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160

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TargetMolキット

カタログ番号	製品名	別名	ターゲット
T5637	Triflumuron		Others
	Triflumuron is an insecticide belonging to the group of so-called insect growth regulators. It inhibits the synthesis of chitin by the insect larvae, causing the die.		Others
T8794	4-MMPB	15-Lipoxygenase Inhibitor 1	Apoptosis , Others , Lipoxygenase
	15-Lipoxygenase Inhibitor 1 is a selective inhibitor of 15-lipoxygenase, with an IC50 of 18 μM. 4-MMPB (15-Lipoxygenase Inhibitor 1) has IC50s of 19.5 μM and 19.1 μM for soybean 15-lipoxygenase (SLO) and human 15-lipoxyg...		Apoptosis , Others , Lipoxygenase
T14496	BAMB-4	ITPKA-IN-C14	Others
	BAMB-4 (ITPKA-IN-C14) is a highly membrane-permeable inhibitor of inositol-1,4,5-trisphosphate-3-kinase A (ITPKA). It acts by suppressing the metastasis-promoting effect of ITPKA in lung tumor cells(with IC50 of 37 μM in...		Others
T22733	DL-AP5		NMDAR
	DL-AP5 is the racemic form of a selective N-methyl-D-aspartate (NMDA) receptor antagonist with anticonvulsant effects.		NMDAR
T60080	TMPH	2,2,6,6-Tetramethylpiperidin-4-yl heptanoate	AChR
	TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.		AChR
T2691	Oritavancin diphosphate	LY333328 diphosphate	Others , Antibacterial , Antibiotic
	Oritavancin diphosphate (LY333328 diphosphate) is a novel semisynthetic glycopeptide antibiotic which is being developed for the treatment of serious Gram-positive bacterial infections.		Others , Antibacterial , Antibiotic
T2051	SKLB4771	FLT3-IN-1,FLT3-IN-1	FLT
	SKLB4771 (FLT3-IN-1) is a novel potent and selective Flt3 inhibitor.		FLT
T7476	AS057278	3-Methylpyrazole-5-carboxylic acid	Others
	AS057278 (3-Methylpyrazole-5-carboxylic acid) is an D-amino acid oxidase (DAAO) inhibitor.		Others
T0171	Norethynodrel	Lynestrol	Estrogen/progestogen Receptor
	Norethynodrel (Lynestrol) is a synthetic progestational hormone with actions and uses similar to those of PROGESTERONE. It has been used in the treatment of functional uterine bleeding and endometriosis. As a contracepti...		Estrogen/progestogen Receptor
T23284	Ryuvidine		Histone Demethylase , Histone Methyltransferase , CDK
	Ryuvidine is a dual inhibitor of KDM5A and SETD8, an inducer of the DNA damage response with potential anticancer activity, inhibition of H4K20 methylation, and inhibition of CDK4, and can be used to study breast cancer ...		Histone Demethylase , Histone Methyltransferase , CDK
T2576	Brivanib (alaninate)	BMS-582664,Brivanib Alaninate	VEGFR , FGFR , Autophagy
	Brivanib Alaninate (BMS-582664) is the alaninate salt of a vascular endothelial growth factor receptor 2 (VEGFR2) inhibitor with potential antineoplastic activity. Brivanib strongly binds to and inhibits VEGFR2, a tyrosi...		VEGFR , FGFR , Autophagy
T15581	Inolitazone	RS5444,Efatutazone,CS-7017	PPAR
	Inolitazone (RS5444) a high-affinity PPARγ agonist. Inolitazone exhibits IC50 for growth inhibition is ~0.8 nM in vitro.		PPAR
T14034	3CAI		Akt
			Akt
T25770	116-9e	MAL-2-11B,MAL2-11B,MAL211B,MAL 2 11B,MAL2 11B	Virus Protease
	116-9e (MAL2-11B) is a potent Hsp70 co-chaperone DNAJA1 inhibitor with antiviral properties, inhibition of simian virus 40 (SV40) replication, inhibition of tumour antigen (TAg) endogenous ATPase activity, and TAg-mediat...		Virus Protease
T11226	ERK1/2 inhibitor 1		ERK
	ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively.		ERK
T60019	VPC-70063	Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-	Apoptosis , PARP , c-Myc
	VPC-70063 (Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-) is an inhibitor of c-Myc-MAX. VPC-70063 exhibits Myc-Max transcriptional activity inhibition of 106% with an IC50 of 8.9 μM and Myc-Max/UBE2C do...		Apoptosis , PARP , c-Myc
T6686	Sulconazole mononitrate	Exelderm,Sulconazole Nitrate,RS 44872	Antibacterial , Antibiotic , Antifungal
	Sulconazole mononitrate (Exelderm) is the nitrate salt form of sulconazole, a synthetic imidazole derivative with the antifungal property. Sulconazole mononitrate inhibits fungal cytochrome P-450 sterol C-14 alpha-demeth...		Antibacterial , Antibiotic , Antifungal
T6244	Cidofovir	HPMPC,GS 0504,(S)-HPMPC	Others , DNA/RNA Synthesis
	Cidofovir ((S)-HPMPC) inhibits virus replication by specific inhibition of viral DNA synthesis.		Others , DNA/RNA Synthesis
T14997	Conteltinib	SY-707,CT-707	FAK , PYK2 , ALK
	Conteltinib (CT-707) is an enzyme inhibitor with antitumor activity targeting FAK, ALK, and Pyk2.Conteltinib exhibits significant inhibition of FAK, overcomes hypoxia-mediated sorafenib resistance in hepatocellular carci...		FAK , PYK2 , ALK
T15044	D609		Apoptosis , Antioxidant
	D609 (Tricyclodecan-9-yl-Xanthogenate) has a wide range of biological activities including antioxidant, antiapoptotic, anticholinergic, antitumor, anti-inflammatory, antiviral, antiproliferative, and neuroprotective acti...		Apoptosis , Antioxidant
T2627	Nolatrexed dihydrochloride	Thymitaq,AG 337	DNA/RNA Synthesis
	Nolatrexed dihydrochloride (Thymitaq) is the dihydrochloride salt of nolatrexed, a water-soluble lipophilic quinazoline folate analog with antineoplastic activity. Nolatrexed occupies the folate binding site of thymidyla...		DNA/RNA Synthesis
T12430	PF-06821497		Histone Methyltransferase
			Histone Methyltransferase
T6831	Etretinate	Retinoid,Tegison,Etretinato,Ethyl etrinoate,Ro 10-9359	Apoptosis , Others
	Etretinate (Ro 10-9359) is an oral aromatic retinoid acid which is effective in psoriasis and other dermatological syndromes. It activates retinoid receptors, causing an induction of cell differentiation, inhibition of c...		Apoptosis , Others
T6536	HJC0350		cAMP
	HJC0350 is an effective and specific EPAC2 inhibitor (IC50: 0.3 μM), and no inhibition of Epac1.		cAMP
T3352	XL413		cholecystokinin , Casein Kinase , Pim , CDK
	XL-413 is an orally bioavailable cell division cycle 7 homolog (CDC7) kinase inhibitor with potential antineoplastic activity. XL-413 binds to and inhibits the activity of CDC7, which may result in the inhibition of DNA ...		cholecystokinin , Casein Kinase , Pim , CDK
T1428	Trifluridine	NSC 529182,Trifluorothymidine,5-Trifluorothymidine,NSC 75520,Viroptic,Trifluridina	Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis , HSV
	Trifluridine (NSC-75520) is a fluorinated thymidine analog with potential antineoplastic activity. Trifluridine is incorporated into DNA and inhibits thymidylate synthase, resulting in inhibition of DNA synthesis, inhibi...		Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis , HSV
T0676	Hydroxyurea	Hydroxycarbamide,nsc32065,nci-c04831	Apoptosis , HIV Protease , DNA/RNA Synthesis , Autophagy
	Hydroxyurea (Hydroxycarbamide), an antineoplastic agent, inhibits DNA synthesis through the inhibition of ribonucleoside diphosphate reductase.		Apoptosis , HIV Protease , DNA/RNA Synthesis , Autophagy
T9360	CRBN ligand-9	2-(2,6-dioxopiperidin-3-yl)-5-nitroisoindoline-1,3-dione	Ligand for E3 Ligase
	CRBN ligand-9 (2-(2,6-dioxopiperidin-3-yl)-5-nitroisoindoline-1,3-dione) exhibit inhibition of CRBN.		Ligand for E3 Ligase
T8694	ML406		Antibacterial , Antibiotic
	ML406 shows anti-tubercular activity via MtbbioA (DAPA synthase) enzyme inhibition(IC50 : 30 nM)		Antibacterial , Antibiotic
T5101	BW-A 78U	BW-A78U	PDE
	BW-A 78U is a PDE4 inhibitor (IC50: 3 μM). It is not inhibition on the lipopolysaccharide (LPS)-induced TNF-α release.		PDE
T1348	Diphenyl phosphate	Phenyl hydrogen phosphate	Others
	Diphenyl phosphate (Phenyl hydrogen phosphate) is capable of gender-specific inhibition of growth and energy metabolism in zebrafish.		Others
T9823	WAY-325398		Others
	WAY-325398 is a furan derivatives. WAY-325398 inhibits osteoclast formation, inhibition rate is 14.11% at 10 μM.		Others
T24214	Phenamacril	JS39919,JS399 19	Myosin , Antifungal
	Phenamacril (JS39919) is acyanoacrylate fungicide, has powerful inhibition against Fusarium species, especially to Fusarium graminearum. Phenamacril is a specific Fusarium myosin I inhibitor.		Myosin , Antifungal
T1625	Lomefloxacin hydrochloride	Lomefloxacin HCl,Okacyn,Maxaquin	Topoisomerase , Antibacterial , Antibiotic
	Lomefloxacin hydrochloride (Okacyn) inhibits DNA gyrase, a type II topoisomerase involved in the induction or relaxation of supercoiling during DNA replication. This inhibition leads to a decrease in DNA synthesis during...		Topoisomerase , Antibacterial , Antibiotic
T71356	Lanperisone HCl
	Lanperisone, also known as NK433, is a muscle relaxant. NK433 inhibited the facilitation of the flexor reflex mediated by group II afferent fibers that was induced by intrathecal administration of noradrenaline-HCl. NK43...
T9345	Aminopeptidase M		Others
	Aminopeptidase M (AMP) inhibition is of interest for several diseases, such as highly vascularized cancer types.		Others
T9015	LY900009		Gamma-secretase
	LY900009 is a small molecule inhibitor of Notch signalling via selective inhibition of the γ-secretase protein.		Gamma-secretase
T2267	BQU57		GTPase , Ras
	BQU57 shows selective inhibition for Ral relative to Ras or Rho and inhibit xenograft tumor growth.		GTPase , Ras
T14673	BMS 299897		Beta Amyloid , Gamma-secretase
	BMS 299897 is a sulfonamide γ-secretase inhibitor. It has an IC50 of 7 nM for Aβ production inhibition in HEK293 cells stably overexpressing amyloid precursor protein (APP).		Beta Amyloid , Gamma-secretase
T24444	Medifoxamine	LG 152,Medifoxamina,LG-152,LG152	Dopamine Receptor , Monoamine Oxidase
	Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.Medifoxamine preferentially inhibits dopamine reuptake.		Dopamine Receptor , Monoamine Oxidase
T1849	Momelotinib	CYT11387,CYT387,LM-1149	Apoptosis , JAK , Autophagy
	Momelotinib (LM-1149) is an orally bioavailable small-molecule inhibitor of Janus kinases 1 and 2 (JAK1/2) with IC50 of 11 nM/18 nM. JAK1/2 inhibitor CYT387 competes with JAK1/2 for ATP binding, which may result in inhib...		Apoptosis , JAK , Autophagy
TNU0022	6-Azauridine	6-Azuridine	Apoptosis
	6-Azauridine (6-Azuridine) is a purine nucleoside analog with a broad spectrum of antitumor activity, targeting malignant tumors of the inert lymphatic system and inducing apoptosis.6-Azuridine's anticancer mechanism is ...		Apoptosis
T6546	IPA-3	IPA3,IPA 3	PAK
			PAK
T6214	Emtricitabine	FTC,Emtriva,BW1592	HIV Protease , Reverse Transcriptase
	Emtricitabine (FTC) (FTC), a nucleoside reverse transcriptase inhibitor, exhibits inhibition activity against human immunodeficiency virus (HIV) and hepatitis B virus.		HIV Protease , Reverse Transcriptase
T12831L	SAR405		PI3K , Autophagy
	SAR-405 is a potent and selective PIK3C3/Vps34 inhibitor (IC50:1.2 nM; Kd:1.5 nM) that prevents autophagy and synergizes with MTOR inhibition in tumor cells. SAR405 treatment also inhibits autophagy induced either by sta...		PI3K , Autophagy
T7142	Cephalosporin C zinc salt		Others
	Cephalosporin C zinc salt was a potent inhibitor of SAMHD1 (IC50 : 1.1 ± 0.1 µM), and this inhibition was largely attributable to the presence of zinc.		Others
T6632	Raltitrexed	ZD1694,D1694,ICI-D1694,Tomudex	Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis
	Raltitrexed (D1694)(IC50 of 9 nM), a thymidylate synthase inhibitor, is used for the inhibition of L1210 cell growth.		Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis
T29170	XU1	Benzo[c][1,8]naphthyridin-6(5h)-One	Aurora Kinase
	XU1（Benzo[c][1,8]naphthyridin-6(5h)-One） is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or modulation of kinase signaling.		Aurora Kinase
T63119	NF-κB/MAPK-IN-1		NF-κB , MAPK
	NF-κB/MAPK-IN-1 is a potent dual inhibitor of the NF-κB and MAPK pathways with potential anti-inflammatory activity, inhibition of NO production, and inhibition of LPS-induced activation of iNOS, COX-2, ERΚ and P38. NF-κ...		NF-κB , MAPK
T3211	Midostaurin	N-Benzoylstaurosporine,PKC412,CGP41231,CGP 41251	Others , PKC
	PKC412(Midostaurin (PKC412); CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor. Midostaurin inhibits protein kinase C alpha (PKCalpha), vascular endothelial growth factor receptor 2 (VEGFR2), c-kit, platel...		Others , PKC

Compounds

Synonym: 15-Lipoxygenase Inhibitor 1

Target: Apoptosis, Others, Lipoxygenase

BAMB-4

T14496

Synonym: ITPKA-IN-C14

Synonym: 2,2,6,6-Tetramethylpiperidin-4-yl heptanoate

Target: AChR

Oritavancin diphosphate

T2691

Synonym: LY333328 diphosphate

Target: Others, Antibacterial, Antibiotic

SKLB4771

T2051

Synonym: FLT3-IN-1,FLT3-IN-1

Target: FLT

AS057278

T7476

Synonym: 3-Methylpyrazole-5-carboxylic acid

Target: Estrogen/progestogen Receptor

Ryuvidine

T23284

Synonym:

Target: Histone Demethylase, Histone Methyltransferase, CDK

Brivanib (alaninate)

T2576

Synonym: BMS-582664,Brivanib Alaninate

Target: VEGFR, FGFR, Autophagy

Inolitazone

T15581

Synonym: RS5444,Efatutazone,CS-7017

Synonym: MAL-2-11B,MAL2-11B,MAL211B,MAL 2 11B,MAL2 11B

Target: Virus Protease

Synonym: Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-

Target: Apoptosis, PARP, c-Myc

Sulconazole mononitrate

T6686

Synonym: Exelderm,Sulconazole Nitrate,RS 44872

Target: Antibacterial, Antibiotic, Antifungal

Cidofovir

T6244

Synonym: HPMPC,GS 0504,(S)-HPMPC

Target: Others, DNA/RNA Synthesis

Conteltinib

T14997

Synonym: SY-707,CT-707

Target: FAK, PYK2, ALK

D609

T15044

Synonym:

Target: Apoptosis, Antioxidant

Nolatrexed dihydrochloride

T2627

Synonym: Thymitaq,AG 337

Target: DNA/RNA Synthesis

PF-06821497

T12430

Synonym:

Target: Histone Methyltransferase

Etretinate

T6831

Synonym: Retinoid,Tegison,Etretinato,Ethyl etrinoate,Ro 10-9359

Target: Apoptosis, Others

Target: cholecystokinin, Casein Kinase, Pim, CDK

Trifluridine

T1428

Synonym: NSC 529182,Trifluorothymidine,5-Trifluorothymidine,NSC 75520,Viroptic,Trifluridina

Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis, HSV

Hydroxyurea

T0676

Synonym: Hydroxycarbamide,nsc32065,nci-c04831

Target: Apoptosis, HIV Protease, DNA/RNA Synthesis, Autophagy

CRBN ligand-9

T9360

Synonym: 2-(2,6-dioxopiperidin-3-yl)-5-nitroisoindoline-1,3-dione

Target: Ligand for E3 Ligase

ML406

T8694

Synonym:

Target: Antibacterial, Antibiotic

Synonym: Phenyl hydrogen phosphate

Synonym: JS39919,JS399 19

Target: Myosin, Antifungal

Lomefloxacin hydrochloride

T1625

Synonym: Lomefloxacin HCl,Okacyn,Maxaquin

Target: Topoisomerase, Antibacterial, Antibiotic

Target: Gamma-secretase

Target: Beta Amyloid, Gamma-secretase

Medifoxamine

T24444

Synonym: LG 152,Medifoxamina,LG-152,LG152

Target: Dopamine Receptor, Monoamine Oxidase

Momelotinib

T1849

Synonym: CYT11387,CYT387,LM-1149

Target: Apoptosis, JAK, Autophagy

Synonym: FTC,Emtriva,BW1592

Target: HIV Protease, Reverse Transcriptase

SAR405

T12831L

Synonym:

Target: PI3K, Autophagy

Cephalosporin C zinc salt

Synonym: ZD1694,D1694,ICI-D1694,Tomudex

Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis

XU1

T29170

Synonym: Benzo[c][1,8]naphthyridin-6(5h)-One

Target: Aurora Kinase

Synonym: N-Benzoylstaurosporine,PKC412,CGP41231,CGP 41251

Target: Others, PKC

カタログ番号	製品名	別名	ターゲット
T5722	Nevadensin	Pedunculin	Anti-infection , Antibacterial
	Nevadensin is an important herb-based constituent inhibiting estragole bioactivation. Nevadensin protects against a methyleugenol-induced marker of hepatocarcinogenicity in male F344 rat. It also exhibits inhibition acti...		Anti-infection , Antibacterial
T5S0384	Rhapontin	Ponticin,Rhaponiticin,Rhaponticin,Rhapontigenin glucoside	Apoptosis , Others
	1. Rhapontin (Ponticin) can alleviate liver steatosis and improve blood glucose and lipid profiles in KK/Ay diabetic mice, indicates that rhaponticin has a noticeable antidiabetic effect and could be potentially used as ...		Apoptosis , Others
T1465	Mupirocin	Pseudomonic acid,BRL-4910A	DNA/RNA Synthesis , Antibacterial , Antibiotic
	Mupirocin (BRL-4910A) is a RNA synthetase inhibitor antibacterial. It has shown excellent activity against gram-positive staphylococci and streptococci.		DNA/RNA Synthesis , Antibacterial , Antibiotic
T8148	Mupirocin calcium hydrate	Mupirocin calcium	Others , Antibacterial , Antibiotic
	Mupirocin calcium hydrate is an antibiotic produced by Pseudomonas fluorescens, showed a high level of activity against staphylococci and streptococci and against certain gram-negative bacteria		Others , Antibacterial , Antibiotic
T10886	Crocetine dimethyl ester	Dimethylcrocetin	Antioxidant
	Crocetine dimethyl ester (Dimethylcrocetin) is a saffronin derivative with antioxidant activity, inhibition of AChE activity, and inhibition of cell growth and differentiation.		Antioxidant
T3880	Silydianin	Silidianin	Phosphatase
	Silydianin (Silidianin) exerts inhibition of UGT in human liver. Silydianin exerts inhibition of OATP1B1, OATP1B3 (unknown origin) expressed in HEK293 cells. Silydianin exerts inhibition of OATP2B1 (unknown origin) expre...		Phosphatase
T3817	Darutigenol		Others
	Darutigenol has obvious antithrombotic effect, its mechanism may be related to inhibition of platelet aggregation and adhesion.		Others
T3899	Calceolarioside B	Desrhamnosyl isoacteoside,Nuomioside A	Aromatase
	Calceolarioside B (Desrhamnosyl isoacteoside) displays inhibition of aromatase. Calceolarioside B displays inhibition of human recombinant PKCalpha.		Aromatase
T3401	Ginsenoside F1	20(S)-Ginsenoside F1	P450 , Endogenous Metabolite
	Ginsenoside F1 (20(S)-Ginsenoside F1) is an enzymatically modified derivative of ginsenoside Rg1, showing competitive inhibition of the activity of CYP3A4 and a weaker inhibition of the activity of CYP2D6.		P450 , Endogenous Metabolite
TN2343	Pseudojervine	Jervin-3-glucoside,O-beta-D-Glucopyranosyljervine	Platelet aggregation
	Pseudojervine (O-beta-D-Glucopyranosyljervine) is derived from Veratrum nigrum L. Pseudojervine exhibits feeble inhibition activity against platelet aggregation.		Platelet aggregation
TN3460	Asebogenin		Antifungal
	Asebogenin is a compound fractionated from Salvia miltiorrhiza with antifungal activity, inhibition of GPVI-induced platelet reactions, and inhibition of NET formation induced by pro-inflammatory stimuli.		Antifungal
TN7125	2-Propen-1-one, 1-(2,6-dimethoxyphenyl)-3-(4-hydroxyphenyl)-		Others
	2-Propen-1-one, 1-(2,6-dimethoxyphenyl)-3-(4-hydroxyphenyl)- can be used in studies about the inhibition against L-phenylalanine ammonia-lyase.		Others
TN1021	Secologanic acid		NO Synthase
	Secologanic acid is a plant growth inhibitor, it shows inhibition of nitric oxide production in lipopolysaccharide-activated macrophages.		NO Synthase
T2S0973	2-Methoxycinnamic acid	AI3-11206,o-Methoxycinnamic acid	Tyrosinase
	1. 2-Methoxycinnamic acid (o-Methoxycinnamic acid) can enhance inhibition of tyrosinase activity.		Tyrosinase
TN1873	Lirinidine		Others
	(+)-Lirinidine has antioxidative activity, and it can significantly inhibit the proliferation of melanoma cells; it also shows potent inhibition of melanogenesis. Lirinidine exhibits significant inhibition of collagen, a...		Others
T19931	Gentisein	NSC 329491,NSC329491,NSC-329491	Serotonin Transporter
	Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency with an IC50 value of 4.7 µM[1][2].		Serotonin Transporter
TN3548	Bulleyanin		Others
	Bulleyanin shows strong inhibition of mouse ehrlich ascites carcinoma (ECA), mouse sarcoma S-180, and mouse liver ascites.		Others
TN1733	Hesperetin 7-O-glucoside		Anti-infection , Antibacterial , HMG-CoA Reductase
	Hesperetin 7-O-glucoside and prunin are direct precursors of naringin and neohesperidin, respectively, in C. aurantium. Hesperetin 7-O-glucoside shows inhibition of human HMG-CoA reductase, it also exhibits effective inh...		Anti-infection , Antibacterial , HMG-CoA Reductase
T3682	(-)-Catechin gallate	(-)-Catechin 3-O-gallate,(-)-Catechin 3-gallate	Others , COX
	(-)-Catechin gallate ((-)-Catechin 3-O-gallate) displays inhibition of 6PGD, IDH. (-)-Catechin gallate ((-)-Catechin 3-O-gallate) displays inhibition of human Beta-secretase. (-)-Catechin gallate ((-)-Catechin 3-O-gallat...		Others , COX
TN1057	Veratrosine	Veratramine 3-glycoside,Veratramine-beta-D-glucoside	Platelet aggregation
	Veratrosine (Veratramine-beta-D-glucoside) is an alkaloid isolated from the herbs of Veratrum nigrum. Veratrosine exhibits feeble inhibition activity against platelet aggregation.		Platelet aggregation
T3S1850	Bayogenin		Others
	Bayogenin is an alfalfa saponin, Bayogenin shows moderate potency of glycogen phosphorylase inhibition.		Others
TN2202	Sempervirine		DNA/RNA Synthesis
	Sempervirine can unwind circular DNA, it shows selective inhibition of in vitro synthesis of cancer DNA .		DNA/RNA Synthesis
T4S1616	Sanggenon D	Sanggenone D	NOS , COX , GABA Receptor
	Sanggenone D represents a new scaffold of positive GABAA receptor modulators, it also inhibits COX-2 activity (IC 50 = 73-100 μM). Sanggenone D has anti-inflammatory activity, it can inhibit NO production from lipopolysa...		NOS , COX , GABA Receptor
T2S2018	7beta-Hydroxylathyrol	7β-Hydroxylathyrol,7-Hydroxylathyrol,7-beta-Hydroxylathyrol	P-gp
	7β-Hydroxylathyrol is a diterpenoid extract from the seed oil of Caper Spurge and displays P-gp inhibition resulting in cytotoxic properties.		P-gp
TN1137	Isobutylshikonin		Others
	Isobutylshikonin exhibits obvious antioxidant activities , it exerts very good radical scavenging activities toward ABTS+ but shows moderate inhibition of DPPH·.		Others
T3668	Galangin	Norizalpinin,3,5,7-Trihydroxyflavone	ERK , P450 , NF-κB , Autophagy
	Galangin (Norizalpinin) is an agonist/antagonist of the arylhydrocarbon receptor, and also shows inhibition of CYP1A1 activity.		ERK , P450 , NF-κB , Autophagy
TQ0070	Luteolin-3-O-beta-D-glucuronide		Others
	Luteolin-3-O-beta-D-glucuronide is active in the inhibition of nitrite production in macrophages.		Others
T6213	Vinorelbine ditartrate	Vinorelbine Tartrate,Nor-5'-anhydrovinblastine ditartrate,KW-2307,Navelbine tartrate	Microtubule Associated , Autophagy
	Vinorelbine ditartrate (KW-2307), a semi-synthetic vinca alkaloid, interacts with tubulin resulting in mitosis inhibition.		Microtubule Associated , Autophagy
T1441	Capreomycin sulfate	Capastat sulfate	ribosome , Antibacterial , Antibiotic
	Capreomycin sulfate (Capastat sulfate) , a cyclic peptide antibiotic, binds to the 70S ribosomal unit leading to inhibition of protein synthesis.		ribosome , Antibacterial , Antibiotic
TN7126	N-Vanillyloctanamide		Others
	N-Vanillyloctanamide is a capsaicinoid from the fruits of Capsicum annuum L. var. annuum. N-Vanillyloctanamide reduces the radical length of Lactuca sativa seedling, this inhibition being dose-dependent.		Others
TN1975	Neosmitilbin	Neoastilbin	Others
	Neosmitilbin (Neoastilbin) may have antioxidant and anti-inflammatory activities, it shows potent inhibition of lens aldose reductase.		Others
T1276	Danofloxacin mesylate	CP 76136-27	DNA/RNA Synthesis , Antibacterial , Antibiotic
	Danofloxacin mesylate (CP 76136-27) is a synthetic antibacterial agent of the fluoroquinolone class, acts principally by the inhibition of bacterial DNA-gyrase.		DNA/RNA Synthesis , Antibacterial , Antibiotic
TN2008	Okanin		NF-κB , TLR
	Okanin shows significant activities on both linoleic acid peroxidation inhibition and DPPH radical scavenging effect.		NF-κB , TLR
TN1995	5,7,8-Trimethoxyflavone	Norwogonin 5,7,8-trimethyl ether	NO Synthase
	5,7,8-Trimethoxyflavone (Norwogonin 5,7,8-trimethyl ether) is a compound extracted from Andrographis paniculata with anti-inflammatory activity and NO inhibition.		NO Synthase
T12651	Rabdosiin	(+)-Rabdosiin	Others
	Rabdosiin ((+)-Rabdosiin) is a natural product, and has anti-allergic activity, anti-HIV activity and inhibition on DNA topoisomerase.		Others
TWS1977	Kamebakaurin	Kamebakaurine	NF-κB
	1. Kamebakaurin (Kamebakaurine) has the ability to protect the liver from APAP-induced hepatotoxicity, presumably by both inhibiting the inflammatory response and oxidative stress. 2. Kamebakaurin inhibits the expression...		NF-κB
T8187	Tetrahydroepiberberine		Others , Influenza Virus , Antifungal
	Tetrahydroepiberberine, an isoquinoline alkaloid, has antifungal and selective inhibition against the PI-3 virus activities.		Others , Influenza Virus , Antifungal
T3S1967	(S)-Indoximod	N-ME-Tryptophan,Abrine,L-Abrine	Others , Indoleamine 2,3-Dioxygenase (IDO)
	(S)-Indoximod (L-Abrine) exhibits inhibition of rabbit small intestine indoleamine 2, 3-dioxygenase, competitive inhibition of IDO, reduction of Foxp3 protein expression in tumor of C57BL/6 mouse allografted with mouse L...		Others , Indoleamine 2,3-Dioxygenase (IDO)
T6413	Bindarit	AF2838	CCR
	Bindarit (AF2838) displays specific inhibition against monocyte chemotactic proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.		CCR
TN4661	Nodosin		IL Receptor , Autophagy
	Nodosin has anti-inflammatory function of Nodosin via inhibition of IL-2. Nodosin perfusion provides a potential protective effect through inducing HO-1 expression to attenuate ischemia/reperfusion injury in liver transp...		IL Receptor , Autophagy
T3S2340	Usaramine	(15E)-Retrorsine,Mucronatine,NISTC15503874	Others , Antibacterial
	Usaramine (Mucronatine) demonstrates phytotoxicity against Lactuca sativa var. Carrascoy (lettuce) assessed as inhibition of seed germination at 50 ug/cm2 after 24 hr.		Others , Antibacterial
T7468	(-)-α-Terpineol	α-Terpineol	Others
	(-)-α-Terpineol has antitumour, anti-inflammatory, and antimicrobial activities, it inhibits the growth of tumour cells through a mechanism that involves inhibition of the NF-kappaB pathway		Others
TN5503	Linaroside		Antibacterial
	Linaroside exhibited 30% inhibition for antimycobacterial activity against Mycobacterium tuberculosis, strain H(37)Rv at 6.25 microg mL(-1) concentration.		Antibacterial
T6S0444	Salvianolic acid A	Dan Phenolic Acid A	MMP
	Salvianolic acid A (Dan Phenolic Acid A) could protect the blood brain barrier through inhibition of matrix metallopeptidase 9 (MMP-9) and anti-inflammation.		MMP
T2S1181	Aloenin	Aloenin A,Aloearbonaside	Beta-Secretase , AChR
	1. Aloenin (Aloenin A) and aloe-emodin are active principles for inhibition of c-ADH and c-ALDH activities in vitro.		Beta-Secretase , AChR
T4S0111	Hupehenine		AChR
	Hupehenine is a steriodal alkaloid extracted from the bulbs of Fritillaria Hupehensis, with the potential for inhibiting acetylcholine, antagonism for muscarinic receptors and cholinesterase inhibition.		AChR
T6S1529	Cynarin	Cyclohexanecarboxylic acid, 1,3-bis[[3-(3,4-dihydroxyphenyl)-1-oxo-2-propen-1-yl]oxy]-4,5-dihydroxy-, (1R,3R,4S,5R)-,Cynarine,1,5-Dicaffeoylquinic acid	Antioxidant , Antiviral , Influenza Virus , Reactive Oxygen Species
	Cynarin (1,5-Dicaffeoylquinic acid) has neuroprotective, and antioxidant effects, it can inhibition of GSK3β as well as the modulation of Bcl-2/Bax.
T5S1952	9-Methoxycamptothecin		Apoptosis , Topoisomerase
	9-Methoxycamptothecin (MCPT) has antitumour activities through topoisomerase inhibition.		Apoptosis , Topoisomerase
T8244	Raspberry ketone glucoside		Others
	Raspberry ketone glucoside is a natural product in raspberry fruit, has lasting effects for the inhibition of melanogenesis and various melanogenic factors after the degradation in the skin.		Others
T13768	(+)-Medicarpin		Estrogen/progestogen Receptor
	(+)-Medicarpin, a pterocarpan, is an isoflavonoid compound derived from multiple medicinal plant species such as Sophora japonica, Zollernia paraensis, Platymiscium yucatamun, Machaerium aristulatum, and Platymiscium flo...		Estrogen/progestogen Receptor
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天然物製品

Nevadensin

T5722

Synonym: Pedunculin

Target: Anti-infection, Antibacterial

Rhapontin

T5S0384

Synonym: Ponticin,Rhaponiticin,Rhaponticin,Rhapontigenin glucoside

Target: Apoptosis, Others

Mupirocin

T1465

Synonym: Pseudomonic acid,BRL-4910A

Target: DNA/RNA Synthesis, Antibacterial, Antibiotic

Mupirocin calcium hydrate

T8148

Synonym: Mupirocin calcium

Target: Others, Antibacterial, Antibiotic

Crocetine dimethyl ester

T10886

Synonym: Dimethylcrocetin

Synonym: Desrhamnosyl isoacteoside,Nuomioside A

Target: Aromatase

Ginsenoside F1

T3401

Synonym: 20(S)-Ginsenoside F1

Target: P450, Endogenous Metabolite

Pseudojervine

TN2343

Synonym: Jervin-3-glucoside,O-beta-D-Glucopyranosyljervine

Target: Platelet aggregation

2-Propen-1-one, 1-(2,6-dimethoxyphenyl)-3-(4-hydroxyphenyl)-

2-Methoxycinnamic acid

T2S0973

Synonym: AI3-11206,o-Methoxycinnamic acid

Synonym: NSC 329491,NSC329491,NSC-329491

Target: Serotonin Transporter

Hesperetin 7-O-glucoside

TN1733

Synonym:

Target: Anti-infection, Antibacterial, HMG-CoA Reductase

(-)-Catechin gallate

T3682

Synonym: (-)-Catechin 3-O-gallate,(-)-Catechin 3-gallate

Target: Others, COX

Veratrosine

TN1057

Synonym: Veratramine 3-glycoside,Veratramine-beta-D-glucoside

Target: Platelet aggregation

Target: DNA/RNA Synthesis

Sanggenon D

T4S1616

Synonym: Sanggenone D

Target: NOS, COX, GABA Receptor

7beta-Hydroxylathyrol

T2S2018

Synonym: 7β-Hydroxylathyrol,7-Hydroxylathyrol,7-beta-Hydroxylathyrol

Synonym: Norizalpinin,3,5,7-Trihydroxyflavone

Target: ERK, P450, NF-κB, Autophagy

Luteolin-3-O-beta-D-glucuronide

TQ0070

Synonym:

Target: Others

Vinorelbine ditartrate

T6213

Synonym: Vinorelbine Tartrate,Nor-5'-anhydrovinblastine ditartrate,KW-2307,Navelbine tartrate

Target: Microtubule Associated, Autophagy

Capreomycin sulfate

T1441

Synonym: Capastat sulfate

Target: ribosome, Antibacterial, Antibiotic

Danofloxacin mesylate

T1276

Synonym: CP 76136-27

Target: DNA/RNA Synthesis, Antibacterial, Antibiotic

5,7,8-Trimethoxyflavone

TN1995

Synonym: Norwogonin 5,7,8-trimethyl ether

Target: NO Synthase

Rabdosiin

T12651

Synonym: (+)-Rabdosiin

Target: Others

Kamebakaurin

TWS1977

Synonym: Kamebakaurine

Target: NF-κB

Tetrahydroepiberberine

T8187

Synonym:

Target: Others, Influenza Virus, Antifungal

(S)-Indoximod

T3S1967

Synonym: N-ME-Tryptophan,Abrine,L-Abrine

Target: Others, Indoleamine 2,3-Dioxygenase (IDO)

Target: IL Receptor, Autophagy

Usaramine

T3S2340

Synonym: (15E)-Retrorsine,Mucronatine,NISTC15503874

Target: Others, Antibacterial

Target: Antibacterial

Salvianolic acid A

T6S0444

Synonym: Dan Phenolic Acid A

Target: MMP

Aloenin

T2S1181

Synonym: Aloenin A,Aloearbonaside

Target: Beta-Secretase, AChR

Synonym: Cyclohexanecarboxylic acid, 1,3-bis[[3-(3,4-dihydroxyphenyl)-1-oxo-2-propen-1-yl]oxy]-4,5-dihydroxy-, (1R,3R,4S,5R)-,Cynarine,1,5-Dicaffeoylquinic acid

Target: Antioxidant, Antiviral, Influenza Virus, Reactive Oxygen Species

9-Methoxycamptothecin

T5S1952

Synonym:

Target: Apoptosis, Topoisomerase

Raspberry ketone glucoside

Target: Estrogen/progestogen Receptor

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Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPK-00782	PLAU/uPA Protein, Mouse, Recombinant (His & Avi)	Mouse	HEK293 Cells
	Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor pro...
TMPY-02078	HtrA2/Omi Protein, Human, Recombinant (His)	Human	E. coli
	Serine protease HTRA2, also known as high-temperature requirement protein A2, Omi stress-regulated endoprotease, Serine protease 25, Serine proteinase OMI and HTRA2, is a single-pass membrane protein that belongs to the ...
TMPY-02483	ATP citrate lyase/ACLY Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	ATP citrate lyase, also known as Acly or Acl, is the primary enzyme responsible for the synthesis of cytosolic acetyl-CoA in many tissues. The enzyme is composed of two polymer chains which are polypeptides in human. ATP...
TMPJ-01172	IL-17 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Interleukin-17 is a potent pro-inflammatory cytokine produced by activated memory T cells. There are at least six members of the IL-17 family in humans and in mice. Mature mouse IL-17A shares 61% and 89% amino acid seque...
TMPY-05176	AMH Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Anti-Mullerian hormone (AMH), a member of the TGF-beta superfamily, is produced by granulosa cells (GCs) of preantral and small antral follicles and plays a role in regulating the recruitment of primordial follicles and ...
TMPY-04830	GAS6 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	The growth arrest-specific 6 gene (GAS6) is a member of the family of plasma vitamin K-dependent proteins, which are able to bind to phospholipids using an N-terminal gamma-carboxyglutamic acid domain. GAS6 is a vitamin ...
TMPY-02219	Influenza A H1N1 (A/Puerto Rico/8/34/Mount Sinai) Non-structural/NS1 Protein (His)	H1N1	E. coli
	The NS1 Influenza protein is created by the internal protein-encoding, linear negative-sense, single-stranded RNA, NS gene segment and which also codes for the nuclear export protein or NEP, formerly referred to as the N...
TMPH-00554	Trypsin inhibitor DE-3 Protein, Erythrina caffra, Recombinant (His)	Erythrina caffra	P. pastoris (Yeast)
	Inhibition of trypsin.
TMPH-02886	SOST Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	Negative regulator of bone growth that acts through inhibition of Wnt signaling and bone formation.
TMPH-01659	MAGEA4 Protein, Human, Recombinant (A173T, His & Myc)	Human	E. coli
	Regulates cell proliferation through the inhibition of cell cycle arrest at the G1 phase. Also negatively regulates p53-mediated apoptosis.
TMPH-01658	MAGEA4 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Regulates cell proliferation through the inhibition of cell cycle arrest at the G1 phase. Also negatively regulates p53-mediated apoptosis.
TMPK-01485	HLA-A*01:01&B2M&DSG3 (YTDNWLAVY) Monomer Protein, Human, MHC (His & Avi)	Human	HEK293 Cells
	DSG3 is overexpressed in head neck cancer and is a potential molecular target for inhibition of oncogenesis. DSG3 is identified overexpressed in HNC, with the degree of overexpression associated with clinicopathologic fe...
TMPH-01715	CHRM2 Protein, Human, Recombinant (His)	Human	E. coli
	The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. ...
TMPY-00729	Cystatin D Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Cystatins are natural inhibitors of papain-like (family C1) and legumain-related (family C13) cysteine peptidases. The mammalian cystatin superfamily members are of three major types, including the type 1 cystatins (stef...
TMPY-02425	Serpin B4, Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	Overexpression of SERPINB4 in tumor cells inhibited recombinant GrM-induced as well as NK cell-mediated cell death and this inhibition depended on the reactive center loop of the serpin.
TMPJ-00604	KIR2DL4 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Killer cell immunoglobulin-like receptor 2DL4(KIR2DL4) is a Single-pass type I membrane protein and contains 2 Ig-like C2-type (immunoglobulin-like) domains.It belongs to the immunoglobulin superfamily. KIR2DL4 is expres...
TMPH-01717	CHRM5 Protein, Human, Recombinant (His)	Human	E. coli
	The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. ...
TMPH-01714	CHRM1 Protein, Human, Recombinant (His)	Human	E. coli
	The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. ...
TMPH-03338	CHRM1 Protein, Rat, Recombinant (His)	Rat	E. coli
	The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. ...
TMPH-01610	LINGO1 Protein, Human, Recombinant (His)	Human	E. coli
	Functional component of the Nogo receptor signaling complex (RTN4R/NGFR) in RhoA activation responsible for some inhibition of axonal regeneration by myelin-associated factors. Is also an important negative regulator of ...
TMPH-01716	CHRM3 Protein, Human, Recombinant (B2M & His)	Human	E. coli
	The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. ...
TMPH-01341	FILIP1L Protein, Human, Recombinant (His)	Human	E. coli
	Acts as a regulator of the antiangiogenic activity on endothelial cells. When overexpressed in endothelial cells, leads to inhibition of cell proliferation and migration and an increase in apoptosis. Inhibits melanoma gr...
TMPK-00553	ADAM9 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	A disintegrin and metalloproteinase 9 (ADAM9) is a member of the transmembrane ADAM family. It is expressed in different types of solid cancer and promotes tumor invasiveness. ADAM9 may be a prognostic marker for vestibu...
TMPK-01095	MEPE Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Matrix extracellular phosphoglycoprotein (MEPE) is expressed in bone and teeth where it has multiple functions. The C-terminus of MEPE contains a mineral-binding, acidic serine- and aspartate-rich motif (ASARM) that is a...
TMPK-00539	PLAU/uPA Protein (active form), Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor pro...
TMPK-00102	SOST Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	SOST, also known as sclerostin, is a member of the cerberus/DAN family, a group of secreted glycoproteins characterized by a cysteine-knot motif. SOST is negative regulator of bone growth that acts through inhibition of ...
TMPK-00783	PLAU/uPA Protein, Mouse, Recombinant (His & Avi), Biotinylated	Mouse	HEK293 Cells
	Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor pro...
TMPK-00103	SOST Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	SOST, also known as sclerostin, is a member of the cerberus/DAN family, a group of secreted glycoproteins characterized by a cysteine-knot motif. SOST is negative regulator of bone growth that acts through inhibition of ...
TMPH-01642	MELK Protein, Human, Recombinant (His & Myc)	Human	E. coli
	Serine/threonine-protein kinase involved in various processes such as cell cycle regulation, self-renewal of stem cells, apoptosis and splicing regulation. Has a broad substrate specificity; phosphorylates BCL2L14, CDC25...
TMPJ-01052	DYNLL1 Protein, Human, Recombinant (His)	Human	E. coli
	Human Dynein Cytoplasmic Light Chain 1 (DYNLL1) has been identified as a protein that interacts with NOS1, leading to NOS1 inhibition. NOS1 dimer is destabilized after binding DYNLL1 a conformation necessary activity, an...
TMPJ-00407	ROBO4 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Roundabout homolog 4(ROBO4) contains 2 fibronectin type-III domains, 2 Ig-like C2-type (immunoglobulin-like) domains and belongs to the immunoglobulin superfamily.The protein is a receptor for slit proteins, at least fo...
TMPJ-00008	CXCL10 Protein, Human, Recombinant (hFc & His)	Human	HEK293 Cells
	Human C-X-C Motif Chemokine Ligand 10 (CXCL10) is a non-ELR chemokine secreted by various cell types, such as monocytes, endothelial cells and fibroblasts, in response to IFN-γ. CXCL10 functions via chemokine receptor CX...
TMPK-01293	SOST Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	SOST, also known as sclerostin, is a member of the cerberus/DAN family, a group of secreted glycoproteins characterized by a cysteine-knot motif. SOST is negative regulator of bone growth that acts through inhibition of ...
TMPH-03733	Zaire ebolavirus (strain Kikwit-95) VP35 Protein (His & Myc)	ZEBOV	HEK293 Cells
	Plays an essential role in viral RNA synthesis and also a role in suppressing innate immune signaling. Acts as a polymerase cofactor in the RNA polymerase transcription and replication complexes. Serves as nucleoprotein/...
TMPH-03732	Zaire ebolavirus (strain Kikwit-95) VP35 Protein (E. col, His & Myc)	ZEBOV	E. coli
	Plays an essential role in viral RNA synthesis and also a role in suppressing innate immune signaling. Acts as a polymerase cofactor in the RNA polymerase transcription and replication complexes. Serves as nucleoprotein/...
TMPK-00428	HER2/ErbB2 Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	ErbB2, also called Neu and Her2 (human epidermal growth factor receptor 2), is a type I membrane glycoprotein that is a member of the ErbB family of tyrosine kinase receptors. ErbB family members serve as receptors for t...
TMPK-00274	PLAU/uPA Protein (active form), Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor pro...
TMPY-04409	GRK6 Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	G protein-coupled receptor kinase 6, also known as G protein-coupled receptor kinase GRK6, GRK6, and GPRK6, is a lipid-anchor protein that belongs to the protein kinase superfamily, AGC Ser/Thr protein kinase family, and...
TMPK-01045	IL-20RA Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	IL-20RA was highly expressed in the tumor tissue of CRC and related to the advanced stage.IL-20RA was involved in regulating oncogenic and immune pathways and affecting the expression of genes related to cell proliferati...
TMPK-00564	TNFR1/CD120a/TNFRSF1A Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Tumour necrosis factor alpha (TNF-α) is a pleiotropic cytokine with both injurious and protective functions, which are thought to diverge at the level of its two cell surface receptors, TNFR1 and TNFR2. In the setting of...
TMPK-00022	Galectin-1 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Galectin 1 (Gal-1), a β-galactoside binding mammalian lectin of 14KDa, is implicated in many signalling pathways, immune responses associated with cancer progression and immune disorders. Inhibition of human Gal-1 has be...
TMPK-00893	PGF Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Placental growth factor (PGF) is another member of the VEGF family of cytokines with pro-angiogenic and pro-inflammatory effects. Retinal inhibition of PGF in combination with VEGF-A prevents vascular leakage and CNV pos...
TMPK-00829	Galectin-1 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	Galectin 1(Gal-1), a β-galactoside binding mammalian lectin of 14KDa, is implicated in many signalling pathways, immune responses associated with cancer progression and immune disorders. Inhibition of human Gal-1 has bee...
TMPJ-00692	GAS7 Protein, Human, Recombinant (His)	Human	E. coli
	Growth Arrest-Specific Protein 7 (GAS7) is expressed primarily in terminalaly differentiated brain cells and predominantly in mature cerebellar Purkinje neurons. GAS7 may play a role in neuronal development by promoting ...
TMPJ-00855	GLUL Protein, Human, Recombinant (His)	Human	E. coli
	Glutamine Synthetase reglutes intracellular concentration of glutamate. Glutamine Synthetase catalyzes the synthesis of glutamine from glutamate and ammonia. Glutamine is an important source of energy and that takes part...
TMPH-02753	LINGO1 Protein, Mouse, Recombinant (His)	Mouse	E. coli
	Functional component of the Nogo receptor signaling complex (RTN4R/NGFR) in RhoA activation responsible for some inhibition of axonal regeneration by myelin-associated factors. Is also an important negative regulator of ...
TMPY-06179	IdeS Protein, Streptococcus pyogenes, Recombinant (His & GST)	Streptococcus pyogenes	E. coli
	IdeS (IgG-degrading enzyme of Streptococcus pyogenes) is a secreted cysteine endopeptidase from the human pathogen S. pyogenes with an extraordinarily high degree of substrate specificity, catalyzing a single proteolytic...
TMPH-03598	Streptopain Protein, S. pyogenes serotype M28, Recombinant (His & SUMO)	Streptococcus pyogenes	E. coli
	Important streptococcal virulence factor which cleaves human fibronectin and degrades vitronectin. Also cleaves human IL1B precursor to form biologically active IL1B. Can induce apoptosis in human monocytes and epithelia...
TMPH-03599	Streptopain Protein, S. pyogenes, Recombinant (His & SUMO)	Streptococcus pyogenes	E. coli
	Important streptococcal virulence factor which cleaves human fibronectin and degrades vitronectin. Also cleaves human IL1B precursor to form biologically active IL1B. Can induce apoptosis in human monocytes and epithelia...
TMPH-01428	TRAP1 Protein, Human, Recombinant (GST)	Human	E. coli
	Chaperone that expresses an ATPase activity. Involved in maintaining mitochondrial function and polarization, downstream of PINK1 and mitochondrial complex I. Is a negative regulator of mitochondrial respiration able to ...
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PLAU/uPA Protein, Mouse, Recombinant (His & Avi)

TMPK-00782

Species: Mouse

Expression System: HEK293 Cells

HtrA2/Omi Protein, Human, Recombinant (His)

TMPY-02078

Species: Human

Expression System: E. coli

ATP citrate lyase/ACLY Protein, Human, Recombinant (His)

TMPY-02483

Species: Human

Expression System: Baculovirus Insect Cells

IL-17 Protein, Mouse, Recombinant (His)

TMPJ-01172

Species: Mouse

Expression System: HEK293 Cells

AMH Protein, Human, Recombinant (His)

TMPY-05176

Species: Human

Expression System: HEK293 Cells

GAS6 Protein, Mouse, Recombinant (His)

TMPY-04830

Species: Mouse

Expression System: HEK293 Cells

Influenza A H1N1 (A/Puerto Rico/8/34/Mount Sinai) Non-structural/NS1 Protein (His)

TMPY-02219

Species: H1N1

Expression System: E. coli

Trypsin inhibitor DE-3 Protein, Erythrina caffra, Recombinant (His)

TMPH-00554

Species: Erythrina caffra

Expression System: P. pastoris (Yeast)

SOST Protein, Mouse, Recombinant (hFc)

TMPH-02886

Species: Mouse

Expression System: HEK293 Cells

MAGEA4 Protein, Human, Recombinant (A173T, His & Myc)

TMPH-01659

Species: Human

Expression System: E. coli

MAGEA4 Protein, Human, Recombinant (His)

TMPH-01658

Species: Human

Expression System: HEK293 Cells

HLA-A*01:01&B2M&DSG3 (YTDNWLAVY) Monomer Protein, Human, MHC (His & Avi)

TMPK-01485

Species: Human

Expression System: HEK293 Cells

CHRM2 Protein, Human, Recombinant (His)

TMPH-01715

Species: Human

Expression System: E. coli

Cystatin D Protein, Human, Recombinant (His)

TMPY-00729

Species: Human

Expression System: HEK293 Cells

Serpin B4, Protein, Human, Recombinant (His)

TMPY-02425

Species: Human

Expression System: Baculovirus Insect Cells

KIR2DL4 Protein, Human, Recombinant (His)

TMPJ-00604

Species: Human

Expression System: HEK293 Cells

CHRM5 Protein, Human, Recombinant (His)

TMPH-01717

Species: Human

Expression System: E. coli

CHRM1 Protein, Human, Recombinant (His)

TMPH-01714

Species: Human

Expression System: E. coli

CHRM1 Protein, Rat, Recombinant (His)

TMPH-03338

Species: Rat

Expression System: E. coli

LINGO1 Protein, Human, Recombinant (His)

TMPH-01610

Species: Human

Expression System: E. coli

CHRM3 Protein, Human, Recombinant (B2M & His)

TMPH-01716

Species: Human

Expression System: E. coli

FILIP1L Protein, Human, Recombinant (His)

TMPH-01341

Species: Human

Expression System: E. coli

ADAM9 Protein, Cynomolgus, Recombinant (His)

TMPK-00553

Species: Cynomolgus

Expression System: HEK293 Cells

MEPE Protein, Mouse, Recombinant (His)

TMPK-01095

Species: Mouse

Expression System: HEK293 Cells

PLAU/uPA Protein (active form), Cynomolgus, Recombinant (His)

TMPK-00539

Species: Cynomolgus

Expression System: HEK293 Cells

SOST Protein, Human, Recombinant (His & Avi)

TMPK-00102

Species: Human

Expression System: HEK293 Cells

PLAU/uPA Protein, Mouse, Recombinant (His & Avi), Biotinylated

TMPK-00783

Species: Mouse

Expression System: HEK293 Cells

SOST Protein, Human, Recombinant (His & Avi), Biotinylated

TMPK-00103

Species: Human

Expression System: HEK293 Cells

MELK Protein, Human, Recombinant (His & Myc)

TMPH-01642

Species: Human

Expression System: E. coli

DYNLL1 Protein, Human, Recombinant (His)

TMPJ-01052

Species: Human

Expression System: E. coli

ROBO4 Protein, Human, Recombinant (hFc)

TMPJ-00407

Species: Human

Expression System: HEK293 Cells

CXCL10 Protein, Human, Recombinant (hFc & His)

TMPJ-00008

Species: Human

Expression System: HEK293 Cells

SOST Protein, Cynomolgus, Recombinant (His)

TMPK-01293

Species: Cynomolgus

Expression System: HEK293 Cells

Zaire ebolavirus (strain Kikwit-95) VP35 Protein (His & Myc)

TMPH-03733

Species: ZEBOV

Expression System: HEK293 Cells

Zaire ebolavirus (strain Kikwit-95) VP35 Protein (E. col, His & Myc)

TMPH-03732

Species: ZEBOV

Expression System: E. coli

HER2/ErbB2 Protein, Human, Recombinant (His & Avi)

TMPK-00428

Species: Human

Expression System: HEK293 Cells

PLAU/uPA Protein (active form), Human, Recombinant (His & Avi), Biotinylated

TMPK-00274

Species: Human

Expression System: HEK293 Cells

GRK6 Protein, Human, Recombinant (His & GST)

TMPY-04409

Species: Human

Expression System: Baculovirus Insect Cells

IL-20RA Protein, Mouse, Recombinant (hFc)

TMPK-01045

Species: Mouse

Expression System: HEK293 Cells

TNFR1/CD120a/TNFRSF1A Protein, Cynomolgus, Recombinant (His)

TMPK-00564

Species: Cynomolgus

Expression System: HEK293 Cells

Galectin-1 Protein, Human, Recombinant (hFc)

TMPK-00022

Species: Human

Expression System: HEK293 Cells

PGF Protein, Human, Recombinant (hFc)

TMPK-00893

Species: Human

Expression System: HEK293 Cells

Galectin-1 Protein, Mouse, Recombinant (hFc)

TMPK-00829

Species: Mouse

Expression System: HEK293 Cells

GAS7 Protein, Human, Recombinant (His)

TMPJ-00692

Species: Human

Expression System: E. coli

GLUL Protein, Human, Recombinant (His)

TMPJ-00855

Species: Human

Expression System: E. coli

LINGO1 Protein, Mouse, Recombinant (His)

TMPH-02753

Species: Mouse

Expression System: E. coli

IdeS Protein, Streptococcus pyogenes, Recombinant (His & GST)

TMPY-06179

Species: Streptococcus pyogenes

Expression System: E. coli

Streptopain Protein, S. pyogenes serotype M28, Recombinant (His & SUMO)

TMPH-03598

Species: Streptococcus pyogenes

Expression System: E. coli

Streptopain Protein, S. pyogenes, Recombinant (His & SUMO)

TMPH-03599

Species: Streptococcus pyogenes

Expression System: E. coli

TRAP1 Protein, Human, Recombinant (GST)

TMPH-01428

Species: Human

Expression System: E. coli

--------- More ---------

カタログ番号	製品名
L7300	Potassium Channel Blocker Library	152 compounds
	A unique collection of 152 potassium channel blockers and agonists for high throughput and high content screening;
L2160	Anti-Cancer Active Compound Library	3188 compounds
	A unique collection of 3188 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
L2150	Anti-Cancer Drug Library	3080 compounds
	A unique collection of 3080 anticancer drugs for high throughput screening (HTS) and high content screening (HCS);
L2120	Anti-Cancer Clinical Compound Library	2545 compounds
	A unique collection of 2545 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
L2100	Anti-Cancer Compound Library	7234 compounds
	A unique collection of 7234 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
L2110	Anti-Cancer Approved Drug Library	1779 compounds
	A unique collection of 1779 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
L8100	Cell Cycle Compound Library	677 compounds
	A unique collection of 677 cell cycle related compounds for high throughput screening (HTS) and high content screening (HCS);
L2180	Anti-Cancer Compound Library Plus	1468 compounds
	Well-chosen 1468 anti-tumor compounds with unique structures;
L9000	Apoptosis Compound Library	1760 compounds
	A unique collection of 1760 apoptosis-related compounds for apoptosis research, research in tumorigenesis, and anti-cancer drug screening;
L5300	Mitochondria-Targeted Compound Library	812 compounds
	A unique collection of 812 promising or approved mitochondria-targeted compounds including Idebenone, the only approved drug targeting mitochondria, for research in mitochondrial medicine;
L8500	HIF-1 Signaling Pathway Compound Library	1336 compounds
	A unique collection of 1336 HIF-1 related small chemicals can be used for drug discovery in ischemic disease and cancer and related mechanism studies；
L7110	Anti-Hypertension Compound Library	678 compounds
	678 hypertension-related small molecules for high-throughput and high-content screening.
L9410	Covalent Inhibitor Library	1920 compounds
	A unique collection of 1920 covalent Inhibitors and other molecules with common warheads like chloroacetyl，2-Chloropropionyl，Acryloyl，sulfonyl fluoride, alkyne，acrylamide, ketocarbonyl，disulfide bond, etc.