2646	AD2646
	AD-2646 is a new quinoline derivative. It also has similar pharmacological properties to tricyclic antidepressants.
T20492	Tetragastrin	Cholecystokinin tetrapeptide,Gastrin tetrapeptide
	Tetragastrin is the C-terminal tetrapeptide of gastrin. It has the same physiological and pharmacological activity as gastrin.
T34819	Tetragastrin HCl	Trp-Met-Asp-Phe hydrochloride,Tetragastrin hydrochloride
	Tetragastrin HCl is the HCl salt of Tetragastrin, the C-terminal tetrapeptide of gastrin. It has the same physiological and pharmacological activity as gastrin.
T30489	BMS 181101	BMS181101,BMS-181101
	BMS-181101 is a novel antidepressant that has pharmacological characteristics as a serotonin reuptake inhibitor and a serotonin 5-HT receptor agonist.
T23710	Watanidipine dihydrochloride
	Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.
T14940	CGP11952		Others
	CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.		Others
T19182	Afegostat D-Tartrate	Isofagomine D-Tartrate,D-Isofagomine D-Tartrate	Others
			Others
T25542	Isamfazone	Isamfazona,Isamfazonum
	Isamfazone is utilized in the chemical and pharmacological studies on substituted pyridazones, the discovery of novel anti-inflammatory agents by aligning screening.
T71600	Benazoline oxalate salt
	Benazoline oxalate salt is a pharmacological active compound that inhibits casein kinase Iε (CKIε) or CKIδ phosphorylation of the PER2 protein.
T19181	Afegostat	D-Isofagomine,Isofagomine	Others
			Others
T29227	ZK-91296	ZK 91296,ZK91296
	ZK-91296 is a GABA receptor agonist. ZK 91296 can reduce anxiety in animals at doses well below those causing sedation. ZK 91296 may possess pharmacological selectivity for a particular type of BZ receptor interaction, p...
T23653	Afegostat HCl	Afegostat,AT-2101,Afegostat hydrochloride,AT2101
	Afegostat is an acid β-glucosidase (GCase) active site inhibitor that acts as a pharmacological chaperone. Afegostat inhibits GCase with K(i) ~30 nM for wild-type and mutant enzymes. Afegostat was an experimental drug fo...
T36664	Dehydro Aripiprazole (hydrochloride)
	Dehydro aripiprazole is the primary, active metabolite of aripiprazole, an atypical antipsychotic. The metabolite is produced from the parent compound by the actions of cytochrome P450 (CYP) isoforms CYP3A4 and CYP2D6. D...
T27210	DRX-065	DRX 065,DRX065,deuterated R-enantiomer of pioglitazone
	DRX-065 is a stabilized and deuterated R-enantiomer of pioglitazone. DRX-065 has pharmacological properties desirable for the treatment of NASH (mitochondrial function modulation, non-steroidal anti-inflammatory effects,...
T75002	Antidepressant agent 3
	Antidepressant agent 3, an orally active compound, showcases multifaceted pharmacological properties including antidepressant, anxiolytic, performance-enhancing, and nootropic activities [1].
T60284	4-(Phenyldiazenyl)benzoic acid
	4-(Phenyldiazenyl)benzoic acid is a photosensitive and photoswitchable TRPA1 agonist that can be used as pharmacological tool to study pain signaling.
T78564	Depramine	GP 31406
	Depramine (GP 31406), a tricyclic antidepressant, exhibits pharmacological activity by inhibiting acetylcholinesterase, Mg^2+-ATPase, and Na^+/K^+ ATPase activity [1] [2].
T38261	Sparstolonin B
	Sparstolonin B is a chemical compound that functions as a selective antagonist for TLR2 and TLR4, specifically targeting TLR2- and TLR4-mediated inflammatory signaling. This compound demonstrates additional pharmacologic...
T39795	Tricarbonyldichlororuthenium(II) dimer	CORM-2
	Tricarbonyldichlororuthenium(II) dimer, a pharmacological CO donor, prevents ischemia/reperfusion (I/R)-induced oxidative damage to the gastric mucosa by enhancing gastric blood flow (GBF) and reducing DNA oxidation and ...
T71160	Levomepromazine HCl
	Levomepromazine HCl is a phenothiazine with pharmacological activity similar to that of both CHLORPROMAZINE and PROMETHAZINE. It has the histamine-antagonist properties of the antihistamines together with CENTRAL NERVOUS...

Compounds

ML365

T4316

Synonym:

Target: Potassium Channel

Spiperone

T0280

Synonym: Spiroperidol,Spiropitan

Target: Dopamine Receptor

N-Acetylcarnosine

TP1088

Synonym: N-Acetyl-L-carnosine

Target: Others

N-Desmethyl-Apalutamide

T12146

Synonym: N-Desmethyl Apalutamide

Target: P450, Androgen Receptor

RO495

T22416

Synonym: CS-2667

Target: Tyrosine Kinases, JAK

Endovion

T15233

Synonym: NS3728

Target: Chloride channel

Synonym: AE-0047,AE 0047,AE0047

Target: Calcium Channel

Pipequaline hydrochloride

T4688

Synonym: PK-8165 hydrochloride

Target: GABA Receptor

GP-82996

T21720

Synonym: Cdk4/6 Inhibitor IV,CINK4

Target: CDK

VU0359595

T21777

Synonym: VU0359595-1,CID-53361951,ML-270

Target: Phospholipase

Olodaterol hydrochloride

T5159

Synonym: BI-1744 HCl,BI 1744 hydrochloride

Target: Adrenergic Receptor

Cimetidine

T0797

Synonym: SKF-92334

Target: Histamine Receptor

Doxepin hydrochloride

T1540

Synonym: Toruan,Doxepin HCl,Aponal,Novoxapin

Target: P450, Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor

Valiglurax

T35028

Synonym: VU2957,VU 0652957,VU 2957,VU-0652957,VU0652957,VU-2957

Synonym: (Rac)-EM-652,EM-343

Target: Estrogen Receptor/ERR

ML353

T67917

Synonym: VU0478006

Target: Potassium Channel

Aspirin

T0005

Synonym: Acetylsalicylate,Acetylsalicylic Acid,ASA

Target: Mitophagy, Virus Protease, COX, Autophagy

Levobupivacaine

T1787

Synonym:

Target: Sodium Channel

7-Chloro-4-(piperazin-1-yl)quinoline

Synonym: HF 1854,LX 100-129

Target: Dopamine Receptor, Adrenergic Receptor, AChR

COR659

T36520

Synonym:

Target: Cannabinoid Receptor, GABA Receptor

ABT-866

T29533

Synonym: ABT 866,A 286666

Target:

Dabequin

T31178

Synonym: dabechin,G 800

Lurasidone metabolite 14326 hydrochloride

T11893L

Synonym: Lurasidone metabolite 14326 hydrochloride (186204-33-1 free base)

Target: Others

SNAP 398299

T28822

Synonym: SNAP-398299,SNAP398299

Target:

NBI-34041

T33607

Synonym: NBI34041,SB 723620,SB-723620,SB723620

Synonym: Cholecystokinin tetrapeptide,Gastrin tetrapeptide

Target:

Tetragastrin HCl

T34819

Synonym: Trp-Met-Asp-Phe hydrochloride,Tetragastrin hydrochloride

Target:

BMS 181101

T30489

Synonym: BMS181101,BMS-181101

Target:

Watanidipine dihydrochloride

Synonym: Isofagomine D-Tartrate,D-Isofagomine D-Tartrate

Target: Others

Isamfazone

T25542

Synonym: Isamfazona,Isamfazonum

Target:

Benazoline oxalate salt

Synonym: D-Isofagomine,Isofagomine

Target: Others

ZK-91296

T29227

Synonym: ZK 91296,ZK91296

Target:

Afegostat HCl

T23653

Synonym: Afegostat,AT-2101,Afegostat hydrochloride,AT2101

Target:

Dehydro Aripiprazole (hydrochloride)

Synonym: DRX 065,DRX065,deuterated R-enantiomer of pioglitazone

Target:

Antidepressant agent 3

T75002

Synonym:

Target:

4-(Phenyldiazenyl)benzoic acid

Tricarbonyldichlororuthenium(II) dimer

カタログ番号	製品名	別名	ターゲット
T5722	Nevadensin	Pedunculin	Anti-infection , Antibacterial
	Nevadensin is an important herb-based constituent inhibiting estragole bioactivation. Nevadensin protects against a methyleugenol-induced marker of hepatocarcinogenicity in male F344 rat. It also exhibits inhibition acti...		Anti-infection , Antibacterial
T4104	Ophiopojaponin C	Ophiopogonin C	Others
	Ophiopogonin C' pharmacological activities may be related to the substances in nucleus mainly.		Others
T3O2709	Bronze Red	Scarlet 808	Others
	Bronze Red, an amide class organic compound, is utilized for content determination, identification, and pharmacological experiments.		Others
TQ0264	Nigakinone		Others
	Nigakinone, isolated from Kumu, is an alkaloid with the pharmacological activity.		Others
T7324	Chelidonine hydrochloride		Others
	Chelidonine hydrochloride is one of the alkaloids of Chelidonium majus, which has broad pharmacological activities		Others
T2837	Chrysin	5, 7-Dihydroxyflavone,NSC 407436,5,7-Dihydroxyflavone	Estrogen Receptor/ERR , Antioxidant
	Chrysin (5,7-Dihydroxyflavone) exhibits many biological activities and pharmacological effects, including antioxidant, anti-inflammatory, anticancer, and antiviral activities.		Estrogen Receptor/ERR , Antioxidant
T3S1251	Neoruscogenin		ROR
	1. Neoruscogenin represents a universal pharmacological tool for RORα research due to its specific selectivity profile versus other nuclear receptors.		ROR
T3362	Eupatilin	NSC 122413	PPAR , Autophagy
	Eupatilin (NSC-122413), a flavone derived from Artemisia princepsPampanini, is a PPARα agonist, with pharmacological activity.		PPAR , Autophagy
T7443	4'-Methoxychalcone		PARP , PPAR
	4'-Methoxychalcone with a variety of pharmacological activities, such as anti-tumor and anti-inflammatory activities.		PARP , PPAR
T4S1659	Xanthotoxol	8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,8-Hydroxypsoralene	Reactive Oxygen Species , 5-HT Receptor , Endogenous Metabolite
	Xanthotoxol (Psoralen) is a biologically active linear furocoumarin, shows strong pharmacological activities as anti-inflammatory, antioxidant, 5-HT antagonistic, and neuroprotective effects.
T2891	Ammonium glycyrrhizinate	Glycamil,Monoammonium glycyrrhizinate,Ammonium Glycyrrhizate,Monoammonium glycyrrhizinate hydrate,Glycyrram	Others
	Ammonium glycyrrhizinate (Glycyrram) has various pharmacological actions such as anti-inflammatory, antiallergic, antigastriculcer, and antihepatitis activities.		Others
TN1714	Grosvenorine	Grosvenorin	Antibacterial
	Grosvenorine (Grosvenorin) exhibits good antibacterial and antioxidant activities, with its metabolites possessing more potent activities, intestinal bacteria play an important role in the gastrointestinal metabolism of ...		Antibacterial
T2817	Picroside II	Vanilloyl catalpol,6-Vanilloylcatalpol	Apoptosis , Others , Influenza Virus , NF-κB , Reactive Oxygen Species
	Picroside II (Vanilloyl catalpol) is the main active ingredient in iridoid glycosides. It has antioxidant, anti-inflammatory, immune regulatory, anti-virus and other pharmacological activities.
T2718	Palmatine chloride		Others , Indoleamine 2,3-Dioxygenase (IDO) , Aurora Kinase
	Palmatine chloride an isoquinoline alkaloid, is an important medicinal herbal extract with diverse pharmacological and biological properties.		Others , Indoleamine 2,3-Dioxygenase (IDO) , Aurora Kinase
T0595	Naringin	Naringoside	Mitophagy , P450 , Endogenous Metabolite , Autophagy
	Naringin (Naringoside), a flavanone glycoside, exerts various of pharmacological effects such as blood lipid lowering, antioxidant activity, anticancer activity, and inhibition of cytochrome P450 enzymes.		Mitophagy , P450 , Endogenous Metabolite , Autophagy
T2746	Sophocarpine monohydrate	Sophocarpine	Apoptosis , Influenza Virus , Akt , PI3K , AMPK , Autophagy
	Sophocarpine monohydrate, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.		Apoptosis , Influenza Virus , Akt , PI3K , AMPK , Autophagy
T5749	10-Deacetyl-7-xylosyl paclitaxel	10-Deacetyl-7-xylosyltaxol,10-Deacetyltaxol 7-Xyloside,7-Xylosyl-10-deacetyltaxol,10-Deacetylpaclitaxel 7-Xyloside	Others , Microtubule Associated
	10-Deacetyl-7-xylosyl paclitaxel (7-Xylosyl-10-deacetyltaxol) is a Paclitaxel derivative with improved pharmacological features and higher water solubility,used in Chinese clinics to treat cancer.		Others , Microtubule Associated
T2866	Echinocystic acid		Apoptosis , Antioxidant , Reactive Oxygen Species
	Echinocystic acid (EA), a natural triterpone enriched in various herbs, shows a range of pharmacological activities including anti-inflammatory and antioxidant effects.		Apoptosis , Antioxidant , Reactive Oxygen Species
T1716	Echinacoside		Reactive Oxygen Species , Wnt/beta-catenin
	Echinacoside is a natural polyphenolic compound with various kinds of pharmacological activities, such as anti-inflammatory, antioxidative, hepatoprotective, neuroprotective, nitric oxide radical-scavenging and vasodilat...		Reactive Oxygen Species , Wnt/beta-catenin
TN7030	Heteroclitin G		Others
	Heteroclitin G was found as potential biomarkers of KIS blood-replenishing activity, and quantitative analysis provided a research basis for further pharmacological research.		Others
T6S1101	Astragalin	Kaempferol 3-D-glucoside,Kaempferol 3-O-glucoside,kaempferol-3-glucoside,3-Glucosylkaempferol,Astragaline,Kaempferol 3-β-D-glucopyranoside	Apoptosis , NF-κB
	Astragalin (Kaempferol 3-O-glucoside) is a biologically active natural flavonoid. It has a variety of pharmacological properties, including antioxidant, anti-inflammatory, anti-cancer, neuroprotective, and cardioprotecti...		Apoptosis , NF-κB
T3373	Columbianadin	Zosimin,2-Butenoic acid	Apoptosis
	Columbianadin (Zosimin), one of the main bioactive constituents of the roots of Angelica pubescens Maxim. f. biserrata Shan et Yuan, has been found to possess obvious pharmacological effects in previous studies.		Apoptosis
T5S1882	Songorine	Napellonine,Zongorine,Bullatine G	Others , GABA Receptor
	Songorine (Napellonine) shows favorable anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.		Others , GABA Receptor
TN1046	Murrayone		Others
	Murrayone, a coumarin-containing compound derived from M. paniculata, stands out as the most bioactive substance within this species, primarily due to its unique pharmacological attributes that notably suppress cancer me...		Others
T4878	Hecogenin	Hocogenin	Others , Antifungal
	Hecogenin (Hocogenin), a steroid saponin derived from Agave sisalana, serves as a specific inhibitor for human UDP-glucuronosyltransferases. Notably, it exhibits a broad range of pharmacological activities, such as anti-...		Others , Antifungal
T5737	Euphol		Others , Lipase , Endogenous Metabolite
	Euphol, an alcohol tetracyclic triterpene, has a wide range of pharmacological properties and is considered to have anti-inflammatory action.		Others , Lipase , Endogenous Metabolite
T1516	Curcumin	Diferuloylmethane,Natural Yellow 3,Indian Saffron,Turmeric yellow	Mitophagy , Epigenetic Reader Domain , Ferroptosis , Influenza Virus , Nrf2 , Histone Acetyltransferase , HDAC , Autophagy
	Curcumin (Natural Yellow 3) is a phenolic natural product, an inhibitor of histone acetyltransferase p300/CREB (IC50=25 μM) with specificity. Curcumin has a wide range of pharmacological activities such as antitumor, ant...
T5764	Alliin	(S)-3-(Allylsulphinyl)-L-alanine	NF-κB , PPAR
	Alliin ((S)-3-(Allylsulphinyl)-L-alanine) is a garlic organosulfur compound that possesses various pharmacological properties.alliin protected against LPS-induced ALI by activating PPARγ, which subsequently inhibited LPS...		NF-κB , PPAR
T8250	2,6,6-Trimethyl-2,4-cycloheptadien-1-one		Others
	2,6,6-Trimethyl-2,4-cycloheptadien-1-one is a terpene compound found in many plants, including parsley, dill and celery. It is an important component of essential oils and has a variety of medicinal and pharmacological p...		Others
T3S1250	Ophiogenin 3-O-α-L-rhamnopyranosyl-(1→2)-β-D-glucopyranoside	Ophiogenin-3-O-alpha-L-rhaMnopyranosyl-(1->2)-beta-D-glucopyranoside	Others
	Ophiogenin 3-O-α-L-rhamnopyranosyl-(1→2)-β-D-glucopyranoside (Ophiogenin-3-O-alpha-L-rhaMnopyranosyl-(1->2)-beta-D-glucopyranoside) is a natural product, and has good pharmacological effects on the cardiovascular system.		Others
TN1966	N-(3-Methoxybenzyl)Oleamide	N-Benzyloleamide,MAC 18:1	Antioxidant
	N-(3-Methoxybenzyl)Oleamide (MAC 18:1), an agmatine isolated from Lepidium meyenii, has pharmacological effects on exercise-induced fatigue, which may be related to the modulation of energy metabolism and improvement of ...		Antioxidant
T3920	Pseudoginsenoside F11	Ginsenoside A1	Others , Endogenous Metabolite
	Pseudoginsenoside F11 (Ginsenoside A1) is a component of Panax quinquefolium (American ginseng) which main pharmacological activities are positive inotropic effect on isolated heart function, good therapeutic effect on m...		Others , Endogenous Metabolite
T4749	Squalene	Nikko Squalane EX,Super Squalene,AddaVax,all-trans-Squalene,trans-Squalene,Spinacene	Reactive Oxygen Species , Endogenous Metabolite , Antifungal
	Squalene (AddaVax) is a natural organic compound originally obtained for commercial purposes primarily from shark liver oil, though there are botanical sources as well, including rice bran, wheat germ, and olives. All hi...
T2729	Scoparone	Escoparone,Scoparon,Aesculetin dimethyl ether,6,7-dimethoxycoumarin,6,7-Dimethylesculetin	Others
	Scoparone (Aesculetin dimethyl ether) can be found in a number of food items such as sweet orange, wild celery, mandarin orange (clementine, tangerine), and lemon. It is found in the Chinese herb Artemisia scoparia and h...		Others
T3030	L-Sophoridine	Sophoridine,Matridin-15-one	Others
	L-Sophoridine (Matridin-15-one) , a natural product obtained from medicinal plants, which has a variety of pharmacological effects, including anti-Y effects, and selectively induces apoptotic cell death in a variety of h...		Others
T6677	Sophocarpine		ERK , p38 MAPK , NF-κB , TLR , COX , HER , JNK , STAT
	Sophocarpine, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.		ERK , p38 MAPK , NF-κB , TLR , COX , HER , JNK , STAT
T2768	Saikosaponin A		NF-κB , Antibacterial , Liver X Receptor
	Saikosaponin A has a variety of pharmacological benefits, including antiepileptic, anti-osteoporosis, antioxidant, anti-in ammatory, immunomodulatory, and anti-bacterial activities. It can effectively attenuate neuropath...		NF-κB , Antibacterial , Liver X Receptor
TN5888	Toddaculin		Others
	Toddaculine may be beneficial for the prevention and treatment of osteoporosis, it can not only inhibit the differentiation of osteoclasts via activation of the NF-κB, ERK 1/2, and p38 MAPK signaling pathways, but can in...		Others
T83601	(+)-Diasyringaresinol
	(+)-Diasyringaresinol, a lignan derived from Aquilaria agallocha seeds [1], exhibits potential pharmacological properties.
T78504	Lavandoside
	Lavandoside, an active compound isolated from the flowers of Lavandula spica [1], exhibits pharmacological properties.
T81195	Schiarisanrin E
	Schisandrin E (compound 5), a lignan extractible from Schisandra chinensis [1], exhibits pharmacological properties.
T82336	Ganoderic acid T
	Ganoderic acid T, a natural compound isolated from Ganoderma lucidum [1], exhibits various pharmacological properties.
T82318	Ginsenoside Rs1
	Ginsenoside Rs1, extracted from the root of Panax ginseng [1], is a chemical compound with potential pharmacological properties.
T38479	3-Hydroxypyridine
	3-Hydroxypyridine, extracted from Bamboo grass, is a structural analogue of vitamin B6. It exhibits diverse pharmacological properties, including antioxidant activity.
TN6584	Pallidol
	Pallidol is a potent and selective singlet oxygen quencher in aqueous systems, it may be used in singlet oxygen-mediated diseases as a pharmacological agent.
T81220	Salvileucantholide
	Salvileucantholide, a diterpenoid extracted from Salvia leucantha [1], exhibits noteworthy pharmacological properties.
T81055	Szechenyin A
	Szechenyin A, a constituent of the Tibetan medicinal plant Gentianae Szechenyii Spray, exhibits various pharmacological properties.
T81907	Lucenin 3
	Lucenin 3, a bioactive flavonoid [1], exhibits pharmacological properties beneficial to health.
TN1378	α-Viniferin	ALPHA-VINIFERIN	P450 , NO Synthase , Prostaglandin Receptor
	α-Viniferin known as 2-arylbenzofuran flavonoids, that are inhibitors of prostaglandin H2 synthetase. α-Viniferin has anti-Alzheimer's disease, anti-tuberculosis, anti-tumor, anti-inflammation, anti-diabetes and other ph...		P450 , NO Synthase , Prostaglandin Receptor
TN5498	6,7,4'-Trihydroxyflavanone		Others
			Others
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天然物製品

Nevadensin

T5722

Synonym: Pedunculin

Target: Anti-infection, Antibacterial

Ophiopojaponin C

T4104

Synonym: Ophiopogonin C

Chelidonine hydrochloride

Synonym: 5, 7-Dihydroxyflavone,NSC 407436,5,7-Dihydroxyflavone

Target: Estrogen Receptor/ERR, Antioxidant

Target: PPAR, Autophagy

Synonym: 8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,8-Hydroxypsoralene

Target: Reactive Oxygen Species, 5-HT Receptor, Endogenous Metabolite

Ammonium glycyrrhizinate

T2891

Synonym: Glycamil,Monoammonium glycyrrhizinate,Ammonium Glycyrrhizate,Monoammonium glycyrrhizinate hydrate,Glycyrram

Target: Antibacterial

Picroside II

T2817

Synonym: Vanilloyl catalpol,6-Vanilloylcatalpol

Target: Apoptosis, Others, Influenza Virus, NF-κB, Reactive Oxygen Species

Palmatine chloride

T2718

Synonym:

Target: Others, Indoleamine 2,3-Dioxygenase (IDO), Aurora Kinase

Naringin

T0595

Synonym: Naringoside

Target: Mitophagy, P450, Endogenous Metabolite, Autophagy

Sophocarpine monohydrate

T2746

Synonym: Sophocarpine

Target: Apoptosis, Influenza Virus, Akt, PI3K, AMPK, Autophagy

10-Deacetyl-7-xylosyl paclitaxel

T5749

Synonym: 10-Deacetyl-7-xylosyltaxol,10-Deacetyltaxol 7-Xyloside,7-Xylosyl-10-deacetyltaxol,10-Deacetylpaclitaxel 7-Xyloside

Target: Others, Microtubule Associated

Echinocystic acid

T2866

Synonym:

Target: Apoptosis, Antioxidant, Reactive Oxygen Species

Echinacoside

T1716

Synonym:

Target: Reactive Oxygen Species, Wnt/beta-catenin

Synonym: Kaempferol 3-D-glucoside,Kaempferol 3-O-glucoside,kaempferol-3-glucoside,3-Glucosylkaempferol,Astragaline,Kaempferol 3-β-D-glucopyranoside

Target: Apoptosis, NF-κB

Columbianadin

T3373

Synonym: Zosimin,2-Butenoic acid

Target: Apoptosis

Songorine

T5S1882

Synonym: Napellonine,Zongorine,Bullatine G

Target: Others, GABA Receptor

Target: Others, Antifungal

euphol

T5737

Synonym:

Target: Others, Lipase, Endogenous Metabolite

Curcumin

T1516

Synonym: Diferuloylmethane,Natural Yellow 3,Indian Saffron,Turmeric yellow

Target: Mitophagy, Epigenetic Reader Domain, Ferroptosis, Influenza Virus, Nrf2, Histone Acetyltransferase, HDAC, Autophagy

Alliin

T5764

Synonym: (S)-3-(Allylsulphinyl)-L-alanine

Target: NF-κB, PPAR

2,6,6-Trimethyl-2,4-cycloheptadien-1-one

T8250

Synonym:

Target: Others

Ophiogenin 3-O-α-L-rhamnopyranosyl-(1→2)-β-D-glucopyranoside

T3S1250

Synonym: Ophiogenin-3-O-alpha-L-rhaMnopyranosyl-(1->2)-beta-D-glucopyranoside

Target: Others

N-(3-Methoxybenzyl)Oleamide

TN1966

Synonym: N-Benzyloleamide,MAC 18:1

Target: Antioxidant

Pseudoginsenoside F11

T3920

Synonym: Ginsenoside A1

Target: Others, Endogenous Metabolite

Squalene

T4749

Synonym: Nikko Squalane EX,Super Squalene,AddaVax,all-trans-Squalene,trans-Squalene,Spinacene

Target: Reactive Oxygen Species, Endogenous Metabolite, Antifungal

Scoparone

T2729

Synonym: Escoparone,Scoparon,Aesculetin dimethyl ether,6,7-dimethoxycoumarin,6,7-Dimethylesculetin

Target: Others

L-Sophoridine

T3030

Synonym: Sophoridine,Matridin-15-one

Target: ERK, p38 MAPK, NF-κB, TLR, COX, HER, JNK, STAT

Saikosaponin A

T2768

Synonym:

Target: NF-κB, Antibacterial, Liver X Receptor

(+)-Diasyringaresinol

Synonym: ALPHA-VINIFERIN

Target: P450, NO Synthase, Prostaglandin Receptor

6,7,4'-Trihydroxyflavanone

TN5498

Synonym:

Target: Others

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Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-03407	NQO1 Protein, Human, Recombinant (His)	Human	E. coli
	NQO1 gene is a member of the NAD(P)H dehydrogenase (quinone) family and encodes a cytoplasmic 2-electron reductase. NQO1 forms homodimers and reduces quinones to hydroquinones. NQO1's enzymatic activity prevents the one-...
TMPY-04483	IRAK4 Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	Interleukin-1 receptor-associated kinase 4, also known as Renal carcinoma antigen NY-REN-64, IRAK-4, and IRAK4, is a member of the protein kinase superfamily, TKL Ser/Thr protein kinase family, and Pelle subfamily. IRAK4...
TMPK-00733	CD200 Protein, Mouse, Recombinant (aa 31-232, His)	Mouse	HEK293 Cells
	CD200 and its receptors are highly expressed in the lung, on epithelial cells and leukocytes, and emerging evidence links dysregulation of the CD200 pathway with asthma. Moreover, pharmacological modulation of CD200 rece...
TMPK-00476	CD200 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	CD200 and its receptors are highly expressed in the lung, on epithelial cells and leukocytes, and emerging evidence links dysregulation of the CD200 pathway with asthma. Moreover, pharmacological modulation of CD200 rece...
TMPJ-00660	IMPase2 Protein, Human, Recombinant (His)	Human	E. coli
	Inositol monophosphatase 2, also known as Inositol-1(or 4)-monophosphatase 2, Myo-inositol monophosphatase A2 and IMPA2, is an enzyme which belongs to the inositol monophosphatase family. IMPA2 catalyzes the dephosphoylr...
TMPY-03499	CARHSP1 Protein, Human, Recombinant (His)	Human	E. coli
	CARHSP1 is a biomarker for diabetic complications. Adenovirus-mediated CARHSP1 overexpression and siRNA-mediated knockdown experiments were performed to characterize the role of CARHSP1 in the regulation of gluconeogen...
TMPY-06821	THRB Protein, Human, Recombinant (His)	Human	E. coli
	Thyroid hormone receptor beta (THRB), also known as TRbeta and NR1A2, belongs to the nuclear hormone receptor family. Featuring an N-terminal transactivation domain, a central DNA-binding domain, and a hormone/ligand-bin...
TMPY-04554	JNK1 Protein, Human, Recombinant (GST)	Human	Baculovirus Insect Cells
	Mitogen-activated protein kinase 8 (MAPK8), also known as JNK1, is a member of the MAP kinase family. MAP kinases act as an integration point for multiple biochemical signals and are involved in a wide variety of cellula...

NQO1 Protein, Human, Recombinant (His)

TMPY-03407

Species: Human

Expression System: E. coli

IRAK4 Protein, Human, Recombinant (His)

TMPY-04483

Species: Human

Expression System: Baculovirus Insect Cells

CD200 Protein, Mouse, Recombinant (aa 31-232, His)

TMPK-00733

Species: Mouse

Expression System: HEK293 Cells

CD200 Protein, Cynomolgus, Recombinant (His)

TMPK-00476

Species: Cynomolgus

Expression System: HEK293 Cells

IMPase2 Protein, Human, Recombinant (His)

TMPJ-00660

Species: Human

Expression System: E. coli

CARHSP1 Protein, Human, Recombinant (His)

TMPY-03499

Species: Human

Expression System: E. coli

THRB Protein, Human, Recombinant (His)

TMPY-06821

Species: Human

Expression System: E. coli

JNK1 Protein, Human, Recombinant (GST)

TMPY-04554

Species: Human

Expression System: Baculovirus Insect Cells

カタログ番号	製品名
L9100	Phosphatase Inhibitor Library	79 compounds
	A collection of 79 phosphatase inhibitors with known activity;
L4150	Featured Novel Bioactive Compound Library	989 compounds
	It is well-selected from Bioactive compound library Plus (D7800), from which 1-15 compounds with the highest scores (activity value, pharmacological properties, structure-diversity, etc.) were chosen. This library consis...
L2700	Adrenergic Receptor-Targeted Compound Library	193 compounds
	A unique collection of 193 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification;
L6150	Covalent Natural Product Library	583 compounds
	Detialed biological information and pharmacological information of the products, providing theoretical direction and research basis for screening.
L3400	Clinical Compound Library	3404 compounds
	A unique collection of 3404 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
L5800	Drug Metabolite/Impurity Library	197 compounds
	A unique collection of 197 drug isomers/metabolites for high throughput screening (HTS) and high content screening (HCS);
L4710	Nonsteroidal Anti-Inflammatory Compound Library	530 compounds
	530 non-steroidal anti-inflammatory compounds for high-throughput and high-content screening.
L1600	Kinase Inhibitor Library	2720 compounds
	A unique collection of 2720 kinase inhibitors/regulators for high throughput screening and high content screening for drug discovery in kinase related diseases;
L6230	Miao medicine Compound Library	534 compounds
	A unique collection of 534 compounds featuring natural product molecules derived from Miao medicine that can be used for high-throughput and high-content screening.
L6000	Natural Product Library for HTS	4533 compounds
	A unique collection of 4533 pure natural products and their derivatives with known biological activity for drug discovery, pharmacological study, stem cell differentiation, fingerprint study and quality research, and can...
L6900	Rare Natural Product Library	693 compounds
	A unique collection of 693 rare natural products, which can be used for high throughput screening (HTS) and high content screening (HCS);
L6110	Alkaloid Natural Product Library	464 compounds
	A unique collection of 464 natural alkaloids can be used for high throughput and high content screening；
L7200	Calcium Channel Compound Library	140 compounds
	A unique collection of 140 calcium channel blockers and agonists for high throughput and high content screening;
L2193	Anti-Liver Cancer Compound Library	1787 compounds
	1787 species of compounds related to liver cancer that can be used in anti-liver cancer drug development and pharmacological studies.
L7400	Sodium Channel Blocker Library	118 compounds
	A unique collection of 118 sodium channel blockers and agonists for high throughput and high content screening;
L2610	Neurotransmitter Receptor Compound Library	1513 compounds
	A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
L6010	Natural Product Library	3840 compounds
	A unique collection of 3840 natural products for high throughput screening (HTS) and high content screening (HCS);
L6400	Marine Natural Product Library	144 compounds
	A unique collection of 144 marine natural products for high throughput screening (HTS) and high content screening (HCS);
L6730	Anti-virus Traditional Chinese Medicine Monomer Library	268 compounds
	A collection of 268 TCM monomers with anti-virus activity. An effective tool for drug development and pharmacological studies.
L9850	Orally Active Compound Library	2427 compounds
	A unique collection of 2427 of orally active compounds for high-throughput screening and high-content screening.
L6220	Traditional Mongolian Medicine Compound Library	950 compounds
	A collection of 950 natural product molecules originated from Mongolian medicine, which can be used for high-throughput and high-content screening.
L7100	Anti-Obesity Compound Library	2247 compounds
	A unique collection of 2247 anti-obesity compounds for high throughput and high content screening;
L6020	Selectable Natural Product Library	16627 compounds
	A unique collection of 16627 pure natural products with diverse structures and sources covering various plant, animal, and microbe species;
L6200	The Yao nationality medicine Library	221 compounds
	A collection of 221 natural product molecules originated from Yao medicine, which can be used for high-throughput and high-content screening.
L2196	Anti-Ovarian Cancer Compound Library	1867 compounds

L6750	PBCRBS Traditional Chinese Medicine Compound Library	580 compounds
	A unique collection of 580 compounds derived from traditional Chinese medicines (TCMs) for promoting blood circulation and removing blood stasis.
L6740	Anti-Colorectal Cancer Traditional Chinese Medicine Compound Library	382 compounds
	A collection of 382 TCM monomers with anti-colorectal activity. An effective tool for drug development and pharmacological studies.
L6800	Chinese Pharmacopoeia Natural Product Library	2051 compounds
	A unique collection of 2051 natural products included in Chinese Pharmacopoeia (CP), a powerful tool for drug development and pharmacological study;
L9410	Covalent Inhibitor Library	1920 compounds
	A unique collection of 1920 covalent Inhibitors and other molecules with common warheads like chloroacetyl，2-Chloropropionyl，Acryloyl，sulfonyl fluoride, alkyne，acrylamide, ketocarbonyl，disulfide bond, etc.