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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T77432 | Anifrolumab | MDX-1333,MEDI-546 | IFNAR |
Anifrolumab(MEDI-546) is a potent type I interferon (IFN) receptor antagonist, a human monoclonal antibody that targets IFN.Anifrolumab inhibits the activity of type I interferon and is used for the prevention and treatm... | |||
T9438 | 2,3,4-Trifluoro-5-Nitro-Benzoic Acid | Others | |
2,3,4-Trifluoro-5-Nitro-Benzoic Acid is a useful intermediate in organic synthesis. It has been used to study the effect of fluorine substitution on the reactivity of organic molecules. It has also been used to study the... | |||
T125462 | Gnetifolin K | GnetifolinK | |
Gnetifolin K (GnetifolinK) is a novel stilbene diglucoside from Gnetum parvifolium with potential neuroprotective activity for the study of DNA damage. | |||
T64167 | Ifebemtinib | IN-10018,BI-853520 | FAK |
Ifebemtinib (BI-853520) is an orally active and potent inhibitor of adhesion plaque kinase (FAK) (IC50=1 nM) with anti-tumour activity that inhibits globule formation and in situ tumour growth in malignant pleural mesoth... | |||
T9269 | N-Chloroacetyl-3,5-bis(trifluoromethyl)aniline | N-(3,5-Bis(trifluoromethyl)phenyl)-2-chloroacetamide | Others |
N-Chloroacetyl-3,5-bis(trifluoromethyl)aniline (KM1954) is an insecticide, it is most active against 1st stage Ae. aegypti larvae with LC50 values of 125μM. | |||
T77702 | 4-Chloro-3-(trifluoromethyl)phenyl isocyanate | Others | |
4-Chloro-3-(trifluoromethyl)phenyl isocyanate is a biochemical reagent that can be produced by a series of reactions between o-chlorobenzotrifluoride and acetic anhydride. | |||
T11200 | Endoxifen (E-isomer) | E-Endoxifen,Endoxifen E-isomer | Estrogen Receptor/ERR |
Endoxifen E-isomer (E-Endoxifen) is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects. | |||
T4350 | Palifosfamide | ZIO-201,Isophosphamide mustard,Isophosphoramide mustard | DNA Alkylator/Crosslinker , DNA Alkylation , Drug Metabolite |
Palifosfamide (Isophosphamide mustard) lysine (ZIO-201) is a stable form of palifosfamide. Palifosfamide lysine has broad activity in sarcoma lines in vitro. The IC50 ranges from 2.25 to 6.75 μM for most cell lines excep... | |||
T1543 | Naftifine hydrochloride | Naftifungin,Naftifine HCl,Naftin,Exoderil | Hedgehog/Smoothened , Antibiotic , Antifungal |
Naftifine Hydrochloride is the hydrochloride salt form of naftifine, an allylamine derivate with synthetic broad-spectrum antifungal activity. Although the exact mechanism through which naftifine hydrochloride exerts its... | |||
T77749 | Upifitamab | Others | |
Upifitamab is a naked antibody to upifitamab rilsodotin, which can be used to synthesize the antibody-coupled active molecule UPRI, which can be used to study cancer. | |||
T7586 | Trifarotene | CD5789 | Retinoid Receptor , Autophagy |
Trifarotene (CD5789) is a potent and selective RARγ agonist with 65-fold and 16-fold selectivitiy for the RARγ (EC50=7.7 nM) over RARα (EC50=500 nM) and RARβ (EC50=125 nM). | |||
T1428 | Trifluridine | NSC 529182,Trifluorothymidine,5-Trifluorothymidine,NSC 75520,Viroptic,Trifluridina | Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis , HSV |
Trifluridine (NSC-75520) is a fluorinated thymidine analog with potential antineoplastic activity. Trifluridine is incorporated into DNA and inhibits thymidylate synthase, resulting in inhibition of DNA synthesis, inhibi... | |||
T67849 | O-Desethyl Dapagliflozin | Empagliflozin-4 | SGLT |
O-Desethyl Dapagliflozin (Empagliflozin-4) is a SGLT2 inhibitor, IC50=33nM. | |||
T23372 | SMIFH2 | Others | |
SMIFH2 is formin homology 2 (FH2) domains inhibitor. | |||
T5819 | Rapastinel Trifluoroacetate | Thr-Pro-Pro-Thr-NH2 Trifluoroacetate,GLYX-13 Trifluoroacetate | NMDAR , iGluR |
Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties. | |||
TP1344 | Luciferase | Others | |
Luciferase is a flavin-dependent monooxygenase found in bioluminescent bacteria. Luciferase is an invaluable tool for identifying and characterizing functional variants, allowing investigations of gene expression, intrac... | |||
T7750 | N-[3,5-bis(trifluoroMethyl)phenyl]-N'-[(9R)-6'-Methoxycinchonan-9-yl]- Thiourea | Others | |
N-[3,5-bis(trifluoroMethyl)phenyl]-N'-[(9R)-6'-Methoxycinchonan-9-yl]- Thiourea is a cinchona alkaloid-derived bifunctional catalyst. | |||
T7384 | Ocifisertib(CFI-400945 free base) | PLK | |
CFI-400945 is an potent, selective and orally active inhibitor of polo-like kinase 4(PLK4; Ki value of 0.26 nM). | |||
T33600L | (Rac)-Naxifylline | (Rac)-Naxifylline((Rac)-166374-49-8) | Others |
(Rac)-Naxifylline may be used to study congestive heart failure. | |||
T29215 | Zifaxaban | TY 602,TY602,TY-602 | Factor Xa |
Zifaxaban (TY-602) is an orally active, competitive and selective inhibitor of factor Xa (FXa) with an IC50 of 11.1 nM for human FXa.Zifaxaban has a very high affinity, more than 10,000-fold higher than that of other ser... | |||
T6271 | Tipifarnib | R115777,Zarnestra,IND 58359 | Transferase |
Tipifarnib (IND 58359) is a nonpeptidomimetic quinolinone with potential antineoplastic activity. Tipifarnib binds to and inhibits the enzyme farnesyl protein transferase, an enzyme involved in protein processing (farnes... | |||
T64391 | Antiproliferative agent-15 | Others | |
Antiproliferative agent-15 is a reagent with anticancer activity. Antiproliferative agent-15 showed antiproliferative activity against human colon cancer (HCT116 and HCT15) and brain cancer (LN-229 and GBM-10). | |||
T38192 | Unifiram | Others | |
Unifiram is a nootropic agent.1It increases acetylcholine (ACh) release in the rat cerebral cortexin vivoand induces a long-lasting increase in the amplitude of field excitatory postsynaptic potentials (fEPSPs) in the ra... | |||
T1501 | Rifabutin | LM-427,Ansamycin | HSP , DNA/RNA Synthesis , Antibacterial , Antibiotic |
Rifabutin (LM-427) inhibits bacterial DNA-dependent RNA polymerase, thereby suppressing the initiation of RNA formation and leading to inhibition of RNA synthesis and transcription. Rifabutin is a semisynthetic ansamycin... | |||
T38655 | Trifludimoxazin | Others | |
Trifludimoxazin is an inhibitor of protoporphyrinogen oxidase and can be used as a herbicide. | |||
T50062 | 2,5-dichloro-4-(difluoromethoxy)-N,N-dimethylbenzene-1-sulfonamide | PDE | |
2,5-dichloro-4-(difluoromethoxy)-N,N-dimethylbenzene-1-sulfonamide is a PDE inhibitor. | |||
T4281 | Endoxifen | (E/Z)-N-desmethyl-4-hydroxy Tamoxifen,(E/Z)-Endoxifen | Estrogen Receptor/ERR , Aromatase , Estrogen/progestogen Receptor , Parasite , Drug Metabolite |
(E/Z)-Endoxifen ((E/Z)-Endoxifen) is an active metabolite of tamoxifen produced by the sequential action of cytochrome P450 (CYP) isoforms, including CYP2D6. It is a strong anti-estrogen, as it has an approximately 100-f... | |||
T5146 | Eptifibatide acetate (148031-34-9 free base) | Eptifibatide acetate | Others |
Eptifibatide acetate (148031-34-9 free base) (Eptifibatide acetate) , an antiplatelet drug of the glycoprotein IIb/IIIa inhibitor class, is a cyclic heptapeptide constructed from 6 amino acids and a mercaptopropionyl res... | |||
T1187 | Bifonazole | Bay H-4502 | P450 , Antibiotic , Antifungal |
Bifonazole (Bay H-4502) acts to destabilize the fungal cytochrome p450 51 enzyme (also known as Lanosterol 14-alpha-demethylase). It works by inhibiting the production of a substance called ergosterol, which is an essent... | |||
T67291 | 2′,2′-Difluorodeoxyuridine | dFdU,2',2'-Difluoro-2'-deoxyuridine | Drug Metabolite |
2′,2′-Difluorodeoxyuridine (dFdU) is the major metabolite of Gemcitabine.2′,2′-Difluorodeoxyuridine has anticancer and antitumor activity, and shows radiosensitization under hypoxic conditions, and can be used to study p... | |||
T1186L | Ifenprodil | RC 61-91,RC-61-91,RC61-91,RC 6191 | Adrenergic Receptor , NMDAR |
Ifenprodil (RC61-91) is an inhibitor of the NMDA receptor, specifically of GluN1 (glycine-binding NMDA receptor subunit 1) and GluN2B (glutamate-binding NMDA receptor subunit 2) subunits. Additionally, Ifenprodil inhibit... | |||
T4420 | 4-Hydroxytamoxifen | ICI 79280,(Z)-4-hydroxy Tamoxifen,trans-4-Hydroxytamoxifen | Estrogen Receptor/ERR , Estrogen/progestogen Receptor |
4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency. 4-Hydroxytamoxifen has antitumor activity and may be used in breast cancer rese... | |||
T0693 | Niflumic acid | Nifluril,Forenol,Landruma | Others , Phospholipase , Chloride channel , COX , Monocarboxylate transporter , UGT |
Niflumic acid (Nifluril) is a Ca2+-activated Cl- channel blocker and an analgesic and anti-inflammatory agent used in the therapy of rheumatoid arthritis. | |||
T60231 | N-[2-nitro-4-(trifluoromethyl)phenyl]piperazine | Others | |
N-[2-nitro-4-(trifluoromethyl)phenyl]piperazine is a biologically active compound belonging to the piperazine group. It is an important synthetic intermediate used in the preparation of a wide range of drugs, agrochemica... | |||
T2004 | Ciproxifan maleate | FUB 359 maleate,FUB 359 | Histamine Receptor |
Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes. | |||
T7217 | Bexagliflozin | THR-1442,EGT1442,EGT0001442 | SGLT |
Bexagliflozin (EGT1442) is a potent, selective sodium glucose co-transporter 2 (SGLT2) inhibitor with IC50 values of 5.6 μM and 2 nM for human SGLT1 and SGLT2, respectively | |||
T77138 | Ragifilimab | INCAGN-01876,INCAGN-1876,CM-701 | TNF |
Ragifilimab (INCAGN-1876) is an agonist monoclonal antibody targeting glucocorticoid-induced TNFR-associated protein (GITR). Ragifilimab can be used in the study of advanced or metastatic solid tumors. | |||
T7866 | Difenoconazole | Others , Antifungal | |
Difenoconazole is a broad-spectrum triazole fungicide that inhibits ergosterol biosynthesis via inhibition of the cytochrome P450-dependent 14α-demethylation of lanosterol, which results in disruption of the fungal cell ... | |||
T60026 | KIF18A-IN-2 | Microtubule Associated | |
KIF18A-IN-2 is an inhibitor of mitotic kinesin Kif18A with IC50 of 28 nM and can be used in studies about chromosomal instability-associated vulnerabilities. | |||
T4503 | Talniflumate | Somalgen | Chloride channel , COX , N-Acetylglucosaminyltransferase , Anion Exchanger |
Talniflumate (Somalgen) is a calcium-activated chloride channel (hCLCA1/mCLCA3) blocker that reduces mucin synthesis and releases in animal models and cell culture. It possesses anti-inflammatory actions via inhibition o... | |||
Fr12535 | 2-(Trifluoromethyl)benzimidazole | ||
Compound Fr12535 is a useful organic compound for research related to life sciences. The catalog number is Fr12535 and the CAS number is 312-73-2. | |||
T7110 | Thifluzamide | Antifungal | |
Thifluzamide is a fungicide widely used to control crop diseases. | |||
T1534 | Darifenacin hydrobromide | Darifenacin HBr,UK-88525 | AChR |
Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome. | |||
T8832 | Eledoisin trifluoroacetate (69-25-0 free base) | Eledoisin trifluoroacetate | Others |
Eledoisin trifluoroacetate (69-25-0 free base) is a peptide extracted from the posterior salivary glands of certain small octopi (Eledone spp., Mollusca), or obtained by synthesis. Its actions resemble those of SUBSTANCE... | |||
T0835 | Tamoxifen Citrate | Tamoxifen Z-isomer citrate,ICI 46474,ICI 46474 Citrate | Apoptosis , Estrogen Receptor/ERR , HSP , Estrogen/progestogen Receptor , Autophagy |
Tamoxifen is an antineoplastic nonsteroidal selective estrogen receptor modulator (SERM). | |||
T5000 | Diflucortolone valerate | Afusona,Diflucortolone 21-valerate | Others , Antibacterial , Antifungal |
Diflucortolone valerate (Diflucortolone 21-valerate) is a corticosteroid esterified with valeric acid. It helps to reduce itching, redness, and swelling. | |||
T3658 | Trifluridine/tipiracil hydrochloride mixture | Trifluridine-tipiracil hydrochloride mixture,TAS102,TAS-102,TAS 102 | Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis |
Trifluridine/tipiracil hydrochloride mixture (TAS-102) is a novel oral combination drug containing trifluridine (TFT) and Tipiracil hydrochloride (TTP) in a molar ratio of 2:1. | |||
T0225 | Pizotifen Malate | Pizotyline (malate),BC-105 (malate),BC-105 | 5-HT Receptor |
Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based on benzocycloheptane. | |||
T9341 | Bemnifosbuvir | AT-511 | Others , HCV Protease , SARS-CoV |
Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV. | |||
T19832 | Acriflavine Hydrochloride | Acriflavine HCl | HIF |
Acriflavine Hydrochloride (Acriflavine HCl) is a HIF-1α inhibitor. It acts by targeting HIF-1α-mediated pathways and decreasing the level of PGK1, VEGF, and HIF-1α in vitro and in vivo. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
TN2430 | Glucodigifucoside | ||
Glucodigifucoside, a cardiac glycoside that can be isolated from digitalis seeds, is specifically cytotoxic to human renal adenocarcinoma cells. | |||
T67685 | 4-Methylumbelliferyl-β-D-xylopyranoside | 4-Methylumbelliferyl-β-D-xyloside | |
4-Methylumbelliferyl-β-D-xylopyranoside (4-Methylumbelliferyl-β-D-xyloside) exhibits bursting steady-state kinetics in biological experiments, which supports the conclusion of rapid hydrolysis of the glycosidic bond of t... | |||
TN2283 | Tripterifordin | HIV Protease | |
Tripterifordin shows anti-HIV replication activity in H9 lymphocyte cells with an EC50 of 1 microgram/ml. | |||
T1186 | Ifenprodil Tartrate | Potassium Channel , NMDAR , iGluR | |
Ifenprodil is a selective NMDA receptor (glutamate) antagonist. | |||
T4587 | Mirificin | BCP10902,Puerarin Apioside | Tyrosinase |
Mirificin (BCP10902) is an active ingredient in Tongmai formula (TMF) which is a well-known Chinese medicinal preparation. Anti-oxidant. | |||
T2S1907 | Coniferaldehyde | Ferulaldehyde,Ferulyl aldehyde,4-HYDROXY-3-METHOXYCINNAMALDEHYDE,Coniferyl aldehyde | Apoptosis , Antioxidant |
Coniferaldehyde (Ferulaldehyde) is a member of the class of cinnamaldehydes that is cinnamaldehyde substituted by a hydroxy group at position 4 and a methoxy group at position 3. It has a role as an antifungal agent and ... | |||
T3768 | Epifriedelanol | Epifriedelinol | Others |
Epifriedelanol (Epifriedelinol) suppresses adriamycin-induced cellular senescence, replicative senescence in human fibroblasts (HDFs) and HUVECs. Because of Epifriedelanol can reduce cellular senescence in human primary ... | |||
T4S0145 | Corylifol A | Corylinin | hCE , STAT , UGT |
1. Corylifol A (Corylinin) displays cytotoxic activity against HepG2 and Hep3B hepatocellular carcinoma cell lines, with IC50 values of 4.6 and 13.5 ug/ml, respectively. 2. Corylifol A and Biochanin A can be the potentia... | |||
T8347 | Rifamycin S | Reactive Oxygen Species , ROS , Antibacterial , Antibiotic | |
Rifamycin S is a potent DNA-dependent RNA polymerase inhibitor,is a quinone and an antibiotic agnet against Gram-positive bacteria | |||
T1391 | 4-Methylumbelliferone | Hymecromone,4-MU | Others |
4-Methylumbelliferone (Hymecromone) is a coumarin derivative possessing properties as a spasmolytic, choleretic and light-protective agent. It is also used in ANALYTICAL CHEMISTRY TECHNIQUES for the determination of NITR... | |||
T2S2211 | Tenuifoliside C | Dehydrogenase | |
Tenuifoliside C, isolated from polygala tenuifolia willd, is a target lactate dehydrogenase inhibitor. It significantly inhibits chlorzoxazone 6-hydroxylation catalyzed by CYP2E1[1]. | |||
T6S1652 | Benzoylpaeoniflorin | COX | |
1. Benzoylpaeoniflorin is active against cyclooxygenase-1 and cyclooxygenase-2 enzymes. | |||
T8384 | Gatifloxacin hydrochloride | AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride) | Topoisomerase , Antibacterial , Antibiotic |
Gatifloxacin hydrochloride (AM-1155 hydrochloride) is an antibiotic of the fourth-generation fluoroquinolone family, which can inhibit the bacterial enzyme DNA rotase and topoisomerase IV. | |||
T11685 | Isolongifolene | (-)-Isolongifolene | Apoptosis , Others |
Isolongifolene ((-)-Isolongifolene), a tricyclic sesquiterpene isolated from Murraya koenigii, exhibits antioxidant, anti-inflammatory, anticancer, and neuroprotective properties. It mitigates Rotenone-induced oxidative ... | |||
T6981 | Nudifloric Acid | Nudifloric Acid | Others |
1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid (Nudifloric Acid) is from Cordyceps bassiana. Nudifloric Acid targets to block AP-1-mediated luciferase activity, implying it has an anti-inflammatory function. | |||
T3369 | Nuciferine | (-)-Nuciferine,VLT 049,Sanjoinine E | Dopamine Receptor , 5-HT Receptor |
Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera. It has a profile of action associated with dopamine receptor blockade. | |||
T3273 | Bifendate | Bifendatatum | HBV , Reverse Transcriptase |
Bifendate (Bifendatatum) is commonly used to treat the transaminase elevation that caused by viral hepatitis and drug-induced liver injury. | |||
TN1174 | Schinifoline | Apoptosis , cell cycle arrest | |
Schinifoline is a quinolone derivative extracted from Zanthoxylum schinifolium Sieb with cytotoxic activity that promotes radiosensitization of cancer cells, affects the cell cycle and apoptosis. | |||
T3012 | Mangiferin | Alpizarin,Chinomin,Hedysarid | Apoptosis , Others , NF-κB , Nrf2 |
Mangiferin (Hedysarid) is used for antidiabetes. Extracted from Mangifera indica L. | |||
TN1012L | Febrifugine dihydrochloride | ISF-2123,Propyldazine hydrochloride,Atensil,(+)-Febrifugine dihydrochloride,Pildralazine dihydrochloride | Parasite |
Febrifugine dihydrochloride (Propyldazine hydrochloride) is a biochemical with therapeutic activity regarding malaria, cancer, fibrosis and inflammatory diseases. | |||
TL0009 | Coniferin | Coniferoside,Abietin | Others , Antifungal |
Coniferin (Abietin) has ATP-dependent transport activity and has anti-oxidation effects. Coniferin has preferred substrates for the coniferin beta-glucosidase, the chromogenic coniferin analogue show the exclusive presen... | |||
TN3849 | Dihydrodehydrodiconiferyl alcohol | TNF | |
Dihydrodehydrodiconiferyl alcohol is the methanolic extract of Liriodendron tulipifera[1]. | |||
T4902 | Isotrifoliin | Isoquercetin,Isoquercitroside | Reactive Oxygen Species |
T3313 | D-Luciferin | Firefly luciferin,D-(-)-Luciferin | Others |
D-Luciferin (D-(-)-Luciferin) is a popular bioluminescent substrate of luciferase in the presence of ATP, used in luciferase-based bioluminescence imaging and cell-based high-throughput screening applications. | |||
T3805 | Prim-O-glucosylcimifugin | Cimifugin beta-D-glucopyranoside,Cimifugin 7-glucoside | TNF , COX , JAK , NO Synthase |
Prim-O-glucosylcimifugin (Cimifugin 7-glucoside) can inhibit the proliferation of SMC(smooth muscle cell) stimulated by TNF-alpha, increase the proportion of G0/G1 phase. | |||
T6430 | Calcifediol | U 32070E,25-hydroxy Vitamin D3,RO 8-8892 | Endogenous Metabolite |
Calcifediol (U 32070E)(Ki of 3.9 μM), a major circulating metabolite of vitamin D3, works as a competitive inhibitor. It (ED50=2 nM)also inhibits PTH secretion and mRNA. | |||
TN7097 | Tetrahydrodehydrodiconiferyl alcohol | Others | |
Tetrahydrodehydrodiconiferyl alcohol is a natural product. | |||
T6S1653 | Albiflorin | Alibiflorin | Reactive Oxygen Species |
1. Albiflorin (Alibiflorin) has anticonvulsant effect for pain relief. 2. Albiflorin and paeoniflorin has neuroprotective action against Glu toxicity. 3. Albiflorin and paeoniflorin significantly ameliorated Glu-induced ... | |||
TN3694 | Coniferaldehyde | NOS , COX , Nrf2 , PKC , Autophagy | |
Coniferaldehyde can significantly inhibit the growth of viability of strains of Oenococcus oeni. Coniferaldehyde exerts anti-inflammatory properties by inducing heme oxygenase-1(HO-1). | |||
T3873 | Griffonilide | Others | |
Griffonilide is an extract from the Semiaquilegia adoxoides root, a traditional anticancer herb. | |||
T3804 | Neomangiferin | Mangiferin 7-glucoside | Phosphatase |
Neomangiferin (Mangiferin 7-glucoside) has beneficial effects on high fat diet-induced nonalcoholic fatty liver disease in rats. Neomangiferin and mangiferin inhibit tartrate-resistant acid phosphatase, a biochemical mar... | |||
T40080 | (±)-Taxifolin | (±)-Dihydroquercetin | Antioxidant , Tyrosinase |
(±)-Taxifolin ((±)-Dihydroquercetin) is the racemate of Taxifolin, a flavonoid commonly found in onion, silymarin, French maritime pine bark, and Douglas fir bark, with anti-tyrosinase and anti-fibrotic activity.Taxifoli... | |||
T1549 | Raloxifene hydrochloride | LY156758 hydrochloride,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl | Estrogen Receptor/ERR , Others , MAO , Estrogen/progestogen Receptor , Autophagy |
Raloxifene hydrochloride (LY156758 hydrochloride) is a second generation selective estrogen receptor modulator (SERM) used to prevent osteoporosis in postmenopausal women. It has estrogen agonist effects on bone and chol... | |||
TN1091 | Dehydronuciferine | AChE | |
Dehydronuciferine is isolated from the leaves of Nelumbo nucifera Gaertn. Dehydronuciferine shows inhibitory of acetylcholinesterase with the IC50 of 25 ug/mL. | |||
TN2260 | Taxifolin 7-O-rhamnoside | Taxifolin 7-O-α-L-rhamnoside | Others |
Taxifolin 7-O-rhamnoside (Taxifolin 7-O-α-L-rhamnoside) is a natural product from Hypericum japonicum. | |||
TN1139L | Tetradehydrothalictrifoline | Others | |
Tetradehydrothalictrifoline is a nature product. | |||
TN1092 | O-Nornuciferine | Potassium Channel , HER | |
O-Nornuciferine reveals distinct in vitro hERG blockages measured in HEK293 cells with the IC50 value of 2.89 uM. | |||
T3383 | Cimifugin | Cimitin | Others |
Cimifugin (Cimitin) inhibits NO production induced by lipopolysaccharide in macrophage cell line RAW 264.7 and for 1, 1-diphenyl-2-picrylhydrazyl free-radical scavenging activity in cell-free bioassay system. | |||
TN7040 | Taxifolin 7-O-β-D-glucoside | Taxifolin 7-Glucoside | Others |
Taxifolin 7-O-β-D-glucoside is a flavonoid mainly found in endosperm and involved in defense against pathogens and UV damage. | |||
T6S1294 | Nicotiflorin | Nictoflorin,Kaempferol-3-O-Rutinoside,Nicotifloroside | Others |
1. Nicotiflorin (Kaempferol-3-O-Rutinoside) has potential therapeutic effects on cerebral ischemic illness. 2. Nicotiflorin has protective effects on reducing memory dysfunction, energy metabolism failure and oxidative s... | |||
TN2156 | Rhombifoline | Antioxidant | |
Rhombifoline is a family of alkaloids isolated from the leaf stems of Anagyrus foetida and Genista tenera. | |||
T4S0969 | Obtusifolin | Antioxidant , NF-κB | |
1. Obtusifolin has antioxidant properties and improves chemically induced diabetes and its complications by modulation of oxidative stress. 2. Obtusifolin suppresses phthalate esters-mediated bone resorption, thus may be... | |||
T3822 | Bellidifolin | Bellidifoline,Bellidifolium | Others , HIV Protease |
Bellidifolin (Bellidifoline) has anti-oxidation, hepatoprotective, anti-inflammatory and antitumor actions, it may contribute to the protective effects associated with nerve injury initiated by hypoxia by mechanisms rela... | |||
T1693 | Umbelliferone | Skimmetine,Hydrangin,Hydrangine,7-Hydroxycoumarin,NSC 19790 | Apoptosis , Antioxidant , Endogenous Metabolite |
Umbelliferone (7-Hydroxycoumarin) is found in anise. Umbelliferone occurs widely in plants including Angelica species Phytoalexin of infected sweet potat. It has been reported to have antioxidant properties. | |||
TN7218 | Diformylphloroglucinol | 2,4,6-Trihydroxyisophthalaldehyde | Antioxidant |
Diformylphloroglucinol (2,4,6-Trihydroxyisophthalaldehyde) is an acyl resorcinol isolated from the leaves of the Eucalyptus nigra tree and is a raw material for the synthesis of resorcinol compounds with antioxidant and ... | |||
TN1736 | Hibifolin | Adenosine deaminase | |
Hibifolin is a flavonol glycoside natural product,is a potential inhibitor of adenosine deaminase (Ki of 49.92 μM). Hibifolin protects neurons against beta-amyloid-induced neurotoxicity. | |||
TN1067 | Galloylpaeoniflorin | 6'-O-Galloyl paeoniflorin | NF-κB , Androgen Receptor , ROS |
Galloylpaeoniflorin (6'-O-Galloyl paeoniflorin) may be developed as a cytoprotector against ROS-mediated oxidative stress. Galloylpaeoniflorin is also an inhibtior of NF-κB and DNA cleavage. | |||
TN7027 | Benzoylalbiflorin | Paeonivayin | Others |
Benzoylalbiflorin (Paeonivayin) is a monoterpenoid isolated from Radix Paeoniae Alba. | |||
T5S2207 | 7-O-Methylmangiferin | Others | |
7-O-MethylMangiferin is an xanthone isolated from the rhizomes of Iris nigricans. | |||
TQ0296L | N-Nornuciferine hydrochloride(4846-19-9 free base) | N-Nornuciferine hydrochloride | P450 |
N-Nornuciferine hydrochloride(4846-19-9 free base) (N-Nornuciferine hydrochloride) is an aporphine alkaloid in lotus leaf, significantly inhibits CYP2D6 (IC50: 3.76 μM, Ki: 2.34 μM). | |||
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カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPY-03221 | Intrinsic Factor Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Gastric intrinsic factor, also known as GIF, belongs to the of the cobalamin transport protein family. It is a glycoprotein produced by the parietal cells of the stomach. Gastric intrinsic factor plays a key role in the ... | |||
TMPH-03273 | Complement factor I Protein, Rat, Recombinant (His & Myc) | Rat | Baculovirus Insect Cells |
Complement factor I Protein, Rat, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 69.2 kDa and the accession number is Q9WUW3. | |||
TMPK-01023 | Complement factor I Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Complement factor I (CFI) is a serine protease which plays a key role in the modulation of complement system and the induced-fit factor responsible for controlling the complement-mediated processes. Complement factor I P... | |||
TMPK-00776 | Complement factor I Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Complement factor I (CFI) is a serine protease which plays a key role in the modulation of complement system and the induced-fit factor responsible for controlling the complement-mediated processes. Complement factor I P... | |||
TMPY-02566 | Interferon alpha 4/IFNA4 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
Interferon alpha 4/IFNA4 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 20.7 kDa and the accession number is P05014. | |||
TMPY-00991 | LIFR Protein, Human, Recombinant (His) | Human | HEK293 Cells |
LIFR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 91 kDa and the accession number is P42702-1. | |||
TMPY-04799 | IFNAR2 Protein, Human, Recombinant (His), Biotinylated | Human | HEK293 Cells |
IFNAR2 Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.2 kDa and the accession number is P48551-1. | |||
TMPY-03467 | IFN-beta Protein, Mouse, Recombinant | Mouse | HEK293 Cells |
IFN-beta Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 20.3 kDa and the accession number is P01575. | |||
TMPY-06983 | IFN gamma Protein, Human, Recombinant (E. coli) | Human | E. coli |
IFN gamma, also known as IFNG, is a secreted protein that belongs to the type II interferon family. IFN gamma is produced predominantly by natural killer and natural killer T cells as part of the innate immune response, ... | |||
TMPY-01151 | IFNGR1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
IFNGR1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.3 kDa and the accession number is A0A0S2Z3Y2. | |||
TMPY-01714 | IFN gamma Protein, Human, Recombinant | Human | CHO Cells |
IFN gamma Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 16.7 kDa and the accession number is A0A7R8GUN6. | |||
TMPY-00265 | Interferon alpha 2/IFNA2 Protein, Human, Recombinant | Human | P. pastoris (Yeast) |
Interferon alpha 2/IFNA2 Protein, Human, Recombinant is expressed in yeast. The predicted molecular weight is 19.3 kDa and the accession number is P01563.1. | |||
TMPY-02647 | IFNAR1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
IFNAR1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 48.6 kDa and the accession number is P17181-1. | |||
TMPY-05493 | LIFR Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
LIFR Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 116.1 kDa and the accession number is P42702-1. | |||
TMPY-01131 | Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA1 Protein(His) | H1N1 | HEK293 Cells |
Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA1 Protein(His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is C3W5S1. | |||
TMPJ-00746 | IFN-alpha 2b/IFNA2 Protein, Human, Recombinant | Human | E. coli |
At least 23 different variants of IFN-α are known. The individual proteins have molecular masses between 19-26 kDa and consist of proteins with lengths of 156-166 and 172 amino acids. All IFN-α subtypes possess a common ... | |||
TMPY-00956 | Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA Protein ( (Native, HA1+HA2, uncleaved),His) | H1N1 | HEK293 Cells |
Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA Protein ( (Native, HA1+HA2, uncleaved),His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number ... | |||
TMPY-00182 | Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA0 Protein | H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA0 Protein is expressed in Baculovirus insect cells. The predicted molecular weight is 61.5 kDa and the accession number is C3W5S1. | |||
TMPY-03532 | LIF Protein, Human, Recombinant (His) | Human | HEK293 Cells |
LIF Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 21.2 kDa and the accession number is P15018. | |||
TMPY-02355 | IFNGR1 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
IFNGR1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.4 kDa and the accession number is P15261. | |||
TMPY-00642 | Influenza A H1N1 (A/California/07/2009) Hemagglutinin/HA Protein (His) | H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/California/07/2009) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59 kDa and the accession number is C3W5X2. | |||
TMPY-02876 | Influenza A H1N1 (A/California/07/2009) Nucleoprotein/NP Protein (His) | H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/California/07/2009) Nucleoprotein/NP Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.4 kDa and the accession number is C6KQ05. | |||
TMPY-00638 | Interferon alpha B/IFNA8 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Interferon alpha B/IFNA8 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 20.9 kDa and the accession number is A0A7R8C381. | |||
TMPY-02515 | Interferon alpha 7/IFNA7 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Interferon alpha 7/IFNA7 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 48 kDa and the accession number is P01567. | |||
TMPY-04578 | Interferon alpha 1/IFNA1 Protein, Human, Recombinant (His) | Human | P. pastoris (Yeast) |
Interferon alpha 1/IFNA1 Protein, Human, Recombinant (His) is expressed in yeast with His tag. The predicted molecular weight is 20.8 kDa and the accession number is L0N195. | |||
TMPY-04588 | Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA-specific B cell probe (His) | H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA-specific B cell probe (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.8 kDa and the accession number is C3W5S1. | |||
TMPY-00007 | Interferon alpha 2/IFNA2 Protein, Mouse, Recombinant | Mouse | P. pastoris (Yeast) |
Interferon alpha 2/IFNA2 Protein, Mouse, Recombinant is expressed in yeast. The predicted molecular weight is 19.4 kDa and the accession number is B1AYH7. | |||
TMPY-03072 | IFN-omega Protein, Human, Recombinant (His) | Human | HEK293 Cells |
IFN-omega Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 21.6 kDa and the accession number is P05000. | |||
TMPY-03356 | IFN gamma Protein, Mouse, Recombinant | Mouse | HEK293 Cells |
IFN gamma Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 15.5 kDa and the accession number is A0A7R8C347. | |||
TMPH-03617 | Miraculin Protein, Synsepalum dulcificum, Recombinant (His) | Synsepalum dulcificum | P. pastoris (Yeast) |
Miraculin has the property of modifying a sour taste into a sweet taste. This alteration of taste perception persists for many minutes. Miraculin Protein, Synsepalum dulcificum, Recombinant (His) is expressed in yeast wi... | |||
TMPY-06407 | Interferon alpha 2/IFNA2 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Interferon alpha 2/IFNA2 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 46.29 kDa and the accession number is P01563-1. | |||
TMPY-02827 | IFN gamma Protein, Rat, Recombinant (hFc) | Rat | HEK293 Cells |
IFN gamma Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.5 kDa and the accession number is P01581. | |||
TMPY-01441 | Influenza A H1N1 (A/California/04/2009) Neuraminidase/NA | H1N1 | HEK293 Cells |
Influenza A H1N1 (A/California/04/2009) Neuraminidase/NA is expressed in HEK293 mammalian cells. The predicted molecular weight is 47.8 kDa and the accession number is C3W5S3. | |||
TMPY-03145 | IFN-beta Protein, Human, Recombinant | Human | CHO Cells |
IFN-beta Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 20 kDa and the accession number is P01574. | |||
TMPY-02344 | Influenza A H1N1 (A/California/04/2009) Neuraminidase/NA (His) | H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/California/04/2009) Neuraminidase/NA (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 50 kDa and the accession number is C3W5S3. | |||
TMPY-04278 | LIF Protein, Mouse, Recombinant | Mouse | HEK293 Cells |
LIF Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 19.9 kDa and the accession number is P09056. | |||
TMPY-00831 | IFN-beta Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
IFN-beta Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 46.7 kDa and the accession number is A0A7R8GV38. | |||
TMPY-04104 | LIF Protein, Human, Recombinant | Human | HEK293 Cells |
LIF Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 19.7 kDa and the accession number is P15018-1. | |||
TMPK-00047 | IFN gamma Protein, Human, Recombinant (His & Avi) | Human | HEK293 Cells |
Interferon-gamma (IFN gamma) is a cytokine that plays physiologically important roles in promoting innate and adaptive immune responses. The absence of IFN gamma production or cellular responsiveness in humans and experi... | |||
TMPJ-00745 | IFN-alpha 2a/IFNA2 Protein, Human, Recombinant | Human | E. coli |
At least 23 different variants of IFN-α are known. The individual proteins have molecular masses between 19-26 kDa and consist of proteins with lengths of 156-166 and 172 amino acids. All IFN-α subtypes possess a common ... | |||
TMPY-03851 | BPIFB1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
BPIFB1, also known as LPLUNC1, belongs to the BPI/LBP/Plunc superfamily, plunc family. BPIFB1 may be involved in the innate immune response to bacterial exposure in the mouth, nasal cavities, and lungs. BPIFB1 is express... | |||
TMPY-03027 | Interferon alpha 4/IFNA4 Protein, Rat, Recombinant (hFc) | Rat | HEK293 Cells |
Interferon alpha 4/IFNA4 Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 47.5 kDa and the accession number is D3ZFH0. | |||
TMPY-03620 | Interferon alpha B/IFNA8 Protein, Cynomolgus, Recombinant (mFc) | Cynomolgus | HEK293 Cells |
Interferon alpha B/IFNA8 Protein, Cynomolgus, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 46 kDa and the accession number is G7PS89. | |||
TMPY-02634 | IFNAR1 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
IFNAR1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 74 kDa and the accession number is P17181-1. | |||
TMPY-06952 | LIF Protein, Cynomolgus, Rhesus, Recombinant (His & Avi), Biotinylated | Cynomolgus,Rhesus | HEK293 Cells |
LIF Protein, Cynomolgus, Rhesus, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 22.96 kDa and the accession number is A0A2K5UCA6. | |||
TMPH-03705 | NfuA Protein, Vibrio vulnificus, Recombinant | Vibrio vulnificus | E. coli |
Involved in iron-sulfur cluster biogenesis. Binds a 4Fe-4S cluster, can transfer this cluster to apoproteins, and thereby intervenes in the maturation of Fe/S proteins. Could also act as a scaffold/chaperone for damaged ... | |||
TMPY-01642 | IFNAR2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
IFNAR2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.2 kDa and the accession number is P48551-1. | |||
TMPY-03375 | IFN-alpha 13/IFNA13 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
IFN-alpha 13/IFNA13 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 20.8 kDa and the accession number is G7NFW4. | |||
TMPY-05527 | Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA Protein (His), Biotinylated | H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/California/04/2009) Hemagglutinin/HA Protein (His), Biotinylated is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59 kDa and the accession number is C3W5S1. | |||
TMPY-03319 | Interferon alpha 2/IFNA2 Protein, Rhesus, Recombinant (mFc) | Rhesus | HEK293 Cells |
Interferon alpha 2/IFNA2 Protein, Rhesus, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 45.9 kDa and the accession number is B6CK11. | |||
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カタログ番号 | 製品名 | ||
---|---|---|---|
L3500 | Histone Modification Compound Library | 469 compounds | |
A unique collection of 469 histone modification related compounds for high throughput screening (HTS) and high content screening (HCS); | |||
L2630 | Neuronal Differentiation Compound Library | 672 compounds | |
L8000 | Stem Cell Differentiation Compound Library | 1197 compounds | |
A unique collection of 1197 stem cell differentiation signaling targeted compounds for high throughput and high content screening; | |||
L8300 | Chromatin Modification Compound Library | 250 compounds | |
A unique collection of 250 compounds targeting chromatin remodeling pathway for high throughput screening (HTS) and high content screening (HCS); | |||
L8500 | HIF-1 Signaling Pathway Compound Library | 1336 compounds | |
A unique collection of 1336 HIF-1 related small chemicals can be used for drug discovery in ischemic disease and cancer and related mechanism studies; | |||
L2140 | Cancer Cell Differentiation Compound Library | 406 compounds | |
A unique collection of 406 cancer cell differentiation inducing compounds for high throughput and high content screening; | |||
L1900 | Anti-Diabetic Compound Library | 683 compounds | |
A unique collection of 683 diabetes related compounds; | |||
L9810 | Anti-Fibrosis Compound Library | 1180 compounds | |
A unique collection of 1180 potential anti-fibrosis compounds, can be used in HTS and HCS; | |||
L8710 | Cuproptosis Compound Library | 400 compounds | |
TargetMol’s Cuproptosis Compound Library is a collection of 400 compounds related to copper-dependent death that can be used to study its mechanism and related diseases. | |||
L8400 | Hematonosis Compound Library | 514 compounds | |
A unique collection of 514 compounds related to hematologic diseases for high throughput screening (HTS) and high content screening (HCS); | |||
L1310 | Cytoskeletal Signaling Pathway Compound Library | 759 compounds | |
A unique collection of 759 cytoskeleton-related compounds, can be used for HTS and HCS; |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
TMIH-0494 | Rifampicin-d3 | ||
Rifampicin-d3 is a deuterated compound of Rifampicin. Rifampicin has a CAS number of 13292-46-1. Rifampicin is an antibacterial drug of the class of rifamycin. | |||
T12329 | Ospemifene D4 | FC-1271a D4 | Estrogen/progestogen Receptor |
Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator of estrogen receptor. | |||
TMIH-0190 | Difamilast-d5 | ||
Difamilast-d5 is a deuterated compound of Difamilast. Difamilast has a CAS number of 937782-05-3. Difamilast is a selective inhibitor of phosphodiesterase-4 (PDE4) with particularly efficient inhibition of subtype B (IC5... | |||
T71300 | Pentoxifylline-d6 | ||
Pentoxifylline-d6 is intended for use as an internal standard for the quantification of pentoxifylline by GC- or LC-MS. Pentoxifylline is a hemorrheologic agent. It increases the deformability of washed isolated human er... | |||
TMIH-0086 | Amifampridine-d3 2HCl | ||
Amifampridine-d3 2HCl is a deuterated compound of Amifampridine 2HCl. Amifampridine 2HCl has a CAS number of 54-96-6. Amifampridine is predominantly in the treatment of a number of rare muscle diseases. Amifampridine wor... | |||
TMIH-0041 | 3,4-Difluoro-4'-(cis-4-propylcyclohexyl)biphenyl-d4 | 3,4-difluoro-4'-((1r,4s)-4-propylcyclohexyl)-1,1'-biphenyl-2',3',5',6'-d4 | |
3,4-Difluoro-4'-(cis-4-propylcyclohexyl)biphenyl-d4 is a deuterated compound of 3,4-Difluoro-4'-(cis-4-propylcyclohexyl)biphenyl. | |||
TMIH-0390 | Nifekalant-d4 | ||
Nifekalant-d4 is a deuterated compound of Nifekalant. Nifekalant has a CAS number of 130636-43-0. | |||
T10661 | Calcifediol-D6 | Others | |
Calcifediol-D6 is the deuterated form of Calcifediol, which is a prehormone that is produced in the liver by hydroxylation of vitamin D3 by the enzyme cholecalciferol 25-hydroxylase. | |||
T10669 | Canagliflozin-d4 | Canagliflozin D4 | Others |
Canagliflozin D4 is a deuterium-labeled Canagliflozin. Canagliflozin is an SGLT2 inhibitor. | |||
T71286 | Guaifenesin-d3 | ||
Guaifenesin-d3 is intended for use as an internal standard for the quantification of guaifenesin by GC- or LC-MS. Guaifenesin is an expectorant. It inhibits production of mucin 5AC (MUC5AC), reduces mucus viscosity and e... | |||
TMIH-0013 | (S)-Empagliflozin-d4 | ||
(S)-Empagliflozin-d4 is a deuterated compound of (S)-Empagliflozin. (S)-Empagliflozin has a CAS number of 864070-44-0. Empagliflozin is a Sodium-Glucose Cotransporter 2 Inhibitor. The mechanism of action of empagliflozin... | |||
T64761 | 5-(Methyl-d3)-dibenzothiophenium, 1,1,1-trifluoromethanesulfonate | ||
5-(Methyl-d3)-dibenzothiophenium, 1,1,1-trifluoromethanesulfonate is a useful organic compound for research related to life sciences and the catalog number is T64761. | |||
TMIH-0495 | Rifampicin-d4 | ||
Rifampicin-d4 is a deuterated compound of Rifampicin. | |||
T12618L | Quetiapine-d4 hemifumarate | Others | |
Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic. | |||
TMIH-0496 | Rifampicin-d8 | ||
Rifampicin-d8 is a deuterated compound of Rifampicin. Rifampicin has a CAS number of 13292-46-1. Rifampicin is an antibacterial drug of the class of rifamycin. | |||
TMID-0025 | Quetiapine-d8 Hemifumarate | ||
Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar... | |||
T11089 | Doxercalciferol-D3 | Others | |
Doxercalciferol-d3 is the deuterated form of Doxercalciferol and ACTS as vitamin D receptor activator (VDRA), which is a vitamin D2 analogue. | |||
T19187 | Aliskiren D6 hemifumarate | CGP 60536 D6 hemifumarate,SPP 100 D6 hemifumarate,CGP60536B D6 hemifumarate | RAAS |
Aliskiren (CGP 60536) D6 hemifumarate is a deuterium-labeled Aliskiren hemifumarate. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM). | |||
T12222 | Nifedipine-d6 | Nifedipine D6,BAY-a-1040 D6 | Others |
Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel. | |||
T12973 | Solifenacin D5 hydrochloride | Others | |
Solifenacin D5 hydrochloride is a deuterium labeled Solifenacin hydrochloride. Solifenacin hydrochloride is an antagonist of muscarinic receptor(pKis of 7.6, 6.9 and 8.0 for M1, M2 and M3 receptors, respectively). | |||
T38638 | 4-Trifluoromethylsalicylic acid-13C6 | 4-Trifluoromethylsalicylic acid-13C6,Desacetyl triflusal-13C6 | |
4-Trifluoromethylsalicylic acid-13C6 is 13C-labeled 4-Trifluoromethylsalicylic acid, mainly used as a quantitative tracer in drug development. 4-Trifluoromethylsalicylic acid is also a platelet aggregation inhibitor. | |||
T13076 | Tamoxifen-d5 | ICI 47699-d5,(Z)-Tamoxifen-d5,trans-Tamoxifen-d5 | HSP |
Tamoxifen-d5 is a deuterium labeled Tamoxifen. Tamoxifen is a selective modulator of estrogen receptor (SERM). Tamoxifen is a potent activator of Hsp90 and enhances the Hsp90 molecular chaperone ATPase activity. | |||
T71293 | Nifuroxazide-d4 | ||
Nifuroxazide-d4 is intended for use as an internal standard for the quantification of nifuroxazide by GC- or LC-MS. Nifuroxazide is a nitrofuran antibiotic. It is active against strains of the enteropathogenic bacteria C... | |||
TMIH-0042 | 3,4-Difluoro-4'-(trans-4-propylcyclohexyl)biphenyl-d4 | 3,4-difluoro-4'-((1s,4r)-4-propylcyclohexyl)-1,1'-biphenyl-2',3',5',6'-d4 | |
3,4-Difluoro-4'-(trans-4-propylcyclohexyl)biphenyl-d4 is a deuterated compound of 3,4-Difluoro-4'-(trans-4-propylcyclohexyl)biphenyl. 3,4-Difluoro-4'-(trans-4-propylcyclohexyl)biphenyl has a CAS number of 85312-59-0. | |||
T10958 | Dapagliflozin-d5 | BMS-512148 D5 | Others |
Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor. | |||
T11694 | Ivabradine-d6 hydrochloride | Ivabradine D6 hydrochloride | Others |
Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D6 hydrochloride is the deuterium labeled Ivabradine hydrochloride. | |||
T11692 | Ivabradine-d3 hydrochloride | Ivabradine D3 Hydrochloride | Others |
Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D3 Hydrochloride is the deuterium labeled Ivabradine hydrochloride. |