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カタログ番号	製品名	別名	ターゲット
T9988	Wnt/β-catenin agonist 3		Wnt/beta-catenin
	Wnt/β-catenin agonist 3 is a Wnt/beta-catenin agonist.		Wnt/beta-catenin
T2320	Indacaterol		Adrenergic Receptor
	Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.		Adrenergic Receptor
T13867	RH01386		Others
	RH01386 is a small molecule that can prevent ER stress-induced β cell dysfunction and death, and inhibits proapoptotic gene expression,has the potential for type 2 diabetes treatment. RH01386 restores ER stress-impaired ...		Others
T2161	Cardiogenol C		Wnt/beta-catenin
	Cardiogenol C is a cardiomyogenesis inducer in embryonic stem cells.		Wnt/beta-catenin
T3635	IQ 1	IQ1,IQ-1	Wnt/beta-catenin
	IQ 1 has multiple roles, such as maintaining the multifunctionality of mouse ESCs, decreasing Wnt-stimulated phosphorylation, blocking PP2A/Nkd interactions, and so on.		Wnt/beta-catenin
T10904	CWP232228		Wnt/beta-catenin
	CWP232228, a potent and selective Wnt / β-catenin signaling inhibitor, antagonizes the binding of β-catenin to T-cell factor (TCF) in the nucleus. CWP232228 inhibits the formation and metastasis of tumors by inhibiting t...		Wnt/beta-catenin
T16079	Mirodenafil	SK3530	PDE
	Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.		PDE
T9713	δ-secretase inhibitor 11		Beta Amyloid , Caspase
	δ-secretase inhibitor 11 is an inhibitor of δ-secretase and can be used as a lead compound for translational development of AD treatment.		Beta Amyloid , Caspase
T8730	BMS986260		TGF-beta/Smad
	BMS-986260 is a selective, and orally bioavailable TGFβR1 inhibitor(IC50 = 1.6 nM).		TGF-beta/Smad
T8233	BRD3308		Apoptosis , HIV Protease , HDAC
	BRD3308 is a highly selective inhibitor of HDAC3(IC50 of 54 nM), attenuating PE-mediated phosphorylation of ERK but not JNK.		Apoptosis , HIV Protease , HDAC
T11571	HLY78	4-Ethyl-5-methyl-5,6-dihydro-[1,3]dioxolo[4,5-j]phenanthridine	Wnt/beta-catenin
	HLY78 (4-Ethyl-5-methyl-5,6-dihydro-[1,3]dioxolo[4,5-j]phenanthridine) targets the DIX domain of Axin, is an activator of the Wnt/β-catenin signaling pathway and can enhance Axin-LRP6 binding to promote Wnt signaling.		Wnt/beta-catenin
T3100	GSK-J4	GSK J4 HCl	Apoptosis , Histone Demethylase
	GSK-J4 (GSK J4 HCl) is a potent H3K27me3 demethylase inhibitor, with IC50s of 8.6 μM and 6.6 μM towards KDM6B and KDM6A respectively. It is the first selective inhibitor of the H3K27 histone demethylase JMJD3 and UTX wit...		Apoptosis , Histone Demethylase
T1239	Indacaterol maleate	QAB149	Adrenergic Receptor
	Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.		Adrenergic Receptor
TQ0126	Mirodenafil dihydrochloride	SK-3530 dihydrochloride	PDE
	Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.		PDE
T8005	Cardiogenol C hydrochloride	Cardiogenol C HCl,Cardiogenol C	Wnt/beta-catenin
	Cardiogenol C hydrochloride (Cardiogenol C) can induces the differentiation of ESCs into cardiomyocytes (EC50= 100 nM).		Wnt/beta-catenin
T4383	GSK-J4 Hydrochloride	GSK J4 HCl,GSK J4 HCl (1373423-53-0 free base)	Histone Demethylase
	GSK-J4 Hydrochloride (GSK J4 HCl) is a cell permeable, potent and selective histone demethylase(JMJD3 )inhibitor. is an ethyl ester derivative of the GSK-J1 with an IC50 value greater than 50 μM in vitro.		Histone Demethylase
T21769L	β-Pompilidotoxin Acetate	β-Pompilidotoxin Acetate(216064-36-7 Free base)	Sodium Channel
	β-Pompilidotoxin Acetate is a wasp venom peptide. β-Pompilidotoxin Acetate can slow sodium channel inactivation and increase steady-state sodium current in cells.		Sodium Channel
T15677	KY1220		Wnt/beta-catenin
	KY1220 destabilizes both β-catenin and Ras by targeting the Wnt/β-catenin pathway. It has an IC50 of 2.1 μM in HEK293 reporter cells.		Wnt/beta-catenin
TP1382L	HAEGTFTSDVS acetate	HAEGTFTSDVS acetate(864915-61-7 free base)	Glucagon Receptor
	HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.		Glucagon Receptor
T3521	γ-Secretase-IN-1	Compound E	Beta Amyloid , Gamma-secretase
	γ-Secretase-IN-1 is a potent γ-secretase inhibitor that displays partial antiproliferative activity on T-47D cells and inhibits β-amyloid(40), β-amyloid(42), and Notch γ-secretase cleavage.		Beta Amyloid , Gamma-secretase
T4022	QS11	QS 11	GTPase
	QS11 is a GTPase activating protein of ADP-ribosylation factor 1 (ARFGAP1) inhibitor. Modulates ARF-GTP levels and synergizes with the Wnt/β-catenin signaling pathway to upregulate β-catenin nuclear translocation. Also r...		GTPase
T14284	β-Amyloid (25-35)	β-Amyloid peptide(25-35),Aβ25-35,Amyloid beta-peptide(25-35)	Beta Amyloid
	β-Amyloid (25-35) (Aβ25-35) is the fragment Aβ(25-35) of the Alzheimer's amyloid β-peptide. Which has shown neurotoxic activities in cultured cells.		Beta Amyloid
TP1263	Fz7-21	(Ac)-LPSDDLEFWCHVMY-NH2	Wnt/beta-catenin
	Fz7-21 ((Ac)-LPSDDLEFWCHVMY-NH2) is a peptide antagonist of FZD7 . It antagonises WNT3A-induced Wnt-β-catenin signalling in HEK293 expressing FZD7. Fz7-21 impairs Wnt/β-catenin signaling in HEK293 cells stimulated with e...		Wnt/beta-catenin
T14673	BMS 299897		Beta Amyloid , Gamma-secretase
	BMS 299897 is a sulfonamide γ-secretase inhibitor. It has an IC50 of 7 nM for Aβ production inhibition in HEK293 cells stably overexpressing amyloid precursor protein (APP).		Beta Amyloid , Gamma-secretase
T23446	TCS 2210		Others
	TCS 2210 is an inducer of neuronal differentiation in mesenchymal stem cells and increases the neuronal markers β-III tubulin expression and neuron-specific enolase expression.		Others
T11447	GNF4877		GSK-3 , DYRK
	GNF4877 is a potent DYRK1A and GSK3β inhibitor (IC50s: 6 nM and 16 nM). It leads to blockade of nuclear factor of activated T-cells (NFATc) nuclear export and increased β-cell proliferation cells.		GSK-3 , DYRK
TP1786L	Amyloid β-Protein 10-20 acetate	Amyloid β-Protein 10-20 acetate(152286-31-2 free base)	Beta Amyloid
	Amyloid β-Protein 10-20 acetate (Amyloid β-Protein 10-20 acetate (152286-31-2 free base)) is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.Amyloid β protein fragment containing the α...		Beta Amyloid
T8400	Pamidronic acid		Wnt/beta-catenin
	Pamidronic acid Leads to Bone Necrosis via Suppression of Wnt/β-Catenin Signaling in Human Bone Marrow Mesenchymal Stem Cells		Wnt/beta-catenin
T11784	KT182		MAGL
	KT182 is a selective and potent inhibitor of α/β-hydrolase domain containing 6 (ABHD6), with an IC50 of 0.24 nM in Neuro2A cells.		MAGL
T29857	Alethine	β-Alethine	TNF
	Alethine (β-Alethine) is a small molecule compound with antitumour activity and is used to treat tumours and infections. The alethine-induced up-regulation of TNFα increases the cytotoxicity of T cells.		TNF
T37450	SSK1		p38 MAPK
	SSK1 is a compound that selectively kills senescent cells and is a precursor for β-galactosidase, which can reduce the inflammatory response of the body. SSK1 can activate the phosphorylation of p38 MAPK and MKK3/MKK6 in...		p38 MAPK
T2310	CHIR-99021	Laduviglusib,CT99021,CHIR-99021	GSK-3 , Wnt/beta-catenin , Autophagy
	CHIR-99021 (CT99021) is an activator of the Wnt/β-catenin signaling pathway and a GSK-3α/β inhibitor (IC50=10/6.7 nM) with selective and oral activity.CHIR-99021 induces cellular autophagy, which enhances self-renewal in...		GSK-3 , Wnt/beta-catenin , Autophagy
TP1125	Insulin(cattle)	Insulin from bovine pancreas	IGF-1R
	Insulin bovine (Insulin from bovine pancreas) is a biologically derived two-chain polypeptide hormone, synthesized in vivo by pancreatic β cells. It is frequently utilized as a growth supplement in cell culture applicati...		IGF-1R
T21867	BI-6015		Others
	BI 6015 is an antagonist of HNF4α. HNF4α is a nuclear receptor that regulates gene expression in the intestine cells, liver cells, and pancreas-β cells.		Others
T14946	Ch55	Ch-55,CH 55,3,5-Di-tert-butylchalcone	Retinoid Receptor
	Ch55 (3,5-Di-tert-butylchalcone) is an effective inducer of the differentiation of HL60 cells (EC50 = 200 nM) and shows high affinity with RAR-α and RAR-β receptors. Ch55 can be used in studies about cancer.		Retinoid Receptor
T24897	TP0427736	TP427736,TP-0427736,TP-427736	TGF-beta/Smad
	TP-0427736 is a novel potent and selective ALK5 inhibitor (IC50: 2.72 nM). P0427736 was 300-fold higher than the inhibitory effect on ALK3. TP0427736 reduces TGF-β induced growth inhibition in human outer root sheath cel...		TGF-beta/Smad
T11048L	DIPQUO hydrochloride	DIPQUO hydrochloride(1269365-82-3 Free base)	Phosphorylase
	DIPQUO hydrochloride is an activator of the bone marker alkaline phosphatase (ALP), with an EC50 of 6.27 μM in C2C12 cells. DIPQUO hydrochloride promotes mouse and human osteoblast differentiation via activation of p38 M...		Phosphorylase
T73415	Miclxin	DS37262926	Wnt/beta-catenin
	Miclxin (DS37262926) is a novel MIC60 inhibitor that induces apoptosis through mitochondrial stress in mutant tumor cells via β-catenin.Miclxin is a potent inhibitor of mutant β-catenin, which is involved in the Wnt sign...		Wnt/beta-catenin
T26869	BMS-986122	BMS 986122	Opioid Receptor
	BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC5...		Opioid Receptor
T2106	WS6		EGFR , IκB/IKK
	WS6, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase pathway.		EGFR , IκB/IKK
T15429	GSK2194069		Others , NADPH , Fatty Acid Synthase
	GSK2194069 is an active β-keto reductase (KR)-specific inhibitor of fatty acid synthase (FASN) with an IC50 of 7.7 nM in an assay for the detection of released CoA.GSK2194069 inhibits the proliferation of FAS in cancer c...		Others , NADPH , Fatty Acid Synthase
T3984	GLP-1(7-36), amide	MKC 253,Human GLP-1-(7-36)-amide,Glucagon-like Peptide 1 (7-36) amide,Glucagon-Like Peptide (GLP) I (7-36), amide, human,GLP-1(7-36),GLP-1-(7-36)-amide	Glucagon Receptor
	GLP-1(7-36), amide (MKC 253) is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays various antidiabetic effects by potentiating glucose-...		Glucagon Receptor
T2055	WS3		EGFR , IκB/IKK
	WS3, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase pathway.		EGFR , IκB/IKK
T3162	IDE1		Others
	IDE1 can induce definitive endoderm from embryonic stem cells. It has been shown to induce the differentiation of Sox17+/FoxA2+-expressing pancreatic progenitors from human and mouse embryonic stems cells (EC50: 125.5 nM...		Others
T1726	SB-431542	SB 431542	ALK , TGF-beta/Smad
	SB-431542 is an inhibitor of ALK5/TGF-β type I Receptor (IC50=94 nM) and is selective. SB 431542 also has inhibitory activity against ALK4 and ALK7 but not other proteins. SB 431542 can be used for induced differentiatio...		ALK , TGF-beta/Smad
T10782	CGP52411	DAPH	EGFR , Beta Amyloid
	CGP52411 is an orally active, and ATP-competitive inhibitor of EGFR (IC50: 0.3 μM). CGP52411 blocks the toxic influx of Ca2+ ions into neuronal cells and dramatically inhibits and reverses the formation of β-amyloid Aβ42...		EGFR , Beta Amyloid
T77701	FL118	FL 118,FL-118,10,11-(Methylenedioxy)-20(S)-camptothecin	Survivin
	FL118 is a novel survivin inhibitor that inhibits cancer stem cell-like properties.FL118 is a novel camptothecin analog with anticancer activity that inhibits epithelial-mesenchymal transition through the Wnt/β-catenin s...		Survivin
T60485	DIF-3
	DIF-3 is a chemical compound that acts by activating GSK-3β to facilitate the degradation of cyclin D1 and c-Myc, resulting in reduced expression levels of these proteins. In addition, DIF-3 inhibits Wnt/β-catenin signal...
T3637	Pifithrin-β hydrobromide	Cyclic PFT-α,PFT-β,Cyclic Pifithrin-α hydrobromide,Pifithrin-β,PFT β (hydrobromide)	Ferroptosis , p53
	Pifithrin-β hydrobromide (Cyclic PFT-α) is an inhibitor of p53; reversibly blocks p53-dependent transcriptional activation and apoptosis. Protects against neuronal death in models of stroke and neurodegenerative disorder...		Ferroptosis , p53
T2310L	CHIR-99021 HCl	CT99021 HCl,Laduviglusib HCl	GSK-3
	CHIR-99021 HCl (Laduviglusib HCl) is a highly potent and selective inhibitor of GSK-3α/β, with IC50 values of 10 nM and 6.7 nM respectively. It demonstrates remarkable selectivity for GSK-3, with over 500-fold selectivit...		GSK-3

Compounds

Wnt/β-catenin agonist 3

T9988

Synonym:

Target: Wnt/beta-catenin

Indacaterol

T2320

Synonym:

Target: Adrenergic Receptor

Target: Wnt/beta-catenin

IQ 1

T3635

Synonym: IQ1,IQ-1

Target: Wnt/beta-catenin

CWP232228

T10904

Synonym:

Target: Wnt/beta-catenin

δ-secretase inhibitor 11

T9713

Synonym:

Target: Beta Amyloid, Caspase

BMS986260

T8730

Synonym:

Target: TGF-beta/Smad

BRD3308

T8233

Synonym:

Target: Apoptosis, HIV Protease, HDAC

HLY78

T11571

Synonym: 4-Ethyl-5-methyl-5,6-dihydro-[1,3]dioxolo[4,5-j]phenanthridine

Target: Wnt/beta-catenin

GSK-J4

T3100

Synonym: GSK J4 HCl

Target: Apoptosis, Histone Demethylase

Indacaterol maleate

T1239

Synonym: QAB149

Target: Adrenergic Receptor

Mirodenafil dihydrochloride

TQ0126

Synonym: SK-3530 dihydrochloride

Target: PDE

Cardiogenol C hydrochloride

T8005

Synonym: Cardiogenol C HCl,Cardiogenol C

Target: Wnt/beta-catenin

GSK-J4 Hydrochloride

T4383

Synonym: GSK J4 HCl,GSK J4 HCl (1373423-53-0 free base)

Target: Histone Demethylase

β-Pompilidotoxin Acetate

T21769L

Synonym: β-Pompilidotoxin Acetate(216064-36-7 Free base)

Target: Sodium Channel

KY1220

T15677

Synonym:

Target: Wnt/beta-catenin

HAEGTFTSDVS acetate

TP1382L

Synonym: HAEGTFTSDVS acetate(864915-61-7 free base)

Target: Glucagon Receptor

γ-Secretase-IN-1

T3521

Synonym: Compound E

Target: Beta Amyloid, Gamma-secretase

Synonym: β-Amyloid peptide(25-35),Aβ25-35,Amyloid beta-peptide(25-35)

Target: Beta Amyloid

Fz7-21

TP1263

Synonym: (Ac)-LPSDDLEFWCHVMY-NH2

Target: Wnt/beta-catenin

BMS 299897

T14673

Synonym:

Target: Beta Amyloid, Gamma-secretase

Amyloid β-Protein 10-20 acetate

TP1786L

Synonym: Amyloid β-Protein 10-20 acetate(152286-31-2 free base)

Target: Wnt/beta-catenin

Synonym: Laduviglusib,CT99021,CHIR-99021

Target: GSK-3, Wnt/beta-catenin, Autophagy

Insulin(cattle)

TP1125

Synonym: Insulin from bovine pancreas

Synonym: Ch-55,CH 55,3,5-Di-tert-butylchalcone

Target: Retinoid Receptor

TP0427736

T24897

Synonym: TP427736,TP-0427736,TP-427736

Target: TGF-beta/Smad

DIPQUO hydrochloride

T11048L

Synonym: DIPQUO hydrochloride(1269365-82-3 Free base)

Target: Phosphorylase

Miclxin

T73415

Synonym: DS37262926

Target: Wnt/beta-catenin

BMS-986122

T26869

Synonym: BMS 986122

Target: Opioid Receptor

WS6

T2106

Synonym:

Target: EGFR, IκB/IKK

GSK2194069

T15429

Synonym:

Target: Others, NADPH, Fatty Acid Synthase

GLP-1(7-36), amide

T3984

Synonym: MKC 253,Human GLP-1-(7-36)-amide,Glucagon-like Peptide 1 (7-36) amide,Glucagon-Like Peptide (GLP) I (7-36), amide, human,GLP-1(7-36),GLP-1-(7-36)-amide

Target: Glucagon Receptor

WS3

T2055

Synonym:

Target: EGFR, IκB/IKK

Target: ALK, TGF-beta/Smad

CGP52411

T10782

Synonym: DAPH

Target: EGFR, Beta Amyloid

FL118

T77701

Synonym: FL 118,FL-118,10,11-(Methylenedioxy)-20(S)-camptothecin

Pifithrin-β hydrobromide

T3637

Synonym: Cyclic PFT-α,PFT-β,Cyclic Pifithrin-α hydrobromide,Pifithrin-β,PFT β (hydrobromide)

Target: Ferroptosis, p53

CHIR-99021 HCl

T2310L

Synonym: CT99021 HCl,Laduviglusib HCl

Target: GSK-3

カタログ番号	製品名	別名	ターゲット
TN2190	Scoulerine		Apoptosis , Beta-Secretase , BACE , Parasite
	Scoulerine is an inhibitor of ß-site amyloid precursor protein cleaving enzyme 1(BACE1). Scoulerine a potent antimitotic compound that inhibits proliferation, arrests cell cycle, and induces apoptosis in cancer cells.		Apoptosis , Beta-Secretase , BACE , Parasite
T13475	β-Aminopropionitrile	3-Aminopropionitrile,BAPN	Others , Endogenous Metabolite
	β-Aminopropionitrile (3-Aminopropionitrile) is a selective inhibitor of lysyl oxidase.		Others , Endogenous Metabolite
TN7108	Urolithin C		Apoptosis , Calcium Channel , Reactive Oxygen Species , IGF-1R , Endogenous Metabolite
	Urolithin C is a gut metabolite of ellagic acid. Urolithin C induces apoptosis in PC12 cells through a mitochondria-mediated pathway.
T1048	Estradiol	E2,17β-Estradiol,17β-Oestradiol,β-Estradiol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	Estradiol (E2) is a naturally occurring steroidal sex hormone that is essential for female fertility and maintenance of secondary sexual characteristics. Estradiol upregulates IL-6 expression through estrogen receptor be...
T2882	Genistin	Genistoside,Genistein glucoside,Genistein 7-glucoside,Genistine,Genistein 7-O-β-D-glucopyranoside	Apoptosis , Estrogen Receptor/ERR , Others
	Genistin (Genistoside) is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-inflammatory and anticancer activities		Apoptosis , Estrogen Receptor/ERR , Others
TN1818	Kaempferol 3-O-β-D-glucuronide	Kaempferol-3-O-glucuronide,Kaempferol-3-beta-O-glucuronide,Kaempferol-3-glucuronide	IL Receptor
	Kaempferol 3-O-β-D-glucuronide (Kaempferol-3-beta-O-glucuronide)e has antioxidant activity. Flavonoid glucuronides can be deconjugated by microsomal α²-glucuronidase from various human cells.		IL Receptor
TN7036	N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide	(9Z,12Z,15Z)-N-[(3-Methoxyphenyl)methyl]-9,12,15-octadecatrienamide,Macamide Impurity 14	Wnt/beta-catenin
	N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide (Macamide Impurity 14) induces osteogenic differentiation and subsequent bone formation of mesenchymal stem cells by activating the canonical Wnt/β-catenin signaling pa...		Wnt/beta-catenin
T5703	β,β-Dimethylacrylalkannin		Others
	β,β-Dimethylacrylalkannin is a natural product isolated from Arnebia nobilis Reichb.f, increases collagen and involucrin content in skin cells.		Others
TMS0484	Episyringaresinol 4'-O-β-D-glncopyranoside	(-)-Syringaresinol 4-O-β-D-glucopyranosi	Others
	Episyringaresinol 4'-O-β-D-glncopyranoside ((-)-Syringaresinol 4-O-β-D-glucopyranosi) inhibits the proliferation of human promyelocytic HL-6 cells through G(1) arrest and induction of apoptosis, may be a potential chemot...		Others
TN2213	Imperialine 3-β-D-glucoside	Sipeimine-3-beta-D-glucoside	Others
	Imperialine 3-β-D-glucoside (Sipeimine-3-beta-D-glucoside) is a natural product. Imperialine 3-β-D-glucoside may exhibit anti-tumor properties against multi-drug resistant tumor cells.		Others
T2S0389	Emodin-1-O-β-D-glucopyranoside	Emodin-1-O-glucoside	Others
	1. Emodin-1-O-β-D-glucopyranoside (Emodin-1-O-glucoside) has neuroprotective and uncoupling activities, and that it may be the a new uncoupler of nNOS-PSD-95. 2. Emodin-1-O-β-D-glucopyranoside shows inhibitory effects on...		Others
TL0008	Gigantol		Wnt/beta-catenin , Glucosidase
	Gigantol is a novel inhibitor of the Wnt/β-catenin pathway. It inhibits Wnt/β-catenin signaling through downregulation of phosphorylated LRP6 and cytosolic β-catenin in breast cancer cells. Gigantol may be developed as a...		Wnt/beta-catenin , Glucosidase
T5646	Cinnamic acid	3-Phenylacrylic acid,β-Phenylacrylic acid	Endogenous Metabolite
	Cinnamic acid (β-Phenylacrylic acid) has potential use in cancer intervention,The concentration causing a 50% reduction of cell proliferation (IC50) ranged from 1 to 4.5 mM in glioblastoma, melanoma, prostate and lung ca...		Endogenous Metabolite
TN4368	Kaempferol-3,7-di-O-β-glucoside	Kaempferol 3,7-di-O-glucoside	Glucosidase , Amylase
	Kaempferol-3,7-di-O-β-glucoside (Kaempferol 3,7-diglucoside) is a flavonol from Morettia philaena, It can inhibit α-amylase, α-glucosidase and Acetylcholinesterase. Kaempferol-3, 7-di-o-β-Glucoside has neuroprotective ac...		Glucosidase , Amylase
T12581	Puerarin-4'-O-β-D-glucopyranoside	Puerarin4'-O-glucoside	Others
	Puerarin-4'-O-β-D-glucopyranoside (Puerarin4'-O-glucoside) is a natural product isolated from Pueraria lobata root having estrogenic activity and anti-proliferation in MCF-7 human breast carcinoma cells.		Others
T4956	Tetrahydroxystilbene-2-O-β-D-glucoside	tetrahydroxyl diphenylethylene-2-o-gluco,EH-201	Others
	Tetrahydroxystilbene-2-O-β-D-glucoside (EH-201) is a low MW inducer of erythropoietin. Tetrahydroxystilbene-2-O-β-D-glucoside induces expression of erythropoietin, PPAR-γ coactivator 1α (PGC-1α) and haemoglobin in astroc...		Others
T3S2344	β,β-Dimethylacrylshikonin	Dimethylacrylshikonin,β, β-Dimethylacrylshikonin	ERK , HIF/HIF Prolyl-Hydroxylase
	1. β,β-Dimethylacrylshikonin (Dimethylacrylshikonin) is a promising agent for developing an improved strategy for radiotherapy against tumors. (a) Injection of Dimethylacrylshikonin combined with IR treatment significant...		ERK , HIF/HIF Prolyl-Hydroxylase
T4869	D-Allose	β-D-Allopyranose,D-(+)-ALLOSE	Others , Endogenous Metabolite
	D-Allose (β-D-Allopyranose) is a rare naturally occurring monosaccharide known to exert anti-proliferative effects on cancer cells. The effects of D-Allose on the cellular membranes of hormone-refractory prostate cancer ...		Others , Endogenous Metabolite
T3769	Tenuifolin		Others , Beta-Secretase , AChE
	Tenuifolin has no inherent toxicity to either the transfected or wild type cells at the effective concentrations, it inhibits amyloid-β secretion in vitro.		Others , Beta-Secretase , AChE
T2820	Glycitin	Glycitein-7-β-O-glucoside,Glycitein 7-O-β-glucoside	Others , Influenza Virus , Antibacterial
	Glycitin (Glycitein 7-O-β-glucoside), a natural isoflavone isolated from legumes, can promote the proliferation of bone marrow stromal cells and osteoblasts and suppresses bone turnover.		Others , Influenza Virus , Antibacterial
T14854	Caerulomycin A	Cerulomycin,Caerulomycin	Antifungal
	Caerulomycin A (Caerulomycin) (Cerulomycin; Caerulomycin) is an antifungal compound. Which induces generation of T cells, enhances TGF-β-Smad3 protein signaling via suppressing interferon-γ-induced STAT1 signaling. Antif...		Antifungal
TN7052	Crocin III	Crocetin-mono-(β-D-gentiobiosyl)-ester	Others
	Crocin III (Crocetin-mono-(β-D-gentiobiosyl)-ester) is a crocin derived from saffron (Crocus sutivus L.). Crocins inhibit the cell growth of tumor cells and have anti-inflammatory activity.		Others
TL0007	Bisdemethoxycurcumin	Curcumin III,Didemethoxycurcumin	Epigenetic Reader Domain , Wnt/beta-catenin
	Bisdemethoxycurcumin (Curcumin III) is a natural demethoxy derivative of curcumin. It is a potent activator of macrophage phagocytosis, interacting with 1α, 25-dihydroxy vitamin D3 to stimulate amyloid-β clearance by mac...		Epigenetic Reader Domain , Wnt/beta-catenin
T2S0618	β-Elemonic Acid	3-oxo Tirucallic Acid,Beta-Elemonic acid,3-Oxotirucallenoic Acid,Elemadienonic Acid	Apoptosis , Reactive Oxygen Species , COX
	β-Elemonic Acid (3-Oxotirucallenoic Acid) exhibits anti-inflammatory effects. Beta-Elemonic acid inhibits proliferation by inducing hypoploid cells and cell apoptosis, the anticancer effects of beta-Elemonic acid are rel...		Apoptosis , Reactive Oxygen Species , COX
T4S1796	Heterophyllin B		PI3K
	Heterophyllin B effectively suppresses the adhesion and invasion of the human esophageal carcinoma cells by mediating the PI3K/AKT/β-catenin pathways and regulating the expression levels of adhesion- and invasion-associa...		PI3K
T0906	Salinomycin	Procoxacin	Wnt/beta-catenin , Antibacterial
	Salinomycin (Procoxacin), a polyether potassium ionophore antibiotic, specifically inhibits the growth of gram-positive bacteria. It acts as a potent inhibitor of Wnt/β-catenin signaling, blocking Wnt-induced LRP6 phosph...		Wnt/beta-catenin , Antibacterial
TP2167	β-CGRP, human acetate	β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate	CGRP Receptor
	β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor (CRLR) (IC50s: 1 nM and 300 nM for CRLR/RAMP1 and CRLR/RAMP...		CGRP Receptor
TN6694	5,6-Benzoflavone	β-Naphthoflavone,beta-NF	Antioxidant
	5,6-Benzoflavone (β-Naphthoflavone) is an exogenous ligand for the aryl hydrocarbon receptor, which disrupts zinc homeostasis in human hepatocellular carcinoma HepG2 cells. 5,6-Benzoflavone (β-Naphthoflavone) possesses a...		Antioxidant
TQ0216	Ercalcitriol	1α,25-Dihydroxy Vitamin D2	Others
	Ercalcitriol (1α,25-Dihydroxy Vitamin D2) is an active metabolite of vitamin D2. Ercalcitriol, as the physiological activated form of vitamin D, can strengthen immunity via regulation of cathelicidin antimicrobial peptid...		Others
T3391	Corosolic acid	Corsolic acid,2α-Hydroxyursolic acid,Glucosol,Colosolic acid,Colosic acid	FAK , Autophagy
	Corosolic acid (Colosic acid) contains anti-angiogenic activity that can suppress FAK signaling induced by angiopoietin-1. Corosolic acid exerts anticancer activities against HCC, colon, and colorectal Y cells, by induci...		FAK , Autophagy
T4915	β-Glycerophosphate disodium salt hydrate		Phosphatase , Endogenous Metabolite
	β-Glycerophosphate is a classical serine-threonine phosphatase inhibitor used in kinase reaction buffers. BGP is often used in combination with other phosphatase/protease inhibitors for broad spectrum inhibition. It func...		Phosphatase , Endogenous Metabolite
TWS1563	Incensole		Others
	1. Incensole has a protective or stimulating effect on β-cells of the rat pancreas, it also can increase the insulin secretion, which evidenced by a significant increase both in body weight and in liver glycogen.		Others
T7044	Norepinephrine	Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol	MMP , Endogenous Metabolite , Adrenergic Receptor , Autophagy
	Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression of vascular endothelial growth factor, matrix metalloprotei...
T3674	Hydroxysafflor yellow A	HSYA,Safflomin A	TGF-beta/Smad
	Hydroxysafflor yellow A (Safflomin A) inhibited adipogenesis by increasing HSL promoter activities. Hydroxysafflor yellow A can effectively protect the liver from long-term alcohol injury by enhancing antioxidant capacit...		TGF-beta/Smad
TN2100	Pratensein		Others , NF-κB
	Pratensein as a novel transcriptional up-regulator of scavenger receptor class B type I in HepG2 cells.		Others , NF-κB
T4S1943	Kirenol	Kirel	Wnt/beta-catenin
	1. Kirenol (Kirel) has anti-oxidant, anti-inflammatory, anti-allergic, and anti-arthritic activities. 2. Kirenol is effective against gram-positive bacteria. 3. Kirenol possesses antitumor action on human chronic myeloid...		Wnt/beta-catenin
T4S0998	Trifolirhizin		TNF , Tyrosinase
	Trifolirhizin exerts varying degrees of inhibition on tyrosinase-dependent melanin biosynthesis, and therefore, are candidates as skin-whitening agents.Trifolirhizin possesses potential anti-inflammatory and anti-cancer ...		TNF , Tyrosinase
T2O2707	D-(+)-Fucose		Others
	1. D-(+)-Fucose is a hexose deoxy sugar found on N-linked glycans that appears on the cell surface of mammalian and plant cells.		Others
T3803	Specnuezhenide	Nuzhenide,Nuezhenide	Others , NF-κB , Wnt/beta-catenin
	Specnuezhenide (Nuezhenide) significantly protects human neuroblastoma SH-SY5Y cells from 6-hydroxydopamine-induced neurotoxicity.Nuezhenide is the main inhibitory compound of fruits, it shows a clear inhibitory effect t...		Others , NF-κB , Wnt/beta-catenin
TN1721	Gypenoside L		ERK , p38 MAPK , Calcium Channel , NF-κB , ROS
	Gypenoside L inhibits autophagic flux and induces cell death in human esophageal cancer cells through endoplasm reticulum stress-mediated Ca2+ release. It also inhibit non-small cell lung carcinoma A549 cell inhibitory a...		ERK , p38 MAPK , Calcium Channel , NF-κB , ROS
T5S0106	Peimisine	Ebeiensine	RAAS , AChR
	1. Peimisine (Ebeiensine) can affect M-receptor, excit β-receptor, restrain the release of internal calcium, and promote to releaseing nitrogen monoxidum in order to relax tracheal smooth muscle and relieve asthma. 2. Pe...		RAAS , AChR
T4S0498	Glaucocalyxin A	Wangzaozin B,Leukamenin F	Apoptosis , Akt , Caspase , PI3K
	1. Glaucocalyxin A (Leukamenin F)-SBE-β-CD could be useful with a better solubility and sustained function in drug delivery. 2. Glaucocalyxin A activates caspase-3, decreases BAD phosphorylation, and reduces the expressi...		Apoptosis , Akt , Caspase , PI3K
T3S1553	Trans-Cinnamaldehyde	Cinnamaldehyde,Cinnamic aldehyde,Cinnamal,Phenylacrolein	COX , Endogenous Metabolite
	1. trans-Cinnamaldehyde (Phenylacrolein) exhibits excellent anti-inflammatory activities and antidepressant-like effects in stressed mid-aged rats as a COX-2 inhibitor. 2. Cinnamic aldehyde induces apoptosis of CML cells...		COX , Endogenous Metabolite
T6491	(-)-(S)-Equol	(−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	(-)-(S)-Equol (4',7-Dihydroxyisoflavan) is an orally bioavailable, non-steroidal estrogen naturally produced by the metabolism of the isoflavonoid daidzein by human intestinal microflora, with potential chemoprotective a...
T23645	Aeroplysinin 1	NSC170364,Aeroplysinin I,NSC 170364,NSC-170364
	Aeroplysinin I is an antibacterial compound from the sponge. It has cytotoxic activity against colon cancer cells by promoting β-catenin degradation.
T13756	Liquiritigenin-7-apiosylglucoside	Liquiritigenin-7-O-β-D-glucopyranosyl-(1→2)-β-D-apiofuranoside	Others
	Liquiritigenin-7-O-β-D-glucopyranosyl-(1→2)-β-D-apiofuranoside, a flavonoid extracted from Glycyrrhiza roots, exhibits lower cytotoxic effects on a variety of tumor and normal cells.		Others
T3S0205	β-Hederin	Beta-Hederin	Parasite
	1. β-Hederin has antileishmanial activity. 2. β-Hederin has apoptotic effect on breast cancer cells, it could be a promising candidate for chemotherapy of breast cancer.		Parasite
TN3129	5-Nonadecylresorcinol		Others
	5-Nonadecylresorcinol shows inhibitory effects on the release of β-hexosaminidase from RBL-2H3 cells.		Others
TN5187	Triptoquinone B		IL Receptor
	Triptoquinone B is a novel interleukin-1 inhibitor, shows extremely potent inhibitory activities against interleukin-lα and β releases for human peripheral mononticlear cells, it shows the significant immunosuppressive a...		IL Receptor
T83344	3-O-β-D-Glucopyranosyl(1→2)-[a-Lrhamnopyranosyl(1→3)]-β-D-glucopyranosyl 28-O-β-D-glucuronopyranoside
	3-O-β-D-Glucopyranosyl(1→2)-[α-L-rhamnopyranosyl(1→3)]-β-D-glucopyranosyl 28-O-β-D-glucuronopyranoside is a saponin compound extracted from Polaskia chichipe Backbg. It demonstrates an 84.2% inhibitory activity on melani...
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天然物製品

Scoulerine

TN2190

Synonym:

Target: Apoptosis, Beta-Secretase, BACE, Parasite

β-Aminopropionitrile

T13475

Synonym: 3-Aminopropionitrile,BAPN

Target: Others, Endogenous Metabolite

Urolithin C

TN7108

Synonym:

Target: Apoptosis, Calcium Channel, Reactive Oxygen Species, IGF-1R, Endogenous Metabolite

Estradiol

T1048

Synonym: E2,17β-Estradiol,17β-Oestradiol,β-Estradiol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite

Genistin

T2882

Synonym: Genistoside,Genistein glucoside,Genistein 7-glucoside,Genistine,Genistein 7-O-β-D-glucopyranoside

Target: Apoptosis, Estrogen Receptor/ERR, Others

Kaempferol 3-O-β-D-glucuronide

TN1818

Synonym: Kaempferol-3-O-glucuronide,Kaempferol-3-beta-O-glucuronide,Kaempferol-3-glucuronide

Target: IL Receptor

N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide

TN7036

Synonym: (9Z,12Z,15Z)-N-[(3-Methoxyphenyl)methyl]-9,12,15-octadecatrienamide,Macamide Impurity 14

Target: Wnt/beta-catenin

β,β-Dimethylacrylalkannin

T5703

Synonym:

Target: Others

Episyringaresinol 4'-O-β-D-glncopyranoside

TMS0484

Synonym: (-)-Syringaresinol 4-O-β-D-glucopyranosi

Target: Others

Imperialine 3-β-D-glucoside

TN2213

Synonym: Sipeimine-3-beta-D-glucoside

Target: Others

Emodin-1-O-β-D-glucopyranoside

T2S0389

Synonym: Emodin-1-O-glucoside

Target: Wnt/beta-catenin, Glucosidase

Cinnamic acid

T5646

Synonym: 3-Phenylacrylic acid,β-Phenylacrylic acid

Target: Endogenous Metabolite

Kaempferol-3,7-di-O-β-glucoside

TN4368

Synonym: Kaempferol 3,7-di-O-glucoside

Target: Glucosidase, Amylase

Puerarin-4'-O-β-D-glucopyranoside

T12581

Synonym: Puerarin4'-O-glucoside

Target: Others

Tetrahydroxystilbene-2-O-β-D-glucoside

T4956

Synonym: tetrahydroxyl diphenylethylene-2-o-gluco,EH-201

Target: Others

β,β-Dimethylacrylshikonin

T3S2344

Synonym: Dimethylacrylshikonin,β, β-Dimethylacrylshikonin

Target: ERK, HIF/HIF Prolyl-Hydroxylase

D-Allose

T4869

Synonym: β-D-Allopyranose,D-(+)-ALLOSE

Target: Others, Endogenous Metabolite

Tenuifolin

T3769

Synonym:

Target: Others, Beta-Secretase, AChE

Glycitin

T2820

Synonym: Glycitein-7-β-O-glucoside,Glycitein 7-O-β-glucoside

Target: Others, Influenza Virus, Antibacterial

Caerulomycin A

T14854

Synonym: Cerulomycin,Caerulomycin

Target: Antifungal

Crocin III

TN7052

Synonym: Crocetin-mono-(β-D-gentiobiosyl)-ester

Target: Others

Bisdemethoxycurcumin

TL0007

Synonym: Curcumin III,Didemethoxycurcumin

Target: Epigenetic Reader Domain, Wnt/beta-catenin

β-Elemonic Acid

T2S0618

Synonym: 3-oxo Tirucallic Acid,Beta-Elemonic acid,3-Oxotirucallenoic Acid,Elemadienonic Acid

Target: Apoptosis, Reactive Oxygen Species, COX

Target: Wnt/beta-catenin, Antibacterial

β-CGRP, human acetate

TP2167

Synonym: β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate

Target: CGRP Receptor

5,6-Benzoflavone

TN6694

Synonym: β-Naphthoflavone,beta-NF

Target: Antioxidant

Ercalcitriol

TQ0216

Synonym: 1α,25-Dihydroxy Vitamin D2

Target: Others

Corosolic acid

T3391

Synonym: Corsolic acid,2α-Hydroxyursolic acid,Glucosol,Colosolic acid,Colosic acid

Target: FAK, Autophagy

β-Glycerophosphate disodium salt hydrate

T4915

Synonym:

Target: Phosphatase, Endogenous Metabolite

Synonym: Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol

Target: MMP, Endogenous Metabolite, Adrenergic Receptor, Autophagy

Hydroxysafflor yellow A

T3674

Synonym: HSYA,Safflomin A

Target: TGF-beta/Smad

Pratensein

TN2100

Synonym:

Target: Others, NF-κB

Kirenol

T4S1943

Synonym: Kirel

Target: Wnt/beta-catenin

Trifolirhizin

T4S0998

Synonym:

Target: TNF, Tyrosinase

Synonym: Nuzhenide,Nuezhenide

Target: Others, NF-κB, Wnt/beta-catenin

Gypenoside L

TN1721

Synonym:

Target: ERK, p38 MAPK, Calcium Channel, NF-κB, ROS

Synonym: Wangzaozin B,Leukamenin F

Target: Apoptosis, Akt, Caspase, PI3K

trans-Cinnamaldehyde

T3S1553

Synonym: Cinnamaldehyde,Cinnamic aldehyde,Cinnamal,Phenylacrolein

Target: COX, Endogenous Metabolite

(-)-(S)-Equol

T6491

Synonym: (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite

Aeroplysinin 1

T23645

Synonym: NSC170364,Aeroplysinin I,NSC 170364,NSC-170364

Target:

Liquiritigenin-7-apiosylglucoside

T13756

Synonym: Liquiritigenin-7-O-β-D-glucopyranosyl-(1→2)-β-D-apiofuranoside

Target: Others

β-Hederin

T3S0205

Synonym: Beta-Hederin

Target: Parasite

5-Nonadecylresorcinol

3-O-β-D-Glucopyranosyl(1→2)-[a-Lrhamnopyranosyl(1→3)]-β-D-glucopyranosyl 28-O-β-D-glucuronopyranoside

T83344

Synonym:

Target:

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Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPJ-00261	TGF beta 2 Protein, Mouse/Rat, Recombinant	Mouse,Rat	HEK293 Cells
	Transforming growth factor beta 2 (TGF-β2) is a member of TGF-beta superfamily that shares a characteristic cysteine knot structure. Mice with TGF-β2 gene deletion show defects in development of cardiac, lung, craniofaci...
TMPJ-00249	TGF beta 1 Protein, Human, Recombinant (Avi), Biotinylated	Human	HEK293 Cells
	Transforming Growth Factor β-1 (TGFβ-1) is a secreted protein which belongs to the TGF-β family. TGFβ-1 is abundantly expressed in bone, articular cartilage and chondrocytes and is increased in osteoarthritis (OA). TGFβ-...
TMPJ-01099	IL-15RA Protein, Human, Recombinant (hFc, Human Cells)	Human	HEK293 Cells
	Interleukin 15 Receptor alpha (IL-15Rα) is a transmembrane glycoprotein that plays a pleiotropic role in immune development and function, including the positive maintenance of lymphocyte homeostasis. IL-15Rα chain can bi...
TMPJ-00651	CD155/PVR Protein, Human, Recombinant (aa 21-343, His)	Human	HEK293 Cells
	Poliovirus Receptor (PVR) is a 70 kDa type I transmembrane single-span glycoprotein that belongs to the nectin-like (Necl) family and was originally identified based on its ability to mediate the cell attachment and entr...
TMPJ-00542	TPSB2 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Tryptases are Trypsin-like Serine Proteases. β-Tryptases are the main isoenzymes in mast cells. Βtryptases form active tetramers with heparin proteoglycan. In the tetramer, the unique arrangement of the active sites faci...
TMPJ-01243	DEFB4 Protein, Human, Recombinant	Human	E. coli
	Defensins are cationic peptides. It is an important ingredient of the innate immune system. β-defensins are expressed on some leukocytes and epithelial surfaces. Four human β-Defensins have been identified to date: BD-1,...
TMPJ-01055	HBA1 Protein, Human, Recombinant (His)	Human	E. coli
	Hemoglobin subunit alpha 1 (HBA1), also known as α2β2, is a hetero-tetramer consisting of two α and two β subunits held together by non-covalent interactions. Each subunit contains a heme group with an iron atom in the F...
TMPJ-00003	DEFB1 Protein, Human, Recombinant	Human	E. coli
	β-Defensin 1 (DEFB1) is a member of the β-defensin family, which is highly expressed by epithelial cells. β-defensins are expressed as the C-terminal portion of precursors and are released by proteolytic cleavage of a si...
TMPJ-00572	Vasorin Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Vasorin is a Type I membrane protein, which is predominantly expressed in vascular smooth muscle cells in a developmentally regulated pattern. The expression level of Vasorin can be down regulated during vessel repair af...
TMPJ-00786	ITGB1 Protein, Human, Recombinant (aa 21-728, His)	Human	HEK293 Cells
	Integrin β-1 (ITGB1) belongs to the integrin β chain family. Integrin family members are membrane receptors involved in cell adhesion and recognition in a variety of processes including embryogenesis, hemostasis, tissue ...
TMPJ-00771	TGF beta 1 Protein, Mouse/Rat, Recombinant	Mouse,Rat	HEK293 Cells
	Transforming growth factor beta 1 (TGFβ1) is the prototype of a growing superfamily of peptide growth factors and plays a prominent role in a variety of cellular processes, including cell-cycle progression, cell differen...
TMPY-03058	SLITL2/VASN Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Vasorin is a typical type I membrane protein. It contains 1 EGF-like domain, 1 fibronectin type-III domain, 10 LRR (leucine-rich) repeats, 1 LRRCT domain and 1 LRRNT domain. Vasorin is predominantly expressed in vascular...
TMPK-00156	DKK1 N terminal Domain Protein, Human, Recombinant (hFc & Avi)	Human	HEK293 Cells
	Dickkopf-1 (Dkk1), the founding and best-studied member of the Dkk family, functions as an antagonist of canonical Wnt/β-catenin. Dkk1 is considered to play a broad role in a variety of biological processes. DKK1 N termi...
TMPK-00158	DKK1 N terminal Domain Protein, Human, Recombinant (hFc & Avi), Biotinylated	Human	HEK293 Cells
	Dickkopf-1 (Dkk1), the founding and best-studied member of the Dkk family, functions as an antagonist of canonical Wnt/β-catenin. Dkk1 is considered to play a broad role in a variety of biological processes. DKK1 N termi...
TMPK-00223	Ephrin B2/EFNB2 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Ephrin-B2 controls platelet-derived growth factor receptor β (PDGFRβ) distribution in the VSMC plasma membrane, endocytosis, and signaling in a fashion that is highly distinct from its role in the endothelium. Ephrin-B2 ...
TMPK-00157	DKK1 C terminal Domain Protein, Human, Recombinant (hFc & Avi), Biotinylated	Human	HEK293 Cells
	Dickkopf-1 (Dkk1), the founding and best-studied member of the Dkk family, functions as an antagonist of canonical Wnt/β-catenin. Dkk1 is considered to play a broad role in a variety of biological processes. DKK1 C termi...
TMPK-00155	DKK1 C terminal Domain Protein, Human, Recombinant (hFc & Avi)	Human	HEK293 Cells
	Dickkopf-1 (Dkk1), the founding and best-studied member of the Dkk family, functions as an antagonist of canonical Wnt/β-catenin. Dkk1 is considered to play a broad role in a variety of biological processes. DKK1 C termi...
TMPK-00925	Noggin/NOG Protein, Mouse, Recombinant	Mouse	HEK293 Cells
	Noggin is an antagonist of bone morphogenetic proteins (BMP), being indispensable for certain developmental events.Noggin expression positively correlated with EGFR expression in both GC cell line models and The Cancer G...
TMPJ-00792	DNA PolymeraseBeta Protein, Human, Recombinant (His)	Human	E. coli
	Human DNA polymerase β is constitutively expressed in cells. It fills in gaps in DNA that are formed following base excision repair. Repair polymerase that plays a key role in base-excision repair. Has 5'-deoxyribose-5-p...
TMPJ-00415	HGFR/c-Met Protein, Human, Recombinant (aa 25-932, His & Avi), Biotinylated	Human	HEK293 Cells
	Hepatocyte growth factor receptor (HGF R) is a glycosylated receptor tyrosine kinase that plays a central role in epithelial morphogenesis and cancer development. HGF R is synthesized as a single chain precursor which un...
TMPJ-00160	EMMPRIN/CD147 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Extracellular Matrix Metalloproteinase Inducer (EMMPRIN) belongs to the immunoglobulin superfamily, which has the homology to both the immunoglobulin V domain and MHC class II antigen β-chain. EMMPRIN is a transmembrane ...
TMPJ-01061	Nucleobindin-2 Protein, Human, Recombinant	Human	E. coli
	Nesfatin-1 is a metabolic polypeptide encoded in the N-terminal region of the precursor protein, Nucleobindin2 (NUCB2). Nesfatin-1 is a neuropeptide produced in the hypothalamus of mammals. It participates in the regulat...
TMPK-00926	Noggin/NOG Protein, Mouse, Recombinant (His & Flag)	Mouse	HEK293 Cells
	Noggin is an antagonist of bone morphogenetic proteins (BMP), being indispensable for certain developmental events.Noggin expression positively correlated with EGFR expression in both GC cell line models and The Cancer G...
TMPK-01065	SEZ6 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Seizure-related protein 6 (Sez6) contributes to chronic pain development as sez6 knockout mice show attenuated pain behaviours after peripheral nerve injury, compared with control mice. The type I transmembrane isoform o...
TMPK-00541	SEZ6 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Seizure-related protein 6 (Sez6) contributes to chronic pain development as sez6 knockout mice show attenuated pain behaviours after peripheral nerve injury, compared with control mice. The type I transmembrane isoform o...
TMPK-00998	SEZ6 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Seizure-related protein 6 (Sez6) contributes to chronic pain development as sez6 knockout mice show attenuated pain behaviours after peripheral nerve injury, compared with control mice. The type I transmembrane isoform o...
TMPK-00997	SEZ6 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Seizure-related protein 6 (Sez6) contributes to chronic pain development as sez6 knockout mice show attenuated pain behaviours after peripheral nerve injury, compared with control mice. The type I transmembrane isoform o...
TMPK-00996	SEZ6 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	Seizure-related protein 6 (Sez6) contributes to chronic pain development as sez6 knockout mice show attenuated pain behaviours after peripheral nerve injury, compared with control mice. The type I transmembrane isoform o...
TMPK-00329	TGFBR2 Protein, Human, Recombinant (mFc & Avi), Biotinylated	Human	HEK293 Cells
	The TGFBR2 gene provides instructions for making a protein called transforming growth factor-beta (TGF-β) receptor type 2. This receptor transmits signals from the cell surface into the cell through a process called sign...
TMPJ-00028	CCL2 Protein, Mouse, Recombinant	Mouse	E. coli
	C-C motif chemokine 2 (CCL2) is a member of the C-C or β chemokine family. Mouse CCL2 shares 82% amino acid (aa) identity with rat CCL2 over the entire sequence, and 58%, 56%, 55%, 53% and 53% aa identity with human, equ...
TMPK-01304	Kremen-2 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Kremen2 (Krm2) plays an important role in embryonic development, bone formation, and tumorigenesis as a crucial regulator of classical Wnt/β-catenin signaling pathway. Compared to para-cancerous tissues, Krm2 was signifi...
TMPK-01093	Kremen-2 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Kremen2 (Krm2) plays an important role in embryonic development, bone formation, and tumorigenesis as a crucial regulator of classical Wnt/β-catenin signaling pathway. Compared to para-cancerous tissues, Krm2 was signifi...
TMPK-01106	Kremen-2 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Kremen2 (Krm2) plays an important role in embryonic development, bone formation, and tumorigenesis as a crucial regulator of classical Wnt/β-catenin signaling pathway. Compared to para-cancerous tissues, Krm2 was signifi...
TMPJ-00457	OGG1 Protein, Human, Recombinant	Human	E. coli
	Human N-Glycosylase/DNA Lyase(OOG1) is a DNA repair enzyme, which belongs to the type-1 OGG1 family. OOG1 incises DNA at 8-oxoG residues, and excises 7,8-dihydro-8-oxoguanine and 2,6-diamino-4-hydroxy-5-N-methylformamido...
TMPJ-01234	IL-36 gamma Protein, Mouse, Recombinant	Mouse	E. coli
	Interleukin-36 gamma (IL-36γ) is a member of the interleukin 1 cytokine family that includes three closely related genes, IL-36α, β, and γ, formerly known as IL-1F6, F8, and F9 respectively. IL-36α has been detected in b...
TMPK-00328	TGFBR2 Protein, Human, Recombinant (mFc & Avi)	Human	HEK293 Cells
	The TGFBR2 gene provides instructions for making a protein called transforming growth factor-beta (TGF-β) receptor type 2. This receptor transmits signals from the cell surface into the cell through a process called sign...
TMPJ-00292	CD36 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Platelet Glycoprotein 4 (CD36) is an integral membrane glycoprotein that has multiple physiological functions. It is broadly expressed on a variety of cell types including microvascular endothelium, adipocytes, skeletal ...
TMPJ-00680	ANGPTL7 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Angiopoietin-like 7 (ANGPTL7) is a secreted glycoprotein that is structurally related to the angiopoietins. Members of this protein family contain an N-terminal coiled coil domain and a C-terminal fibrinogen-like domain....
TMPK-00499	HGFR/c-Met Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	c-Met, also called tyrosine-protein kinase Met or hepatocyte growth factor receptor (HGFR), is a protein that in humans is encoded by the MET gene.The protein possesses tyrosine kinase activity. The primary single chain ...
TMPK-00457	HGFR/c-Met Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	c-Met, also called tyrosine-protein kinase Met or hepatocyte growth factor receptor (HGFR), is a protein that in humans is encoded by the MET gene.The protein possesses tyrosine kinase activity. The primary single chain ...
TMPJ-00993	CCL5 Protein, Rat, Recombinant (E. coli, His)	Rat	E. coli
	C-C motif chemokine 5(CCL5) is a β-chemokine that plays a primary role in the inflammatory immune response by means of its ability to attract and activate leukocytes. CCL5 is secreted by many cell types at inflammatory s...
TMPJ-00933	PRDX5 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Peroxisomes are essential organelles that participate in multiple important metabolic processes, including the β-oxidation of fatty acids, plasmalogen synthesis, and the metabolism of reactive oxygen species (ROS). Perox...
TMPY-03627	CREB3L1 Protein, Human, Recombinant (aa 396-519, His)	Human	HEK293 Cells
	CREB3L1, also known as OASIS, is a cellular transcription factor synthesized as a membrane-bound precursor. It is a putative endoplasmic reticulum (ER) stress sensor in astrocytes with a mechanism of activation. OASIS mR...
TMPJ-00100	Artemin Protein, Human, Recombinant	Human	E. coli
	Human Artemin is a GDNF family ligand that is distantly related to the TGF-β superfamily of molecules. It is synthesized as a preproprotein, and contains a variable length pre-, or signal sequence, plus a 68 amino acid (...
TMPY-03861	Amelotin Protein, Human, Recombinant (mFc)	Human	HEK293 Cells
	Amelotin (AMTN) is a tooth enamel protein which is expressed in maturation-stage ameloblasts and also in the internal basal lamina of junctional epithelium, a unique epithelial structure attached to the tooth surface whi...
TMPJ-00304	ALK-1 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	Activin Receptor-Like Kinase 1 (ALK-1) is a type I cell-surface receptor for the TGF-β superfamily of ligands, which mediates signaling of BMP9 (bone morphogenetic protein) and BMP10. ALK1 signaling is necessary for angi...
TMPJ-00238	Lefty-A Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Left-right determination factor 2(LEFTY2) is a secreted protein which belongs to the TGF-beta family. Lefty was first identified in a screen for undifferentiated cell-specific cDNAs from the P19 mouse embryonal carcinoma...
TMPY-01052	R-Cadherin/CDH4 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	The cadherin superfamily is a large family that engage in both homo- and heterotypic, calcium-dependent, cell-cell adhesion events, and can be divided into at least four subfamilies based on the extracellular (EC) region...
TMPY-03341	ASF1B Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	The histone chaperone anti-silencing factor 1a (ASF1a) interacts with MDC1 and is recruited to sites of DSBs to facilitate the interaction of phospho-ATM with MDC1 and phosphorylation of MDC1, which are required for the ...
TMPY-00681	BMP-5 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Bone Morphogenetic Protein 5 (BMP-5) is a member of the structurally and functionally related bone morphogenetic proteins (BMPs) which constitute a novel subfamily of the transforming growth factor β (TGF-β) superfamily....
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TGF beta 2 Protein, Mouse/Rat, Recombinant

TMPJ-00261

Species: Mouse,Rat

Expression System: HEK293 Cells

TGF beta 1 Protein, Human, Recombinant (Avi), Biotinylated

TMPJ-00249

Species: Human

Expression System: HEK293 Cells

IL-15RA Protein, Human, Recombinant (hFc, Human Cells)

TMPJ-01099

Species: Human

Expression System: HEK293 Cells

CD155/PVR Protein, Human, Recombinant (aa 21-343, His)

TMPJ-00651

Species: Human

Expression System: HEK293 Cells

TPSB2 Protein, Human, Recombinant (His)

TMPJ-00542

Species: Human

Expression System: HEK293 Cells

DEFB4 Protein, Human, Recombinant

TMPJ-01243

Species: Human

Expression System: E. coli

HBA1 Protein, Human, Recombinant (His)

TMPJ-01055

Species: Human

Expression System: E. coli

DEFB1 Protein, Human, Recombinant

TMPJ-00003

Species: Human

Expression System: E. coli

Vasorin Protein, Human, Recombinant (His)

TMPJ-00572

Species: Human

Expression System: HEK293 Cells

ITGB1 Protein, Human, Recombinant (aa 21-728, His)

TMPJ-00786

Species: Human

Expression System: HEK293 Cells

TGF beta 1 Protein, Mouse/Rat, Recombinant

TMPJ-00771

Species: Mouse,Rat

Expression System: HEK293 Cells

SLITL2/VASN Protein, Human, Recombinant (His)

TMPY-03058

Species: Human

Expression System: HEK293 Cells

DKK1 N terminal Domain Protein, Human, Recombinant (hFc & Avi)

TMPK-00156

Species: Human

Expression System: HEK293 Cells

DKK1 N terminal Domain Protein, Human, Recombinant (hFc & Avi), Biotinylated

TMPK-00158

Species: Human

Expression System: HEK293 Cells

Ephrin B2/EFNB2 Protein, Human, Recombinant (hFc)

TMPK-00223

Species: Human

Expression System: HEK293 Cells

DKK1 C terminal Domain Protein, Human, Recombinant (hFc & Avi), Biotinylated

TMPK-00157

Species: Human

Expression System: HEK293 Cells

DKK1 C terminal Domain Protein, Human, Recombinant (hFc & Avi)

TMPK-00155

Species: Human

Expression System: HEK293 Cells

Noggin/NOG Protein, Mouse, Recombinant

TMPK-00925

Species: Mouse

Expression System: HEK293 Cells

DNA PolymeraseBeta Protein, Human, Recombinant (His)

TMPJ-00792

Species: Human

Expression System: E. coli

HGFR/c-Met Protein, Human, Recombinant (aa 25-932, His & Avi), Biotinylated

TMPJ-00415

Species: Human

Expression System: HEK293 Cells

EMMPRIN/CD147 Protein, Human, Recombinant (His)

TMPJ-00160

Species: Human

Expression System: HEK293 Cells

Nucleobindin-2 Protein, Human, Recombinant

TMPJ-01061

Species: Human

Expression System: E. coli

Noggin/NOG Protein, Mouse, Recombinant (His & Flag)

TMPK-00926

Species: Mouse

Expression System: HEK293 Cells

SEZ6 Protein, Mouse, Recombinant (His)

TMPK-01065

Species: Mouse

Expression System: HEK293 Cells

SEZ6 Protein, Cynomolgus, Recombinant (His)

TMPK-00541

Species: Cynomolgus

Expression System: HEK293 Cells

SEZ6 Protein, Human, Recombinant (His)

TMPK-00998

Species: Human

Expression System: HEK293 Cells

SEZ6 Protein, Human, Recombinant (hFc)

TMPK-00997

Species: Human

Expression System: HEK293 Cells

SEZ6 Protein, Human, Recombinant (His & Avi), Biotinylated

TMPK-00996

Species: Human

Expression System: HEK293 Cells

TGFBR2 Protein, Human, Recombinant (mFc & Avi), Biotinylated

TMPK-00329

Species: Human

Expression System: HEK293 Cells

CCL2 Protein, Mouse, Recombinant

TMPJ-00028

Species: Mouse

Expression System: E. coli

Kremen-2 Protein, Cynomolgus, Recombinant (His)

TMPK-01304

Species: Cynomolgus

Expression System: HEK293 Cells

Kremen-2 Protein, Mouse, Recombinant (His)

TMPK-01093

Species: Mouse

Expression System: HEK293 Cells

Kremen-2 Protein, Human, Recombinant (His)

TMPK-01106

Species: Human

Expression System: HEK293 Cells

OGG1 Protein, Human, Recombinant

TMPJ-00457

Species: Human

Expression System: E. coli

IL-36 gamma Protein, Mouse, Recombinant

TMPJ-01234

Species: Mouse

Expression System: E. coli

TGFBR2 Protein, Human, Recombinant (mFc & Avi)

TMPK-00328

Species: Human

Expression System: HEK293 Cells

CD36 Protein, Human, Recombinant (hFc)

TMPJ-00292

Species: Human

Expression System: HEK293 Cells

ANGPTL7 Protein, Human, Recombinant (His)

TMPJ-00680

Species: Human

Expression System: HEK293 Cells

HGFR/c-Met Protein, Cynomolgus, Recombinant (His)

TMPK-00499

Species: Cynomolgus

Expression System: HEK293 Cells

HGFR/c-Met Protein, Human, Recombinant (His & Avi)

TMPK-00457

Species: Human

Expression System: HEK293 Cells

CCL5 Protein, Rat, Recombinant (E. coli, His)

TMPJ-00993

Species: Rat

Expression System: E. coli

PRDX5 Protein, Human, Recombinant (His)

TMPJ-00933

Species: Human

Expression System: HEK293 Cells

CREB3L1 Protein, Human, Recombinant (aa 396-519, His)

TMPY-03627

Species: Human

Expression System: HEK293 Cells

Artemin Protein, Human, Recombinant

TMPJ-00100

Species: Human

Expression System: E. coli

Amelotin Protein, Human, Recombinant (mFc)

TMPY-03861

Species: Human

Expression System: HEK293 Cells

ALK-1 Protein, Mouse, Recombinant (hFc)

TMPJ-00304

Species: Mouse

Expression System: HEK293 Cells

Lefty-A Protein, Human, Recombinant (His)

TMPJ-00238

Species: Human

Expression System: HEK293 Cells

R-Cadherin/CDH4 Protein, Human, Recombinant (His)

TMPY-01052

Species: Human

Expression System: HEK293 Cells

ASF1B Protein, Human, Recombinant (His)

TMPY-03341

Species: Human

Expression System: Baculovirus Insect Cells

BMP-5 Protein, Human, Recombinant (hFc)

TMPY-00681

Species: Human

Expression System: HEK293 Cells

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カタログ番号	製品名
L4100	TGF-beta/Smad Compound Library	184 compounds
	A unique collection of 184 TGF-beta/Smad signaling targeted compounds for high throughput and high content screening;
L7900	Osteogenesis Compound Library	317 compounds
	A unique collection of 317 osteogenesis related compounds for high throughput and high content screening;
L7700	Neural Regeneration Compound Library	524 compounds
	A unique collection of 149 neuroregeneration related compounds for high throughput and high content screening;
L9840	Anti-Alzheimer's Disease Compound Library	986 compounds
	A unique collection of 986 compounds with anti-AD activities or acting on main drug targets of AD can be used for HTS and HCS.

ライブラリー

TGF-beta/Smad Compound Library

L4100

Compounds: 184

Osteogenesis Compound Library

L7900

Compounds: 317

Neural Regeneration Compound Library

L7700

Compounds: 524

Anti-Alzheimer's Disease Compound Library

L9840

Compounds: 986