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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T10432L | AZD-8529 mesylate | GluR | |
AZD-8529 mesylate is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: 285 nM). It shows no positive allosteric modulator responses at 20-25 M on the mGluR1, 3, 4, 5, 6, 7, and 8 ... | |||
T7099 | Gefarnate | Others | |
Gefarnate is a synthetic compound used for the treatment of gastric ulcers,and also used in the treatment of dry eye syndrome. | |||
T9806 | NVP-DKY709 | Others | |
NVP-DKY709 is a potent IKZF2 inhibitor for the treatment of cancers. | |||
T60099 | RBN013209 | CD38 | |
RBN013209 is a potent CD38 inhibitor. RBN013209 is useful in the treatment of cancer. | |||
T19379 | Ipsalazide | Autophagy | |
Ipsalazide is a novel salicylazosulfapyridine analog for the treatment of inflammatory bowel disease. | |||
T68128 | Picumast | Others | |
Picumast shows antiallergic activity and can be utilized in the treatment of asthma. Picumast may be used in the treatment of therapeutic allergic airway diseases. | |||
T28665 | Saviprazole | Hoe731,Hoe 731,Hoe-731 | Proton pump |
Saviprazole (Hoe-731), a proton pump inhibitor, is used potentially for treatment of gastric ulcer. | |||
T28226 | Octahydroaminoacridine succinate | Others | |
Octahydroaminoacridine succinate, an acetylcholinesterase inhibitor, is used potentially for the treatment of Alzheimer's disease. | |||
T0151 | Efloxate | Angorlisin | Adrenergic Receptor |
Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency. | |||
T25364L | Efegatran sulfate | LY294468 sulfate,GYKI-14766 sulfate,LY 294468 sulfate,LY-294468 sulfate | Thrombin |
Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders. | |||
T60014 | SHEN26 | Antiviral | |
SHEN26 has antiviral activity and can be used in research on the treatment of viral infections. | |||
T4549 | Tibolone | tibolonum,tibolona | Estrogen/progestogen Receptor |
Tibolone is an estrogen-like compound used for the treatment of the symptoms associated with menopausal transition (i.e., climacteric symptoms) and also for the treatment of osteoporosis. | |||
T4557 | Amylmetacresol | 5-Methyl-2-Pentylphenol | Others , HIV Protease |
Amylmetacresol (5-Methyl-2-Pentylphenol) is used in the treatment of sore throat or 'acute sore throat', pharyngitis, tonsillitis and laryngitis. As well as in the treatment of influenza A and SARS-CoV. | |||
T11220L | UK 227786 | hydrochloride(150452-18-9 Free base),1-[4-(1,3-Benzodioxol-5a-ylmethylamino)-6-chloroquinazolin-2-yl]piperidine-4-carboxylic acid;hydrochloride(150452-18-9 Free base),1-[4-(1,3-Benzodioxol-5a-ylmethylamino)-6-chloroquinazolin-2-yl]piperidine-4-carboxylic acid | PDE |
UK 227786 is an inhibitor of phosphodiesterase 5 (PDE5), used for treatment of prostatic diseases. | |||
T1383 | Bitoscanate | p-Phenylene diisothiocyanate,Biscomate,PDITC,1,4-Diisothiocyanatobenzene | Parasite |
Bitoscanate (PDITC) is used in the treatment of hookworms. | |||
T26524 | ABT-080 | VML530,VML-530,VML 530,ABT080 | Leukotriene Receptor |
ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma. | |||
T14551 | Bevenopran | CB-5945,ADL-5945 | Opioid Receptor |
Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction. | |||
T68119 | Ontazolast | BIRM-270 | LTR |
Ontazolast is a small molecule leukotriene B4 receptor (LTB4R) antagonist for the treatment of immune system disorders and respiratory diseases.Ontazolast is a candidate compound for the treatment of asthma. | |||
T27599 | Imiloxan | RS-21361,RS 21361,RS21361 | Adrenergic Receptor |
Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder. | |||
T90596 | Sivifene | Others | |
Sivifene is a antitumor agent. Sivifene can be used for research on the treatment of cutaneous metastases from cancer. | |||
T27087 | Cronidipine | LF 2.0254,LF-20254,LF20254,LF 20254 | Calcium Channel |
Cronidipine (LF 20254), a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia. | |||
T31668 | Eribaxaban | PD 348292,PD0348292,PD-0348292,PD-348292,PD 0348292,PD348292 | Factor Xa |
Eribaxaban (PD348292) is an orally available factor Xa inhibitor for the prevention and treatment of venous thromboembolism. | |||
T9852 | MUN36378 | Others | |
MUN36378 is a FTO inhibitor for treatment of leukemia. | |||
T11305 | Flurofamide | Others | |
Flurofamide is an effective bacterial urease inhibitor and has potential in the treatment of infected urinary calculi. | |||
T6390 | Anagrelide hydrochloride | BMY 26538-01,Anagrelide HCl,Agrylin,BL4162A | PDE |
Anagrelide hydrochloride (BL4162A) serves as a treatment for essential thrombocytosis. | |||
T77457 | Emicizumab | ACE 910,RO 5534262 | Others |
Emicizumab(ACE 910) is a humanized monoclonal antibody that bridges activated factor IX and activated factor X to mimic the function of activated factor VIII. Emicizumab is used for the prevention and treatment of hemoph... | |||
T16427 | Padsevonil | UCB-0942,UCB1415943-000 | GABA Receptor |
Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy. | |||
T6957 | PRT-060318 | P142-76,PRT318,PRT-060318 2HCl | Syk |
PRT-060318 (P142-76) is a novel selective inhibitor of the Syk tyrosine kinase, as an approach to HIT treatment. | |||
T35300 | Zeniplatin | Zeniplatinum | Others |
Zeniplatin (Zeniplatinum) is a new cisplatin complex with anticancer activity for the treatment of metastatic melanoma and kidney cancer. | |||
T0338 | Minaprine | Cantor,Minaprine dihydrochloride,Minaprina,Minaprinum | MAO , Dopamine Receptor , 5-HT Receptor , AChR , AChE , Monoamine Oxidase |
Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states. | |||
T27864 | LX-2931 | LX 3305,LX2931,LX-3305,ACB20034,LX 2931,LX3305 | S1P Receptor |
LX-2931(LX-3305) is a sphingosine-1-phosphate cleavage enzyme (S1P) inhibitor for the treatment of rheumatoid arthritis. | |||
T27845 | Losigamone | ADD-137022,AO33,AO 33,ADD 137022,AO-33,ADD137022;Losigamone | GABA Receptor |
Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures. | |||
T27865 | LX-6171 | LX6171 | Others |
LX-6171, a proline transporter (SLC6A7) inhibitor, is used potentially for the treatment of schizophrenia and Alzheimer's disease. | |||
T16106 | ML224 | NCGC00242364,ANTAG3 | TSH Receptor |
ML224 (NCGC00242364) is a TSHR antagonist for the treatment of Graves' orbital disease and Graves' hyperthyroidism. | |||
T39250 | Bevurogant | ROR | |
Bevurogant is an antagonist of RORγt receptor and can be used in studies about the treatment of chronic inflammatory diseases. | |||
T28686 | SB-237376 HCl | SB-237376 hydrochloride | Calcium Channel , Sodium Channel |
SB-237376 HCl (SB-237376 hydrochloride) is a calcium and potassium channel antagonist used in the treatment of cardiac arrhythmias. | |||
T0367 | Fluocinolone (Acetonide) | Fluocinolone acetonide,Flucort-N | Glucocorticoid Receptor |
Fluocinolone Acetonide (Flucort-N) is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, gel, lotion, or ointment. It has also been used topically in... | |||
T6469 | Dichlorphenamide | Diclofenamide,Daranide,Antidrasi | Carbonic Anhydrase |
Dichlorphenamide (Diclofenamide) is a carbonic anhydrase inhibitor that is used in the treatment of glaucoma. | |||
T7712L | Disomotide TFA 181477-43-0(free base) | Others | |
Disomotide TFA is an oligopeptide for the treatment of melanoma. | |||
T33386 | Milveterol HCl | Milveterol,GSK-159797,GSK 159797,GSK159797 | Adrenergic Receptor |
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD). | |||
T15253 | CCX354 | CCR1 antagonist 1,CCX-354,CCX 354 | CCR |
CCX354 (CCR1 antagonist 1) is a potent small molecule CCR1 antagonist with anti-inflammatory activity for the treatment of rheumatoid arthritis. | |||
T26526 | Abt-288 | ABT 288,ABT288 | Histamine Receptor |
ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia. | |||
T21060L | NPC 567 acetate | NPC 567 acetate(109333-26-8 Free base) | Bradykinin Receptor |
NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease. | |||
T34648 | Sinitrodil | ITF296,ITF-296,ITF 296 | Guanylate cyclase |
Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of myocardial ischemia and angina pectoris. | |||
T27932 | LY-2300559 | LY2300559 | GluR |
LY-2300559 is an agonist of metabotropic glutamate receptor 2 (mGluR2) and can be used in studies about the treatment of migraine. | |||
T77691 | Cyclopentyl phenyl ketone | Benzoylcyclopentane | Others |
Cyclopentyl phenyl ketone (Benzoylcyclopentane) is used for the prevention and treatment of traumatic stress. | |||
T1466 | Nadifloxacin | OPC7251 | Antibacterial , Antibiotic |
Nadifloxacin (OPC7251) has been used in trials studying the treatment of Acne Vulgaris. | |||
T22835 | H2L5186303 | ZINC33388081 | LPA Receptor |
H2L5186303 is an LPA2 antagonist and can be used in studies about asthma treatment. | |||
T13329L | Vofopitant dihydrochloride | GR 205171A,Vofopitant 2HCl | Neurokinin receptor |
Vofopitant dihydrochloride (GR 205171A) is an orally available, selective tachykinin NK1 receptor antagonist that inhibits [3H]SP binding to NK1 with pKi values of 9.5 and 10.6, respectively.Vofopitant dihydrochloride is... | |||
T19659 | Annaosanchun | YC6,YC-6,YC 6 | Others , AMPK |
Annaosanchun (YC-6) is potentially for the treatment of acute ischemic stroke (AIS). |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T4001 | Euxanthone | 1,7-Dihydroxyxanthone | Autophagy |
Euxanthone (1,7-Dihydroxyxanthone), an xanthone derivative extracted from the roots of Polygala tenuifolia Willd, has antitumour, neuroprotective and vasorelaxant activities, and attenuates Aβ1-42-induced oxidative stres... | |||
T3S0128 | Hydroprotopine | Others | |
Hydroprotopine, treatment for coronary heart disease and angina, and the treatment effect is remarkable. | |||
TWS1613 | Erioside | mulberroside B | Others |
Erioside (mulberroside B) can antitussive, antiasthmatic, hypoglycemic, anti-tumor, treatment of gout. | |||
T3501 | Colistimethate Sodium | Colistin-1,3,5,9-tetramethanesulfonic A acid | Others |
Colistin-1,3,5,9-tetramethanesulfonic A acid is used for the treatment of serious infections due to selected aerobic Gram-negative pathogens in patients with limited treatment options. | |||
T24403 | Folinic acid | HSDB 6544,Leucovorin | Endogenous Metabolite , Antifolate |
Folinic acid (Leucovorin) is a biofolic acid that can be used in the treatment of methotrexate, often in combination with Methotrexate (MTX) to reduce MTX-induced toxicity, and can be used as an adjuvant treatment for co... | |||
TN5031 | Sitostenone | Others | |
Sitostenone has antioxidation activity. Stigmasta-4-en-3-one(Sitostenone) can be used for the treatment of androgen-dependent diseases, especially for the treatment of benign prostatic hyperplasia. | |||
T3S0640 | Triolein | Glycerol trioleate,Glycerine Trioleate | MMP , Others , Endogenous Metabolite |
Glyceryl Trioleate has been investigated for the treatment of Adrenoleukodystrophy. | |||
T1382 | Griseofulvin | Fulvicin,Amudane,Grisactin | Apoptosis , Microtubule Associated , Antibiotic , Antifungal |
Griseofulvin (Fulvicin) is an antifungal agent used in the treatment of TINEA infections. | |||
T8304 | Anisodamine Hydrobromide | 6-Hydroxyhyoscyamine | Adrenergic Receptor , AChR |
Anisodamine Hydrobromide (6-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock. | |||
T1273 | Diacerein | Diacerhein,Fisiodar,Diacetylrhein | IL Receptor , Interleukin |
Diacerein (Fisiodar) is a prodrug which is metabolized to rhein. It is currently approved in France for the treatment of osteoarthritis although the use of diacerein is restricted due to the side effects including sevre ... | |||
T5S0802 | Palmatine | Berbericinine,Burasaine | Indoleamine 2,3-Dioxygenase (IDO) , AChR , AChE , Aurora Kinase |
1. Palmatine (Burasaine) is an inhibitor of dopamine generation. 2. Palmatine could potentially be developed for the treatment of flavivirus infections. 3. Palmatine has been used in the treatment of jaundice, dysentery,... | |||
T1134 | Clofoctol | Antibacterial , Antibiotic | |
Clofoctol is a bacteriostatic antibiotic with activity against Gram-positive bacteria, used in the treatment of upper and lower respiratory tract infections. | |||
T19687 | Phenylethyl isothiocyanate | JC 5411,JC5411,JC-5411 | HDAC |
Phenylethyl isothiocyanate (JC5411) is an HDAC inhibitor. It potentially for the treatment of benign prostatic hypertrophy. | |||
T7849 | Norspermine | Others | |
Norspermine is a polyamine analogue ,used in the treatment of non-small cell lung carcinoma and breast cancer. | |||
TN1803 | Isoscoparin | Antioxidant , TNF , NO Synthase , Fatty Acid Synthase | |
Isoscoparin is derived from Gentiana algida Pall with antioxidant and anti-adipogenic activities. Isoscoparin can be used in stuides about the prevention and treatment of obesity. | |||
T6401 | Azithromycin | Zithromax,CP 62993,XZ-450 | Others , Antibacterial , Antibiotic , Autophagy |
Azithromycin (CP 62993) is an antibiotic by inhibiting protein synthesis, used for the treatment of bacterial infections. | |||
TL0002 | Liquiritin apioside | Others | |
Liquiritin Apioside is one of the main active components in Suan-Zao-Ren decoction as a treatment for insomnia. | |||
T3820 | Iridin | Lridin | Others |
Iridin (Lridin) is major active ingredient of Iris dichotoma which could be used as the drug for pain, inflammation treatment | |||
TN1076 | Oleonuezhenide | Others | |
Oleonuezhenide is a natural product from Chinese formula Ligustrum lucidum, exerts neuroprotective effects and also considered as treatment of osteoporosis. | |||
TN1997 | Notoginsenoside FP2 | Others | |
Notoginsenoside FP2 is a natural product isolated from the fruit pedicels of Panax notoginseng and can be used in studies about the treatment of cardiovascular diseases. | |||
T4S0398 | Rosin | p38 MAPK | |
Rosin is a natural product,may have therapeutic potential for the treatment of inflammation | |||
T1680 | Tolazoline hydrochloride | Imidaline hydrochloride,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride) | Adrenergic Receptor |
Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn. | |||
T6460 | Cysteamine hydrochloride | 2-Mercaptoethylamine Hydrochloride,β-Mercaptoethylamine Hydrochloride,Thioethanolamine Hydrochloride,2-Aminoethanethiol Hydrochloride,Cysteamine HCl,Bekaptan | Apoptosis , Others , Reactive Oxygen Species , Endogenous Metabolite , Autophagy |
Cysteamine hydrochloride (Thioethanolamine Hydrochloride) is an agent for the treatment of nephropathic cystinosis and an antioxidant. | |||
T12139 | N-(3-Methoxybenzyl)Palmitamide | FAAH | |
N-(3-Methoxybenzyl)Palmitamide is a promising FAAH inhibitor, treatment of pain, inflammation and CNS degenerative disorders. | |||
T4987 | NSC 42196 | Calcium α-D-heptagluconate hydrate,Calcium glucoheptonate | Others , Endogenous Metabolite |
NSC 42196 (Calcium glucoheptonate) is the calcium salt of (2xi)-D-gluco-heptonic acid. NSC 42196 is used as a calcium supplement for treatment of hypocalcemia. | |||
T1330 | Acitretin | Ro 10-1670,Etretin | Apoptosis , Retinoid Receptor , Autophagy |
Acitretin (Ro 10-1670) is a second-generation, systemic retinoid that has been used in the treatment of psoriasis. | |||
T7117 | Sapropterin dihydrochloride | Sapropterin Hydrochloride,6R-Tetrahydro-L-biopterin dihydrochloride,6R-BH4 dihydrochloride | Hydroxylase |
Sapropterin dihydrochloride (6R-BH4 dihydrochloride) is phenylalanine hydroxylase agonist that is approved for the treatment of BH4 responsive PKU. | |||
T5297 | 3-Indolepropionic acid | Indolepropionic acid,IPA,indole-3-propionic acid | Antioxidant , Reactive Oxygen Species , Endogenous Metabolite |
3-Indolepropionic acid (Indolepropionic acid) is shown to be a powerful antioxidant with potential in the treatment for Alzheimer’s disease. | |||
T20699 | Daunomycinone | Daunomycinon,Leukaemomycinone C,NSC 109351,NSC-109351,NSC109351 | Antibiotic |
Daunomycinone (NSC-109351) is a glycan of daunomycin, which belongs to the antibiotic class and is a representative glycan of tumour-inhibiting anthracyclines, used in the treatment of cancer and leukaemia. | |||
T1156 | Palonosetron hydrochloride | RS 25259 197,Palonosetron HCl,RS 25259 | 5-HT Receptor |
Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting. | |||
T4644 | Tapinarof | GSK2894512,Benvitimod,WBI 1001 | AhR , Aryl Hydrocarbon Receptor |
Tapinarof (Benvitimod) is targeted as a topical cream treatment for psoriasis, a chronic autoimmune skin disease. | |||
T2570 | Vitamin K4 | Kapilin,Menadiol Diacetate,acetomenaphthone | Apoptosis , Endogenous Metabolite |
Vitamin K4 (Menadiol Diacetate) is a vitamin medicine for the treatment of blood coagulation disorders that caused by the lack of VK4. | |||
T22293 | Chondroitine sulfate | Chondroitine sulfate (From cattle) | Others |
Chondroitin sulfate is an important structural component of cartilage and has been used as a dietary supplement for the treatment of joint discomfort. | |||
T0970 | Racanisodamine | Anisodamine,7β-Hydroxyhyoscyamine,Raceanisodamine | Adrenergic Receptor , AChR |
Racanisodamine (7β-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock. | |||
T2726 | Sinomenine | Cucoline,Kukoline | Apoptosis , Others , NF-κB , Opioid Receptor , Autophagy |
Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis. | |||
T7908 | DL-Methionine Methylsulfonium Chloride | Others | |
DL-Methionine Methylsulfonium Chloride is a natural product, used in the treatment of peptic ulcers, colitis, and gastritis. | |||
T0896 | Furaltadone hydrochloride | Furaltadone HCl | Antibacterial , Antibiotic , Parasite |
Furaltadone hydrochloride (Furaltadone HCl) is an antibacterial and shows distinct curative effect in the treatment of coccidiosis. | |||
T1068 | Dithranol | 1,8,9-trihydroxyanthracene,cignoline,Anthralin | Others , DNA/RNA Synthesis |
Dithranol (cignoline) is an anthracene derivative that disrupts MITOCHONDRIA function and structure and is used for the treatment of DERMATOSES, especially PSORIASIS. It may cause FOLLICULITIS. | |||
TQ0152 | Dalfopristin | RP54476 | Antibacterial , Antibiotic |
Dalfopristin (RP54476) is a semi-synthetic streptogramin antibiotic. Quinupristin/Dalfopristin (Q/D) is used for the treatment of multi-drug resistant Enterococcus faecium infections. | |||
T2968 | Hyodeoxycholic acid | NSC 60672,α-Hyodeoxycholic Acid,HDCA | FXR , Endogenous Metabolite , GPCR19 |
Hyodeoxycholic acid (NSC 60672) has been used in trials studying the treatment of Hypercholesterolemia. | |||
T1419 | Azithromycin hydrate | CP-62993 dihydrate,Azithromycin dihydrate | ribosome , Antibacterial , Antibiotic , Autophagy |
Azithromycin hydrate (CP-62993 dihydrate) is a semi-synthetic macrolide antibiotic structurally related to ERYTHROMYCIN. It has been used in the treatment of Mycobacterium avium intracellulare infections, toxoplasmosis, ... | |||
T3S1944 | Darutoside | Darutin | Others |
1. Darutoside (Darutin) can as an appropriate treatment for wounds. 2. Darutoside can improve skin elasticity, surface appearance and stretch mark removal, through soothing the skin, decreasing inflammation, restoring co... | |||
T0788 | Spectinomycin dihydrochloride | Spectinomycin 2HCl,Actinospectacin | ribosome , Antibacterial , Antibiotic |
Spectinomycin dihydrochloride (Actinospectacin) is an antibiotic produced by Streptomyces spectabilis. It is active against gram-negative bacteria and used for the treatment of gonorrhea. | |||
T2839 | Orsellinic acid | Apoptosis , Others | |
Orsellinic acid, a compound obtained by treatment of Lecanoric acidy with alcohols, inhibits platelet-activating factor (PAF)-mediated neuronal apoptosis. | |||
TN5538 | 6-Methoxykaempferol | Others | |
6-Methoxykaempferol is a flavonoid found in brazilian propolis. 6-Methoxykaempferol has anti-proliferative activity against cancer cells, neuroprotective effects on isolated rat brain synaptosomes and reduces glutathione... | |||
TN1520 | Isoforskolin | Coleonol B | IL Receptor , TNF |
Isoforskolin is derived from Coleus forskohlii and reduces the secretion of TNF-α, IL-1β, IL-6 and IL-8 in human mononuclear leukocytes. Isoforskolin can be used in studies about the treatment of Lyme arthritis. | |||
T7131 | Antineoplaston A10 | NSC-648539 | Apoptosis , Endogenous Metabolite , Ras |
Antineoplaston A10 (NSC-648539) is a Ras inhibitor potentially for the treatment of glioma, lymphoma, astrocytoma and breast cancer. | |||
T1694 | Oxypurinol | Oxipurinol | ROS , Xanthine Oxidase , Endogenous Metabolite |
Oxypurinol is a xanthine oxidase inhibitor. Oxipurinol is potentially used for the treatment of congestive heart failure. | |||
TN6457 | N-trans-caffeoyltyramine | Trans-N-Caffeoyltyramine,N-(E)-Caffeoyl-lambda-tyramine,N-cis-Caffeoyltyramine,Typheramide | Immunology/Inflammation related |
N-trans-caffeoyltyramine (Trans-N-Caffeoyltyramine) is a modulator of inflammatory responses and can be used in studies about treatment for chronic inflammatory diseases. | |||
T1152 | Albendazole | SKF-62979 | HIF/HIF Prolyl-Hydroxylase , Microtubule Associated , Antibiotic , Parasite |
Albendazole (SKF-62979) is used as a drug indicated for the treatment of a variety of worm infestations. | |||
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カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPH-01863 | PIEZO1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
PIEZO1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 33.6 kDa and the accession number is Q92508. | |||
TMPY-00539 | GSTA1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
GSTA1 (Glutathione S-Transferase Alpha 1) is a Protein Coding gene. This gene encodes a member of a family of enzymes that function to add glutathione to target electrophilic compounds. Glutathione S-transferases (GSTs) ... | |||
TMPY-00117 | FGF-16 Protein, Human, Cynomolgus, Recombinant | Human,Cynomolgus | Baculovirus Insect Cells |
Fibroblast growth factor 16 (FGF16) is preferentially expressed in the heart after birth, suggesting its regulation is associated with tissue-specific chromatin remodeling and DNA-protein interactions. Mutation of the ME... | |||
TMPY-02078 | HtrA2/Omi Protein, Human, Recombinant (His) | Human | E. coli |
Serine protease HTRA2, also known as high-temperature requirement protein A2, Omi stress-regulated endoprotease, Serine protease 25, Serine proteinase OMI and HTRA2, is a single-pass membrane protein that belongs to the ... | |||
TMPY-01736 | COX-2 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
PTGS2, also known as COX-2, is s component of Prostaglandin-endoperoxide synthase (PTGS). PTGS, also known as cyclooxygenase, is the key enzyme in prostaglandin biosynthesis, and acts both as a dioxygenase and as a perox... | |||
TMPK-01369 | S100B Protein, Canine, Recombinant (hFc) | Canine | HEK293 Cells |
S100B, a calcium-binding protein of the EF-hand type exerts both intracellular and extracellular functions.The intracellular, and extracellular, roles of S100B are attractive therapeutic targets for the treatment of both... | |||
TMPY-00319 | GIP Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Glucose-dependent insulinotropic polypeptide (GIP) is an incretin that plays an important role in fat accumulation. GIP is involved in fat accumulation and insulin resistance with aging. Glucose-dependent insulinotropic ... | |||
TMPY-00176 | FNDC4 Protein, Human, Recombinant (mFc) | Human | HEK293 Cells |
FNDC4 acts as an anti-inflammatory factor on macrophages and improves mouse model of induced colitis. FNDC4 could suppress osteoclast formation via NF-kappaB pathway and downregulation of CXCL10. Analysis of binding of F... | |||
TMPK-00994 | FNDC1 Protein, Human, Recombinant (His) | Human | E. coli |
Fibronectin type III domain‑containing protein 1 (FNDC1) is a protein that contains a major component of the structural domain of fibronectin.FNDC1 was highly upregulated and acted as an oncogene in BC. Therefore, target... | |||
TMPK-01310 | Syndecan-1 Protein, Rabbit, Recombinant (His) | Rabbit | HEK293 Cells |
CD138 (syndecan-1, Sdc-1) is a member of the syndecan family that comprises heparan sulfate proteoglycans. CD138 is significant for cell-cell and cell-matrix interactions.CD138 plays a crucial role in carcinogenesis and ... | |||
TMPK-00935 | APLP2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Amyloid β precursor-like protein 2 (APLP2) has been determined to serve an important role in the progression of a number of cancer types. APLP2 expression was significantly associated with disease-specific survival (P<0.... | |||
TMPK-00553 | ADAM9 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
A disintegrin and metalloproteinase 9 (ADAM9) is a member of the transmembrane ADAM family. It is expressed in different types of solid cancer and promotes tumor invasiveness. ADAM9 may be a prognostic marker for vestibu... | |||
TMPK-01230 | CLEC2D Protein, Human, Recombinant (hFc & Avi) | Human | HEK293 Cells |
C-type lectin domain family 2, member D (CLEC2D) is implicated in the immune response. Pre-eclampsia and HIV infection have opposing immune responses. The contrasting expression of CLEC2D in HIV infection and pre-eclamps... | |||
TMPK-00842 | CD21 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
CD21 mRNA expression, an EBV-entry receptor, was transiently detected in NK cells after exosome treatment, and levels decreased after further culture. CD21 protein expression was also transiently transferred to NK cells ... | |||
TMPK-01276 | CD161 Protein, Cynomolgus, Recombinant (His & Avi) | Cynomolgus | HEK293 Cells |
CD161 (NKRP1) is a lectin-like receptor present on NK cells and rare T-cell subsets. We have observed CD161 expression in some cases of T-cell prolymphocytic leukemia (T-PLL) and found it to be useful in follow-up and de... | |||
TMPK-00955 | CD161 Protein, Human, Recombinant (His & Avi), Biotinylated | Human | HEK293 Cells |
CD161 (NKRP1) is a lectin-like receptor present on NK cells and rare T-cell subsets. We have observed CD161 expression in some cases of T-cell prolymphocytic leukemia (T-PLL) and found it to be useful in follow-up and de... | |||
TMPK-01277 | CD161 Protein, Cynomolgus, Recombinant (His & Avi), Biotinylated | Cynomolgus | HEK293 Cells |
CD161 (NKRP1) is a lectin-like receptor present on NK cells and rare T-cell subsets. We have observed CD161 expression in some cases of T-cell prolymphocytic leukemia (T-PLL) and found it to be useful in follow-up and de... | |||
TMPJ-01028 | Claudin-18.2 Protein, Human, Recombinant (Twin strep & Flag) | Human | HEK293 Cells |
Claudin-18 (CLDN18) is a protein that in humans is encoded by the CLDN18 gene. It belongs to the group of claudins. CLDN18 belongs to the large claudin family of proteins, which form tight junction strands in epithelial ... | |||
TMPK-00392 | FGFR1 beta (IIIc) Protein, Human, Recombinant (His & Avi) | Human | HEK293 Cells |
Fibroblast growth factor receptor 1 (FGFR1) transmits signals through the plasma membrane regulating essential cellular processes like division, motility, metabolism, and death. Overexpression of FGFR1 is observed in num... | |||
TMPK-00828 | Mucin-1/MUC1 Isoform Y Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
MUC1, the transmembrane glycoprotein Mucin 1, is usually found to be overexpressed in a variety of epithelial cancers playing an important role in disease progression. MUC1 isoforms such as MUC1/Y, which lacks the entire... | |||
TMPK-00759 | IgG1 Fc Protein, Human, Recombinant | Human | HEK293 Cells |
IgG1 is most abundant in serum among the four IgG subclasses (IgG1, 2, 3 and 4) and binds to Fc receptors (FcγR) on phagocytic cells with high affinity. Fc fragment is demonstrated to mediate phagocytosis, trigger inflam... | |||
TMPK-00394 | FGFR1 beta (IIIc) Protein, Human, Recombinant (His & Avi), Biotinylated | Human | HEK293 Cells |
Fibroblast growth factor receptor 1 (FGFR1) transmits signals through the plasma membrane regulating essential cellular processes like division, motility, metabolism, and death. Overexpression of FGFR1 is observed in num... | |||
TMPK-00956 | CD161 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
CD161 (NKRP1) is a lectin-like receptor present on NK cells and rare T-cell subsets. We have observed CD161 expression in some cases of T-cell prolymphocytic leukemia (T-PLL) and found it to be useful in follow-up and de... | |||
TMPK-01229 | IL-19 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Interleukin-19 (IL-19) has been shown to be involved in coronary artery diseases and atherosclerosis, while its expression in myocardial infarction is poorly understood. In this study, the dynamic increase in circulating... | |||
TMPK-00022 | Galectin-1 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Galectin 1 (Gal-1), a β-galactoside binding mammalian lectin of 14KDa, is implicated in many signalling pathways, immune responses associated with cancer progression and immune disorders. Inhibition of human Gal-1 has be... | |||
TMPY-01843 | SEMA6A Protein, Human, Recombinant (His) | Human | HEK293 Cells |
SEMA6A, the first identified class 6 semaphorin, is contributed to regulate vascular development and adult angiogenesis. SEMA6A could inhibit proliferation, migration, and invasion in different glioma cell lines. That SE... | |||
TMPK-00829 | Galectin-1 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
Galectin 1(Gal-1), a β-galactoside binding mammalian lectin of 14KDa, is implicated in many signalling pathways, immune responses associated with cancer progression and immune disorders. Inhibition of human Gal-1 has bee... | |||
TMPK-00893 | PGF Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Placental growth factor (PGF) is another member of the VEGF family of cytokines with pro-angiogenic and pro-inflammatory effects. Retinal inhibition of PGF in combination with VEGF-A prevents vascular leakage and CNV pos... | |||
TMPK-01057 | CLEC9A Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
CLEC9A expression was significantly higher in psoriatic skin compared with healthy donor. In psoriatic skin and PsA ST, CLEC9A() cells were in close proximity to TUNEL() cells. SF CLEC9A levels were significantly lower c... | |||
TMPY-03989 | PFDN1 Protein, Human, Recombinant (His) | Human | E. coli |
PFDN1 expression positively correlated with tumor size and tumor invasion. The inhibitory effect of PFDN1 on tumor cell growth and motility was partially due to G2/M cell cycle blockage and cytoskeletal deficiency. PFDN1... | |||
TMPY-02046 | PFDN1 Protein, Mouse, Recombinant (His) | Mouse | E. coli |
PFDN1 expression positively correlated with tumor size and tumor invasion. The inhibitory effect of PFDN1 on tumor cell growth and motility was partially due to G2/M cell cycle blockage and cytoskeletal deficiency. PFDN1... | |||
TMPY-00607 | PSMB6 Protein, Mouse, Recombinant (His) | Mouse | E. coli |
PSMB6 subunit belongs to the 20S proteasomal subunit family, which plays an importance role in the antigen presentation by MHC class I molecular. Proteasome subunit beta type 6 (PSMB6) is a member of 20S proteasomal subu... | |||
TMPY-03386 | ART3 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
ART3 is an arginine-specific ADP-ribosyltransferase which belongs to the Arg-specific ADP-ribosyltransferase family. ART3 catalyzes a reversible reaction which modifies proteins by the addition or removal of ADP-ribose t... | |||
TMPK-00455 | IGF1R/CD221 Protein, Human, Recombinant (His & Avi) | Human | HEK293 Cells |
The type 1 IGF receptor (IGF1R) is a transmembrane tyrosine kinase that is frequently overexpressed by tumours, and mediates proliferation and apoptosis protection. IGF signalling also influences hypoxia signalling, prot... | |||
TMPK-00548 | CLEC12A/MICL/CLL-1 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
CLEC12A has recently been identified as an antigen, expressed on leukemic stem cells and leukemic blasts. Given the fact that this expression profile seems stable throughout diagnosis, treatment and relapse on leukemic b... | |||
TMPK-01158 | Kallikrein 5/KLK5 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
The inhibition of kallikrein 5 (KLK5) has been identified as a potential strategy for treatment of the genetic skin disorder Netherton syndrome, in which loss-of-function mutations in the SPINK5 gene lead to down-regulat... | |||
TMPK-00728 | PSCA Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Gastric cancer is a deadly malignancy and is a prognostically unfavorable entity with restricted therapeutic strategies available. Prostate stem cell antigen (PSCA) is a glycosylphosphatidylinositol (GPI)-anchored cell s... | |||
TMPK-01005 | CLEC12A/MICL/CLL-1 Protein, Human, Recombinant (His), FITC-Labeled | Human | HEK293 Cells |
CLEC12A has recently been identified as an antigen, expressed on leukemic stem cells and leukemic blasts. Given the fact that this expression profile seems stable throughout diagnosis, treatment and relapse on leukemic b... | |||
TMPK-01006 | CLEC12A/MICL/CLL-1 Protein, Human, Recombinant (aa 65-265, His) | Human | HEK293 Cells |
CLEC12A has recently been identified as an antigen, expressed on leukemic stem cells and leukemic blasts. Given the fact that this expression profile seems stable throughout diagnosis, treatment and relapse on leukemic b... | |||
TMPK-00658 | IGF1R/CD221 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
The type 1 IGF receptor (IGF1R) is a transmembrane tyrosine kinase that is frequently overexpressed by tumours, and mediates proliferation and apoptosis protection. IGF signalling also influences hypoxia signalling, prot... | |||
TMPK-01375 | PRLR Protein, Canine, Recombinant (hFc) | Canine | HEK293 Cells |
Prolactin receptor (PRLR) is highly expressed in a subset of human breast cancer and prostate cancer, which makes it a potential target for cancer treatment. In clinical trials, the blockade of PRLR was shown to be safe ... | |||
TMPK-00995 | CLEC12A/MICL/CLL-1 Protein, Mouse, Recombinant (aa 65-267, His) | Mouse | HEK293 Cells |
CLEC12A has recently been identified as an antigen, expressed on leukemic stem cells and leukemic blasts. Given the fact that this expression profile seems stable throughout diagnosis, treatment and relapse on leukemic b... | |||
TMPK-01002 | CLEC12A/MICL/CLL-1 Protein, Human, Recombinant (hFc & Avi), Biotinylated | Human | HEK293 Cells |
CLEC12A has recently been identified as an antigen, expressed on leukemic stem cells and leukemic blasts. Given the fact that this expression profile seems stable throughout diagnosis, treatment and relapse on leukemic b... | |||
TMPK-00547 | PRLR Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
Prolactin receptor (PRLR) is highly expressed in a subset of human breast cancer and prostate cancer, which makes it a potential target for cancer treatment. In clinical trials, the blockade of PRLR was shown to be safe ... | |||
TMPK-00906 | PSCA Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
Gastric cancer is a deadly malignancy and is a prognostically unfavorable entity with restricted therapeutic strategies available. Prostate stem cell antigen (PSCA) is a glycosylphosphatidylinositol (GPI)-anchored cell s... | |||
TMPK-01004 | CLEC12A/MICL/CLL-1 Protein, Human, Recombinant (aa 65-265, hFc) | Human | HEK293 Cells |
CLEC12A has recently been identified as an antigen, expressed on leukemic stem cells and leukemic blasts. Given the fact that this expression profile seems stable throughout diagnosis, treatment and relapse on leukemic b... | |||
TMPK-00456 | IGF1R/CD221 Protein, Human, Recombinant (aa 31-932, His & Avi), Biotinylated | Human | HEK293 Cells |
The type 1 IGF receptor (IGF1R) is a transmembrane tyrosine kinase that is frequently overexpressed by tumours, and mediates proliferation and apoptosis protection. IGF signalling also influences hypoxia signalling, prot... | |||
TMPY-03329 | DPEP1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Dehydropeptidase-I, also known as DPEP1, is a kidney membrane enzyme. Its expression in normal colonic mucosa is very low, but it is highly expressed in colorectal adenoma and cancer specimens and is negatively correl... | |||
TMPJ-00711 | GADD45G Protein, Human, Recombinant (His) | Human | E. coli |
Growth Arrest and DNA Damage-Inducible Protein GADD45 Υ (GADD45G) is a nuclear protein which belongs to the GADD45 family. GADD45G is highly expressed in placenta. GADD45G interacts with various proteins whose transcript... | |||
TMPK-01003 | CLEC12A/MICL/CLL-1 Protein, Human, Recombinant (His, Avi), Biotinylated | Human | HEK293 Cells |
CLEC12A has recently been identified as an antigen, expressed on leukemic stem cells and leukemic blasts. Given the fact that this expression profile seems stable throughout diagnosis, treatment and relapse on leukemic b... | |||
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カタログ番号 | 製品名 | ||
---|---|---|---|
L8400 | Hematonosis Compound Library | 514 compounds | |
A unique collection of 514 compounds related to hematologic diseases for high throughput screening (HTS) and high content screening (HCS); | |||
L9410 | Covalent Inhibitor Library | 1920 compounds | |
A unique collection of 1920 covalent Inhibitors and other molecules with common warheads like chloroacetyl,2-Chloropropionyl,Acryloyl,sulfonyl fluoride, alkyne,acrylamide, ketocarbonyl,disulfide bond, etc. | |||
L2151 | Chemotherapy Drug Library | 48 compounds | |
48 Chemotherapeutic drugs that can be used for high-throughput and high-content screening. | |||
L6140 | Saccharide and Glycoside Natural Product Library | 595 compounds | |
A unique collection of 595 saccharides and glycosides compounds can be used for HTS and HCS; | |||
L4520 | Anti-Bacterial Compound Library | 904 compounds | |
A unique collection of 904 antibacterial bioactive compounds, a powerful tool for antibacterial drug development; | |||
L1800 | Anti-Infection Compound Library | 2938 compounds | |
A unique collection of 2938 anti-infective compounds including anti-bacterial, anti-fungi, anti-Human Cytomegalovirus (HCMV), anti-HIV, anti-SARS, anti-influenza, etc; | |||
L2520 | Glycometabolism Compound Library | 702 compounds | |
702 glycometabolism-related comounds, can be used for HTS and HCT; | |||
L4600 | Selected Plant-Sourced Compound Library | 3048 compounds | |
A unique collection of 3048 plant-sourced compounds that derived from 277 plant species for high throughput screening (HTS) and high content screening (HCS); | |||
L4660 | Anti-Nervous System Disease Library | 1246 compounds | |
Well-chosen 1246 compounds with unique structures targeting nervous system; | |||
L3900 | DNA Damage & Repair Compound Library | 910 compounds | |
A unique collection of 910 DNA Damage & Repair related compounds for high throughput screening (HTS) and high content screening (HCS); | |||
L6100 | Polyphenolic Natural Product Library | 635 compounds | |
A unique collection of 635 natural polyphenolic compounds for high throughput screening (HTS) and high content screening (HCS); | |||
L4400 | Antibiotics Library | 692 compounds | |
A unique collection of 692 compounds with antibiotic activity for new antibacterial drug screening; | |||
L2152 | Targeted Therapy Drug Library | 119 compounds | |
119 tumor-targeted drugs that can be used for high-throughput and high-content screening. | |||
L2010 | Highly Selective Inhibitor Library | 575 compounds | |
L9210 | Pediatric Drug Library | 972 compounds | |
A unique collection of 972 pediatric drugs for high-throughput screening and high-content screening. | |||
L2190 | Anti-Lung Cancer Compound Library | 1702 compounds | |
A unique collection of 1702 compounds with anti-lung cancer therapeutic activity or targeting lung cancer’s major signaling pathways, can be used for anti-lung cancer drug discovery and mechanism study; | |||
L3980 | DNA Damage and Repair Compound Library Plus | 667 compounds | |
Well-chosen 667 compounds with unique structures targeting DNA damage & repair; | |||
L6500 | Microbial Natural Product Library | 550 compounds | |
A unique collection of 550 microbial natural products for high throughput screening (HTS) and high content screening (HCS); | |||
L6720 | Anti-COVID-19 Traditional Chinese Medicine Compound Library | 1147 compounds | |
A unique collection of 1147 monomers from 60 TCM plants, a powerful tool for anti-COVID-19 drug discovery, can be used for HTS and HCS screening; | |||
L1610 | FDA-Approved Kinase Inhibitor Library | 263 compounds | |
A unique collection of 263 kinase inhibitors/regulators for specific targeting of kinases, ready for high-throughput screening and high-content screening. | |||
L2192 | Anti-Pancreatic Cancer Compound Library | 2238 compounds | |
A unique collection of 2238 pancreatic cancer related compounds can be used in HTS and HCS; | |||
L4500 | Anti-Fungal Compound Library | 252 compounds | |
A unique collection of 252 antifungal compounds effective for drug repurposing screening, combination screening and biological investigation. | |||
L6600 | Anti-Gastroenteritis Natural Product Library | 219 compounds | |
A unique collection of 219 natural products related to gastroenteritis for high throughput screening (HTS) and high content screening (HCS); | |||
L8300 | Chromatin Modification Compound Library | 250 compounds | |
A unique collection of 250 compounds targeting chromatin remodeling pathway for high throughput screening (HTS) and high content screening (HCS); | |||
L6230 | Miao medicine Compound Library | 534 compounds | |
A unique collection of 534 compounds featuring natural product molecules derived from Miao medicine that can be used for high-throughput and high-content screening. | |||
L8110 | Reprogramming Compound Library | 1813 compounds | |
A unique collection of 1813 reprogramming signaling pathway-related bioactive small molecule compounds for high-throughput, high-content screening. | |||
L5900 | CNS-Penetrant Compound Library | 509 compounds | |
A unique collection of 509 CNS-Penetrant compounds for high throughput screening (HTS) and high content screening (HCS); | |||
L8000 | Stem Cell Differentiation Compound Library | 1197 compounds | |
A unique collection of 1197 stem cell differentiation signaling targeted compounds for high throughput and high content screening; | |||
L1720 | Nucleotide Compound Library | 334 compounds | |
A unique collection of 334 nucleoside and nucleotide analogues, can be used for research and development of anti-viral, anti-tumor, anti-fungal, and anti-depressive drugs; | |||
L9860 | Antidepressant Compound Library | 1163 compounds | |
1163 compounds associated with depression that can be used for high-throughput and high-content screening | |||
L1100 | Protease Inhibitor Library | 343 compounds | |
A unique collection of 343 protease and proteasome inhibitors for research in chemical genomics, and drug screening; | |||
L2600 | Neuronal Signaling Compound Library | 2540 compounds | |
A unique collection of 2540 compounds targeting CNS signaling for high throughput screening (HTS) and high content screening (HCS) for new drugs; | |||
L7400 | Sodium Channel Blocker Library | 118 compounds | |
A unique collection of 118 sodium channel blockers and agonists for high throughput and high content screening; | |||
L2191 | Anti-Breast Cancer Compound Library | 1939 compounds | |
A unique collection of 1939 compounds with anti-breast cancer therapeutic activity or targeting breast cancer’s major signaling pathways, can be used for anti-breast cancer drug discovery and mechanism study; | |||
L6700 | Anti-Tumor Natural Product Library | 1772 compounds | |
A unique collection of 1772 natural products with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS); | |||
L2196 | Anti-Ovarian Cancer Compound Library | 1867 compounds | |
L6730 | Anti-virus Traditional Chinese Medicine Monomer Library | 268 compounds | |
A collection of 268 TCM monomers with anti-virus activity. An effective tool for drug development and pharmacological studies. | |||
L2510 | Lipid Metabolism Compound Library | 492 compounds | |
A unique collection of 492 compounds targeting lipid metabolism, can be used for high-throughput screening (HTS) and high-content screening (HCS). | |||
L9600 | Peptide Compound Library | 791 compounds | |
791 peptides can be used in peptide drug development and signaling transduction and mechanism study; | |||
L2610 | Neurotransmitter Receptor Compound Library | 1513 compounds | |
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening; | |||
L9700 | Endoplasmic Reticulum Stress Compound Library | 193 compounds | |
A unique collection of 193 endoplasmic reticulum stress (ER stress) related compounds used for high throughput screening (HTS) and high content screening (HCS); | |||
L4700 | Immunology/Inflammation Compound Library | 4720 compounds | |
A unique collection of 4720 anti-inflammation compounds effective for high throughput screening and high content screening. | |||
L9830 | Anti-Parkinson's Disease Compound Library | 857 compounds | |
A unique collection of 857 compounds with anti-PD activities or acting on main drug targets of PD can be used for HTS and HCS. | |||
L7110 | Anti-Hypertension Compound Library | 678 compounds | |
678 hypertension-related small molecules for high-throughput and high-content screening. | |||
L7100 | Anti-Obesity Compound Library | 2247 compounds | |
A unique collection of 2247 anti-obesity compounds for high throughput and high content screening; | |||
L9420 | Exosome Compound Library | 76 compounds | |
76 exosome-related compounds that can be used for high-throughput and high-content screening. | |||
L6030 | Natural Product Derivatives Library for CADD | 163000 compounds | |
Large quantity: contains 163,000 natural product derivatives and the number is continuously updating; | |||
L7600 | Chemokine Inhibitor Library | 59 compounds | |
A unique collection of 59 chemokines or chemokine receptors targeted compounds for high throughput and high content screening; | |||
L2170 | Immuno-Oncology Compound Library | 449 compounds | |
A unique collection of 449 compounds acting on immune-oncology therapeutic targets can be used for high throughput and high content screening; | |||
L2630 | Neuronal Differentiation Compound Library | 672 compounds | |
L6620 | Antiparasitic Natural Product Library | 253 compounds | |
A unique collection of 253 natural products with antiparasitic activity, a powerful tool for high throughput screening (HTS) and high content screening (HCS); | |||
L8500 | HIF-1 Signaling Pathway Compound Library | 1336 compounds | |
A unique collection of 1336 HIF-1 related small chemicals can be used for drug discovery in ischemic disease and cancer and related mechanism studies; | |||
L6750 | PBCRBS Traditional Chinese Medicine Compound Library | 580 compounds | |
A unique collection of 580 compounds derived from traditional Chinese medicines (TCMs) for promoting blood circulation and removing blood stasis. | |||
L2550 | Glutamine Metabolism Compound Library | 565 compounds | |
A unique collection of 565 glutamine metabolism related compounds can be used for high throughput screening (HTS) and high content screening (HCS), and also is an effective tool for research in glutamine metabolism and ... | |||
L6740 | Anti-Colorectal Cancer Traditional Chinese Medicine Compound Library | 382 compounds | |
A collection of 382 TCM monomers with anti-colorectal activity. An effective tool for drug development and pharmacological studies. | |||
L6820 | Tobacco Monomer Library | 747 compounds | |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T14687 | Deucravacitinib | BMS-986165 | Tyrosine Kinases , JAK , IFNAR , Interleukin |
Deucravacitinib (BMS-986165) inhibits IL-12/23 and type I IFN pathways[1][2]. BMS-986165 is a highly selective, orally bioavailable allosteric TYK2 inhibitor for the treatment of autoimmune diseases. Which selectively bi... | |||
T27098 | Ivacaftor-D9 | deutivacaftor,CTP-656 | |
CTP-656, a cystic fibrosis transmembrane conductance regulator (CFTR) channel activator, is used potentially for the treatment of cystic fibrosis. | |||
T11867 | Loperamide-d6 hydrochloride | R-18553 D6 hydrochloride | Others |
Loperamide D6 hydrochloride, a deuterium-labeled variant of Loperamide hydrochloride, acts as an opioid receptor agonist utilized for diarrhea treatment. | |||
T31108 | CTP-347 | CTP347,CTP 347 | |
CTP-347, a deuterated version of paroxetine, is potentially the best non-hormonal drug in its class for the treatment of hot flashes. | |||
T13023 | Sulfadiazine-d4 | Sulfadiazine D4 | Others |
Sulfadiazine D4 is a deuterium labeled Sulfadiazine. Sulfadiazine used for the treatment of toxoplasmosis. | |||
T19548 | Repaglinide D5 | AG-EE 623ZW D5 | Others |
Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus. | |||
T12701 | (rel)-Tranylcypromine D5 hydrochloride | 2-Phenylcyclopropylamine D5 hydrochloride | Histone Demethylase |
(rel)-Tranylcypromine D5 hydrochloride is a deuterium labeled (rel)-Tranylcypromine hydrochloride. (rel)-Tranylcypromine hydrochloride is an irreversible, nonselective inhibitor of monoamine oxidase (MAO) used in the tre... | |||
T17047 | Tetrabenazine-d6 | Ro 1-9569 D6 | Others |
Tetrabenazine D6 is the deuterium-labeled Tetrabenazine. Tetrabenazine is a VMAT-inhibitor used for the treatment of hyperkinetic movement disorder. | |||
T13155 | Tiaprofenic acid D3 | Others | |
Tiaprofenic acid D3 is a deuterium-labeled Tiaprofenic acid. Tiaprofenic acid is a nonsteroidal anti-inflammatory drug and treatment of rheumatic diseases. | |||
T19305 | Eldecalcitol-d6 | Others | |
Eldecalcitol is an orally active analogue of active vitamin D used in the treatment of osteoporosis. Eldecalcitol-d6 is the deuterium labeled Eldecalcitol. | |||
T10528 | Bexarotene D4 | LGD1069 D4 | Others |
Bexarotene D4 is a deuterium-labeled Bexarotene (LGD1069). Bexarotene is a selective RXR agonist used in the treatment of cutaneous T-cell lymphoma. | |||
T11247 | Etravirine D4 | R-165335 D4,TMC-125 D4 | Others |
Etravirine is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used for the treatment of HIV. Etravirine D4 is the deuterium labeled Etravirine. | |||
T19183 | Albendazole-d3 | Albendazole D3 | Others |
Albendazole D3 is the deuterium-labeled Albendazole. Albendazole is used as a drug indicated for the treatment of a variety of worm infestations. | |||
T34589 | SD-1077 | d3-L-DOPA,deuldopa,deuterated levodopa,SD1077 | |
SD-1077, also known as d3-L-DOPA, is a deuterium containing levodopa. SD-1077 has been shown in preclinical models to improve the half-life of dopamine in the brain resulting in a prolonged treatment effect. | |||
T13282 | Valsartan-d9 | CGP-48933 D9 | Others |
Valsartan D9 is a deuterium-labeled valsartan. Valsartan is an antagonist of the angiotensin II receptor and for the treatment of high blood pressure and heart failure. | |||
T10229 | Acebutolol D7 | Others | |
Acebutolol D7 is a deuterium-labeled Acebutolol. Acebutolol is a selective antagonist of the β1 adrenergic receptor used in the treatment of angina pectoris, hypertension, and cardiac arrhythmias. | |||
T12363 | Paricalcitol-D6 | Others | |
Paricalcitol-D6 is the deuterated form of Paricalcitol, which is used for the prevention and treatment of secondary hyperparathyroidism (excessive secretion of parathyroid hormone) associated with chronic renal failure. | |||
T27210 | DRX-065 | DRX 065,DRX065,deuterated R-enantiomer of pioglitazone | |
DRX-065 is a stabilized and deuterated R-enantiomer of pioglitazone. DRX-065 has pharmacological properties desirable for the treatment of NASH (mitochondrial function modulation, non-steroidal anti-inflammatory effects,... | |||
TMID-0053 | Amisulpride-d5 | ||
Amisulpride-d5 is a deuterated compound of Amisulpride. Amisulpride has a CAS number of 71675-85-9. Amisulpride (trade name Solian) is an antipsychotic drug sold by Sanofi-Aventis. It is not approved for use in the Unite... | |||
T11113 | Duloxetine D3 hydrochloride | (S)-Duloxetine D3 hydrochloride,LY248686 D3 hydrochloride | Others |
Duloxetine D3 hydrochloride is a serotonin-norepinephrine reuptake inhibitor (SNRI) with a Ki of 4.6 nM, used for treatment of major depressive disorder and generalized anxiety disorder (GAD).Duloxetine D3 hydrochloride ... | |||
T73716 | Miglustat-d9 HCl | ||
Miglustat-d 9 (hydrochloride), a deuterium-labeled variant of Miglustat (hydrochloride), functions as a glucosylceramide synthase inhibitor. Its primary application is in the treatment of Type I Gaucher disease (GD1) [1]... | |||
T10118 | 3-O-Methyltolcapone D7 | Ro 40-7591 D7 | Transferase |
3-O-Methyltolcapone D7 (Ro 40-7591 D7) is a deuterium labeled 3-O-Methyltolcapone. 3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor. Tolcapone crosses the blood-brain barrier... | |||
TMID-0035 | Naratriptan-d3 | ||
Naratriptan-d3 is a deuterated compound of Naratriptan. Naratriptan has a CAS number of 121679-13-8. Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches. | |||
TMIH-0609 | Zafirlukast-d7 | ||
Zafirlukast-d7 is a deuterated compound of Zafirlukast. Zafirlukast has a CAS number of 107753-78-6. Zafirlukast is an orally available leukotriene receptor antagonist which is widely used for the prophylaxis and chronic... | |||
TMID-0042 | Rac-Paroxetine-d4 Hydrochloride | ||
rac-Paroxetine-d4 Hydrochloride is a deuterated compound of rac-Paroxetine Hydrochloride. rac-Paroxetine Hydrochloride has a CAS number of 78246-49-8. Paroxetine hydrochloride is a serotonin uptake inhibitor that is effe... | |||
TMIJ-0012 | Trans-Diethyl-1,1,1’,1’-Stilbestrol-3,3’,5,5’-d8 | ||
Trans-Diethyl-1,1,1’,1’-Stilbestrol-3,3’,5,5’-d8 is a deuterated compound of Trans-Diethyl-Stilbestrol. Trans-Diethyl-Stilbestrol has a CAS number of 56-53-1. Diethylstilbestrol is used in the treatment of menopausal and... | |||
TMIH-0469 | Quinidine-d3 | ||
Quinidine-d3 is a deuterated compound of Quinidine. Quinidine has a CAS number of 56-54-2. Quinidine is a stereoisomer of the antimalarial agent quinine and a class Ia antiarrhythmic agent. for the treatment of abnormal ... | |||
TMIH-0283 | Ipratropium-d3 Bromide | ||
Ipratropium-d3 Bromide is a deuterated compound of Ipratropium Bromide. Ipratropium Bromide has a CAS number of 22254-24-6. Ipratropium is a synthetic anticholinergic agent that is used as an inhalant for treatment of ac... | |||
TMIH-0024 | 10,11-Dihydro-10-hydroxycarbamazepine-d4 | rac-Licarbazepine-d4 | |
10,11-Dihydro-10-hydroxycarbamazepine-d4 is a deuterated compound of 10,11-Dihydro-10-hydroxycarbamazepine. 10,11-Dihydro-10-hydroxycarbamazepine has a CAS number of 29331-92-8. Licarbazepine is the pharmacologically act... | |||
TMID-0025 | Quetiapine-d8 Hemifumarate | ||
Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar... | |||
T71893 | Clobetasol Propionate-d5 | ||
Clobetasol propionate-d5 is intended for use as an internal standard for the quantification of clobetasol propionate by GC- or LC-MS. Clobetasol propionate is a corticosteroid. It binds to glucocorticoid receptors in a c... | |||
TMIH-0427 | Perospirone hydrochloride-d8 | ||
Perospirone hydrochloride-d8 is a deuterated compound of Perospirone hydrochloride. Perospirone hydrochloride has a CAS number of 129273-38-7. Perospirone hydrochloride is an atypical antipsychotic agent for the treatmen... | |||
TMIH-0605 | Vortioxetine-d8 2HBr | ||
Vortioxetine-d8 2HBr is a deuterated compound of Vortioxetine 2HBr. Vortioxetine 2HBr has a CAS number of 508233-74-7. Vortioxetine is a serotonergic antidepressant used for major depression disorders. Vortioxetine has b... | |||
TMIH-0591 | Vadadustat-13C2-15N | ||
Vadadustat-13C2-15N is 13C and 15N labeled Vadadustat. Vadadustat has a CAS number of 1000025-07-9. Vadadustat is a novel, titratable, oral hypoxia-inducible factor prolyl hydroxylase (HIF-PH) inhibitor in development fo... | |||
T71329 | Theophylline-d6 | ||
Theophylline-d6 is intended for use as an internal standard for the quantification of theophylline by GC- or LC-MS. Theophylline is an inhibitor of phosphodiesterase. It is also an adenosine A1 and A2 receptor antagonist... | |||
T71065 | Quinapril-d5 | ||
Quinapril-d5 is intended for use as an internal standard for the quantification of quinapril by GC- or LC-MS. Quinapril is a prodrug form of the angiotensin converting enzyme (ACE) inhibitor quinaprilat. In vivo, quinapr... | |||
TMIH-0602 | Vonoprazan-d4 | ||
Vonoprazan-d4 is a deuterated compound of Vonoprazan. Vonoprazan has a CAS number of 881681-00-1. Vonoprazan is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduoden... | |||
TMIH-0524 | Sofosbuvir-13C-d3 | ||
Sofosbuvir-13C-d3 is the 13C and deuterated compound of Sofosbuvir. Sofosbuvir has a CAS number of 1190307-88-0. Sofosbuvir is a uridine monophosphate analog inhibitor of hepatitis C virus (HCV) polymerase NS5B that is u... | |||
TMIH-0601 | Vonoprazan-d3 | ||
Vonoprazan-d3 is a deuterated compound of Vonoprazan. Vonoprazan has a CAS number of 881681-00-1. Vonoprazan is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduoden... | |||
T71286 | Guaifenesin-d3 | ||
Guaifenesin-d3 is intended for use as an internal standard for the quantification of guaifenesin by GC- or LC-MS. Guaifenesin is an expectorant. It inhibits production of mucin 5AC (MUC5AC), reduces mucus viscosity and e... | |||
T71206 | Tiagabine-d6 hydrochloride | ||
Tiagabine-d6 is intended for use as an internal standard for the quantification of tiagabine by GC- or LC-MS. Tiagabine is an inhibitor of GABA transporter 1. It inhibits seizures induced by DMCM in mice. Tiagabine reduc... | |||
T70035 | Tasimelteon-d5 | ||
Tasimelteon-d5 is intended for use as an internal standard for the quantification of tasimelteon by GC- or LC-MS. Tasimelteon is a melatonin (MT) receptor agonist. It selectively binds MT1 and MT2 receptors over a panel ... | |||
T71984 | Enrofloxacin-d5 | ||
Enrofloxacin-d5 is intended for use as an internal standard for the quantification of enrofloxacin by GC- or LC-MS. Enrofloxacin is a fluoroquinolone antibiotic. It is active against panels of Campylobacter, E. coli, and... | |||
T71205 | Fosinopril-d7 sodium salt | ||
Fosinopril-d7 is intended for use as an internal standard for the quantification of fosinopril by GC- or LC-MS. Fosinopril is a prodrug form of the angiotensin-converting enzyme inhibitor fosinoprilat. Oral administratio... | |||
T71288 | Phenylbutazone-d9 | ||
Phenylbutazone-d9 is intended for use as an internal standard for the quantification of phenylbutazone by GC- or LC-MS. Phenylbutazone is a non-steroidal anti-inflammatory drug and an inhibitor of the peroxidase activity... | |||
T71306 | Gemfibrozil-d6 | ||
Gemfibrozil-d6 is intended for use as an internal standard for the quantification of gemfibrozil by GC- or LC-MS. Gemfibrozil is a peroxisome proliferator-activated reporter α and PPARγ agonist. In vivo, gemfibrozil redu... | |||
T71145 | Racecadotril-d5 | ||
Racecadotril-d5 is intended for use as an internal standard for the quantification of racecadotril by GC- or LC-MS. Racecadotril is a prodrug form of the neprilysin (NEP) inhibitor thiorphan. In vivo, racecadotril reduce... | |||
T71211 | Rizatriptan-d6 benzoate salt | ||
Rizatriptan-d6 is intended for use as an internal standard for the quantification of rizatriptan by GC- or LC-MS. Rizatriptan is an agonist of the serotonin receptor subtypes 5-HT1B and 5-HT1D. It is selective for 5-H... | |||
T68918 | Phenytoin-d10 | ||
Phenytoin-d10 is intended for use as an internal standard for the quantification of phenytoin by GC- or LC-MS. Phenytoin is an anticonvulsant agent and active metabolite of fosphenytoin. Phenytoin is formed from fospheny... | |||
T69758 | Flutamide-d7 | ||
Flutamide-d7 is intended for use as an internal standard for the quantification of flutamide by GC- or LC-MS. Flutamide is an androgen receptor antagonist and prodrug form of 2-hydroxy flutamide. Flutamide is converted ... | |||
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