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天然化合物

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同位体標識化合物

カタログ番号	製品名	別名	ターゲット
T35628	AN-7		Others
	α-Lipoic acid is a cyclic disulfide antioxidant that interconverts with its reduced dithiol form. It is an essential cofactor for decarboxylation reactions of the citric acid cycle and acts as a general antioxidant. AN-7...		Others
T39658	RMC-4630	SHP2-IN-7,RMC-4630	Phosphatase
	RMC-4630 (SHP2-IN-7) is an inhibitor of SHP2.		Phosphatase
T9752	3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile		Androgen Receptor
	3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.		Androgen Receptor
T25859	Necrostatin-7	Necrostatin 7,Necrostatin7,Nec 7,Nec-7,Nec7	Apoptosis
	Necrostatin-7 (Necrostatin 7) is an inhibitor of necrotic apoptosis with cardioprotective effects, inhibits RANK-NFATc1 signaling, and attenuates macrophage differentiation into osteoblasts.		Apoptosis
T9068	Cucurbit[7]uril		Others
	Cucurbit[7]uril is an emerging candidate for pharmaceutical excipients.Cucurbit[7]uril enhances photosensitization of porphyrins in Neuroblastoma cells		Others
T21588	Olomoucine		ERK , CDK
	Olomoucine is an ATP competitive inhibitor of Cdk2/cyclin A, Cdc2/CyclinB, CDK2/CyclinE, CDK5/p35, and ERK1/p44 MAP kinase with IC50s of 7, 7, 7, 3 and 25 µM, respectively. Olomoucine regulates cell cycle and exhibits an...		ERK , CDK
T81633	Nurr1 agonist 7		Others
	Nurr1 agonist 7 (compound 110) is an agonist targeting the Nurr1 receptor and exhibits an EC50 of 0.12 μM [1].		Others
T4140	IRAK4-IN-1		IRAK
	IRAK4-IN-1 is an interleukin-1 receptor associated kinase 4 (IRAK4) inhibitor with an IC50 of 7 nM.		IRAK
T67781	SD49-7	HNASH	Histone Demethylase
	SD49-7 is an inhibitor of histone lysine demethylase 4 (KDM4) with an IC50 of 0.19 µM.		Histone Demethylase
T26399	7-Methyl-6-mercaptopurine	7-Methyl-6-thiopurine,6-Mercapto-7-methylpurine	Others
	7-Methyl-6-mercaptopurine (7-Methyl-6-thiopurine) is an inhibitor of PRPP aminotransferase, inhibits IMP metabolism and prevents purine, DNA and RNA synthesis.		Others
T1364	7-Aminodeacetoxycephalosporanic acid	7-ADCA,Cephalexin Impurity B,Cefalexine EP IMpurity B,Deacetoxycephalosporanic Acid,7-Aminodesacetoxycephalosporanic acid	Antibiotic
	7-Aminodeacetoxycephalosporanic acid (Cefalexine EP IMpurity B) is used as an antibiotic.		Antibiotic
T15427	GSK2033		Liver X Receptor
	GSK2033 is an antagonist of LXR (pIC50s: 7 and 7.4 for LXRα or LXRβ, respectively).		Liver X Receptor
T9896	7-Methoxy-1-naphthylacetonitrile		Others
	7-Methoxy-1-naphthylacetonitrile is one of the impurities of agomelatine, an antidepressant.		Others
T9898	2-(7-Methoxy-1-naphthyl)ethylamine HCl		Others
	2-(7-Methoxy-1-naphthyl)ethylamine hydrochloride is the impurity of Agomelatine, an antidepressant.		Others
T14388	AZD 4017		Dehydrogenase
			Dehydrogenase
T10325	ANI-7		Chk
	ANI-7 is an activator of aryl hydrocarbon receptor (AhR) pathway. ANI-7 inhibits the growth of multiple cancer cells and potently and selectively inhibits the growth of MCF-7 breast cancer cells (GI50: 0.56 μM).		Chk
T11638	Ilorasertib hydrochloride	ABT-348 hydrochloride	Aurora Kinase
	Ilorasertib hydrochloride (ABT-348 hydrochloride) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora C, Aurora B, and Aurora A (IC50s: 1 nM, 7 nM, 120 nM). It also suppresses RET tyrosine kinase,...		Aurora Kinase
TQ0057	AVE 0991		Others
	AVE 0991, a nonpeptide analog of angiotensin-(1-7) [Ang-(1-7)], is an orally active Mas agonist with inhibitory effects on [125I]-Ang-(1-7) binding to bovine aortic endothelial cell membranes, and inhibits astrocyte-medi...		Others
T6846	Vesatolimod	GS-9620	Apoptosis , HCV Protease , HBV , TLR , HIV Protease
	Vesatolimod (GS-9620) is an effective and specific orally active agonist of Toll-like receptor 7.		Apoptosis , HCV Protease , HBV , TLR , HIV Protease
T9238	KI-7		Adenosine Receptor
	KI-7 is an adenosine A2B receptor positive allosteric modulator.		Adenosine Receptor
T77517	URAT1 inhibitor 7		OAT
	URAT1 inhibitor 7 is a novel and potent inhibitor of the human uric acid transporter protein URAT1 (IC50:12 nM).URAT1 inhibitor 7 inhibits CYP2C9 with an IC50 of 4.2 μM.URAT1 inhibitor 7 can be used to study hyperuricemi...		OAT
T23077L	Novokinin acetate	Novokinin acetate (358738-77-9 free base)	RAAS
	Novokinin acetate exhibited an affinity for the AT2 receptor with Ki of 7 nM, and its antihypertensive and vasorelaxing activities were blocked by PD123319, an AT2 receptor antagonist.		RAAS
T5887	7-Hydroxy-3,4-dihydro-2(1H)-quinolinone	3,4-Dihydro-7-hydroxy-2(1H)-quinolinone	MAO , Monoamine Oxidase
	7-Hydroxy-3,4-dihydro-2(1H)-quinolinone is a weak MAO-A inhibitor(with an IC50 of 183 μM) .		MAO , Monoamine Oxidase
TP1376	GLP-1(7-37) acetate(106612-94-6 free base)	GLP-1(7-37) acetate	Others , Glucagon Receptor
	Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.		Others , Glucagon Receptor
T10245	ACY-957	HDAC Inhibitor C001	HDAC
	ACY-957 (HDAC Inhibitor C001) is an orally active and selective inhibitor of HDAC1 and HDAC2 (IC50s: 7 nM, 18 nM, and 1300 nM against HDAC1/2/3) and shows no inhibition on HDAC4/5/6/7/8/9.		HDAC
T12642	(R)-Simurosertib	(R)-TAK-931	CDK
	(R)-Simurosertib ((R)-TAK-931) is an inhibitor of the ATP-competitive cell division cycle 7 (CDC7) kinase.		CDK
T4427	PF-06409577	PF 06409577	AMPK
	PF-06409577 is an effective, orally active, and specific allosteric activator of AMPK (EC50: 7 nM, for α1β1γ1).		AMPK
T67736	ALW-II-49-7		Ephrin Receptor
	ALW-II-49-7 is a selective and potent inhibitor of EphB2 kinase with an EC50 value of 40 nM in cell.		Ephrin Receptor
T13323	VU6012962		GluR
			GluR
T63896	BE1218		Liver X Receptor
	BE1218 is a liver X receptor (LXR) inverse agonist active on LXRα and LXRβ with an IC50 of 9 nM and 7 nM, respectively.		Liver X Receptor
T39669	TLR7/8/9-IN-1	TLR7/8/9-IN-1	TLR
	TLR7/8/9-IN-1 is a potent inhibitor of Toll-like receptors 7/8/9 (TLR7/8/9) with an IC50 of 43 nM.		TLR
T11850	LIN28 inhibitor LI71		Others
	LIN28 inhibitor LI71 is a potent and cell-permeable LIN28 inhibitor, which abolishes LIN28-mediated oligouridylation with an IC50 of 7 uM.		Others
T9541	CTB	Cholera Toxin B subunit	Epigenetic Reader Domain
	CTB (Cholera Toxin B subunit) is an activator of p300 histone acetyltransferase and induces apoptosis in MCF-7 cells.		Epigenetic Reader Domain
T17032	Telratolimod	MEDI9197,3M-052	TLR
	Telratolimod (MEDI9197) is a toll-like receptors 7/8 agonist. It has an antitumor activity.		TLR
T60155	PBRM1-BD2-IN-7		Epigenetic Reader Domain
	PBRM1-BD2-IN-7, a selective and cell-active inhibitor targeting the polybromo-1 (PBRM1) bromodomain, demonstrates inhibitory efficacy against PBRM1-BD2 with an IC50 value of 0.29 μM. This compound is utilized in cancer r...		Epigenetic Reader Domain
T8742	G5-7	JAK2 inhibitor G5-7	Apoptosis , JAK
	JAK2 inhibitor G5-7 (JAK2 inhibitor G5-7) is an orally active JAK2 inhibitor, selectively inhibits JAK2–mediated phosphorylation and activation of EGFR (Tyr1068) and STAT3 by binding to JAK2. G5-7 has the potential for g...		Apoptosis , JAK
T23910	Cosalane	NSC 658586,NSC-658586,NSC 640067	HIV Protease
	Cosalane (NSC 658586) is an HIV replication inhibitor, an inhibitor of chemokine receptor 7 (CCR7) signalling in humans and mice, with antiviral activity that blocks the binding of CCR7 to its natural ligands, CCL19 and ...		HIV Protease
T5490	AK-7		Sirtuin
	AK-7 is a brain-permeable SIRT2 inhibitor and to characterize its cholesterol-reducing properties in neuronal models with an IC50 of 15.5 μM.		Sirtuin
T15578	Indotecan	NSC-724998,LMP-400	Topoisomerase
	Indotecan (LMP-400) is an effective inhibitor of topoisomerase 1(Top1) (IC50: 300, 1200, 560 nM for P388, HCT116, MCF-7 cell lines, respectively).		Topoisomerase
T14364	AZ-Dyrk1B-33	3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine	DYRK
	AZ-Dyrk1B-33 (3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine) is a potent and selective Dyrk1B kinase inhibitor with an IC50 of 7 nM.		DYRK
T9565	OSBPL7-IN-1		Others
	OSBPL7-IN-1 is an orally active inhibitor of oxysterol binding protein like 7 (OSBPL7). OSBPL7-IN-1 promotes an increase of ABCA1 at the plasma membrane without affecting mRNA expression[1].		Others
T69567L	UCB7362 hydrochloride	UCB7362 hydrochloride(2610631-17-7 Free base),UCB7362 HCl	Parasite
	UCB7362 hydrochloride （UCB7362 HCl） is an orally active plasmepsin X (PMX) inhibitor (IC50: 7 nM) with antimalarial activity that inhibits parasite growth.		Parasite
T9897	7-Methoxy-1-naphthaleneacetic acid		Others
	7-Methoxy-1-naphthaleneacetic acid is an inhibitor of auxin action in plants. 7-Methoxy-1-naphthaleneacetic acid inhibits polar auxin transport and tropic responses associated with asymmetric auxin distribution in Arabid...		Others
T14673	BMS 299897		Beta Amyloid , Gamma-secretase
	BMS 299897 is a sulfonamide γ-secretase inhibitor. It has an IC50 of 7 nM for Aβ production inhibition in HEK293 cells stably overexpressing amyloid precursor protein (APP).		Beta Amyloid , Gamma-secretase
T9287	Hydroxychloroquine	2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol	SARS-CoV , TLR , Parasite , Autophagy
	Hydroxychloroquine (2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol) (HCQ) is an alkalinizing lysosomatropic drug that acts by inducing apoptosis of renal cancer cells in vitro and inhibiting TLR7/9. It i...		SARS-CoV , TLR , Parasite , Autophagy
T4426	CEP-40783	CEP 40783,RXDX-106	c-Met/HGFR , TAM Receptor
	CEP-40783 (RXDX-106) is an effective, specific and orally active AXL/c-Met inhibitor (IC50: 7/12 nM). It also inhibits MER and TYRO3 (IC50: 29/19 nM).		c-Met/HGFR , TAM Receptor
T0134	Imiquimod	R 837,IMQ,S-26308	SARS-CoV , TLR , Autophagy , HSV
	Imiquimod (R 837) is an immune response modifier that acts as a toll-like receptor 7 agonist.		SARS-CoV , TLR , Autophagy , HSV
TQ0059	Ilorasertib	ABT-348	VEGFR , FLT , c-RET , PDGFR , Aurora Kinase
	Ilorasertib (ABT-348) (ABT-348) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora A/Aurora B/Aurora C (IC50s: 120 nM/7 nM/1 nM). It also suppresses RET tyrosine kinase, PDGFRβ, and Flt1 (IC50s: ...		VEGFR , FLT , c-RET , PDGFR , Aurora Kinase
T9890	HIF1-IN-3	Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-	HIF
	HIF1-IN-3 (Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-) is an effective inhibitor of HIF-1 (EC50 = 0.9 μM) and can be used in anticancer studies.		HIF
T5860	CK-869		Microtubule Associated
	CK-869 is an Actin-Related Protein 2/3 (ARP2/3) complex inhibitor(IC50 of 7 μM),and is useful tools for the investigation of the Arp2/3 complex.		Microtubule Associated

Compounds

Synonym: SHP2-IN-7,RMC-4630

Target: Phosphatase

3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile

T9752

Synonym:

Target: Androgen Receptor

Necrostatin-7

T25859

Synonym: Necrostatin 7,Necrostatin7,Nec 7,Nec-7,Nec7

Target: Histone Demethylase

7-Methyl-6-mercaptopurine

T26399

Synonym: 7-Methyl-6-thiopurine,6-Mercapto-7-methylpurine

Target: Others

7-Aminodeacetoxycephalosporanic acid

T1364

Synonym: 7-ADCA,Cephalexin Impurity B,Cefalexine EP IMpurity B,Deacetoxycephalosporanic Acid,7-Aminodesacetoxycephalosporanic acid

Target: Liver X Receptor

7-Methoxy-1-naphthylacetonitrile

T9896

Synonym:

Target: Others

2-(7-Methoxy-1-naphthyl)ethylamine HCl

Target: Dehydrogenase

Ilorasertib hydrochloride

T11638

Synonym: ABT-348 hydrochloride

Target: Aurora Kinase

Target: Apoptosis, HCV Protease, HBV, TLR, HIV Protease

KI-7

T9238

Synonym:

Target: Adenosine Receptor

Synonym: Novokinin acetate (358738-77-9 free base)

Target: RAAS

7-Hydroxy-3,4-dihydro-2(1H)-quinolinone

T5887

Synonym: 3,4-Dihydro-7-hydroxy-2(1H)-quinolinone

Target: MAO, Monoamine Oxidase

GLP-1(7-37) acetate(106612-94-6 free base)

TP1376

Synonym: GLP-1(7-37) acetate

Target: Others, Glucagon Receptor

ACY-957

T10245

Synonym: HDAC Inhibitor C001

Target: Ephrin Receptor

Target: Liver X Receptor

TLR7/8/9-IN-1

T39669

Synonym: TLR7/8/9-IN-1

Synonym: Cholera Toxin B subunit

Target: Epigenetic Reader Domain

Telratolimod

T17032

Synonym: MEDI9197,3M-052

Target: Epigenetic Reader Domain

G5-7

T8742

Synonym: JAK2 inhibitor G5-7

Target: Apoptosis, JAK

Cosalane

T23910

Synonym: NSC 658586,NSC-658586,NSC 640067

Synonym: NSC-724998,LMP-400

Target: Topoisomerase

AZ-Dyrk1B-33

T14364

Synonym: 3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine

UCB7362 hydrochloride

T69567L

Synonym: UCB7362 hydrochloride(2610631-17-7 Free base),UCB7362 HCl

Target: Parasite

7-Methoxy-1-naphthaleneacetic acid

Target: Beta Amyloid, Gamma-secretase

Hydroxychloroquine

T9287

Synonym: 2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol

Target: SARS-CoV, TLR, Parasite, Autophagy

CEP-40783

T4426

Synonym: CEP 40783,RXDX-106

Target: c-Met/HGFR, TAM Receptor

Imiquimod

T0134

Synonym: R 837,IMQ,S-26308

Target: SARS-CoV, TLR, Autophagy, HSV

Ilorasertib

TQ0059

Synonym: ABT-348

Target: VEGFR, FLT, c-RET, PDGFR, Aurora Kinase

HIF1-IN-3

T9890

Synonym: Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-

Target: Microtubule Associated

カタログ番号	製品名	別名	ターゲット
T0543	7-Methylxanthine	Heteroxanthine,Heteroxanthin	Nucleoside Antimetabolite/Analog , Endogenous Metabolite , Adenosine Receptor
	7-Methylxanthine is a methyl derivative of xanthine, the purine component of human urinary calculi.7-Methylxanthine has an affinity for adenosine receptors.7-Methylxanthine is a methyl derivative of xanthine, the purine ...
T11047	DiosMetin 7-O-β-D-Glucuronide		Others , Antioxidant
	DiosMetin 7-O-β-D-Glucuronide is an antioxidant component found in lucerne.		Others , Antioxidant
T5S2207	7-O-Methylmangiferin		Others
	7-O-MethylMangiferin is an xanthone isolated from the rhizomes of Iris nigricans.		Others
T3388	Calycosin-7-O-β-D-glucoside	calycosin-7-O-beta-D-glucopyranoside,Calycosin-7-O-beta-D-glucoside	MMP , Reactive Oxygen Species
	Calycosin-7-O-β-D-glucoside (calycosin-7-O-beta-D-glucopyranoside) possesses a protective effect on rat hepatocytes, an inhibitory effect on COX-2 activity. Calycosin 7-O-β-D-glucoside has antimicrobial activity. Calycos...		MMP , Reactive Oxygen Species
T7327	7-Methoxyisoflavone		AMPK
	7-Methoxyisoflavone is an activator of adenosine monophosphate-activated protein kinase (AMPK).		AMPK
TN1621	Eriodictyol-7-O-glucoside		Nrf2
	Eriodictyol-7-O-glucoside is an Nrf2 activator conferring protection against Cisplatin-induced toxicity. Eriodictyol-7-O-glucoside is a flavonoid and a free radical scavenger with antioxidant activity in pistachio skin.		Nrf2
TN1333	7-O-Methylbiochanin A	4',7-Dimethoxy-5-hydroxyisoflavone
	7-O-Methylbiochanin A (4',7-Dimethoxy-5-hydroxyisoflavone) is an isoflavone derivative that can be isolated from the roots of Lotus polyphyllos and other plants of the water lily family.
T0989	7-Aminocephalosporanic acid	7-ACA	Others , HSP , Antibacterial , Antibiotic
	7-Aminocephalosporanic acid is an HSP90β inhibitor used in the synthesis of cephalosporin antibiotics and their intermediates.		Others , HSP , Antibacterial , Antibiotic
T3801	(Rac)-Byakangelicin	Bjacangelicin,Bjakangelicin,Biacangelicin,7H-Furo[3,2-g][1]benzopyran-7-one, 9-(2,3-dihydroxy-3-methylbutoxy)-4-methoxy-,Byakangelicin	Others
	(Rac)-Byakangelicin (7H-Furo[3,2-g][1]benzopyran-7-one, 9-(2,3-dihydroxy-3-methylbutoxy)-4-methoxy-) is an antineoplastic agent.		Others
T10191L	7-Chlorokynurenic acid	7-chloro-4-hydroxy-2-carboxyquinoline,7-CKA	GluR , NMDAR
	7-Chlorokynurenic acid (7-chloro-4-hydroxy-2-carboxyquinoline) is an effecitve and selective antagonist of NMDA receptor with IC50 of 0.56 μM for the glycine B coagonist site. 7-Chlorokynurenic acid inhibits the reuptake...		GluR , NMDAR
T3376	Cynaroside	Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,Luteolin 7-glucoside	Others , Influenza Virus , DNA/RNA Synthesis
	Cynaroside (Luteolin 7-O-Glucoside) is a flavone, a flavonoid-like chemical compound. It has an anti-oxidant effect, inhibiting lipid and protein oxidation.		Others , Influenza Virus , DNA/RNA Synthesis
T6S0270	Ononin	Formononetin 7-O-β-D-glucopyranoside,Formononetin glucoside,Ononoside,Formononetin 7-O-glucoside	Antibacterial
	1. Ononin (Formononetin 7-O-glucoside) can inhibit the growth of pathogen. 2. Ononin plays an important role in human nutrition as health promoting natural chemicals and are established to be the beneficial components.		Antibacterial
T12796	S-Dihydrodaidzein	(3S)-7-hydroxy-3-(4-hydroxyphenyl)-2,3-dihydrochromen-4-one	Others
	S-Dihydrodaidzein ((3S)-7-hydroxy-3-(4-hydroxyphenyl)-2,3-dihydrochromen-4-one) is an enantiomer of dihydrodaidzein which is involved in equol biosynthesis in a lactic acid bacterium, Lactococcus sp. strain.		Others
T75429	(±)-Liquiritigenin	(±)-4',7-Dihydroxyflavanone	Apoptosis , Calcium Channel
	(±)-Liquiritigenin ((±)-4',7-Dihydroxyflavanone), a flavonoid extracted from Angelica keiskei, inhibits the calcium-activated chloride channel TMEM16A.(±)-Liquiritigenin induces an increase in apoptosis and an enhancemen...		Apoptosis , Calcium Channel
T83321	4-Demethyldeoxypodophyllotoxin		Chk
	4-Demethyldeoxypodophyllotoxin, an aryl tetrahydronaphthalenyl lignan analog from the roots of Podophyllum peltatum, has anticancer activity and modulates the Chk-2 signaling pathway in MCF-7 breast cancer cells.		Chk
TN7041	(-)-Epipodophyllotoxin		Apoptosis
	(-)-Epipodophyllotoxin (2) is an antiproliferative agent against cancer cells with GI50s of 0.36 and 0.24 μM in HeLa cells and MCF-7 cells, respectively. (-)-Epipodophyllotoxin can inhibit mitotic spindle assembly in vit...		Apoptosis
T3798	Ziyuglycoside I	Gouguside 7,Ziyu-glycoside I,3-O-alpha-L-Arabinopyranosylpomolic acid beta-D-glucopyranosyl ester,Zigu-glucoside I,Kudinoside H	Apoptosis , Others
	Ziyuglycoside I (Gouguside 7) has anti-inflammatory activity, could be used as an active ingredient for cosmetics.		Apoptosis , Others
T0945	Cyclosporin A	Cyclosporine A,Ciclosporin,Cyclosporine	Phosphatase , Antibiotic , Complement System
	Cyclosporin A is a naturally occurring cyclic polypeptide that is the active metabolite of a fungus. Cyclosporin A is an immunosuppressant that binds to procyclins and inhibits calcineurin (IC50=7 nM).		Phosphatase , Antibiotic , Complement System
T8038	7-Ethoxy-4-Methylcoumarin		Others
	7-Ethoxy-4-Methylcoumarin is considered an inhibitor of enzymes in cells and has been used in studies of enzyme inhibition and has been used to study the effects of various drugs on the human body.		Others
T4S0094	Hydroxygenkwanin	Luteolin 7-methylether,7-O-Methylluteolin	Antioxidant
	1. Hydroxygenkwanin (Luteolin 7-methylether) possesses significant the antioxidative activity . 2. Hydroxygenkwanin has cytotoxicity, may be an effective natural product to treat glioma, and the combination of Apigenin a...		Antioxidant
T22308	Dimboa	2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one	Others , Antibacterial , Antibiotic , Antifungal
	Dimboa (2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one) is an antifungal compound used in crops.		Others , Antibacterial , Antibiotic , Antifungal
T2789	Scutellarin	Breviscapin,Breviscapinun,Breviscapine,Scutellarein-7-glucuronide	Akt , HIV Protease , STAT
	Scutellarin (Scutellarein-7-glucuronide), an active flavone isolated from Scutellaria baicalensis, can inhibit RANKL-mediated MAPK and NF-κB signaling pathway in osteoclasts, and down-regulate the STAT3/Girdin/Akt signal...		Akt , HIV Protease , STAT
T5724	Neogambogic acid	neo-gambogic acid	Apoptosis , Others , Antibacterial
	Neogambogic acid, an active ingredient in garcinia, can inhibit the growth of some solid tumors and result in an anticancer effect, it may be responsible for the inhibition of proliferation of human breast cancer cell li...		Apoptosis , Others , Antibacterial
T2205	Acefylline	Theophylline-7-acetic acid,Carboxymethyltheophylline,acetyloxytheophylline,Theophyllineacetic acid	TNF , PAD , PKA , HDAC , PDE , Adenosine Receptor
	Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist. It is combined with diphenhydramine in the pharmaceutical preparation Etanautine to help...		TNF , PAD , PKA , HDAC , PDE , Adenosine Receptor
T4519	Alisol A	Alisol-A	Autophagy
	Alisol A (Alisol-A) may be an autophagic inducer, it has anti-cancer activity, it presents inhibitory effects on cancer cell lines tested(HepG2, MDA-MB-231, and MCF-7 cells).		Autophagy
T3818	Fraxinol		Others , P450
	Fraxinol is a predicted metabolite generated by BioTransformer¹ that is produced by the metabolism of 5, 7-dimethoxy-2h-chromen-2-one. It is generated by cyp1a2, cyp2a6, cyp2b6, cyp2c9, cyp2c19, and cyp2e1 enzymes via an...		Others , P450
TN6985	Anhydronotoptol		NO Synthase
	Anhydronotoptol (4-{[(2E,5E)-3,7-dimethylocta-2,5,7-trien-1-yl]oxy}-7H-furo[3,2-g]chromen-7-one), a natural compound extracted from the umbelliferae plant Qiangwu, is a potent inhibitor of nitric oxide production, inhibi...		NO Synthase
TN1727	Helichrysetin		Apoptosis , HIV Protease
	Helichrysetin has mild anti-HIV-1 PR activity. Helichrysetin has great potentials for development as an anticancer agent, it has cytotoxic effect on four selected cancer cell lines, A549, MCF-7, Ca Ski, and HT-29.		Apoptosis , HIV Protease
T3363	Jervine	Iervin,11-Ketocyclopamine,Jerwiny	Hedgehog/Smoothened , Smo
	The biological activity of Jervine (Jerwiny) is mediated via its interaction with the 7 passes transmembrane protein Smoothened. Jervine binds with and inhibits smoothened, which is an integral part of the Hedgehog signa...		Hedgehog/Smoothened , Smo
T21165	Pellitorine	AI3-19560,Pellitorin	TRP/TRPV Channel
	Pellitorine (Pellitorin) is an extract of Tetradium daniellii, and acts as a TRPV1 antagonist.		TRP/TRPV Channel
T2S1865	Octyl gallate	Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8	Antioxidant , Influenza Virus , Reactive Oxygen Species , Antibacterial , Antifungal , HSV
	1. Octyl Gallate is an antioxidant approved by the US Food and Drug Administration (FDA) as a food additive. 2. Octyl Gallate has antimetastatic activity. 3. Octyl Gallate shows antimicrobial activity against H. pylori, ...
TJS0387	Desoxyrhaponticin	Deoxyrhapontin,Deoxyrhaponticin	Apoptosis , Fatty Acid Synthase
	1. Desoxyrhaponticin (Deoxyrhaponticin) is an agent that is potentially effective in controlling postprandial hyperglycemia in diabetes, the in vivo antidiabetic action of this compound can be explained, in part at least...		Apoptosis , Fatty Acid Synthase
T6491	(-)-(S)-Equol	(−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol	Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Endogenous Metabolite
	(-)-(S)-Equol (4',7-Dihydroxyisoflavan) is an orally bioavailable, non-steroidal estrogen naturally produced by the metabolism of the isoflavonoid daidzein by human intestinal microflora, with potential chemoprotective a...
TN1853	Lariciresinol		VEGFR , Antifection
	Lariciresinol is an enterolignan precursor, it possesses fungicidal activities by disrupting the fungal plasma membrane and therapeutic potential as a novel antifungal agent for the treatment of fungal infectious disease...		VEGFR , Antifection
TN3972	Epimedokoreanin B		Apoptosis , Others , Antibacterial
	Epimedokoreanin B (EKB), an isoprenylated flavonoid isolated from Korean Epimedium, exhibited anticancer activity in human non-small cell lung cancer (NSCLC) A549 and NCI-H292 cells.Epimedokoreanin B also possesses anti-...		Apoptosis , Others , Antibacterial
T4115	Auraptene	7-geranyloxycoumarin	MMP , BACE
	Auraptene is a coumarin derived from citrus plants that bears a geranyloxyl moiety at its C-7. It has anti-inflammatory, anti-carcinogenic, anti-bacterial, neuroprotective, and hepatoprotective activities. It inhibits le...		MMP , BACE
TN2254	Taccalonolide A		Apoptosis , Microtubule Associated
	Taccalonolide A is the first microtubule stabilizing agent to be discovered from a plant since identification of the mechanism of action of paclitaxel and it is the first natural product steroid identified to have these ...		Apoptosis , Microtubule Associated
T10990	Dehydrocorydaline chloride	13-Methylpalmatine chloride	BCL , PARP , p38 MAPK , Caspase , Parasite , Autophagy
	Dehydrocorydaline chloride (13-Methylpalmatine chloride) is an alkaloid with anti-inflammatory and anti-cancer activity. Can improve the activation of p38 MAPK.		BCL , PARP , p38 MAPK , Caspase , Parasite , Autophagy
T6S1684	8-Gingerol		Antioxidant , Antibacterial , TRP/TRPV Channel
	1. 8-Gingerol has antioxidant activity. 2. 8-Gingerol has antimycobacterial activity. 3. 8-Gingerol could be used as an effective skin-whitening agent. 4. 8-Gingerol shows antipyretic and anti-inflammation characteristic...		Antioxidant , Antibacterial , TRP/TRPV Channel
T3S1416	Decursin	Decursinol angelate,(+)-Decursin	Apoptosis , PKC
	1. Decursin (Decursinol angelate) is able to attenuate kainic acid-induced seizures and could have potential as an antiepileptic drug. 2. Decursin exhibits hepatoprotective effects , potentially by inhibiting the TGF-β1 ...		Apoptosis , PKC
T3S2344	β,β-Dimethylacrylshikonin	Dimethylacrylshikonin,β, β-Dimethylacrylshikonin	ERK , HIF/HIF Prolyl-Hydroxylase
	1. β,β-Dimethylacrylshikonin (Dimethylacrylshikonin) is a promising agent for developing an improved strategy for radiotherapy against tumors. (a) Injection of Dimethylacrylshikonin combined with IR treatment significant...		ERK , HIF/HIF Prolyl-Hydroxylase
T0486L	Irinotecan Hydrochloride	Camptothecin 11 hydrochloride,CPT-11 hydrochloride	Topoisomerase , Autophagy
	Irinotecan Hydrochloride (CPT-11 hydrochloride) is the hydrochloride salt of a semisynthetic derivative of camptothecin. Irinotecan, a prodrug, is converted to a biologically active metabolite 7-ethyl-10-hydroxy-camptoth...		Topoisomerase , Autophagy
T3S1612	Kuwanon G	Moracenin B,Kuwanone G	Phosphatase , Antibacterial , Bombesin Receptor , AChR , AChE , Glucosidase
	1. Kuwanon G (Moracenin B) as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective treatment for Type II diabetes mellitus. 2. Kuwanon G has a...
T3729	Ethyl gallate	Nipagallin A,Phyllemblin,gallic acid ethyl ester	MMP , NF-κB , Akt , Antibacterial
	Ethyl gallate (gallic acid ethyl ester) obviously decreases cell proliferation in MDA-MB-231 and MCF-7 cells in a dose- and time-dependent manner, exhibits cytotoxicity in a dose-dependent manner. Ethyl gallate can inhib...		MMP , NF-κB , Akt , Antibacterial
T3S2259	Methyl eugenol	4-allylveratrole,eugenyl methyl ether,O-methyleugenol,Eugenol Methyl ether	GABA Receptor
	1. Methyl eugenol (4-allylveratrole) is a natural constituent of the essential oils of a number of plants widely used in foodstuffs as flavouring agents, in view of the carcinogenic potential of ME, the need to check its...		GABA Receptor
T4S0797	Berberine	Berberin,Umbellatine	Reactive Oxygen Species , Topoisomerase , Endogenous Metabolite , Antibacterial , Antibiotic , Autophagy
	1. Berberine (Umbellatine) is a potent oral hypoglycemic agent with beneficial effects on lipid metabolism. 2. Berberine may as a broad-spectrum anti-microbial medicine, a complementary therapeutic agent for HIV/AIDS. 3....
T83061	Anti-inflammatory agent 29
	Compound 29 (Compound 7) is an anti-inflammatory agent that exhibits hepatoprotective activity [1].
TN4222	Homoeriodictyol 7-O-β-D-glucoside	Homoeriodictyol 7-O-glucoside	Others , Platelet aggregation
	Homoeriodictyol 7-O-β-D-glucoside (Homoeriodictyol 7-O-glucoside) is a natural product from Viscum coloratum(Kom.)Nakai. Homoeriodictyol 7-O-β-D-glucoside is an antagonist of platelet-activating factor (PAF).		Others , Platelet aggregation
T83240	7-O-Methyl-6-Prenylnaringenin
	7-O-Methyl-6-Prenylnaringenin, an active compound, can be isolated from Humulus lupulus [1].
T83228	9-O-Methylstecepharine
	9-O-Methylstecepharine (compound 7), an alkaloid present in Stephania cepharantha [1], is a naturally occurring compound.
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天然物製品

7-Methylxanthine

T0543

Synonym: Heteroxanthine,Heteroxanthin

Target: Nucleoside Antimetabolite/Analog, Endogenous Metabolite, Adenosine Receptor

DiosMetin 7-O-β-D-Glucuronide

T11047

Synonym:

Target: Others, Antioxidant

Calycosin-7-O-β-D-glucoside

T3388

Synonym: calycosin-7-O-beta-D-glucopyranoside,Calycosin-7-O-beta-D-glucoside

Target: MMP, Reactive Oxygen Species

Eriodictyol-7-O-glucoside

TN1621

Synonym:

Target: Nrf2

7-O-Methylbiochanin A

TN1333

Synonym: 4',7-Dimethoxy-5-hydroxyisoflavone

Target:

7-Aminocephalosporanic acid

T0989

Synonym: 7-ACA

Target: Others, HSP, Antibacterial, Antibiotic

(Rac)-Byakangelicin

T3801

Synonym: Bjacangelicin,Bjakangelicin,Biacangelicin,7H-Furo[3,2-g][1]benzopyran-7-one, 9-(2,3-dihydroxy-3-methylbutoxy)-4-methoxy-,Byakangelicin

Target: Others

7-Chlorokynurenic acid

T10191L

Synonym: 7-chloro-4-hydroxy-2-carboxyquinoline,7-CKA

Target: GluR, NMDAR

Cynaroside

T3376

Synonym: Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,Luteolin 7-glucoside

Target: Others, Influenza Virus, DNA/RNA Synthesis

Ononin

T6S0270

Synonym: Formononetin 7-O-β-D-glucopyranoside,Formononetin glucoside,Ononoside,Formononetin 7-O-glucoside

Target: Antibacterial

S-Dihydrodaidzein

T12796

Synonym: (3S)-7-hydroxy-3-(4-hydroxyphenyl)-2,3-dihydrochromen-4-one

Target: Others

(±)-Liquiritigenin

T75429

Synonym: (±)-4',7-Dihydroxyflavanone

Target: Apoptosis, Calcium Channel

4-Demethyldeoxypodophyllotoxin

T83321

Synonym:

Target: Chk

(-)-Epipodophyllotoxin

Synonym: Gouguside 7,Ziyu-glycoside I,3-O-alpha-L-Arabinopyranosylpomolic acid beta-D-glucopyranosyl ester,Zigu-glucoside I,Kudinoside H

Target: Apoptosis, Others

Cyclosporin A

T0945

Synonym: Cyclosporine A,Ciclosporin,Cyclosporine

Target: Phosphatase, Antibiotic, Complement System

7-Ethoxy-4-Methylcoumarin

Synonym: Luteolin 7-methylether,7-O-Methylluteolin

Target: Antioxidant

Dimboa

T22308

Synonym: 2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one

Target: Others, Antibacterial, Antibiotic, Antifungal

Scutellarin

T2789

Synonym: Breviscapin,Breviscapinun,Breviscapine,Scutellarein-7-glucuronide

Target: Akt, HIV Protease, STAT

Neogambogic acid

T5724

Synonym: neo-gambogic acid

Target: Apoptosis, Others, Antibacterial

Acefylline

T2205

Synonym: Theophylline-7-acetic acid,Carboxymethyltheophylline,acetyloxytheophylline,Theophyllineacetic acid

Target: TNF, PAD, PKA, HDAC, PDE, Adenosine Receptor

Target: Apoptosis, HIV Protease

Jervine

T3363

Synonym: Iervin,11-Ketocyclopamine,Jerwiny

Target: Hedgehog/Smoothened, Smo

Pellitorine

T21165

Synonym: AI3-19560,Pellitorin

Target: TRP/TRPV Channel

Octyl gallate

T2S1865

Synonym: Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8

Target: Antioxidant, Influenza Virus, Reactive Oxygen Species, Antibacterial, Antifungal, HSV

Desoxyrhaponticin

TJS0387

Synonym: Deoxyrhapontin,Deoxyrhaponticin

Target: Apoptosis, Fatty Acid Synthase

(-)-(S)-Equol

T6491

Synonym: (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite

Lariciresinol

TN1853

Synonym:

Target: VEGFR, Antifection

Epimedokoreanin B

TN3972

Synonym:

Target: Apoptosis, Others, Antibacterial

Auraptene

T4115

Synonym: 7-geranyloxycoumarin

Target: Apoptosis, Microtubule Associated

Dehydrocorydaline chloride

T10990

Synonym: 13-Methylpalmatine chloride

Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy

8-Gingerol

T6S1684

Synonym:

Target: Antioxidant, Antibacterial, TRP/TRPV Channel

Decursin

T3S1416

Synonym: Decursinol angelate,(+)-Decursin

Target: Apoptosis, PKC

β,β-Dimethylacrylshikonin

T3S2344

Synonym: Dimethylacrylshikonin,β, β-Dimethylacrylshikonin

Target: ERK, HIF/HIF Prolyl-Hydroxylase

Irinotecan Hydrochloride

T0486L

Synonym: Camptothecin 11 hydrochloride,CPT-11 hydrochloride

Target: Topoisomerase, Autophagy

kuwanon G

T3S1612

Synonym: Moracenin B,Kuwanone G

Target: Phosphatase, Antibacterial, Bombesin Receptor, AChR, AChE, Glucosidase

Ethyl gallate

T3729

Synonym: Nipagallin A,Phyllemblin,gallic acid ethyl ester

Target: MMP, NF-κB, Akt, Antibacterial

Methyl eugenol

T3S2259

Synonym: 4-allylveratrole,eugenyl methyl ether,O-methyleugenol,Eugenol Methyl ether

Target: GABA Receptor

Berberine

T4S0797

Synonym: Berberin,Umbellatine

Target: Reactive Oxygen Species, Topoisomerase, Endogenous Metabolite, Antibacterial, Antibiotic, Autophagy

Anti-inflammatory agent 29

T83061

Synonym:

Target:

Homoeriodictyol 7-O-β-D-glucoside

TN4222

Synonym: Homoeriodictyol 7-O-glucoside

Target: Others, Platelet aggregation

7-O-Methyl-6-Prenylnaringenin

T83240

Synonym:

Target:

9-O-Methylstecepharine

T83228

Synonym:

Target:

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Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-00365	GALNT7 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	GalNAc-transferase-7 (GALNT7) is essential for the regulation of cell proliferation and has been implicated in tumorigenesis. Colorectal cancer (CRC) arises in a multistep molecular network process, which is from either ...
TMPY-06036	FGFR1 Protein, Human, Recombinant (alpha (IIIb), His)	Human	HEK293 Cells
	FGFR1 Protein, Human, Recombinant (alpha (IIIb), His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40.5 kDa and the accession number is P11362-7.
TMPK-00394	FGFR1 beta (IIIc) Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	Fibroblast growth factor receptor 1 (FGFR1) transmits signals through the plasma membrane regulating essential cellular processes like division, motility, metabolism, and death. Overexpression of FGFR1 is observed in num...
TMPK-00392	FGFR1 beta (IIIc) Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	Fibroblast growth factor receptor 1 (FGFR1) transmits signals through the plasma membrane regulating essential cellular processes like division, motility, metabolism, and death. Overexpression of FGFR1 is observed in num...
TMPK-01331	TSLPR Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Thymic stromal lymphopoietin (TSLP) is an interleukin-7 (IL-7) like cytokine, which plays an important role in the regulation of immune responses to allergens. TSLP binds to a heterodimeric receptor complex composed of t...
TMPJ-01397	Siglec-7 Protein,Human,Recombinant(aa 19-353, His）	Human	HEK293 Cells
	Siglecs (sialic acid binding Ig-like lectins) are I-type (Ig-type) lectins belonging to the Ig superfamily. They are characterized by an N-terminal Ig-like V-type domain which mediates sialic acid binding, followed by va...
TMPY-03623	NKp80/KLRF1 Protein, Cynomolgus, Recombinant (hFc)	Cynomolgus	HEK293 Cells
	NKp80, also known as KLRF1, is an activating homodimeric C-type lectin-like receptor that is expressed on nearly all-natural killer cells and stimulates their cytotoxicity and cytokine release. NKp80 stimulates cytotoxic...
TMPH-00573	DAPA aminotransferase Protein, E. coli, Recombinant (His & Myc)	E. coli	E. coli
	Catalyzes the transfer of the alpha-amino group from S-adenosyl-L-methionine (SAM) to 7-keto-8-aminopelargonic acid (KAPA) to form 7,8-diaminopelargonic acid (DAPA). It is the only animotransferase known to utilize SAM a...
TMPJ-01289	TIMP-4 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Metalloproteinase inhibitor 4 is an enzyme that in humans is encoded by the TIMP4 gene, belongs to the protease inhibitor I35 (TIMP) family. The protein complexes with metalloproteinases (such as collagenases) and irreve...
TMPK-00953	CDH17 Domain 6-7 Protein, Human, Recombinant (mFc)	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPK-00949	CDH17 Domain 7 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPH-03434	BIO3 Protein, S. cerevisiae, Recombinant (His & Myc)	Saccharomyces cerevisiae	E. coli
	Catalyzes the transfer of the alpha-amino group from S-adenosyl-L-methionine (SAM) to 7-keto-8-aminopelargonic acid (KAPA) to form 7,8-diaminopelargonic acid (DAPA). It is the only aminotransferase known to utilize SAM a...
TMPK-00950	CDH17 Domain 6-7 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPJ-00703	Gankyrin Protein, Human, Recombinant	Human	E. coli
	Gankyrin is a multicatalytic proteinase oncoprotein consists of 7 ankyrin repeats. Gankyrin overexpressed in most hepatocellular carcinomas. Gankyrin is involved in theregulation of the phosphorylation of the retinoblast...
TMPJ-00692	GAS7 Protein, Human, Recombinant (His)	Human	E. coli
	Growth Arrest-Specific Protein 7 (GAS7) is expressed primarily in terminalaly differentiated brain cells and predominantly in mature cerebellar Purkinje neurons. GAS7 may play a role in neuronal development by promoting ...
TMPY-03614	PSME3 Protein, Human, Recombinant (His)	Human	E. coli
	PSME3, also known as PA28-gamma, is a subunit of proteasome. The 26S proteasome multicatalytic proteinase complex has a highly ordered structure composed of 2 complexes, a 2S core and a 19S regulator. The 2S core is comp...
TMPY-03612	PSME1 Protein, Human, Recombinant (His)	Human	E. coli
	PA28A, also known as PSME1, is a subunit of proteasome. The 26S proteasome multicatalytic proteinase complex has a highly ordered structure composed of 2 complexes, a 2S core and a 19S regulator. The 2S core is composed ...
TMPJ-00770	Granzyme B/GZMB Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Granzyme B(GZMB) contains 1 peptidase S1 domain and belongs to the peptidase S1 family. This enzyme is necessary for target cell lysis in cell-mediated immune responses. It cleaves after Asp and seems to be linked to an...
TMPY-03610	PSME2 Protein, Human, Recombinant (His)	Human	E. coli
	PSME2, also known as PA28b, is a subunit of proteasome. The 26S proteasome multicatalytic proteinase complex has a highly ordered structure composed of 2 complexes, a 2S core and a 19S regulator. The 2S core is composed ...
TMPK-00951	CDH17 Domain 5-7 Protein (Primary Amine Labeling), Human, Recombinant (His), Biotinylated	Human	HEK293 Cells
	Liver-intestine cadherin (CDH17) has been known to function as a tumor stimulator and diagnostic marker for almost two decades.In vivo studies showed CDH17 knockout resulted in apoptotic PC tumor death through activating...
TMPY-02800	CGB7 Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	CGB7 (chorionic gonadotropin, beta polypeptide 7) belongs to the glycoprotein hormones subunit beta family. Glycoprotein hormones are heterodimers consisting of a common alpha subunit and an unique beta subunit which con...
TMPY-02802	GNG13 Protein, Human, Recombinant (His)	Human	E. coli
	GNG13 is a subunit of heterotrimeric G proteins which consist of alpha, beta, and gamma subunits. Heterotrimeric G proteins are membrane-bound GTPases that are linked to 7-TM receptors. They function as signal transducer...
TMPK-00296	LILRA1/LIR-6/CD85i Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	LILRA1, also known as CD85i and LIR-6, is an approximately 70 kDa variably glycosylated transmembrane protein that regulates immune cell activation. Mature human LILRA1 consists of a 445 amino acid (aa) extracellular dom...
TMPK-00297	LILRA1/LIR-6/CD85i Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	LILRA1, also known as CD85i and LIR-6, is an approximately 70 kDa variably glycosylated transmembrane protein that regulates immune cell activation. Mature human LILRA1 consists of a 445 amino acid (aa) extracellular dom...
TMPJ-00386	ACE2/ACEH Protein, Human, Recombinant (HEK293, His & Avi), Biotinylated	Human	HEK293 Cells
	Angiotensin-Converting Enzyme 2 (ACE-2) is an integral membrane protein and a zinc metalloprotease of the ACE family, the ACE family includes somatic and germinal ACE. ACE-2 cleaves angiotensins I and II as a carboxypept...
TMPJ-00507	EIF4E Protein, Human, Recombinant	Human	E. coli
	Eukaryotic translation initiation factor 4E is a 217 amino acids protein that belongs to the eukaryotic initiation factor 4E family. eIF4F is a multi-subunit complex, the composition of which varies with external and int...
TMPY-02805	GNGT1 Protein, Human, Recombinant (His)	Human	E. coli
	GNGT1 is a subunit of transducin. Heterotrimeric G proteins consist of alpha, beta, and gamma subunits. They are membrane-bound GTPases that are linked to 7-TM receptors. They function as signal transducers for the 7-tra...
TMPJ-00285	IL-7R alpha/CD127 Protein, Human, Recombinant (hFc & His)	Human	HEK293 Cells
	Interleukin 7 Receptor alpha (IL-7Rα), also known as CD127, is a 75 kDa hematopoietin receptor superfamily member that plays an important role in lymphocyte differentiation, proliferation, and survival. IL-7Rα is majorly...
TMPJ-00284	IL-7R alpha/CD127 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	Interleukin 7 Receptor alpha (IL-7Rα), also known as CD127, is a 75 kDa hematopoietin receptor superfamily member that plays an important role in lymphocyte differentiation, proliferation, and survival. IL-7Rα is majorly...
TMPJ-00824	Ig lambda constant 2 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Immunoglobulin lambda constant region is constant region of immunoglobulin light chains. Immunoglobulins, also known as antibodies, are membrane-bound or secreted glycoproteins produced by B lymphocytes. In the recogniti...
TMPJ-01166	IGFBP-7 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Insulin-like growth factor-binding protein 7(IGFBP-7) is a secreted glycosylated protein that contains three protein domain modules. IGFBP7 contains an N-terminal IGFBP domain, followed by a Kazal-type serine proteinase ...
TMPY-03417	ACBD7 Protein, Human, Recombinant (His)	Human	E. coli
	ACBD7, acyl-CoA-binding domain-containing protein 7, is a small (1 Kd) protein that contains 1 ACB (acyl-CoA-binding) domain. The ACB domain consists of four alpha-helices arranged in a bowl shape with a highly exposed ...
TMPJ-00585	Complement C8 gamma Protein, Human, Recombinant (His)	Human	E. coli
	Complement component C8 is a constituent of the membrane attack complex, C8 alpha, C8 beta and C8G. C8G is a secreted protein and comsists a disulfide-linked C8 alpha-gamma heterodimer and a non-covalently associated C8 ...
TMPY-03456	SRFBP1 Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	SRFBP1 contains 7 WD repeats and belongs to the WD repeat STRAP family. SRFBP1 may play a role in the cellular distribution of the SMN complex. The SMN complex plays an essential role in spliceosomal snRNP assembly in th...
TMPJ-00718	AIF Protein, Human, Recombinant (His)	Human	E. coli
	Apoptosis-Inducing Factor 1, Mitochondrial (AIFM1) is a flavoprotein essential for nuclear disassembly in apoptotic cells that is found in the mitochondrial intermembrane space in healthy cells. During apoptosis, it is t...
TMPJ-00760	CXCL7 Protein, Human, Recombinant	Human	E. coli
	Human Chemokine (C-X-C motif) Ligand 7 (CXCL7), also known as neutrophil activating peptide 2 (NAP-2), is a member of the CXC chemokines containing an ELR domain (Glu-Leu-Arg tripeptide motif). Similar to other ELR domai...
TMPJ-01294	SOST Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Sclerostin (SOST) is a member of the cerberus/DAN family, a group of secreted glycoproteins characterized by a cysteine-knot motif. Cerberus/DAN family members are putative BMP antagonists, and include Dan, Cerberus, Gre...
TMPY-02597	IL-37 Protein, Human, Recombinant	Human	E. coli
	Interleukin 1 family member 7, or interleukin 37 (IL1F7 / IL37 / IL-1H4) is a secretory protein belonging to the Interleukin 1 family. IL-1F7 was localized in human peripheral monocytic cells. It has been localized the e...
TMPY-04558	NEK7 Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	NIMA (never in mitosis gene a)-related kinase 7, NEK7 belongs to the NIMA subfamily, NEK Ser/Thr protein kinase family, protein kinase superfamily. NEKs (NIMA-related kinases) are mammalian serine/threonine (Ser/Thr) pro...
TMPJ-00680	ANGPTL7 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Angiopoietin-like 7 (ANGPTL7) is a secreted glycoprotein that is structurally related to the angiopoietins. Members of this protein family contain an N-terminal coiled coil domain and a C-terminal fibrinogen-like domain....
TMPH-00672	Metalloprotease stcE Protein, E. coli O157:H7, Recombinant (His)	E. coli	E. coli
	Virulence factor that contributes to intimate adherence of enterohemorrhagic E.coli (EHEC) O157:H7 to host cells. Is able to cleave the secreted human mucin 7 (MUC7) and the glycoprotein 340 (DMBT1/GP340). Also cleaves h...
TMPH-00789	Hamster polyomavirus (HaPyV) VP1 Protein (His & Myc)	HaPyV	E. coli
	Forms an icosahedral capsid with a T=7 symmetry and a 40 nm diameter. The capsid is composed of 72 pentamers linked to each other by disulfide bonds and associated with VP2 or VP3 proteins. Interacts with sialic acids on...
TMPK-01371	IGFBP-7 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	IGFBP-7, also known as Mac25/Angiomodulin (AGM), GFBP-rp1, tumor-derived adhesion factor (TAF) and prostacyclin-stimulating factor (PSF), is a secreted protein that contains three protein domain modules. Human IGFBP-rp1 ...
TMPH-01516	FCGRT Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Cell surface receptor that transfers passive humoral immunity from the mother to the newborn. Binds to the Fc region of monomeric immunoglobulin gamma and mediates its selective uptake from milk. IgG in the milk is bound...
TMPY-01824	Caspase-14 Protein, Human, Recombinant (His)	Human	E. coli
	Caspase 14 is a member of the caspase family. Caspases are a kind of cysteine proteinase consisting of a prodomain plus large and small catalytic subunits, that play a central role in cell apoptosis. Caspase 14 possesses...
TMPY-01948	COQ7 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Ubiquinone biosynthesis protein COQ7 homolog, also known as Coenzyme Q biosynthesis protein 7 homolog, Timing protein clk-1 homolog and COQ7, is a mitochondrion inner membrane and peripheral membrane protein which bel...
TMPH-01517	FCGRT Protein, Human, Recombinant (GST)	Human	E. coli
	Cell surface receptor that transfers passive humoral immunity from the mother to the newborn. Binds to the Fc region of monomeric immunoglobulin gamma and mediates its selective uptake from milk. IgG in the milk is bound...
TMPJ-00685	BAI3 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Human Brain-Specific Angiogenesis Inhibitor 3 (BAI3) is a 177 kDa seven-span transmembrane (TM) protein, which is thought to be a member of the secretin receptor family. It is synthesized by neurons of the CNS and likely...
TMPK-00828	Mucin-1/MUC1 Isoform Y Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	MUC1, the transmembrane glycoprotein Mucin 1, is usually found to be overexpressed in a variety of epithelial cancers playing an important role in disease progression. MUC1 isoforms such as MUC1/Y, which lacks the entire...
TMPK-00395	FGFR1 alpha (IIIc) Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	FGFR1 alpha (IIIc) Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 42 kDa and the accession number is P11362-7.
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GALNT7 Protein, Human, Recombinant (His)

TMPY-00365

Species: Human

Expression System: HEK293 Cells

FGFR1 Protein, Human, Recombinant (alpha (IIIb), His)

TMPY-06036

Species: Human

Expression System: HEK293 Cells

FGFR1 beta (IIIc) Protein, Human, Recombinant (His & Avi), Biotinylated

TMPK-00394

Species: Human

Expression System: HEK293 Cells

FGFR1 beta (IIIc) Protein, Human, Recombinant (His & Avi)

TMPK-00392

Species: Human

Expression System: HEK293 Cells

TSLPR Protein, Cynomolgus, Recombinant (His)

TMPK-01331

Species: Cynomolgus

Expression System: HEK293 Cells

Siglec-7 Protein,Human,Recombinant(aa 19-353, His）

TMPJ-01397

Species: Human

Expression System: HEK293 Cells

NKp80/KLRF1 Protein, Cynomolgus, Recombinant (hFc)

TMPY-03623

Species: Cynomolgus

Expression System: HEK293 Cells

DAPA aminotransferase Protein, E. coli, Recombinant (His & Myc)

TMPH-00573

Species: E. coli

Expression System: E. coli

TIMP-4 Protein, Human, Recombinant (His)

TMPJ-01289

Species: Human

Expression System: HEK293 Cells

CDH17 Domain 6-7 Protein, Human, Recombinant (mFc)

TMPK-00953

Species: Human

Expression System: HEK293 Cells

CDH17 Domain 7 Protein, Human, Recombinant (hFc)

TMPK-00949

Species: Human

Expression System: HEK293 Cells

BIO3 Protein, S. cerevisiae, Recombinant (His & Myc)

TMPH-03434

Species: Saccharomyces cerevisiae

Expression System: E. coli

CDH17 Domain 6-7 Protein, Human, Recombinant (hFc)

TMPK-00950

Species: Human

Expression System: HEK293 Cells

Gankyrin Protein, Human, Recombinant

TMPJ-00703

Species: Human

Expression System: E. coli

GAS7 Protein, Human, Recombinant (His)

TMPJ-00692

Species: Human

Expression System: E. coli

PSME3 Protein, Human, Recombinant (His)

TMPY-03614

Species: Human

Expression System: E. coli

PSME1 Protein, Human, Recombinant (His)

TMPY-03612

Species: Human

Expression System: E. coli

Granzyme B/GZMB Protein, Mouse, Recombinant (His)

TMPJ-00770

Species: Mouse

Expression System: HEK293 Cells

PSME2 Protein, Human, Recombinant (His)

TMPY-03610

Species: Human

Expression System: E. coli

CDH17 Domain 5-7 Protein (Primary Amine Labeling), Human, Recombinant (His), Biotinylated

TMPK-00951

Species: Human

Expression System: HEK293 Cells

CGB7 Protein, Human, Recombinant (His)

TMPY-02800

Species: Human

Expression System: Baculovirus Insect Cells

GNG13 Protein, Human, Recombinant (His)

TMPY-02802

Species: Human

Expression System: E. coli

LILRA1/LIR-6/CD85i Protein, Human, Recombinant (His & Avi)

TMPK-00296

Species: Human

Expression System: HEK293 Cells

LILRA1/LIR-6/CD85i Protein, Human, Recombinant (His & Avi), Biotinylated

TMPK-00297

Species: Human

Expression System: HEK293 Cells

ACE2/ACEH Protein, Human, Recombinant (HEK293, His & Avi), Biotinylated

TMPJ-00386

Species: Human

Expression System: HEK293 Cells

EIF4E Protein, Human, Recombinant

TMPJ-00507

Species: Human

Expression System: E. coli

GNGT1 Protein, Human, Recombinant (His)

TMPY-02805

Species: Human

Expression System: E. coli

IL-7R alpha/CD127 Protein, Human, Recombinant (hFc & His)

TMPJ-00285

Species: Human

Expression System: HEK293 Cells

IL-7R alpha/CD127 Protein, Mouse, Recombinant (hFc)

TMPJ-00284

Species: Mouse

Expression System: HEK293 Cells

Ig lambda constant 2 Protein, Human, Recombinant (His)

TMPJ-00824

Species: Human

Expression System: HEK293 Cells

IGFBP-7 Protein, Mouse, Recombinant (His)

TMPJ-01166

Species: Mouse

Expression System: HEK293 Cells

ACBD7 Protein, Human, Recombinant (His)

TMPY-03417

Species: Human

Expression System: E. coli

Complement C8 gamma Protein, Human, Recombinant (His)

TMPJ-00585

Species: Human

Expression System: E. coli

SRFBP1 Protein, Human, Recombinant (His & GST)

TMPY-03456

Species: Human

Expression System: Baculovirus Insect Cells

AIF Protein, Human, Recombinant (His)

TMPJ-00718

Species: Human

Expression System: E. coli

CXCL7 Protein, Human, Recombinant

TMPJ-00760

Species: Human

Expression System: E. coli

SOST Protein, Mouse, Recombinant (His)

TMPJ-01294

Species: Mouse

Expression System: HEK293 Cells

IL-37 Protein, Human, Recombinant

TMPY-02597

Species: Human

Expression System: E. coli

NEK7 Protein, Human, Recombinant (His & GST)

TMPY-04558

Species: Human

Expression System: Baculovirus Insect Cells

ANGPTL7 Protein, Human, Recombinant (His)

TMPJ-00680

Species: Human

Expression System: HEK293 Cells

Metalloprotease stcE Protein, E. coli O157:H7, Recombinant (His)

TMPH-00672

Species: E. coli

Expression System: E. coli

Hamster polyomavirus (HaPyV) VP1 Protein (His & Myc)

TMPH-00789

Species: HaPyV

Expression System: E. coli

IGFBP-7 Protein, Human, Recombinant (hFc)

TMPK-01371

Species: Human

Expression System: HEK293 Cells

FCGRT Protein, Human, Recombinant (His)

TMPH-01516

Species: Human

Expression System: HEK293 Cells

Caspase-14 Protein, Human, Recombinant (His)

TMPY-01824

Species: Human

Expression System: E. coli

COQ7 Protein, Human, Recombinant (His)

TMPY-01948

Species: Human

Expression System: HEK293 Cells

FCGRT Protein, Human, Recombinant (GST)

TMPH-01517

Species: Human

Expression System: E. coli

BAI3 Protein, Human, Recombinant (His)

TMPJ-00685

Species: Human

Expression System: HEK293 Cells

Mucin-1/MUC1 Isoform Y Protein, Human, Recombinant (hFc)

TMPK-00828

Species: Human

Expression System: HEK293 Cells

FGFR1 alpha (IIIc) Protein, Human, Recombinant (His & Avi), Biotinylated

TMPK-00395

Species: Human

Expression System: HEK293 Cells

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カタログ番号	製品名
L2800	Serotonin Receptor-Targeted Compound Library	268 compounds
	A unique collection of 268 compounds targeting serotonin receptors for high throughput screening and high content screening;
L2620	Anti-Neurodegenerative Disease Compound Library	2154 compounds
	A unique collection of 2154 compounds related to neurodegenerative diseases can be used for HTS or HCS；
L2192	Anti-Pancreatic Cancer Compound Library	2238 compounds
	A unique collection of 2238 pancreatic cancer related compounds can be used in HTS and HCS;
L6700	Anti-Tumor Natural Product Library	1772 compounds
	A unique collection of 1772 natural products with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);

ライブラリー

Serotonin Receptor-Targeted Compound Library

L2800

Compounds: 268

Anti-Neurodegenerative Disease Compound Library

L2620

Compounds: 2154

Anti-Pancreatic Cancer Compound Library

L2192

Compounds: 2238

Anti-Tumor Natural Product Library

L6700

Compounds: 1772

Isotope Products

カタログ番号	製品名	別名	ターゲット
T13235	Tyk2-IN-7		Others
	Tyk2-IN-7 is an inhibitor of TYK2 JH2, binds to the TYK2 JH2 domain (IC50: 0.00053 μM; Ki.app: 0.00007 μM).		Others
TMID-0022	Spironolactone-d3
	Spironolactone-d3 is a deuterated compound of Spironolactone. Spironolactone has a CAS number of 52-01-7. Spironolactone is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antago...
TMID-0015	Bendazac-d7
	Bendazac-d7 is a deuterated compound of Bendazac. Bendazac has a CAS number of 20187-55-7. Bendazac is an anticataract drug. It may act by preventing protein denaturation.
TMID-0021	Fruquintinib-d3
	Fruquintinib-d3 is a deuterated compound of Fruquintinib. Fruquintinib has a CAS number of 1194506-26-7. Fruquintinib is an orally available, small molecule inhibitor of vascular endothelial growth factor receptors (VEGF...
TMIH-0325	MefenaMic Acid-d4
	MefenaMic Acid-d4 is a deuterated compound of MefenaMic Acid. MefenaMic Acid has a CAS number of 61-68-7. Mefenamic acid is a non-steroidal anti-inflammatory agent with analgesic, anti-inflammatory, and antipyretic prope...
T73246	EZH2-IN-7
	EZH2-IN-7, a potent inhibitor of EZH2, addresses overexpression or mutations in the SET region (Y641F, Y641N, A687V, A677G point mutations) that cause an abnormal increase in H3K27me3, contributing to the proliferation o...
TMIH-0146	Chloroquine-d5
	Chloroquine-d5 is a deuterated compound of Chloroquine. Chloroquine has a CAS number of 54-05-7. Chloroquine is an autophagy and toll-like receptors (TLRs) inhibitor. Chloroquine is an antimalarial and anti-inflammatory ...
TMIH-0427	Perospirone hydrochloride-d8
	Perospirone hydrochloride-d8 is a deuterated compound of Perospirone hydrochloride. Perospirone hydrochloride has a CAS number of 129273-38-7. Perospirone hydrochloride is an atypical antipsychotic agent for the treatmen...
TMIH-0222	Esomeprazole sodium-d6
	Esomeprazole sodium-d6 is a deuterated compound of Esomeprazole sodium. Esomeprazole sodium has a CAS number of 161796-78-7. Esomeprazole Sodium is the S-isomer of omeprazole with selective and irreversible proton pump i...
TMIH-0109	Bempedoic acid-d4
	Bempedoic acid-d4 is a deuterated compound of Bempedoic acid. Bempedoic acid has a CAS number of 738606-46-7. ETC-1002, also known as ESP-55016 and Bempedoic acid, is an orally available, once-daily LDL-C lowering small ...
T71293	Nifuroxazide-d4
	Nifuroxazide-d4 is intended for use as an internal standard for the quantification of nifuroxazide by GC- or LC-MS. Nifuroxazide is a nitrofuran antibiotic. It is active against strains of the enteropathogenic bacteria C...
T35698	Octanoic Acid-13C
	Octanoic acid-13C is intended for use as an internal standard for the quantification of octanoic acid by GC- or LC-MS. Octanoic acid is a medium-chain saturated fatty acid. It has been found in Teleme cheeses made from g...
T35591	Guanfacine-13C,15N3	Guanfacine-13C,15N3
	Guanfacine-13C,15N3is intended for us as an internal standard for the quantification of guanfacine by GC- or LC-MS. Guanfacine is an α2-adrenergic receptor (α2-AR) agonist with Kivalues of 93, 1,380, and 3,890 nM for α2A...
T35791	Palmitic acid-13C
	Palmitic acid-13C is intended for use as an internal standard for the quantification of palmitic acid by GC- or LC-MS. Palmitic acid-13C contains 13C at the C2 position and has been used in the study of free fatty acid i...