12905
3351
13181
50
3
260
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T28589 | Ro 41-5253 | Ro-41-5253,Ro 415253 | Apoptosis , Retinoid Receptor |
Ro 41-5253 is an orally active RARα antagonist, ligand and partial agonist of peroxisome proliferator-activated receptor (PPAR)-γ. It exhibits antitumor activity, inhibits proliferation and induces apoptosis in MCF-7 and... | |||
T16773 | Ro 90-7501 | RO-90-7501 | Apoptosis , Phosphatase , ATM/ATR , Gamma-secretase |
Ro 90-7501 is an amyloid β42 (Aβ42) protofibrillar and TPR-dependent PP5 inhibitor, a novel radiosensitiser for cervical cancer cells, which inhibits ATM phosphorylation, promotes apoptosis, and induces cell-cycle arrest... | |||
T16771 | RO-5963 | Mdm2 , p53 | |
RO-5963 is a dual inhibitor of p53-MDM2 and p53-MDMX (IC50s: ~17 nM and ~24 nM, respectively). | |||
T6643 | Ro 31-8220 Mesylate | Ro 31-8220 methanesulfonate,Bisindolylmaleimide IX,Bisindolylmaleimide IX mesylate | PKC |
Ro 31-8220 Mesylate (Bisindolylmaleimide IX mesylate) is a pan-PKC inhibitor for PKC-α/βI/βII/γ/ε (IC50: 5/24/14/27/24 nM), and also shows potent inhibition against MSK1, MAPKAP-K1b, S6K1, and GSK3β. | |||
T9223 | RO-0335 | Reverse Transcriptase | |
RO-0335 is a potent diphenylether nonnucleoside reverse transcriptase inhibitor. RO-0335 inhibits Wt HIV-1 (IC50 = 1.1 nM) and retained activity (IC50< 100 nM) against 92% of a large number of NNRTI-resistant clinical is... | |||
T2356 | Ro-3306 | Apoptosis , ERK , SGK , PKA , CDK , PKC | |
RO-3306 is a selectivity ATP-competitive CDK1 inhibitor (Ki: 20 nM). The selectivity of RO-3306 for CDK1 is >15-fold higher than a diverse panel of human kinases. | |||
T19706 | Ro 20-1724 | Ro-20-1724,4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone,Ro20-1724 | PDE |
Ro 20-1724 (4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone) is a widely used inhibitor of cyclic nucleotide phosphodiesterase with IC50 of 2.0 μM and Ki of 3.1 μM. | |||
T3194 | Ro 46-2005 | Endothelin Receptor | |
Ro 46-2005 is a synthetic non-peptide endothelin receptor antagonist, inhibits the specific binding of 125I-ET-1 to human vascular smooth muscle cells (ETA receptor, IC50: 220 nM). | |||
T1896 | Ro 61-8048 | Hydroxylase | |
Ro 61-8048 is a potent and selective inhibitor of kynurenine hydroxylase with an IC50 value of 37 nM. | |||
T12758 | Ro 25-6981 | NMDAR | |
T3474 | RO 46-8443 | Endothelin Receptor | |
RO 46-8443 is the first non-peptide endothelin ETB receptor selective antagonist. RO 46-8443 displays up to 2000-fold selectivity for ETB receptors both in terms of binding inhibitory potency and functional inhibition. | |||
T16766 | Ro 08-2750 | Others | |
Ro 08-2750 is a non-peptide and reversible nerve growth factor (NGF) inhibitor which binds to NGF, and with an IC50 of ~ 1 µM. Ro 08-2750 is a selective MSI RNA-binding activity inhibitor, with an IC50 of 2.7 μM. Ro 08-2... | |||
T3478 | Ro 67-7476 | GluR | |
Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors. No activity at human mGlu1 receptors. Potentiates glutamate-induced calcium release with EC 50 of 60.1 nM. | |||
T12761 | Ro 10-5824 dihydrochloride | Dopamine Receptor | |
Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM). | |||
T5513 | RO-3 | P2X Receptor | |
RO3 is a selective antagonist of homomeric P2X3 and heteromeric P2X2/3 receptor | |||
T1771 | Ro 48-8071 fumarate | Others | |
Ro 48-8071 fumarate is an inhibitor of OSC(Oxidosqualene cyclase; IC50=6.5 nM) that has low-density lipoprotein (LDL) cholesterol lowering activity. | |||
T9357 | Ro 5212773 | Epptb | Others |
Ro 5212773 (Epptb) is a selective TAAR1 antagonist. | |||
T6971 | Ro 5126766 | CH5126766,Avutometinib,VS-6766,RO5126766 | Raf , MEK |
RO5126766 (CH5126766) is a dual RAF/MEK inhibitor with IC50 of 8.2 nM, 19 nM, 56 nM, and 160 nM for BRAF V600E, BRAF, CRAF, and MEK1, respectively. Phase 1. | |||
T12758L | Ro 25-6981 Maleate | Others | |
Ro 25-6981 Maleate is a potent and selective activity-dependent NMDA receptors blocker containing the NR2B subunit.(IC50 values are 0.009 and 52 μM for cloned receptor subunit combinations NR1C/NR2B and NR1C/NR2A respect... | |||
T2634 | Ro3280 | RO 3280,Ro5203280 | PLK |
Ro3280 (Ro5203280) is an effective, specific inhibitor of PLK1(IC50=3, Kd=0.09 nM). | |||
T4141 | RG7713 | RO 5028442 | Vasopressin Receptor |
RG7713 (RO 5028442) has been used in trials studying Autistic Disorder. | |||
T68134 | Ro-3201195 | p38 MAPK | |
Ro-3201195 is a novel orally available p38 MAPK inhibitor with high selectivity. | |||
T4687 | Ro5-3335 | CBFβ-Runx1 inhibitor II,Ro 5-3335 | DNA/RNA Synthesis |
Ro5-3335 (CBFβ-Runx1 inhibitor II) is core binding factor (CBF) inhibitor; preferentially kills human leukemia cell lines with CBF fusion proteins (IC50 = 1.1 μM). Ro5-3335 represses RUNX1/CBFβ-dependent transactivation ... | |||
T23245 | Ro-51 | Ro 51 | Others |
dual P2X3 and P2X2/3 antagonist | |||
T8447 | Ro 8-4304 | Ro 8-4304 Hydrochloride | NMDAR |
Ro 8-4304 Hydrochloride is an antagonist of NMDA receptor with IC50 of 0.4 μM | |||
T34364 | Ro 5-6669 | Ro-5-6669,Ro 56669 | Others |
Ro 5-6669 is bioactive chemical. | |||
T28576 | Ro 24-6392 | Ro 246392,Ro-24-6392 | Others |
Ro 24-6392 is an ester-linked co-drug combining ciprofloxacin and desacetylcefotaxime. Ro 24-6392 demonstrats activity against a wide spectrum of aerobic bacteria. | |||
T28566 | Ro 22-8515 | Ro 228515,Ro-22-8515 | Others |
Ro 22-8515 is the ligand of benzodiazepine receptor. | |||
T28577 | Ro 24-6778 | Ro 246778,Ro-24-6778 | Others |
Ro 24-6778 is a dual action cephalosporin with antimicrobial activity. | |||
T28593 | Ro 61-1448 | Ro-61-1448,Ro 611448 | Others |
Ro 61-1448 is a metabolite of tolcapone, a catechol-O-methyltransferase inhibitor. | |||
T24718 | Ro 5-5453 | Ro 55453,Ro 5 5453 | Others |
Ro 5-5453 is an inhibitor of monoamine oxidase. | |||
T34347 | Ro 12-9150 | Ro-129150,Ro-12-9150 | Others |
Ro 12-9150 is a bio-active agent. | |||
T28571 | RO 23-6152 | RO 236152,RO-23-6152 | Others |
RO 23-6152, a new calcium antagonist, can inhibit platelet aggregation in vitro associated with occlusive coronary thrombus formation. | |||
T28586 | Ro 31-8830 | Ro-31-8830,Ro 318830 | Others |
Ro 31-8830, a derivative of Ro 31-8425, has in vivo anti-inflammatory activity. | |||
T34357 | Ro 31-0313 | Ro 310313,Ro-31-0313 | Others |
Ro 31-0313 is a metabolite of Ro 03-8799, radiation sensitizing agent. | |||
T34339 | Ro 03-8800 | Ro-03-8800,Ro 038800 | Others |
Ro 03-8800 is a bio-active chemical. | |||
T28583 | Ro 31-7837 | Ro-31-7837,Ro 317837 | Others |
Ro 31-7837 is an opener of potassium channel. | |||
T28580 | Ro 31-1118 | Ro 311118,Ro-31-1118 | Others |
Ro 31-1118 is a partial agonist of beta-adrenoceptor. | |||
T28588 | Ro 41-1879 | Ro-41-1879,Ro 411879 | Others |
Ro 41-1879 is a catechol cephalosporin with antimicrobial activity. | |||
T28569 | Ro 23-3423 | Ro 233423,Ro-23-3423 | Others |
Ro 23-3423 is a specific inhibitor of thromboxane synthetase. | |||
T28581 | Ro 31-2201 | Ro 312201,Ro-31-2201 | Others |
Ro 31-2201 is a potent inhibitor of angiotensin converting enzyme. | |||
T34353 | Ro 19-7728 | Ro-19-7728,Ro 197728 | Others |
Ro 19-7728 is a metabolite of fleroxacin. | |||
T28562 | Ro 18-3981 | Ro-18-3981,Ro 183981 | Others |
Ro 18-3981 is an inhibition of myocardial Ca2+ channels. The KD value of Ro 18-3981 (1.0 nM) was similar to the IC50 value for blockade of ICa at a Vh of -20 mV (2.3 nM), i.e. at a level of near-maximal depolarization. | |||
T28563 | Ro 18-5364 | Ro-18-5364,Ro 185364 | Others |
Ro 18-5364 is a potent inhibitor of the gastric (H+ + K+)-ATPase with an apparent Ki of 0.1 μM at pH 6. | |||
T34374 | RO5203648 HCl | RO5203648,RO-5203648,RO 5203648 | Others |
RO5203648 HCl is a partial agonist of trace amine-related receptor 1 (TAAR1) with antipsychotic and antidepressant-like activities. RO5203648 HCl can be used in studies about neuropsychiatric therapeutics. | |||
T28595 | Ro-0505124 | Ro0505124,Ro 0505124 | Others |
Ro-0505124 is a potent, selective and ATP-competitive inhibitor of cyclin-dependent kinase 4 (CDK4). | |||
T28574 | Ro 24-4383 | Ro 244383 | Others |
Ro 24-4383 is a carbamate-linked dual-action antibacterial agent. | |||
T34340 | Ro 03-9310 | Ro 03 9310,Ro-03-9310 | Others |
Ro 03-9310 is a bio-active chemical. | |||
T28592 | Ro 48-8587 | Ro 488587 | Others |
Ro 48-8587 is a competitive antagonist of AMPA receptor. | |||
T26104 | Ro 28-2653 | Ro 28 2653,Ro-28-2653,Ro282653 | Others |
Ro 28-2653 is a matrix-metalloproteinases (MMPs) inhibitor with high selectivity for MMP2, MMP9 and membrane type 1-MMP. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T28551 | Ro 09-0680 | Ro-09-0680,Ro 09 0680 | |
Ro 09-0680, a compound derived from Salvia miltiorrhiza, is a potent inhibitor of collagen-induced platelet aggregation in rabbits with potential anti-inflammatory activity for the study of cardiovascular disease. | |||
T3915 | Ginsenoside Ro | Chikusetsusaponin 5,Polysciasaponin P3,Chikusetsusaponin V | Calcium Channel , Reductase , Prostaglandin Receptor |
Ginsenoside Ro (Chikusetsusaponin V) can reduce TXA2 production, weakly reduce COX-1 and TXAS activities, and has antiplatelet effects as a Ca2+ antagonist with an IC50 of 155 μM. | |||
T1589 | D-Cycloserine | RO-1-9213 | Others , Antibacterial , Antibiotic , iGluR |
D-Cycloserine (RO-1-9213) is a broad spectrum antibiotic used as a second line agent for treatment of drug resistant tuberculosis, always in combination with other antituberculosis agents. | |||
T6402 | Azomycin | 2-Nitroimidazole,Ro 05-9129,Amicin | Antibacterial , Antibiotic |
Azomycin (Ro 05-9129) is an antimicrobial antibiotic produced by a strain of Nocardia mesenterica. | |||
T1468 | Lornoxicam | Ro 13-9297,Chlortenoxicam,TS110 | COX , Endogenous Metabolite |
Lornoxicam (Chlortenoxicam) (chlortenoxicam) is a new nonsteroidal anti-inflammatory drug (NSAID) of the oxicam class with analgesic, anti-inflammatory, and antipyretic properties. Lornoxicam differs from other oxicam co... | |||
T1330 | Acitretin | Ro 10-1670,Etretin | Apoptosis , Retinoid Receptor , Autophagy |
Acitretin (Ro 10-1670) is a second-generation, systemic retinoid that has been used in the treatment of psoriasis. | |||
T1556 | Ornidazole | Tiberal,Ornidazolum,NSC 95075,Ro 7-0207 | Antibacterial , Antibiotic , Parasite |
Ornidazole (Tiberal) is a nitroimidazole antiprotozoal agent used in ameba and trichomonas infections. It is partially plasma-bound and also has radiation-sensitizing action. | |||
T0986 | Flucytosine | 5-Fluorocytosine,Ro 2-9915,Fluorocytosine,NSC 103805 | DNA/RNA Synthesis , Antibiotic , Antifungal |
Flucytosine (NSC 103805) is a pyrimidine compound and a fluorinated cytosine analog exhibiting antifungal activity. | |||
T6430 | Calcifediol | U 32070E,25-hydroxy Vitamin D3,RO 8-8892 | Endogenous Metabolite |
Calcifediol (U 32070E)(Ki of 3.9 μM), a major circulating metabolite of vitamin D3, works as a competitive inhibitor. It (ED50=2 nM)also inhibits PTH secretion and mRNA. | |||
T6316 | Calcitriol | Topitriol,Rocaltrol,Calcijex,RO215535,1,25-Dihydroxyvitamin D3 | Endogenous Metabolite |
Calcitriol (1,25-Dihydroxyvitamin D3) is a metabolite of vitamin D and a vitamin D receptor (VDR) agonist (IC50=0.4 nM). Calcitriol increases intestinal absorption of calcium and phosphorus, and increases bone resorption... | |||
TQ0262 | Dihomo-γ-linolenic acid | Diroleuton,all-cis-8,11,14-Eicosatrienoic acid,Ro 12-1989 | Others |
Ro 12-1989 can be converted into prostaglandin E1 (PGE1). Ro 12-1989 competes with arachidonic acid for COX and lipoxygenase, inhibiting the production of arachidonic acid's eicosanoids. | |||
T4950 | 1,2-Dipalmitoyl-sn-glycerol | (S)-1,2-Dipalmitin | Endogenous Metabolite , PKC |
1,2-Dipalmitoyl-sn-glycerol ((S)-1,2-Dipalmitin) is an analog of the PKC-activating second messenger diacylglycerol (DAG). It weakly activates PKC. | |||
T36581 | Glucocerebrosides | Others | |
Glucocerebrosides is a natural product. | |||
TN1824 | Kaempferol 3-sophoroside-7-glucoside | Antioxidant | |
Kaempferol 3-sophoroside-7-glucoside is a bioactive ingredient in the Lei leaves, belonging to the flavonoid group, which has antioxidant and anti-obesity activities. | |||
TN4919 | Rosthornin A | Others | |
Rosthornin A is a kind of natural product derived from the herbs of Rabdosia rosthornii. | |||
T13514 | 5-MethoxyPinocembroside | Others | |
5-MethoxyPinocembroside is a flavonoid isolated from leaves of Moringa oleifera. | |||
T31467 | Dihydrocyclosporin A | Dihydrocyclosporin-A | Others |
Dihydrocyclosporin A (Dihydrocyclosporin-A) is closely related co-metabolite of cyclosporin A. Dihydrocyclosporin A significantly inhibits promastigotes and intracellular amastigotes. | |||
TN7029 | (2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol | Others | |
(2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol is a useful research compound for many research applications, including the fields of chemistry and life sciences, among others. | |||
T7937 | 2-Amino-4'-fluorobenzophenone | Others | |
2-Amino-4'-fluorobenzophenone is a derivative of benzophenone. It is used in the synthesis of p-fluorobenzoyl chloride and has also been used as a fluorescent probe for biochemical studies such as DNA and RNA detection. | |||
TMA1122 | N-Feruloylserotonin | (E/Z)-Moschamine,Moschamine | Antioxidant |
N-Feruloylserotonin ((E/Z)-Moschamine) is a selective FAAH inhibitor that inhibits [H]-AEA uptake and cell proliferation at low concentrations. | |||
T36473 | Trans-Nerolidol | Antifungal | |
trans-Nerolidol is a sesquiterpene alcohol isolated from the above-ground parts of the Saharan Valerian plant with antifungal activity. trans-Nerolidol inhibits cell proliferation in a dose-dependent manner, and induces ... | |||
T4879 | 12-Hydroxydodecanoic acid | 12-hydroxylauric acid | Others , Endogenous Metabolite |
12-Hydroxydodecanoic acid (12-hydroxylauric acid) is the substrate of the human glutathione-dependent formaldehyde dehydrogenase. | |||
TN2019 | Orobol | 3'-Hydroxygenistein,3’,4’,5,7-tetrahydroxy-isoflavon | BCL , Caspase , PI3K |
Orobol (3’,4’,5,7-tetrahydroxy-isoflavon) is an inhibitor of tyrosine-specific protein kinase and phosphatidylinositol turnover. Orobol inhibits PI3K isoforms with IC50s of 3.46-5.27 μM for PI3K α/β/γ/K/δ. Orobol exhibit... | |||
TN7159 | Methyl 2-benzoylamino-3-phenylpropyionate | Others | |
methyl 2-benzoylamino-3-phenylpropyionate is a natural product found in Aspergillus flavipes. | |||
TN6864 | Prosaikogenin F | Others | |
Prosaikogenin F ((2R,3R,4S,5R,6R)-2-{[(1S,2R,4S,5R,8R,9S,10R,13S,14R,17S,18R)-2-hydroxy-9-(hydroxymethyl)-4,5,9,13,20,20-hexamethyl-24-oxahexacyclo[15.5.2.01,1?.0?,1?.0?,1?.0?,13]tetracos-15-en-10-yl]oxy}-6-methyloxane-3... | |||
TN1957 | Mulberrofuran Q | MulberrofuranQ | |
Mulberrofuran Q is an active compound that inhibits the formation of 12-hydroxy-5,8,10-heptadecatrienoic acid (HHT) and thromboxane B2 (cyclooxygenase product) , which protects neuronal cells from hypoxia-glycorrhoea-def... | |||
TN6788 | 5-hydroxy-3,7-dimethoxy-2-phenylchromen- | 3,7-Dimethylgalangin,5-hydroxy-3,7-dimethoxy-2-phenylchromen-4-one,Galangin 3,7-dimethyl ether,4H-1-Benzopyran-4-one, 5-hydroxy-3,7-dimethoxy-2-phenyl- | Others |
5-hydroxy-3,7-dimethoxy-2-phenylchromen- (4H-1-Benzopyran-4-one, 5-hydroxy-3,7-dimethoxy-2-phenyl-),a natural product obtained from the resinous exudate of Heliotropium huascoense. | |||
T2803 | Monocrotaline | Crotaline | TGF-beta/Smad |
Monocrotaline (Crotaline) is a pyrrolizidine alkaloid and a toxic plant constituent that poisons livestock and humans through the ingestion of contaminated grains and other foods. The alkaloid causes pulmonary artery hyp... | |||
TN2215 | Taurochenodeoxycholic acid sodium | Sodium taurochenodeoxycholate | Apoptosis , Endogenous Metabolite |
Taurochenodeoxycholic acid sodium (Sodium taurochenodeoxycholate) is one of the main bioactive substances of animals' bile acid. Taurochenodeoxycholic acid sodium induces apoptosis and shows obvious anti-inflammatory and... | |||
T3850 | Luteolin 7-O-glucuronide | Luteolin-7-glucuronide | MMP |
Luteolin 7-O-glucuronide (Luteolin-7-glucuronide) possesses antioxidant activities. | |||
T0973L | Pyridoxine hydrochloride | Pyridoxine HCl,Pyridoxol (hydrochloride),Vitamin B6 (hydrochloride),Vitamin B6 | Nrf2 , Endogenous Metabolite |
Pyridoxine hydrochloride (Vitamin B6) is the 4-methanol form of vitaminB6 which is converted to pyridoxal phosphate which is a coenzyme for synthesis of amino acids, neurotransmitters (serotonin, norepinephrine), sphingo... | |||
T2738 | Dehydroandrographolide | NOS , Influenza Virus | |
Dehydroandrographolide is a natural compound extracted from herbal medicine Andrographis paniculata (Burm f) Nees. | |||
TN7246 | 3-Sulfopropanoic acid | 3-SPA | Drug Metabolite |
3-Sulfopropanoic acid, a major metabolite of treprostinil and its prodrug ALZ-801, is an endogenous molecule present in the cerebrospinal fluid (CSF) of AD patients that inhibits the formation of Aβ42 oligomers. | |||
T4S1312 | Gypsogenin-3-O-glucuronide | Methyl gypsogenin 3-O-beta-D-glucuronopy | Others |
1. Gypsogenin-3-O-glucuronide (Methyl gypsogenin 3-O-beta-D-glucuronopy) shows inhibitory activity toward pancreatic lipase with IC5 value of .29 mM, and the free carboxylic acid groups in position 28 within its chemical... | |||
T3005 | 4-Hydroxychalcone | P-Cinnamoylphenol | Others , NF-κB |
4-Hydroxychalcone (P-Cinnamoylphenol) attenuates hyperaldosteronism, inflammation, and renal injury in cryptochrome-null mice. | |||
T6917 | Oleuropein | Apoptosis , Aromatase , ROS , PPAR | |
Oleuropein is an antioxidant polyphenol isolated from olive leaf. | |||
T19529 | Proteinase | Others | |
Proteinases are enzymes that catalyse the breakdown of proteins. Proteinases are involved in many biological functions, including the digestion of ingested proteins, the breakdown of old proteins, and cell signalling. Th... | |||
T9719 | 3-Hydroxyoctanoic Acid | GPR | |
3-Hydroxyoctanoic Acid is one of the hydroxy-carboxylic acids (HCAs) that serve as intermediates of energy metabolism. It is an agonist of the orphan receptor GPR109B. | |||
T5497 | AMAROGENTIN | Apoptosis , AMPK | |
Amarogentin is mainly extracted from Swertia and Gentiana roots. It plays cemopreventive/therapeutic role during liver carcinogenesis through modulation of cell cycle and apoptosis | |||
T7442 | 4-Isopropylbenzyl Alcohol | Cuminic alcohol,Cuminyl alcohol,Cumic alcohol | Others |
4-Isopropylbenzyl Alcohol (Cuminic alcohol) is a natural product,with insecticidal effect. | |||
T19433 | Monocrotaline N-Oxide | Others | |
Monocrotaline N-Oxide is a monocrotaline metabolite. | |||
T7324 | Chelidonine hydrochloride | Others | |
Chelidonine hydrochloride is one of the alkaloids of Chelidonium majus, which has broad pharmacological activities | |||
T8023 | 2,3,4-Trihydroxybenzoic acid | Others | |
2,3,4-Trihydroxybenzoic acid is natural compound,with antioxidant activity | |||
T4773 | 3-Ethoxy-3-oxopropanoic acid | Monoethyl malonic acid,Ethyl hydrogen malonate | Others , Endogenous Metabolite |
3-Ethoxy-3-oxopropanoic acid (Monoethyl malonic acid) belongs to the class of organic compounds known as dicarboxylic acids and derivatives. These are organic compounds containing exactly two carboxylic acid groups. 3-Et... | |||
TMA0432 | Octahydroisoindole | Others | |
Octahydroisoindole is a natural product and a reference standard. | |||
TMO2685 | 10-Hydroxydecanoic Acid | NSC 15139 | Antibacterial |
10-Hydroxydecanoic Acid (NSC 15139) has antibacterial, anti - cancer and anti - radiation activity. | |||
T0345 | Estropipate | Piperazine estrone sulfate,Pipestrone,Estrone sulfate piperazine salt | Estrogen Receptor/ERR , Estrogen/progestogen Receptor |
Estropipate (Piperazine estrone sulfate) is a natural estrogenic substance composed of estrone sulfate and piperazine. | |||
T3751 | 2',4'-Dihydroxyacetophenone | Resacetophenone,1-(2,4-Dihydroxyphenyl)ethanone,2,4-Dihydroxyacetophenone,4-Acetylresorcinol | Others , Endogenous Metabolite |
2',4'-Dihydroxyacetophenone (Resacetophenone) is a member of the class of compounds known as alkyl-phenylketones. | |||
T2943 | 5-Hydroxymethylfurfural | 2-Hydroxymethyl-5-furfural,2-Formyl-5-hydroxymethylfuran,5-Hydroxymethyl-2-furaldehyde,5-(Hydroxymethyl)furan-2-carbaldehyde | Others , Antifungal |
5-Hydroxymethylfurfural (2-Formyl-5-hydroxymethylfuran) is found from various carbohydrates. | |||
T4880 | L-Dihydroorotic acid | Others , Endogenous Metabolite | |
L-Dihydroorotic acid, also known as (S)-4,5-dihydroorotate or dihydro-L-orotate, belongs to the class of organic compounds known as alpha amino acids and derivatives. Within the cell, L-dihydroorotic acid is primarily lo... | |||
------------------------ More ------------------------ |
カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPY-05306 | TRIM21 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
TRIM21 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 56.5 kDa and the accession number is P19474-1. | |||
TMPY-03259 | Calreticulin Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Calreticulin Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 47.4 kDa and the accession number is P27797. | |||
TMPY-06327 | Calreticulin Protein, Human, Recombinant | Human | HEK293 Cells |
Calreticulin Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 45.99 kDa and the accession number is P27797. | |||
TMPY-03258 | Calreticulin Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Calreticulin Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 73 kDa and the accession number is P27797. | |||
TMPY-01403 | VNN1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
VNN1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 53.7 kDa and the accession number is O95497. | |||
TMPY-01928 | IL-18 Protein, Rhesus, Recombinant (His) | Rhesus | E. coli |
IL-18 Protein, Rhesus, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 23.7 kDa and the accession number is Q9BGI5. | |||
TMPY-00888 | MMP-9 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
MMP-9 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 77.7 kDa and the accession number is P14780. | |||
TMPY-00955 | Influenza B (B/Florida/4/2006) Hemagglutinin/HA Protein (His) | Influenza B | HEK293 Cells |
Influenza B (B/Florida/4/2006) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60 kDa and the accession number is B1AG46. | |||
TMPY-04753 | IRE1 Protein, Human, Recombinant (aa 465-977) | Human | Baculovirus Insect Cells |
IRE1 Protein, Human, Recombinant (aa 465-977) is expressed in Baculovirus insect cells. The predicted molecular weight is 58.3 kDa and the accession number is O75460-1. | |||
TMPY-04262 | B7-H3 Protein, Human, Recombinant (His), Biotinylated | Human | HEK293 Cells |
B7-H3 Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 48 kDa and the accession number is Q5ZPR3-1. | |||
TMPY-01296 | HGFR/c-Met Protein, Human, Recombinant (His) | Human | HEK293 Cells |
HGFR/c-Met Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 103 kDa and the accession number is A0A024R759. | |||
TMPY-04069 | Neurotrophin 3 Protein, Human, Recombinant | Human | E. coli |
NTF3 (Neurotrophin 3) is a Protein Coding gene. The protein encoded by this gene is a member of the neurotrophin family, that controls the survival and differentiation of mammalian neurons. This protein is closely relate... | |||
TMPY-05455 | CD3E & CD3G Heterodimer Protein, Cynomolgus, Recombinant (hFc) | Cynomolgus | HEK293 Cells |
CD3E & CD3G Heterodimer Protein, Cynomolgus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 74.9 kDa and the accession number is Q95LI5.2&NP_001270839.1. | |||
TMPY-01993 | IL-13 Protein, Human, Recombinant | Human | CHO Cells |
IL-13 Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 12.5 kDa and the accession number is AAK53823.1. | |||
TMPY-06094 | PVRIG Protein, Cynomolgus, Rhesus, Recombinant (His) | Cynomolgus,Rhesus | HEK293 Cells |
PVRIG Protein, Cynomolgus, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 15.3 kDa and the accession number is XP_005549281.1&XP_014989941.2. | |||
TMPY-04116 | KRAS Protein,Human,Recombinant(G12C & Q61H, His) | Human | E. coli |
KRAS Protein,Human,Recombinant(G12C & Q61H, His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 23.3 kDa and the accession number is P01116-2. | |||
TMPY-02483 | ATP citrate lyase/ACLY Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
ATP citrate lyase, also known as Acly or Acl, is the primary enzyme responsible for the synthesis of cytosolic acetyl-CoA in many tissues. The enzyme is composed of two polymer chains which are polypeptides in human. ATP... | |||
TMPY-02365 | HER3/ERBB3 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
HER3/ERBB3 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 70 kDa and the accession number is Q61526. | |||
TMPY-04090 | Influenza A H7N9 (A/Shanghai/2/2013) Hemagglutinin/HA Protein (HEK293, His) | H7N9 | HEK293 Cells |
Influenza A H7N9 (A/Shanghai/2/2013) Hemagglutinin/HA Protein (HEK293, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 57.6 kDa. | |||
TMPY-04064 | B7-H3 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
B7-H3 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 24.9 kDa and the accession number is A6MDC5. | |||
TMPY-00357 | HNT/NTM Protein, Human, Recombinant (His) | Human | HEK293 Cells |
HNT/NTM Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 32.3 kDa and the accession number is Q9P121-3. | |||
TMPY-05090 | CD25/IL2R alpha Protein, Rat, Recombinant (His) | Rat | Baculovirus Insect Cells |
CD25/IL2R alpha Protein, Rat, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 25.9 kDa and the accession number is A6JLS0. | |||
TMPY-02632 | SIRP alpha Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
SIRP alpha Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 39.4 kDa and the accession number is BAA20376.1. | |||
TMPY-00484 | Cerberus 1/CER1 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
Cerberus 1/CER1 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 29.6 kDa and the accession number is AAH69371.1. | |||
TMPY-06021 | CD28 Protein, Human, Cynomolgus, Rhesus, Recombinant (His) | Human,Cynomolgus,Rhesus | HEK293 Cells |
CD28 Protein, Human, Cynomolgus, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.6 kDa and the accession number is Q0PDN3. | |||
TMPY-00891 | Neuropilin-1 Protein, Human, Recombinant (V179A, hFc) | Human | HEK293 Cells |
Neuropilin-1 Protein, Human, Recombinant (V179A, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 96.5 kDa and the accession number is O14786-2. | |||
TMPY-03466 | PLGF/PGF Protein, Mouse, Recombinant | Mouse | HEK293 Cells |
PLGF/PGF Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 16.6 kDa and the accession number is P49764. | |||
TMPY-01691 | Clusterin Protein, Human, Recombinant (CLU34, His) | Human | HEK293 Cells |
Clusterin Protein, Human, Recombinant (CLU34, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 51.5 kDa and the accession number is P10909-2. | |||
TMPY-04870 | Zika virus (ZIKV) (strain Zika SPH2015) ZIKV-NS1 protein (His) | ZIKV | HEK293 Cells |
Zika virus NS1 antigen is one of seven non-structural proteins. NS1 is involved in RNA replication. The possible effects of NS1 on hosts include: localizes to host cell surface and secreted extracellularly, modulates sig... | |||
TMPY-05021 | Influenza B (B/Brisbane/60/2008) Hemagglutinin/HA Protein | Influenza B | Baculovirus Insect Cells |
Influenza B (B/Brisbane/60/2008) Hemagglutinin/HA Protein is expressed in Baculovirus insect cells. The predicted molecular weight is 61.7kDa and the accession number is C0LT35. | |||
TMPY-05302 | CD79 Protein, Human, Recombinant (Flag & His) | Human | HEK293 Cells |
CD79 Protein, Human, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 37.5 kDa and the accession number is NP_001774.1&NP_000617.1. | |||
TMPJ-01467 | Oncostatin M/OSM Protein, Human, Recombinant (E. coli, His) | Human | E. coli |
Oncostatin M (OSM) is a glycoprotein belonging to the interleukin-6 family of cytokines that includes leukemia-inhibitory factor, granulocyte colony-stimulating factor, and interleukin 6. OSM encodes a growth regulator, ... | |||
TMPY-02130 | Argonaute-2 Protein, Mouse, Recombinant (His) | Mouse | Baculovirus Insect Cells |
Argonaute-2 Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 99 kDa and the accession number is Q8CJG0. | |||
TMPY-06986 | FGF-8b Protein, Human, Recombinant | Human | E. coli |
In mammalian embryos, transient Fgf8 expression defines the developing isthmic region, lying between the midbrain and the first rhombomere, but there has been uncertainty about the existence of a distinct isthmic segment... | |||
TMPY-02824 | IL-18R alpha Protein, Rat, Recombinant (hFc) | Rat | HEK293 Cells |
IL-18R alpha Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 62.5kDa and the accession number is A0A8I6A1C2. | |||
TMPY-01376 | IL-18R alpha Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
IL-18R alpha Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 36.8 kDa and the accession number is Q61098. | |||
TMPY-02566 | Interferon alpha 4/IFNA4 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
Interferon alpha 4/IFNA4 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 20.7 kDa and the accession number is P05014. | |||
TMPY-01694 | Clusterin Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Clusterin Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.8 kDa and the accession number is Q06890. | |||
TMPY-00988 | Lipocalin-2/LCN2 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Lipocalin-2/LCN2 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 22.3 kDa and the accession number is P11672. | |||
TMPY-01870 | IL-9 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
IL-9 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 15.5 kDa and the accession number is P15248. | |||
TMPY-00890 | Noggin/NOG Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Noggin/NOG Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 49.8 kDa and the accession number is Q13253. | |||
TMPY-01774 | TREM-1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
TREM-1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 21.8 kDa and the accession number is Q38L15. | |||
TMPY-00772 | DC-SIGN Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
DC-SIGN Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 65.8 kDa and the accession number is Q9NNX6-1. | |||
TMPY-03235 | BST2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
BST2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 14.9 kDa and the accession number is Q10589. | |||
TMPY-02429 | Human coronavirus HKU1 (isolate N1) (HCoV-HKU1) Spike S1 Protein (His) | HCoV-HKU1 | HEK293 Cells |
Human coronavirus HKU1 (isolate N1) (HCoV-HKU1) Spike S1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 85.8 kDa and the accession number is Q5MQD0. | |||
TMPY-03432 | KEAP1 Protein, Human, Recombinant | Human | Baculovirus Insect Cells |
KEAP1 Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 69.7 kDa and the accession number is Q14145. | |||
TMPY-04211 | Latent TGF beta 1 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
Latent TGF beta 1 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.7 kDa. | |||
TMPY-06022 | FOLR1 Protein, Cynomolgus, Rhesus, Recombinant (His) | Cynomolgus,Rhesus | HEK293 Cells |
FOLR1 Protein, Cynomolgus, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.3 kDa and the accession number is A0A2K5UR19&NP_001181576.1. | |||
TMPY-00443 | EPO/Erythropoietin Protein, Mouse, Recombinant | Mouse | HEK293 Cells |
EPO/Erythropoietin Protein, Mouse, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 18.6 kDa and the accession number is P07321. | |||
TMPY-02336 | Influenza A H3N2 (A/Babol/36/2005) Neuraminidase/NA Protein (His) | H3N2 | HEK293 Cells |
Influenza A H3N2 (A/Babol/36/2005) Neuraminidase/NA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 49.6 kDa and the accession number is C0LU95. | |||
------------------------ More ------------------------ |
カタログ番号 | 製品名 | ||
---|---|---|---|
L6160 | RO5 Drug-like Natural Product Library | 2703 compounds | |
A unique collection of 2703 natural product monomers that meet the "Lipinski's Rule of Five", a powerful tool for HTS and HCS screening; | |||
L6900 | Rare Natural Product Library | 693 compounds | |
A unique collection of 693 rare natural products, which can be used for high throughput screening (HTS) and high content screening (HCS); | |||
L8710 | Cuproptosis Compound Library | 400 compounds | |
TargetMol’s Cuproptosis Compound Library is a collection of 400 compounds related to copper-dependent death that can be used to study its mechanism and related diseases. | |||
NY1000 | Natural Product Derivatives Library | 4000 compounds | |
The library consists of more than 4,000 members belonging 22 scaffolds (average 180 compounds per scaffold). | |||
L6010 | Natural Product Library | 3840 compounds | |
A unique collection of 3840 natural products for high throughput screening (HTS) and high content screening (HCS); | |||
L2200 | Tyrosine Kinase Inhibitor Library | 1016 compounds | |
A unique collection of 1016 tyrosine kinase inhibitors for high throughput screening and high content screening for drug discovery in tyrosine kinase related diseases; | |||
L2195 | Anti-Prostate Cancer Compound Library | 2070 compounds | |
2070 compounds associated with prostate cancer that can be used for high-throughput and high-content screening. | |||
L2110 | Anti-Cancer Approved Drug Library | 1779 compounds | |
A unique collection of 1779 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS); | |||
L6700 | Anti-Tumor Natural Product Library | 1772 compounds | |
A unique collection of 1772 natural products with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS); | |||
L6500 | Microbial Natural Product Library | 550 compounds | |
A unique collection of 550 microbial natural products for high throughput screening (HTS) and high content screening (HCS); | |||
L6150 | Covalent Natural Product Library | 583 compounds | |
Detialed biological information and pharmacological information of the products, providing theoretical direction and research basis for screening. | |||
L1110 | Microtubule-Targeted Compound Library | 142 compounds | |
A unique collection of 142 microtubule-targeted compounds can be used in HTS and HCS; | |||
L2630 | Neuronal Differentiation Compound Library | 672 compounds | |
L6001 | Mini Fungal Metabolite Natural Product Screening Library | Inquiry | |
L7860 | Mini Electrophilic Heterocyclic Fragment Library | 369 compounds | |
369 compounds in total in the Highly Solubility Covalent Heterocyclic Fragment Library | |||
L9810 | Anti-Fibrosis Compound Library | 1180 compounds | |
A unique collection of 1180 potential anti-fibrosis compounds, can be used in HTS and HCS; | |||
L7820 | High Solubility Micro Fragment Library | 1081 compounds | |
The compound library of highly soluble micro-fragments consists of 1081 low-molecular-weight fragments. | |||
L6400 | Marine Natural Product Library | 144 compounds | |
A unique collection of 144 marine natural products for high throughput screening (HTS) and high content screening (HCS); | |||
L6020 | Selectable Natural Product Library | 16627 compounds | |
A unique collection of 16627 pure natural products with diverse structures and sources covering various plant, animal, and microbe species; | |||
L8700 | Ferroptosis Compound Library | 779 compounds | |
A unique collection of 779 ferroptosis signaling pathway related compounds, a powerful tool for new target identification, drug discovery, and mechanism study; | |||
L7810 | High Solubility Polyfunctional Group Fragment Library | 1159 compounds | |
Highly soluble multifunctional fragment library contains 1159 kinds of fragment molecules. | |||
L6620 | Antiparasitic Natural Product Library | 253 compounds | |
A unique collection of 253 natural products with antiparasitic activity, a powerful tool for high throughput screening (HTS) and high content screening (HCS); | |||
L6610 | Anti-infective Natural Product Library | 1060 compounds | |
A unique collection of 1060 species of natural products with anti-infective activity for high throughput screening (HTS) and high content screening (HCS); | |||
L1000 | Approved Drug Library | 2808 compounds | |
A unique collection of 2808 approved drugs for high throughput screening (HTS) and high content screening (HCS); | |||
L2540 | Gut Microbial Metabolite Library | 614 compounds | |
A unique collection of 614 gut microbial metabolites which can be used for HTS and HCS; | |||
L6600 | Anti-Gastroenteritis Natural Product Library | 219 compounds | |
A unique collection of 219 natural products related to gastroenteritis for high throughput screening (HTS) and high content screening (HCS); | |||
L9300 | Macrocyclic Compound Library | 210 compounds | |
210 macrocyclic compounds of known activity for high-throughput, high-content screening; | |||
L6100 | Polyphenolic Natural Product Library | 635 compounds | |
A unique collection of 635 natural polyphenolic compounds for high throughput screening (HTS) and high content screening (HCS); | |||
L6110 | Alkaloid Natural Product Library | 464 compounds | |
A unique collection of 464 natural alkaloids can be used for high throughput and high content screening; | |||
L2800 | Serotonin Receptor-Targeted Compound Library | 268 compounds | |
A unique collection of 268 compounds targeting serotonin receptors for high throughput screening and high content screening; | |||
L8720 | Pyroptosis Compound Library | 1066 compounds | |
1066 types of active small molecules associated with pyroptosis for high-throughput and high-content screening. | |||
L6030 | Natural Product Derivatives Library for CADD | 163000 compounds | |
Large quantity: contains 163,000 natural product derivatives and the number is continuously updating; | |||
L1100 | Protease Inhibitor Library | 343 compounds | |
A unique collection of 343 protease and proteasome inhibitors for research in chemical genomics, and drug screening; | |||
L2600 | Neuronal Signaling Compound Library | 2540 compounds | |
A unique collection of 2540 compounds targeting CNS signaling for high throughput screening (HTS) and high content screening (HCS) for new drugs; | |||
L8300 | Chromatin Modification Compound Library | 250 compounds | |
A unique collection of 250 compounds targeting chromatin remodeling pathway for high throughput screening (HTS) and high content screening (HCS); | |||
L6120 | Flavonoid Natural Product Library | 514 compounds | |
A unique collection of 514 flavonoids can be used for high throughput and high content screening; | |||
L1010 | FDA-Approved & Pharmacopeia Drug Library | 3158 compounds | |
3158 compounds from marketed drugs for high throughput screening (HTS) and high content screening (HCS); | |||
L2610 | Neurotransmitter Receptor Compound Library | 1513 compounds | |
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening; | |||
L6130 | Terpene Natural Product Library | 622 compounds | |
A unique collection of 622 natural terpenes and terpenoids can be used for high throughput and high content screening; | |||
L1020 | EMA Approved Drug Library | 657 compounds | |
L2620 | Anti-Neurodegenerative Disease Compound Library | 2154 compounds | |
A unique collection of 2154 compounds related to neurodegenerative diseases can be used for HTS or HCS; | |||
L4200 | FDA-Approved Drug Library | 1729 compounds | |
A unique collection of 1729 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS); | |||
L8110 | Reprogramming Compound Library | 1813 compounds | |
A unique collection of 1813 reprogramming signaling pathway-related bioactive small molecule compounds for high-throughput, high-content screening. | |||
L6800 | Chinese Pharmacopoeia Natural Product Library | 2051 compounds | |
A unique collection of 2051 natural products included in Chinese Pharmacopoeia (CP), a powerful tool for drug development and pharmacological study; | |||
L4710 | Nonsteroidal Anti-Inflammatory Compound Library | 530 compounds | |
530 non-steroidal anti-inflammatory compounds for high-throughput and high-content screening. | |||
L6000 | Natural Product Library for HTS | 4533 compounds | |
A unique collection of 4533 pure natural products and their derivatives with known biological activity for drug discovery, pharmacological study, stem cell differentiation, fingerprint study and quality research, and can... | |||
L5100 | Fluorochemical Library | 574 compounds | |
A unique collection of 574 fluorochemicals that can be used for high through-put screening (HTS) and high content screening (HCS); | |||
L1610 | FDA-Approved Kinase Inhibitor Library | 263 compounds | |
A unique collection of 263 kinase inhibitors/regulators for specific targeting of kinases, ready for high-throughput screening and high-content screening. | |||
L6140 | Saccharide and Glycoside Natural Product Library | 595 compounds | |
A unique collection of 595 saccharides and glycosides compounds can be used for HTS and HCS; | |||
L1520 | Membrane Protein-targeted Compound Library | 4175 compounds | |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T13181 | Tolcapone D7 | Ro 40-7592 D7 | Transferase |
Tolcapone D7 is a deuterium-labeled Tolcapone. Tolcapone is a selective and orally active inhibitor of COMT. | |||
T10118 | 3-O-Methyltolcapone D7 | Ro 40-7591 D7 | Transferase |
3-O-Methyltolcapone D7 (Ro 40-7591 D7) is a deuterium labeled 3-O-Methyltolcapone. 3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor. Tolcapone crosses the blood-brain barrier... | |||
T17047 | Tetrabenazine-d6 | Ro 1-9569 D6 | Others |
Tetrabenazine D6 is the deuterium-labeled Tetrabenazine. Tetrabenazine is a VMAT-inhibitor used for the treatment of hyperkinetic movement disorder. | |||
T13031 | Sulfamethoxazole-d4 | Ro 4-2130 D4 | Others |
Sulfamethoxazole D4 is a deuterium labeled Sulfamethoxazole (Ro 4-2130). Sulfamethoxazole is a sulfonamide bacteriostatic antibiotic. | |||
T11679 | Isavuconazole-d4 | BAL-4815 D4,RO-0094815 D4,Isavuconazole D4 | Others |
Isavuconazole D4 is a deuterium labeled Isavuconazole. Isavuconazole is a triazole prodrug with antifungal activity against yeasts, molds, and dimorphic fungi. | |||
T12571 | PSI-6206 13C,d3 | Sofosbuvir metabolite GS-331007 13CD3,RO-2433 13CD3,PSI-6206 13CD3,GS-331007 13CD3 | Others |
PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor. | |||
T73712 | Metformin-d6 hydrochloride | 1,1-Dimethylbiguanide-d6 hydrochloride | AMPK , Autophagy |
Metformin-d6 hydrochloride (Metformin-d6 hydrochloride) is a deuterated form of Metformin that can be used to study Metformin metabolism in vivo, and is often used as an internal standard for Metformin.ccc_R08 can be use... | |||
T39441 | L-Arginine-15N4 hydrochloride | L-Arginine-15N4 hydrochloride,(S)-(+)-Arginine-15N4 hydrochloride | |
L-Arginine-15N4 ((S)-(+)-Arginine-15N4) hydrochloride, the 15N-labeled variant of L-Arginine hydrochloride ((S)-(+)-Arginine hydrochloride), serves as the nitrogen donor in the synthesis of nitric oxide. This potent vaso... | |||
T37119 | 1,2,3-Trioctanoyl-rac-glycerol-13C3 | 1,2,3-Trioctanoyl-rac-glycerol-13C3 | |
1,2,3-Trioctanoyl-rac-glycerol-13C3 is intended for use as an internal standard for the quantification of 1,2,3-trioctanoyl-rac-glycerol by GC- or LC-MS. 1,2,3-Trioctanoyl-rac-glycerol is a triacylglycerol that contains ... | |||
T13135 | Tetrahydrocurcumin D6 | HZIV 81-2 D6 | Others |
Tetrahydrocurcumin D6 is a deuterium labeled Tetrahydrocurcumin. Tetrahydrocurcumin displays inhibitory activity for CYP2C9 and CYP3A4. | |||
T19201 | Banoxantrone-d12 dihydrochloride | AQ4N D12 dihydrochloride | Others |
Banoxantrone D12 (AQ4N D12) dihydrochloride is the deuterium-labeled Banoxantrone. Banoxantrone is a bioreductive agent that can be reduced to a stable, DNA-affinity compound AQ4, which is a topoisomerase II inhibitor. | |||
TMIH-0197 | DL-Metanephrine-d3 Hydrochloride | ||
DL-Metanephrine-d3 Hydrochloride is a deuterated compound of DL-Metanephrine Hydrochloride. | |||
TMIH-0129 | Bupropion Morpholinol-d8 | ||
Bupropion Morpholinol-d8 is a deuterated compound of Bupropion Morpholinol. | |||
TMIH-0161 | Clencyclohexerol-d10 | ||
Clencyclohexerol-d10 is a deuterated compound of Clencyclohexerol. | |||
TMIH-0054 | 4-Bromobenzoic acid-d4 | ||
4-Bromobenzoic acid-d4 is a deuterated compound of 4-Bromobenzoic acid. 4-Bromobenzoic acid has a CAS number of 586-76-5. | |||
T73711 | Atomoxetine-d3 hydrochloride | ||
Atomoxetine-d3 hydrochloride, the deuterium-labeled form of Atomoxetine hydrochloride, acts as a potent and selective noradrenalin re-uptake inhibitor with Ki values of 5, 77, and 1451 nM for the inhibition of radioligan... | |||
TMIH-0027 | 1-Bromo-4-nitrobenzene-d4 | ||
1-Bromo-4-nitrobenzene-d4 is a deuterated compound of 1-Bromo-4-nitrobenzene. | |||
T10458 | Banoxantrone (D12) | Banoxantrone D12,AQ4N D12 | Others |
Banoxantrone D12 (AQ4N D12) is the deuterium-labeled Banoxantrone. Banoxantrone is a bioreductive agent that can be reduced to a stable, DNA-affinity compound AQ4, which is a topoisomerase II inhibitor. | |||
TMIH-0548 | Tacrolimus-13C-d2 | ||
Tacrolimus-13C-d2 is the 13C and deuterated compound of Tacrolimus. | |||
TMIH-0256 | Glycopyrrolate-d5 | Glycopyrronium Bromide-d5 | |
Glycopyrrolate-d5 is a deuterated compound of Glycopyrrolate. Glycopyrrolate has a CAS number of 596-51-0. Glycopyrrolate is a muscarinic antagonist used as an antispasmodic, in some disorders of the gastrointestinal tra... | |||
TMIH-0195 | DL-4-Hydroxy-3-methoxymandelic-d3 acid | ||
DL-4-Hydroxy-3-methoxymandelic-d3 acid is a deuterated compound of DL-4-Hydroxy-3-methoxymandelic acid. | |||
TMIH-0562 | Testosterone propionate-d3 | ||
Testosterone propionate-d3 is a deuterated compound of Testosterone propionate. | |||
T12487 | Piroxicam D3 | CP-16171 D3 | Others |
Piroxicam D3 is deuterium labeled Piroxicam. Piroxicam is a COX inhibitor(human monocyte COX-1 and COX-2 with IC50s of 47, 25 μM , respectively) . | |||
T12550 | Propranolol-d7 hydrochloride | Propranolol D7 hydrochloride | Others |
Propranolol D7 hydrochloride is a deuterium labeled Propranolol hydrochloride. Propranolol hydrochloride is a nonselective antagonist of β-adrenergic receptor (βAR). | |||
T12800 | (S)-(+)-Ibuprofen D3 | (S)-Ibuprofen D3 | COX |
(S)-(+)-Ibuprofen D3 is a deuterium labeled (S)-(+)-Ibuprofen. (S)-(+)-Ibuprofen is the S(+)-enantiomer of Ibuprofen ,it is an inhibitor of COX-1 and COX-2 activity (IC50s of 2.1 μM and 1.6 μM). | |||
T10181 | 6-beta-Naloxol D5 hydrochloride | 6β-Naloxol D5 hydrochloride | Others |
6-beta-Naloxol D5 hydrochloride is a deuterium-labeled opioid antagonist, closely related to naloxone, that serves as an effective compound in the field of chemical research. | |||
T10282 | Aliskiren D6 Hydrochloride | SPP 100 D6 Hydrochloride,CGP60536B D6 Hydrochloride,CGP 60536 D6 Hydrochloride | Others |
Aliskiren (CGP 60536) D6 Hydrochloride is a deuterium-labeled Aliskiren. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM). | |||
TMIH-0383 | N-Despropyl Macitentan-d4 | ||
N-Despropyl Macitentan-d4 is a deuterated compound of N-Despropyl Macitentan. N-Despropyl Macitentan has a CAS number of 1103522-45-7. Aprocitentan is ETA and ETB antagonist . | |||
TMIH-0268 | Hydroxy Tetramethylpyrazine-d11 | ||
Hydroxy Tetramethylpyrazine-d11 is a deuterated compound of Hydroxy Tetramethylpyrazine. | |||
T71328 | Theobromine-d6 | ||
Theobromine-d6 is intended for use as an internal standard for the quantification of theobromine by GC- or LC-MS. Theobromine is a methylxanthine alkaloid and derivative of caffeine that has been found in cocoa beans and... | |||
T12545 | Proguanil D6 | Others | |
Proguanil D6 is the deuterium labeled Proguanil, and is an agent of prophylactic antimalarial. | |||
T11252 | Ezetimibe phenoxy glucuronide-D4 | Ezetimibe β-D-glucuronide-D4,Ezetimibe glucuronide-D4 | Others |
Ezetimibe phenoxy glucuronide-D4 (Ezetimibe glucuronide-D4) is the deuterium labeled Ezetimibe phenoxy glucuronide. | |||
T11585 | Hydroxy Itraconazole D8 | R-63373 D8 | Others |
Hydroxy Itraconazole D8 is the deuterium-labeled Hydroxy Itraconazole. Hydroxy Itraconazole is an active metabolite of Itraconazole, which is a triazole antifungal agent. | |||
TMIH-0273 | Hydroxyzine dihydrochloride-d10 | (R)-2-(2-(4-((4-chlorophenyl)(phenyl)methyl)pi perazin-1-yl-2,2,3,3,5,5,6,6-d8)ethoxy)ethan-1, 1-d2-1-ol dihydrochloride | |
Hydroxyzine dihydrochloride-d10 is a deuterated compound of Hydroxyzine dihydrochloride. | |||
T11604 | Ibuprofen-d3 | Ibuprofen D3,(±)-Ibuprofen D3 | Others |
Ibuprofen D3 is a deuterium labeled Ibuprofen. Ibuprofen is a COX-1 and COX-2 inhibitor (IC50s: 13 μM and 370 μM). | |||
TMIH-0366 | Nandrolone-d3 | ||
Nandrolone-d3 is a deuterated compound of Nandrolone. | |||
TMIH-0475 | Rac threo-Dihydro Bupropion-d9 Hydrochloride | ||
rac threo-Dihydro Bupropion-d9 Hydrochloride is a deuterated compound of rac threo-Dihydro Bupropion Hydrochloride. rac threo-Dihydro Bupropion Hydrochloride has a CAS number of 1396889-62-5. | |||
T64761 | 5-(Methyl-d3)-dibenzothiophenium, 1,1,1-trifluoromethanesulfonate | ||
5-(Methyl-d3)-dibenzothiophenium, 1,1,1-trifluoromethanesulfonate is a useful organic compound for research related to life sciences and the catalog number is T64761. | |||
T30599 | BS3-d4 Deuterated Crosslinker | Deuterated Crosslinker BS3-d4,BS3-d4,D4-BS3 | |
BS3-d4 Deuterated Crosslinker or Bis(Sulfosuccinimidyl) 2,2,7,7-suberate-d4, is a water-soluble and membrane impermeable protein crosslinking agent. | |||
T71206 | Tiagabine-d6 hydrochloride | ||
Tiagabine-d6 is intended for use as an internal standard for the quantification of tiagabine by GC- or LC-MS. Tiagabine is an inhibitor of GABA transporter 1. It inhibits seizures induced by DMCM in mice. Tiagabine reduc... | |||
TMIH-0457 | Proguanil-d6 HCl | ||
Proguanil-d6 HCl is a deuterated compound of Proguanil HCl. Proguanil HCl has a CAS number of 637-32-1. Proguanil Hydrochloride is a biguanide compound which metabolizes in the body to form cycloguanil, an anti-malaria a... | |||
TMIH-0482 | Ractopamine-d5 Hydrochloride | ||
Ractopamine-d5 Hydrochloride is a deuterated compound of Ractopamine Hydrochloride. | |||
TMIH-0146 | Chloroquine-d5 | ||
Chloroquine-d5 is a deuterated compound of Chloroquine. Chloroquine has a CAS number of 54-05-7. Chloroquine is an autophagy and toll-like receptors (TLRs) inhibitor. Chloroquine is an antimalarial and anti-inflammatory ... | |||
TMIH-0016 | (S)-Metoprolol-d7 | ||
(S)-Metoprolol-d7 is a deuterated compound of (S)-Metoprolol. (S)-Metoprolol has a CAS number of 37350-58-6. | |||
TMIH-0031 | 25-Hydroxy vitamin D2-d3 | ||
25-Hydroxy vitamin D2-d3 is a deuterated compound of 25-Hydroxy vitamin D2. | |||
TMIH-0467 | Pyridoxine-d3 Hydrochloride | ||
Pyridoxine-d3 Hydrochloride is a deuterated compound of Pyridoxine Hydrochloride. | |||
TMIH-0561 | Testosterone-d5 | ||
Testosterone-d5 is a deuterated compound of Testosterone. | |||
TMIH-0151 | Cimbuterol-d9 | ||
Cimbuterol-d9 is a deuterated compound of Cimbuterol. | |||
T19252 | Cyantraniliprole-d3 | DPX-HGW86 D3,HGW-86 D3 | Others |
Cyantraniliprole D3 is deuterium-labeled Cyantraniliprole, which is a Ryan-like insecticide. | |||
T19273 | Debutyldronedarone D7 | SR-35021 D7 | Others |
Debutyldronedarone D7 is deuterium-labeled Debutyldronedarone, which is the main circulating active metabolite of dronedarone in the body. | |||
------------------------ More ------------------------ |