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Histone Demethylase 5-HT Receptor DNA/RNA Synthesis Sodium Channel NMDAR AChR

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カタログ番号	製品名	別名	ターゲット
T0802	Procaine hydrochloride	Novocaine HCl,Procaine HCl	Histone Demethylase , 5-HT Receptor , DNA/RNA Synthesis , Sodium Channel , NMDAR , AChR
	Procaine hydrochloride (Novocaine HCl) is the hydrochloride salt form of procaine, a benzoic acid derivative with local anesthetic and antiarrhythmic properties. Procaine binds to and inhibits voltage-gated sodiumchannel...
T0029	Procaine	Duracaine,Spinocaine,Novocaine,Vitamin H3	Histone Demethylase , DNA/RNA Synthesis , Sodium Channel
	Procaine (Vitamin H3) is a local anesthetic of the ester type that has a slow onset and a short duration of action. It is mainly used for infiltration anesthesia, peripheral nerve block, and spinal block.		Histone Demethylase , DNA/RNA Synthesis , Sodium Channel
T8598	CHEMBL241987	2-PHENYL-2,5-DIHYDRO-4H-PYRAZOLO[3,4-C]QUINOLIN-4-ONE	Adenosine Receptor
	CHEMBL241987 targets the Adenosine receptor A3 (human)		Adenosine Receptor
T19241	Cloquintocet-mexyl		Others
	Cloquintocet-mexyl, a herbicide, targets and controls coarse annual grasses within the Poaceae family.		Others
T19849L	2-PADQZ hydrochloride	2-PADQZ hydrochloride (60547-97-9 Free base)	Antiviral , Influenza Virus
	2-PADQZ hydrochloride shows antiviral activity and targets influenza A virus RNA promoter.		Antiviral , Influenza Virus
T8635	CI 75300		P2X Receptor
	CI 75300 targets the P2X purinoceptor 7 (human).		P2X Receptor
T8912	5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE		PLK
	5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE targets PLK1.		PLK
T16546	PK 11195	RP 52028	Others
	PK 11195 is a ligand of translocator protein. It targets Leishmania chemotherapy (IC50s of 14.2 μM, 8.2 μM, 3.5 μM for L. amazonensis, L. major and L. braziliensis, respectively).		Others
T9827	Carfenazine		Dopamine Receptor
	carfenazine targets the Dopamine receptor and is used for schizophrenia research.		Dopamine Receptor
T8913	1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID		GRK
	1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.		GRK
T9061	EN4	EN4 MYC inhibitor	c-Myc
	EN4 (EN4 MYC inhibitor) MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits MYC transcriptional activity, downregulates MYC targets, an...		c-Myc
T8672	2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE	BisOPP-A	Thyroid hormone receptor(THR)
	2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE is targets the thyroid stimulating hormone receptor (human)		Thyroid hormone receptor(THR)
T9884	EN523		Others
	EN523 targets non-catalytic allosteric cysteine C23 in K48 ubiquitin-specific deuquitinase OTUB1.		Others
T9751	Transfluthrin		Others
	Transfluthrin is a volatile pyrethroid insecticide that targets insect voltage-gated sodium channels (VGSC).		Others
T62620	ZY-444
	ZY-444 is a small molecule that inhibits the progression of breast cancer and targets pyruvate carboxylase.
T5173	SBI-0640756	SBI 0640756,SBI-756	PERK , Autophagy
	SBI-0640756 (SBI-756) (SBI-756) is a first-in-class inhibitor that targets eIF4G1 and disrupts the eIF4F complex.		PERK , Autophagy
T0998	Diazinon	Dimpylate	AChE , Parasite
	Diazinon (Dimpylate) is a thiophosphoric acid ester, functioning as a nonsystemic organophosphate insecticide that effectively targets and controls a variety of pests including cockroaches, silverfish, ants, and fleas.		AChE , Parasite
T6094	MK-2461	MK2461	c-Met/HGFR
	MK-2461 is a novel inhibitor that targets multiple proteins and competitively binds to ATP sites, specifically inhibiting the activated c-Met protein with an average inhibitory concentration (IC50) of 2.5 nM.		c-Met/HGFR
T8584	6-Phenyldihydropyrimidine-2,4(1h,3h)-dione	2,4(1H,3H)-Pyrimidinedione,dihydro-6-phenyl-	Others
	6-Phenyldihydropyrimidine-2,4(1h,3h)-dione targets the polypyrimidine tract-binding protein 1 isoform a (human)		Others
T10232	Acetophenazine dimaleate		Dopamine Receptor
	Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.		Dopamine Receptor
TNU0436	2-Thiocytidine		Apoptosis , Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis
	2-Thiocytidine is a purine nucleoside analog that targets malignant tumors of the inert lymphatic system and has a broad spectrum of antitumor activity.2-Thiocytidine induces apoptosis by inhibiting DNA synthesis.2-Thioc...
T8602	2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA6-BENZO[D]ISOTHIAZOL-3-ONE		Serine Protease
	2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA6-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).		Serine Protease
T22418	S-99		Others
	S-99 is a high purity chemical that targets ASK and is important for Immunology, Inflammation, Cancer research.		Others
T19206	β-Lactamase-IN-1	4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one,beta-lactamase-IN-1	Antibacterial
	β-Lactamase-IN-1 (4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one) is a β-Lactamase inhibitor and targets the infection of Neisseria gonorrhoeae.		Antibacterial
T16925	SQ109	NSC 722041	Others , Parasite
	SQ109 (NSC-722041) is an effective inhibitor of the trypomastigote form of the parasite (IC50 = 50 nM). SQ109 is an antitubercular agent and targets MmpL3.		Others , Parasite
T33296	Merodantoin		Apoptosis
	Merodantoin is an apoptosis inducer and triggers cell apoptosis associated with ROS-dependent autophagy. Merodantoin targets cancer cells expressing KRAS mutations involved in Akt-dependent ROS production.		Apoptosis
T8603	ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE		Prostaglandin Receptor
	ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE targets the prostaglandin E2 receptor EP2 subtype (human)		Prostaglandin Receptor
T9901	Adalimumab		TNF
	Adalimumab (anti-TNF-alpha) is the first fully human recombinant IgG1 monoclonal antibody that specifically targets human TNF-alpha.		TNF
T7330	Nucleozin		Influenza Virus
	Nucleozin targets influenza A nucleoprotein (NP), a multifunctional, RNA-binding protein necessary for virus replication.		Influenza Virus
T1801	SR9243		Liver X Receptor
	SR9243, an LXR inverse agonist, can induce LXR-corepressor interaction; shows anticancer activity and selectively targets the lipogenesis and Warburg effect.		Liver X Receptor
T40811	Eflornithine	RMI71782,α-difluoromethylornithine,DFMO,MDL71782
	Eflornithine is an irreversible inhibitor that specifically targets the enzyme ornithine decarboxylase. It serves as a therapeutic medication for two conditions: the treatment of African trypanosomiasis and the managemen...
T35544	ML115		STAT
	ML115 is a potent and selective activator of transcription 3 (STAT3), with abn EC50 of 2.0 nM, and is inactive against the related STAT1 and NFκB anti-targets.		STAT
T5345	V-9302		Others
	V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uM).		Others
TQ0064	Peretinoin	NIK333	HCV Protease , Retinoid Receptor , S1P Receptor , Autophagy
	Peretinoin (NIK333) is an oral acyclic retinoid with a vitamin A-like structure that targets retinoid nuclear receptors such as RXR and RAR.		HCV Protease , Retinoid Receptor , S1P Receptor , Autophagy
T6562	Latrepirdine dihydrochloride	Dimebolin dihydrochloride,Latrepirdine,Latrepirdine 2HCl,Dimebolin	Beta Amyloid , 5-HT Receptor , Adrenergic Receptor , GluR , Autophagy , Histamine Receptor
	Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors, GluR, and 5-HT receptors, used as an antihistamine drug.
T15373	Gboxin		ATPase , Mitochondrial Metabolism
	Gboxin is an inhibitor of oxidative phosphorylation that targets glioblastoma,inhibits the activity of F0F1 ATP synthase, with antitumour activity.		ATPase , Mitochondrial Metabolism
T77768	BAY 1892005		p53
	BAY 1892005 is a p53 protein modulator that targets the p53 condenser for the study of diseases associated with misfolded p53 protein		p53
T5396	Letermovir	AIC246,MK-8828	Others , HCV Protease
	Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.		Others , HCV Protease
T16128	MP-A08		S1P Receptor
	MP-A08 is a highly selective ATP competitive inhibitor of sphingosine kinase (SPHK1) that targets both SphK1 and SphK2 (Ki: 6.9 ± 0.8 μM and 27 ± 3 μM, respectively).		S1P Receptor
T16560	Poloxin		PLK
	Poloxin is a non-ATP competitive Polo-like Kinase 1 inhibitor. It targets the polo-box domain (IC50: appr 4.8 μM).		PLK
T6824	EAI045		EGFR
	EAI045, an allosteric inhibitor, targets towards drug-resistant EGFR mutants but avoids the wild-type receptor.		EGFR
T4665	Temsavir	BMS626529	HIV Protease
	Temsavir (BMS626529) is a novel attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T cells.		HIV Protease
T77945	TriGalNAc CBz		LYTACs
	TriGalNAc CBz is a GalNAc derivative. As an ASGPR ligand, tri-GalNAc targets lysosomes in mRNA drug delivery and LYTAC studies.L-DABA hydrobromide.		LYTACs
T15675	Tirbanibulin Mesylate	KX2-391 Mesylate,KX01 Mesylate	Microtubule Associated , Src
	Tirbanibulin Mesylate (KX01 Mesylate) is an inhibitor of Src that targets the peptide substrate site of Src (GI50: 9-60 nM in cancer cell lines).		Microtubule Associated , Src
T9914	Vedolizumab		Integrin
	Vedolizumab is a humanized monoclonal antibody that targets the α4β7 integrin for the treatment of Crohn's disease and ulcerative colitis.		Integrin
T9230	KM 91104		ATPase
	KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.		ATPase
T1948	AZD4547		VEGFR , FGFR
	AZD4547, a new-type specific FGFR inhibitor, targets for FGFR1/2/3 (IC50: 0.2/2.5/1.8 nM in cell-free assays).		VEGFR , FGFR
T74140	β-D-Glucan		Others
	β-D-Glucan is a compound that targets tumor-associated macrophages with antitumor activity and modulates the immune response in necrotizing pancreatitis.		Others
T8925	Glu-urea-Lys
	Glu-urea-Lys is a molecular scaffold that targets PSMA and can be used as a prostate cancer imaging agent to study prostate-specific membrane antigens.
T8587	EcDsbB-IN-12	4,5-dichloro-2-[(2-chlorophenyl)methyl]pyridazin-3-one	Others
	EcDsbB-IN-12 (4,5-dichloro-2-[(2-chlorophenyl)methyl]pyridazin-3-one) targets disulfide bond forming enzyme,and is a novel potent specific inhibitor of EcDsbB.		Others

Compounds

Procaine hydrochloride

T0802

Synonym: Novocaine HCl,Procaine HCl

Target: Histone Demethylase, 5-HT Receptor, DNA/RNA Synthesis, Sodium Channel, NMDAR, AChR

Procaine

T0029

Synonym: Duracaine,Spinocaine,Novocaine,Vitamin H3

Target: Histone Demethylase, DNA/RNA Synthesis, Sodium Channel

CHEMBL241987

T8598

Synonym: 2-PHENYL-2,5-DIHYDRO-4H-PYRAZOLO[3,4-C]QUINOLIN-4-ONE

Target: Adenosine Receptor

2-PADQZ hydrochloride

T19849L

Synonym: 2-PADQZ hydrochloride (60547-97-9 Free base)

Target: Antiviral, Influenza Virus

5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE

Target: Dopamine Receptor

1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID

Synonym: EN4 MYC inhibitor

Target: c-Myc

2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE

T8672

Synonym: BisOPP-A

Target: Thyroid hormone receptor(THR)

Synonym: SBI 0640756,SBI-756

Target: PERK, Autophagy

Diazinon

T0998

Synonym: Dimpylate

Target: AChE, Parasite

6-Phenyldihydropyrimidine-2,4(1h,3h)-dione

T8584

Synonym: 2,4(1H,3H)-Pyrimidinedione,dihydro-6-phenyl-

Target: Others

Acetophenazine dimaleate

T10232

Synonym:

Target: Dopamine Receptor

2-Thiocytidine

TNU0436

Synonym:

Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis

2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE

T8602

Synonym:

Target: Serine Protease

Synonym: 4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one,beta-lactamase-IN-1

Target: Antibacterial

SQ109

T16925

Synonym: NSC 722041

Target: Others, Parasite

ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE

T8603

Synonym:

Target: Prostaglandin Receptor

Target: Influenza Virus

SR9243

T1801

Synonym:

Target: Liver X Receptor

Eflornithine

T40811

Synonym: RMI71782,α-difluoromethylornithine,DFMO,MDL71782

Target: HCV Protease, Retinoid Receptor, S1P Receptor, Autophagy

Latrepirdine dihydrochloride

T6562

Synonym: Dimebolin dihydrochloride,Latrepirdine,Latrepirdine 2HCl,Dimebolin

Target: Beta Amyloid, 5-HT Receptor, Adrenergic Receptor, GluR, Autophagy, Histamine Receptor

Gboxin

T15373

Synonym:

Target: ATPase, Mitochondrial Metabolism

Synonym: AIC246,MK-8828

Target: Others, HCV Protease

Tirbanibulin Mesylate

T15675

Synonym: KX2-391 Mesylate,KX01 Mesylate

Target: Microtubule Associated, Src

Synonym: 4,5-dichloro-2-[(2-chlorophenyl)methyl]pyridazin-3-one

Target: Others

カタログ番号	製品名	別名	ターゲット
T8229	5,7,3',4'-Tetramethoxyflavone		Antibacterial , Parasite , Antifungal
	5,7,3',4'-Tetramethoxyflavone (TMF), a prominent polymethoxyflavone (PMF) derived from M. exotica, displays a range of notable bioactivities. These include anti-malarial, anti-fungal, anti-mycobacterial, and anti-inflamm...		Antibacterial , Parasite , Antifungal
T2831	Glycocholic acid	Glycocholate,cholylglycine	Others , Endogenous Metabolite
	Glycocholic acid (Glycocholate) is a bile acid with anticancer activity. Glycocholic acid targets against pump resistance-related and non-pump resistance-related pathways.		Others , Endogenous Metabolite
T3021	Bulleyaconitine A	Bulleyaconi cine A	Sodium Channel
	Bulleyaconitine A (Bulleyaconi cine A), an analgesic and antiinflammatory drug isolated from Aconitum plants, has several potential targets, such as voltage-gated Na+ channels.		Sodium Channel
T17048	Tetradecanoylcarnitine	L-Myristoylcarnitine,Myristoyl-L-(-)-carnitine	Endogenous Metabolite
	Tetradecanoylcarnitine (L-Myristoylcarnitine) is an acylcarnitine involved in the beta-oxidation of long-chain fatty acids, and is a potential marker for very-long-chain coenzyme A dehydrogenase deficiency. alpha-Dihydro...		Endogenous Metabolite
TN2373	(E/Z)-Ginkgolic acid C17:2	Ginkgolic Acid C17:2	Dehydrogenase
	(E/Z)-Ginkgolic acid C17:2 (Ginkgolic Acid C17:2) is a natural product that can be extracted from Ginkgo biloba and targets human dihydroorotic acid dehydrogenase (DHODH).		Dehydrogenase
TN1403	Arjunolic acid		IL Receptor , TNF , Reactive Oxygen Species , JNK , AChE
	Arjunolic acid has antioxidant, anti-inflammatory, antinociceptive and anticholinesterasic (AChE and BuChE) activities, it may as promising targets for the development of innovative multi-functional medicines for Alzheim...		IL Receptor , TNF , Reactive Oxygen Species , JNK , AChE
T1558	Resveratrol	trans-Resveratrol,SRT 501	Apoptosis , Mitophagy , IκB/IKK , Lipoxygenase , Sirtuin , COX , NADPH , DNA/RNA Synthesis , Nrf2 , Antibacterial , Antibiotic , Autophagy , Antifungal
	Resveratrol (SRT 501) is a polyphenolic natural product, a plant antitoxin with antioxidant and chemopreventive activities. Resveratrol has a wide range of targets including COX, SIRT, LOC, etc. Resveratrol induces autop...
T14046	Anandamide	(5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide	Cannabinoid Receptor , Endogenous Metabolite
	Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but also other targets (e.g., GPR18/GPR55) in the central nervous sy...		Cannabinoid Receptor , Endogenous Metabolite
T14304	Aphidicolin		Others
	Aphidicolin, an antibiotic derived from the mold Cephalosporium aphidicola, is a potent inhibitor of DNA (deoxyribonucleic acid) synthesis, effectively hindering the proliferation of herpes simplex virus[2]. It targets D...		Others
TN1249	3-Epiursolic acid		Cysteine Protease , Immunology/Inflammation related
	3-Epiursolic acid may have antiinflammatory activity, it shows inhibition on Cathepsins L (catL), the IC50 value of 6.5 μM, cathepsins L (catL) and B play an important role in tumor progression and have been considered p...		Cysteine Protease , Immunology/Inflammation related
T6981	1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid	Nudifloric Acid	Others
	1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid (Nudifloric Acid) is from Cordyceps bassiana. Nudifloric Acid targets to block AP-1-mediated luciferase activity, implying it has an anti-inflammatory function.		Others
T4808	Agmatine sulfate	Agmatine sulfate salt	Endogenous Metabolite , NO Synthase , Imidazoline Receptor
	Agmatine sulfate (Agmatine sulfate salt) is a bioactive metabolite of the arginine amino acid. It exerts modulatory action at multiple molecular targets, such as neurotransmitter systems, ion channels and nitric oxide sy...		Endogenous Metabolite , NO Synthase , Imidazoline Receptor
TN1015	Meranzin		Adrenergic Receptor , Immunology/Inflammation related
	Meranzin, a bioactive compound derived from the Traditional Chinese Medicine (TCM) Chaihu-Shugan-San (CSS) and isolated from Murraya exotica L. leaves, targets the alpha 2-adrenoceptor and engages the AMPA-ERK1/2–BDNF si...		Adrenergic Receptor , Immunology/Inflammation related
TN1620	Eriocalyxin B		Apoptosis , cAMP , NF-κB , STAT
	Eriocalyxin B induces apoptosis and cell cycle arrest in pancreatic adenocarcinoma cells through caspase- and p53-dependent pathways, should be considered a candidate for pancreatic cancer treatment; it is a specific inh...		Apoptosis , cAMP , NF-κB , STAT
T4900	(±)-Methyl Jasmonate	(±)-Jasmonic Acid methyl ester,Methyl 2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate	Others , Endogenous Metabolite
	Methyl 2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate ((±)-Jasmonic Acid methyl ester)induces the synthesis of proteinase inhibitors in plant leaves. In cancer cells, it suppresses proliferation and induces apoptosis. Mo...		Others , Endogenous Metabolite
T2S1792	Lycobetaine	Ungeremine	Antibacterial
	1. Lycobetaine (Ungeremine) is a potential biofungicide against Penicillium roqueforti and Aspergillus niger.2. Lycobetaine have strong antibacterial activity against Flavobacterium columnare . 3. Lycobetaine effectively...		Antibacterial
T25664	Lepidiline A	Macaline A	Others
	Lepidiline A (Macaline A) is a flavonoid lignin with anti-inflammatory activity. Lepidiline A showed cytotoxic activity against HL-60 cells with IC50 of 32.3 μM. It is the active ingredient of Lepidium meyenii Walpers, a...		Others
T3729	Ethyl gallate	Nipagallin A,Phyllemblin,gallic acid ethyl ester	MMP , NF-κB , Akt , Antibacterial
	Ethyl gallate (gallic acid ethyl ester) obviously decreases cell proliferation in MDA-MB-231 and MCF-7 cells in a dose- and time-dependent manner, exhibits cytotoxicity in a dose-dependent manner. Ethyl gallate can inhib...		MMP , NF-κB , Akt , Antibacterial
T5S2343	Acetylshikonin	Acetyl shikonin	Others , P450 , AChE
	1. Acetylshikonin exhibits weak cytotoxicity against human umbilical vein endothelial cells (HUVECs) with IC5 of over 2 microM, exhibits the antiangiogenic and antitumorigenic effects by suppressing proliferation and ang...		Others , P450 , AChE
T40298	Phallacidin
	Phallacidin, a phallotoxin family member, targets and binds to F-actin in mushroom toxins.
T11274	Ferulenol		Others
			Others
T39918	(±)-Phrymarolin II
	(±)-Phrymarolin II is a promising class of inhibitors that targets the tobacco mosaic virus, representing a novel approach in plant virus suppression.
TN1550	Danshenxinkun A		Others
	Danshenxinkun A, Danshenxinkun B and Neocryptotanshinone may intervene thrombotic diseases by adjusting the targets mainly involved in pathways of endocrine system, signal transduction, signaling molecules and interactio...		Others
T80779	WDB002
	WDB002, a natural product belonging to the FK506/rapamycin family, targets CEP250 and may be employed in COVID-19 research [1].
TN4860	Pueroside B		COX , PPAR
	Pueroside B may can treat coronary heart disease, it can interact with two or more targets[peroxisome proliferator activated receptor γ (PPAR-γ), angiotensin-converting enzyme (ACE), hydroxymethylglutaryl coenzyme A rece...		COX , PPAR
TN2360	Falcarinol	Falcarinol,Panaxynol	HSP
	Falcarinol, also known as Panaxynol, is a naturally occurring compound that acts as an orally active inhibitor of Hsp90. It effectively targets both the N-terminal and C-terminal regions of Hsp90, displaying high selecti...		HSP
T38441	Manzamine A hydrochloride
	Manzamine A hydrochloride is an orally active beta-carboline alkaloid that exhibits specific inhibitory effects on GSK-3β (IC50 = 10.2 μM) and CDK-5 (IC50 = 1.5 μM). Additionally, it targets vacuolar ATPases, leading to ...
T75489	Mildiomycin
	Mildiomycin, an antibiotic produced by Streptoverticillium rimofaciens, effectively targets powdery mildew in barley. It also suppresses the growth of certain Mycobacterium and Rhodotorula species, though it is ineffecti...
T82326	Genkwadaphnin
	Genkwadaphnin, a daphnane diterpenoid, targets importin-β1, reducing the nuclear accumulation of CRPC drivers and suppressing downstream oncogenic signaling. Demonstrating potent anti-tumor effects, it inhibits castratio...
T75686	Enfumafungin
	Enfumafungin, a triterpene glycoside extracted from Hormonema carpetanum fungus, acts as an antifungal by inhibiting (1,3)-beta-D-glucan synthase, crucial for fungal cell wall synthesis. It selectively targets yeasts and...
T75333	Quinine hemisulfate hydrate
	Quinine hemisulfate hydrate, an alkaloid extracted from the cinchona tree bark, serves as an anti-malarial agent and potassium channel inhibitor. It specifically targets and inhibits WT mouse Slo3 (K Ca 5.1) channel curr...
T75491	3-(2-Hydroxyethyl) thio withaferin A
	3-(2-Hydroxyethyl) thio withaferin A, a derivative of Withaferin A, is a steroidal lactone that inhibits NF-kB activation and targets vimentin, showcasing potent anti-inflammatory and anticancer properties. It also acts ...
T73072	PTP1B-IN-20
	PTP1B-IN-20 is a selective PTP1B (protein tyrosine phosphatase 1B) inhibitor, exhibiting an IC50 of 1.05 μM, and demonstrates selectivity over TCPTP (T-cell protein tyrosine phosphatase), which has an IC50 of 78.0 μM. Th...
TN5369	Dehydroleucodine	Dehydroleucodin
	Dehydroleucodine has antidiarrheal, anti-inflammatory, anti-microbial, embryotoxicity, gastric cytoprotective, anti-cancer activities. Dehydroleucodine has an important inhibitory effect in cellular pathways regulating a...
T73206	Wikstrol A
	Wikstrol A, a potent antifungal, antimitotic, and anti-HIV-1 agent, demonstrates significant effects across various biological targets. It induces morphological deformation in P. oryzae mycelia, with a minimum morphologi...
T35770	Cylindrospermopsin
	Cylindrospermopsin, a tricyclic uracil derivative, is a cyanobacterial toxin that was first discovered in an algal bloom contaminating a local drinking supply on Palm Island in Queensland, Australia after an outbreak of ...
TN4286	Isodunnianol		NOS , NF-κB , ROS , AChR
	Isodunnianol exhibits anti-AChE activity with an IC50 value of 13.0 uM; it also exhibits neurite outgrowth-promoting activity at the concentration ranging from 0.1 to 10 uM in the primary cultured rat cortical neurons. I...		NOS , NF-κB , ROS , AChR
T75540	Ipomoeassin F
	Ipomoeassin F, a selective and potent inhibitor of endoplasmic reticulum (ER) protein translocation, targets the Sec61 complex's pore-forming subunit (Sec61α) at the ER membrane. It inhibits the ER membrane translocation...
T36563	(E)-Guggulsterone
	Bile acids are essential for solubilization and transport of dietary lipids, are the major products of cholesterol catabolism, and are physiological ligands for farnesoid X receptor (FXR), a nuclear receptor that regulat...

天然物製品

5,7,3',4'-Tetramethoxyflavone

T8229

Synonym:

Target: Antibacterial, Parasite, Antifungal

Glycocholic acid

T2831

Synonym: Glycocholate,cholylglycine

Target: Others, Endogenous Metabolite

Bulleyaconitine A

T3021

Synonym: Bulleyaconi cine A

Target: Sodium Channel

Tetradecanoylcarnitine

T17048

Synonym: L-Myristoylcarnitine,Myristoyl-L-(-)-carnitine

Target: Endogenous Metabolite

(E/Z)-Ginkgolic acid C17:2

TN2373

Synonym: Ginkgolic Acid C17:2

Target: Dehydrogenase

Arjunolic acid

TN1403

Synonym:

Target: IL Receptor, TNF, Reactive Oxygen Species, JNK, AChE

Resveratrol

T1558

Synonym: trans-Resveratrol,SRT 501

Target: Apoptosis, Mitophagy, IκB/IKK, Lipoxygenase, Sirtuin, COX, NADPH, DNA/RNA Synthesis, Nrf2, Antibacterial, Antibiotic, Autophagy, Antifungal

Anandamide

T14046

Synonym: (5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide

Target: Cannabinoid Receptor, Endogenous Metabolite

Target: Cysteine Protease, Immunology/Inflammation related

1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid

T6981

Synonym: Nudifloric Acid

Target: Others

Agmatine sulfate

T4808

Synonym: Agmatine sulfate salt

Target: Endogenous Metabolite, NO Synthase, Imidazoline Receptor

Meranzin

TN1015

Synonym:

Target: Adrenergic Receptor, Immunology/Inflammation related

Eriocalyxin B

TN1620

Synonym:

Target: Apoptosis, cAMP, NF-κB, STAT

(±)-Methyl Jasmonate

T4900

Synonym: (±)-Jasmonic Acid methyl ester,Methyl 2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate

Target: Others, Endogenous Metabolite

Lycobetaine

T2S1792

Synonym: Ungeremine

Target: Antibacterial

Synonym: Nipagallin A,Phyllemblin,gallic acid ethyl ester

Target: MMP, NF-κB, Akt, Antibacterial

Acetylshikonin

T5S2343

Synonym: Acetyl shikonin

Target: Others, P450, AChE

Synonym: Falcarinol,Panaxynol

Target: HSP

Manzamine A hydrochloride

Quinine hemisulfate hydrate

T75333

Synonym:

Target:

3-(2-Hydroxyethyl) thio withaferin A

Synonym: Dehydroleucodin

Target: NOS, NF-κB, ROS, AChR

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-02801	PHGDH Protein, Human, Recombinant (His)	Human	E. coli
	PHGDH is a member of the D-isomer specific 2-hydroxyacid dehydrogenase family. This new family consists of D-isomer-stereospecific enzymes. The conserved residues in this family appear to be the residues involved in the ...
TMPY-02779	Thyroid peroxidase Protein, Human, Recombinant (S257A & P725T, His)	Human	Baculovirus Insect Cells
	Thyroid peroxidase is a membrane-bound glycoprotein which belongs to the peroxidase family, XPO subfamily. It contains 1 EGF-like domain and 1 Sushi (CCP/SCR) domain. Thyroid Peroxidase represents one of the main autoant...
TMPJ-00051	IL-3 Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Interleukin 3 is a pleiotropic factor produced primarily by activated T cells that can stimulate the proliferation and differentiation of pluripotent hematopoietic stem cells as well as various lineage committed progenit...
TMPJ-00042	TSLP Protein, Human, Recombinant	Human	E. coli
	Thymic stromal lymphopoietin (TSLP) is a novel member of the hemopoietic cytokine family that promotes the development of B cells and shares overlapping activity with IL-7. The human TSLP protein comprises a 28 amino aci...
TMPK-01369	S100B Protein, Canine, Recombinant (hFc)	Canine	HEK293 Cells
	S100B, a calcium-binding protein of the EF-hand type exerts both intracellular and extracellular functions.The intracellular, and extracellular, roles of S100B are attractive therapeutic targets for the treatment of both...
TMPY-02760	CALML3 Protein, Human, Recombinant (His)	Human	E. coli
	Calmodulin-like protein 3 (CALML3) is similar to that of authentic calmodulin and may actually compete with calmodulin by binding, with different affinity, to cellular substrates. Calmodulin-like protein 3 (CALML3) is a ...
TMPY-05099	GBA/glucocerebrosidase Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Mutations in the GBA gene, encoding the lysosomal hydrolase glucocerebrosidase (GCase), are the most common known genetic risk factor for Parkinson's disease (PD) and dementia with Lewy bodies (DLB). ASAH1 (acid ceramida...
TMPK-00280	B7-H6 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	B7-H6 is a glycosylated member of the B7 family of immune co‑stimulatory proteins. which is a ligand for the NK cell activating receptor NKp30, was targeted to create a CAR that targets multiple tumor types. B7H6 is expr...
TMPH-03369	SEMA3A Protein, Rat, Recombinant (His)	Rat	E. coli
	May be involved in guiding growing axons towards their targets by forming a molecular boundary that instructs axons to engage in the formation of specific nerve tracts. Binds to neuropilin. Involved in the development of...
TMPJ-01335	MOB1A Protein, Human, Recombinant (His)	Human	E. coli
	MOB Kinase Activator 1A (MOB1A) belongs to the MOB1/phocein family, which acts as an activator of LATS1/2 in the Hippo signaling pathway, plays a key role in organ size control and tumor suppression by restricting prolif...
TMPK-00060	IL-17B Protein, Mouse, Recombinant (His)	Mouse	E. coli
	IL-17A, the prototypic member of the IL-17 family, several experimental findings strongly support the role of the IL-17B/IL-17 receptor B (IL-17RB) pathway in tumorigenesis and resistance to anticancer therapies. IL-17B/...
TMPK-00044	SKP1 Protein, Human, Recombinant (His, Avi)	Human	HEK293 Cells
	The S-phase Kinase-Associated Protein 1 (SKP1) is a core component of the SKP1, Cullin 1, F-box protein (SCF) complex, an E3 ubiquitin ligase that serves to poly-ubiquitinate a vast array of protein targets as a signal f...
TMPK-00957	MFAP5 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Human basal-like breast cancer (BLBC) is an aggressive malignancy with poor prognosis. Since most current treatments are ineffective, there is an urgent need to identify therapeutic targets for BLBC. Microfibrillar-assoc...
TMPJ-01069	Serpin A1e Protein, Mouse, Recombinant (His)	Mouse	HEK293 Cells
	Alpha-1-antitrypsin 1-5(SERPIN A1) is a secreted protein and belongs to the serpin family. Serpins bind the protease active site resulting in a major conformational rearrangement that traps the enzyme in a covalent acyl-...
TMPK-01217	MFAP5 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	Human basal-like breast cancer (BLBC) is an aggressive malignancy with poor prognosis. Since most current treatments are ineffective, there is an urgent need to identify therapeutic targets for BLBC. Microfibrillar-assoc...
TMPK-00045	SKP1 Protein, Human, Recombinant (His, Avi), Biotinylated	Human	HEK293 Cells
	The S-phase Kinase-Associated Protein 1 (SKP1) is a core component of the SKP1, Cullin 1, F-box protein (SCF) complex, an E3 ubiquitin ligase that serves to poly-ubiquitinate a vast array of protein targets as a signal f...
TMPK-01384	SARS PLpro/papain-like protease Protein (His)	SARS	E. coli
	The coronaviral proteases, papain-like protease (PLpro) and 3C-like protease (3CLpro), are attractive antiviral drug targets because they are essential for coronaviral replication. Although the primary function of PLpro ...
TMPY-06864	GLP1R Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	Glucagon-like peptide (GLP)-1 receptor is encoded by GLP1R. GLP1R plays a critical role in mediating the biological actions of GLP1 in mammals and fish. The neuronal GLP1Rs mediate body weight and anorectic effects of li...
TMPH-01855	PEX19 Protein, Human, Recombinant (GST)	Human	E. coli
	Necessary for early peroxisomal biogenesis. Acts both as a cytosolic chaperone and as an import receptor for peroxisomal membrane proteins (PMPs). Binds and stabilizes newly synthesized PMPs in the cytoplasm by interacti...
TMPH-01235	APOBEC3A Protein, Human, Recombinant (His & SUMO)	Human	E. coli
	DNA deaminase (cytidine deaminase) with restriction activity against viruses, foreign DNA and mobility of retrotransposons. Exhibits antiviral activity against adeno-associated virus (AAV) and human T-cell leukemia virus...
TMPH-01522	HIV-2 (subtype A, isolate ROD) Protein Vpx (His)	HIV-2	P. pastoris (Yeast)
	Plays a role in nuclear translocation of the viral pre-integration complex (PIC), thus is required for the virus to infect non-dividing cells. Targets specific host proteins for degradation by the 26S proteasome. Acts by...
TMPK-01352	SARS-CoV-2 PLpro/papain-like protease Protein (His & Avi)	SARS	E. coli
	The coronaviral proteases, papain-like protease (PLpro) and 3C-like protease (3CLpro), are attractive antiviral drug targets because they are essential for coronaviral replication. Although the primary function of PLpro ...
TMPH-01222	DGKA Protein, Human, Recombinant (His)	Human	E. coli
	Diacylglycerol kinase that converts diacylglycerol/DAG into phosphatidic acid/phosphatidate/PA and regulates the respective levels of these two bioactive lipids. Thereby, acts as a central switch between the signaling pa...
TMPY-00371	STC1 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Stanniocalcin-1 (STC1) is a paracrine factor associated with inflammation and carcinogenesis. STC1 is a secreted glycoprotein hormone and involved in various types of human malignancies. Stanniocalcin-1 (STC1), which has...
TMPJ-01386	STUB1 Protein, Human, Recombinant	Human	E. coli
	E3 Ubiquitin-Protein Ligase CHIP is a cytoplasmic protein. CHIP is highly expressed in skeletal muscle, heart, pancreas, brain and placenta. CHIP interacts with the molecular chaperones Hsc70-Hsp70 and Hsp90 through its ...
TMPJ-01074	PKCE Protein, Human, Recombinant (His)	Human	E. coli
	Protein Kinase C Epsilon type is a member of the serine- and threonine-specific protein kinase family that can be activated by calcium and the second messenger diacylglycerol. Protein Kinase C Epsilon contains these doma...
TMPJ-00505	Serpin A1 Protein, Human, Recombinant (aa 25-418, His)	Human	HEK293 Cells
	Serpin A1 is a prototype member of the Serpin superfamily of the serine protease inhibitors. As one of the most abundant proteinase inhibitors in the circulation, it is synthesized in hepatocytes, and to a lesser extent,...
TMPY-05800	IKB beta/NFKBIB Protein, Human, Recombinant (GST)	Human	E. coli
	NFKBIB (NFKB Inhibitor Beta) is a Protein Coding gene. The protein encoded by this gene belongs to the NF-kappa-B inhibitor family, which inhibits NF-kappa-B by complexing with and trapping it in the cytoplasm. Phosphory...
TMPJ-01431	SARS-CoV-2 Papain-Like Protease Protein	SARS-CoV-2	E. coli
	Replication of severe acute respiratory syndrome (SARS) coronavirus (SARS-CoV) requires proteolytic processing of the replicase polyprotein by two viral cysteine proteases, a chymotrypsin-like protease (3CLpro) and a pap...
TMPH-01269	SMURF2 Protein, Human, Recombinant (His)	Human	E. coli
	E3 ubiquitin-protein ligase which accepts ubiquitin from an E2 ubiquitin-conjugating enzyme in the form of a thioester and then directly transfers the ubiquitin to targeted substrates. Interacts with SMAD7 to trigger SMA...
TMPY-04267	MSH2 Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	MSH2 is a key DNA mismatch repair protein, which plays an important role in genomic stability. In addition to its DNA repair function, MSH2 serves as a sensor for DNA base analogs-provoked DNA replication errors and bind...
TMPJ-00323	Nectin-2 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	CD112 is a type I transmembrane glycoprotein belonging to the Immunoglobulin superfamily. It comprises one Ig-like V-type domain and two Ig-like C2-type domains in the extracellular region. The V domain is believed to me...
TMPJ-00630	B7-1 Protein, Cynomolgus, Recombinant (hFc)	Cynomolgus	HEK293 Cells
	Cynomologous Cluster of Differentiation 80, also called B7-1, is a member of cell surface immunoglobulin superfamily.It is expressed on the surface of antigen-presenting cells including activated B cells, macrophages and...
TMPH-03289	EIF3I Protein, Rat, Recombinant (E. coli, His)	Rat	E. coli
	Component of the eukaryotic translation initiation factor 3 (eIF-3) complex, which is required for several steps in the initiation of protein synthesis. The eIF-3 complex associates with the 40S ribosome and facilitates ...
TMPH-03288	EIF3I Protein, Rat, Recombinant (His)	Rat	Baculovirus Insect Cells
	Component of the eukaryotic translation initiation factor 3 (eIF-3) complex, which is required for several steps in the initiation of protein synthesis. The eIF-3 complex associates with the 40S ribosome and facilitates ...
TMPH-02690	PLA2G10 Protein, Mouse, Recombinant (His & Myc)	Mouse	E. coli
	Secretory calcium-dependent phospholipase A2 that primarily targets extracellular phospholipids. Hydrolyzes the ester bond of the fatty acyl group attached at sn-2 position of phospholipids with preference for phosphatid...
TMPY-02081	PDE2A Protein, Human, Recombinant (aa 215-900, His)	Human	Baculovirus Insect Cells
	cGMP-dependent 3',5'-cyclic phosphodiesterase, also known as cyclic GMP-stimulated phosphodiesterase and PDE2A, is a peripheral membrane protein that belongs to the cyclic nucleotide phosphodiesterase family and PDE2 sub...
TMPY-01771	Latexin Protein, Mouse, Recombinant (His)	Mouse	E. coli
	Latexin, also known as endogenous carboxypeptidase inhibitor, tissue carboxypeptidase inhibitor, TCI, ECI, and LXN, is a cytoplasm protein that belongs to the protease inhibitor I47 (latexin) family. It is highly express...
TMPY-02386	PTP4A2 Protein, Human, Recombinant (GST)	Human	E. coli
	PRL-2 (Protein-tyrosine phosphatase of regenerating liver 2), also known as PTP4A2 (Protein tyrosine phosphatase type IVA, member 2), is a member of PTP family and has an important function in controlling cell growth. PR...
TMPY-04423	CAMKI gamma/CAMK1G Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	Calmodulin-Dependent Protein Kinase (CaM Kinase) is a kind of protein phosphorylate multiple downstream targets. Concentration of cytosolic calcium functions as a second messenger that mediates a wide range of cellular r...
TMPY-03442	MOB4A/MOB1B Protein, Human, Recombinant (GST)	Human	E. coli
	MST1 and MST2 are the mammalian Ste2-related protein kinases most closely related to Drosophila Hippo, a major regulator of cell proliferation and survival during development. Overexpression of MST1 or MST2 in mammalian ...
TMPY-01406	REG3G Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Regenerating gene (Reg), first isolated from a regenerating islet cDNA library, encodes a secretory protein with a growth stimulating effect on pancreatic beta cells. Reg and Reg-related genes which were expressed in var...
TMPH-03037	Alpha-cobratoxin Protein, Naja kaouthia, Recombinant (GST & His & Myc)	Naja kaouthia	E. coli
	Monomer: binds with high affinity to muscular (alpha-1-beta-1-gamma-delta/CHRNA1-CHRNB1-CHRNG-CHRND) nAChR (tested on Torpedo californica, Kd=0.2-4.5 nM) and neuronal alpha-7/CHRNA7 nicotinic acetylcholine receptors (Kd=...
TMPY-04387	AKT2 Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	AKT (AK mouse plus Transforming or Thymoma) is a frequent oncogene expressed in most tissues which includes three isoforms AKT1, AKT2, and AKT3. Hyperactivation of AKT signaling is a central key in many human cancer prog...
TMPH-02317	YTHDF1 Protein, Human, Recombinant (His)	Human	P. pastoris (Yeast)
	Specifically recognizes and binds N6-methyladenosine (m6A)-containing mRNAs, and regulates their stability. M6A is a modification present at internal sites of mRNAs and some non-coding RNAs and plays a role in mRNA stabi...
TMPY-04456	PKC nu Protein, Human, Recombinant (GST)	Human	Baculovirus Insect Cells
	Serine/threonine-protein kinase D3, also known as Protein kinase C nu type, Protein kinase EPK2, PRKD3, EPK2 and PRKCN, is a cytoplasm and membrane protein that belongs to the protein kinase superfamily, CAMK Ser/Thr pro...
TMPY-02228	P53 Protein, Cynomolgus, Recombinant	Cynomolgus	E. coli
	p53, also known as Tp53, is a DNA-binding protein which belongs to the p53 family. It contains transcription activation, DNA-binding, and oligomerization domains. p53 protein is expressed at low level in normal cells and...
TMPH-01692	MAPK3 Protein, Human, Recombinant (His)	Human	E. coli
	Serine/threonine kinase which acts as an essential component of the MAP kinase signal transduction pathway. MAPK1/ERK2 and MAPK3/ERK1 are the 2 MAPKs which play an important role in the MAPK/ERK cascade. They participate...
TMPH-02633	TRIM21 Protein, Mouse, Recombinant (His)	Mouse	Baculovirus Insect Cells
	E3 ubiquitin-protein ligase whose activity is dependent on E2 enzymes, UBE2D1, UBE2D2, UBE2E1 and UBE2E2. Forms a ubiquitin ligase complex in cooperation with the E2 UBE2D2 that is used not only for the ubiquitination of...
TMPH-02632	TRIM21 Protein, Mouse, Recombinant (E. coli, His)	Mouse	E. coli
	E3 ubiquitin-protein ligase whose activity is dependent on E2 enzymes, UBE2D1, UBE2D2, UBE2E1 and UBE2E2. Forms a ubiquitin ligase complex in cooperation with the E2 UBE2D2 that is used not only for the ubiquitination of...
------------------------ More ------------------------

PHGDH Protein, Human, Recombinant (His)

TMPY-02801

Species: Human

Expression System: E. coli

Thyroid peroxidase Protein, Human, Recombinant (S257A & P725T, His)

TMPY-02779

Species: Human

Expression System: Baculovirus Insect Cells

IL-3 Protein, Mouse, Recombinant (His)

TMPJ-00051

Species: Mouse

Expression System: HEK293 Cells

TSLP Protein, Human, Recombinant

TMPJ-00042

Species: Human

Expression System: E. coli

S100B Protein, Canine, Recombinant (hFc)

TMPK-01369

Species: Canine

Expression System: HEK293 Cells

CALML3 Protein, Human, Recombinant (His)

TMPY-02760

Species: Human

Expression System: E. coli

GBA/glucocerebrosidase Protein, Human, Recombinant (His)

TMPY-05099

Species: Human

Expression System: HEK293 Cells

B7-H6 Protein, Human, Recombinant (His & Avi), Biotinylated

TMPK-00280

Species: Human

Expression System: HEK293 Cells

SEMA3A Protein, Rat, Recombinant (His)

TMPH-03369

Species: Rat

Expression System: E. coli

MOB1A Protein, Human, Recombinant (His)

TMPJ-01335

Species: Human

Expression System: E. coli

IL-17B Protein, Mouse, Recombinant (His)

TMPK-00060

Species: Mouse

Expression System: E. coli

SKP1 Protein, Human, Recombinant (His, Avi)

TMPK-00044

Species: Human

Expression System: HEK293 Cells

MFAP5 Protein, Human, Recombinant (hFc)

TMPK-00957

Species: Human

Expression System: HEK293 Cells

Serpin A1e Protein, Mouse, Recombinant (His)

TMPJ-01069

Species: Mouse

Expression System: HEK293 Cells

MFAP5 Protein, Mouse, Recombinant (hFc)

TMPK-01217

Species: Mouse

Expression System: HEK293 Cells

SKP1 Protein, Human, Recombinant (His, Avi), Biotinylated

TMPK-00045

Species: Human

Expression System: HEK293 Cells

SARS PLpro/papain-like protease Protein (His)

TMPK-01384

Species: SARS

Expression System: E. coli

GLP1R Protein, Human, Recombinant (His & Avi)

TMPY-06864

Species: Human

Expression System: HEK293 Cells

PEX19 Protein, Human, Recombinant (GST)

TMPH-01855

Species: Human

Expression System: E. coli

APOBEC3A Protein, Human, Recombinant (His & SUMO)

TMPH-01235

Species: Human

Expression System: E. coli

HIV-2 (subtype A, isolate ROD) Protein Vpx (His)

TMPH-01522

Species: HIV-2

Expression System: P. pastoris (Yeast)

SARS-CoV-2 PLpro/papain-like protease Protein (His & Avi)

TMPK-01352

Species: SARS

Expression System: E. coli

DGKA Protein, Human, Recombinant (His)

TMPH-01222

Species: Human

Expression System: E. coli

STC1 Protein, Human, Recombinant (His)

TMPY-00371

Species: Human

Expression System: HEK293 Cells

STUB1 Protein, Human, Recombinant

TMPJ-01386

Species: Human

Expression System: E. coli

PKCE Protein, Human, Recombinant (His)

TMPJ-01074

Species: Human

Expression System: E. coli

Serpin A1 Protein, Human, Recombinant (aa 25-418, His)

TMPJ-00505

Species: Human

Expression System: HEK293 Cells

IKB beta/NFKBIB Protein, Human, Recombinant (GST)

TMPY-05800

Species: Human

Expression System: E. coli

SARS-CoV-2 Papain-Like Protease Protein

TMPJ-01431

Species: SARS-CoV-2

Expression System: E. coli

SMURF2 Protein, Human, Recombinant (His)

TMPH-01269

Species: Human

Expression System: E. coli

MSH2 Protein, Human, Recombinant (His & GST)

TMPY-04267

Species: Human

Expression System: Baculovirus Insect Cells

Nectin-2 Protein, Mouse, Recombinant (hFc)

TMPJ-00323

Species: Mouse

Expression System: HEK293 Cells

B7-1 Protein, Cynomolgus, Recombinant (hFc)

TMPJ-00630

Species: Cynomolgus

Expression System: HEK293 Cells

EIF3I Protein, Rat, Recombinant (E. coli, His)

TMPH-03289

Species: Rat

Expression System: E. coli

EIF3I Protein, Rat, Recombinant (His)

TMPH-03288

Species: Rat

Expression System: Baculovirus Insect Cells

PLA2G10 Protein, Mouse, Recombinant (His & Myc)

TMPH-02690

Species: Mouse

Expression System: E. coli

PDE2A Protein, Human, Recombinant (aa 215-900, His)

TMPY-02081

Species: Human

Expression System: Baculovirus Insect Cells

Latexin Protein, Mouse, Recombinant (His)

TMPY-01771

Species: Mouse

Expression System: E. coli

PTP4A2 Protein, Human, Recombinant (GST)

TMPY-02386

Species: Human

Expression System: E. coli

CAMKI gamma/CAMK1G Protein, Human, Recombinant (His & GST)

TMPY-04423

Species: Human

Expression System: Baculovirus Insect Cells

MOB4A/MOB1B Protein, Human, Recombinant (GST)

TMPY-03442

Species: Human

Expression System: E. coli

REG3G Protein, Human, Recombinant (His)

TMPY-01406

Species: Human

Expression System: HEK293 Cells

Alpha-cobratoxin Protein, Naja kaouthia, Recombinant (GST & His & Myc)

TMPH-03037

Species: Naja kaouthia

Expression System: E. coli

AKT2 Protein, Human, Recombinant (His & GST)

TMPY-04387

Species: Human

Expression System: Baculovirus Insect Cells

YTHDF1 Protein, Human, Recombinant (His)

TMPH-02317

Species: Human

Expression System: P. pastoris (Yeast)

PKC nu Protein, Human, Recombinant (GST)

TMPY-04456

Species: Human

Expression System: Baculovirus Insect Cells

p53 Protein, Cynomolgus, Recombinant

TMPY-02228

Species: Cynomolgus

Expression System: E. coli

MAPK3 Protein, Human, Recombinant (His)

TMPH-01692

Species: Human

Expression System: E. coli

TRIM21 Protein, Mouse, Recombinant (His)

TMPH-02633

Species: Mouse

Expression System: Baculovirus Insect Cells

TRIM21 Protein, Mouse, Recombinant (E. coli, His)

TMPH-02632

Species: Mouse

Expression System: E. coli

--------- More ---------

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L3980	DNA Damage and Repair Compound Library Plus	667 compounds
	Well-chosen 667 compounds with unique structures targeting DNA damage & repair;
L3900	DNA Damage & Repair Compound Library	910 compounds
	A unique collection of 910 DNA Damage & Repair related compounds for high throughput screening (HTS) and high content screening (HCS);
L3410	Preclinical Compound Library	701 compounds
	A unique collection of 701 preclinical compounds for high throughput screening (HTS) and high content screening (HCS);
L3400	Clinical Compound Library	3404 compounds
	A unique collection of 3404 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
L9500	Target-Focused Phenotypic Screening Library	1796 compounds
	A unique collection of 1796 annotated bioactive compounds with clear targets, suitable for phenotypic screening；
L2152	Targeted Therapy Drug Library	119 compounds
	119 tumor-targeted drugs that can be used for high-throughput and high-content screening.
L2191	Anti-Breast Cancer Compound Library	1939 compounds
	A unique collection of 1939 compounds with anti-breast cancer therapeutic activity or targeting breast cancer’s major signaling pathways, can be used for anti-breast cancer drug discovery and mechanism study；
L4010	Bioactive Compounds Library Max	22555 compounds
	A collection of 22555 bioactive compounds for high-throughput screening, high-content screening, cell induction and target identification.
L6150	Covalent Natural Product Library	583 compounds
	Detialed biological information and pharmacological information of the products, providing theoretical direction and research basis for screening.
L6900	Rare Natural Product Library	693 compounds
	A unique collection of 693 rare natural products, which can be used for high throughput screening (HTS) and high content screening (HCS);
L8800	Drug-Fragment Library	1119 compounds
	1119 drug fragments，a must-have tool for FBDD;
L4000	Bioactive Compound Library	14439 compounds
	A collection of 14439 small molecule compounds with validated activity for high throughput screening (HTS), high content screening (HCS), cell induction, and target identification;
L2700	Adrenergic Receptor-Targeted Compound Library	193 compounds
	A unique collection of 193 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification;
L2195	Anti-Prostate Cancer Compound Library	2070 compounds
	2070 compounds associated with prostate cancer that can be used for high-throughput and high-content screening.
L4200	FDA-Approved Drug Library	1729 compounds
	A unique collection of 1729 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS);
L7820	High Solubility Micro Fragment Library	1081 compounds
	The compound library of highly soluble micro-fragments consists of 1081 low-molecular-weight fragments.
L4150	Featured Novel Bioactive Compound Library	989 compounds
	It is well-selected from Bioactive compound library Plus (D7800), from which 1-15 compounds with the highest scores (activity value, pharmacological properties, structure-diversity, etc.) were chosen. This library consis...
L7860	Mini Electrophilic Heterocyclic Fragment Library	369 compounds
	369 compounds in total in the Highly Solubility Covalent Heterocyclic Fragment Library
L7870	Carboxylic Acid Fragment Library With Solubility	1806 compounds

L2170	Immuno-Oncology Compound Library	449 compounds
	A unique collection of 449 compounds acting on immune-oncology therapeutic targets can be used for high throughput and high content screening；
L4660	Anti-Nervous System Disease Library	1246 compounds
	Well-chosen 1246 compounds with unique structures targeting nervous system;
L9840	Anti-Alzheimer's Disease Compound Library	986 compounds
	A unique collection of 986 compounds with anti-AD activities or acting on main drug targets of AD can be used for HTS and HCS.
L2000	Inhibitor Library	8328 compounds
	A unique collection of 8328 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
L9400	PPI Inhibitor Library	485 compounds
	A unique collection of 485 PPI-related compounds for drug screening;
L2010	Highly Selective Inhibitor Library	575 compounds

L2194	Anti-Colorectal Cancer Compound Library	1545 compounds
	1545 compounds associated with colorectal cancer that can be used for high-throughput and high-content screening.
L2620	Anti-Neurodegenerative Disease Compound Library	2154 compounds
	A unique collection of 2154 compounds related to neurodegenerative diseases can be used for HTS or HCS；
L1710	Anti-COVID-19 Compound Library	1133 compounds
	A unique collection of 1133 compounds with confirmed anti-SARS-CoV-2 activity or potential activity and part of them are broad-spectrum antiviral agents；
L9830	Anti-Parkinson's Disease Compound Library	857 compounds
	A unique collection of 857 compounds with anti-PD activities or acting on main drug targets of PD can be used for HTS and HCS.
LF1000	Pre-plated Diversity Sets	50000 compounds
	For your convenience, there are Diversity Sets of 5,000, 10,000, 15,000, and 20,000 compounds with no structure overlap.
L9300	Macrocyclic Compound Library	210 compounds
	210 macrocyclic compounds of known activity for high-throughput, high-content screening;
L8700	Ferroptosis Compound Library	779 compounds
	A unique collection of 779 ferroptosis signaling pathway related compounds, a powerful tool for new target identification, drug discovery, and mechanism study；
L8110	Reprogramming Compound Library	1813 compounds
	A unique collection of 1813 reprogramming signaling pathway-related bioactive small molecule compounds for high-throughput, high-content screening.
L9860	Antidepressant Compound Library	1163 compounds
	1163 compounds associated with depression that can be used for high-throughput and high-content screening
L2180	Anti-Cancer Compound Library Plus	1468 compounds
	Well-chosen 1468 anti-tumor compounds with unique structures;
L2193	Anti-Liver Cancer Compound Library	1787 compounds
	1787 species of compounds related to liver cancer that can be used in anti-liver cancer drug development and pharmacological studies.
L7200	Calcium Channel Compound Library	140 compounds
	A unique collection of 140 calcium channel blockers and agonists for high throughput and high content screening;
L2130	Anti-Cancer Metabolism Compound Library	1268 compounds
	A unique collection of 1268 cancer cellular metabolism related compounds for cancer research and high throughput screening (HTS) and high content screening (HCS);
L2610	Neurotransmitter Receptor Compound Library	1513 compounds
	A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
L2510	Lipid Metabolism Compound Library	492 compounds
	A unique collection of 492 compounds targeting lipid metabolism, can be used for high-throughput screening (HTS) and high-content screening (HCS).
L6730	Anti-virus Traditional Chinese Medicine Monomer Library	268 compounds
	A collection of 268 TCM monomers with anti-virus activity. An effective tool for drug development and pharmacological studies.
L1310	Cytoskeletal Signaling Pathway Compound Library	759 compounds
	A unique collection of 759 cytoskeleton-related compounds, can be used for HTS and HCS；
L5300	Mitochondria-Targeted Compound Library	812 compounds
	A unique collection of 812 promising or approved mitochondria-targeted compounds including Idebenone, the only approved drug targeting mitochondria, for research in mitochondrial medicine;
L9700	Endoplasmic Reticulum Stress Compound Library	193 compounds
	A unique collection of 193 endoplasmic reticulum stress (ER stress) related compounds used for high throughput screening (HTS) and high content screening (HCS);
L3800	NF-κB Signaling Compound Library	729 compounds
	A unique collection of 729 compounds targeting NF-κB signaling for high throughput screening and high content screening;
L6610	Anti-infective Natural Product Library	1060 compounds
	A unique collection of 1060 species of natural products with anti-infective activity for high throughput screening (HTS) and high content screening (HCS);
L7600	Chemokine Inhibitor Library	59 compounds
	A unique collection of 59 chemokines or chemokine receptors targeted compounds for high throughput and high content screening;
L8500	HIF-1 Signaling Pathway Compound Library	1336 compounds
	A unique collection of 1336 HIF-1 related small chemicals can be used for drug discovery in ischemic disease and cancer and related mechanism studies；
L4800	Angiogenesis related Compound Library	1353 compounds
	A unique collection of 1353 proangiogenic and antiangiogenic compounds for new targets identification, research in mechanisms of angiogenesis, and high throughput screening (HTS) and high content screening (HCS);
L6750	PBCRBS Traditional Chinese Medicine Compound Library	580 compounds
	A unique collection of 580 compounds derived from traditional Chinese medicines (TCMs) for promoting blood circulation and removing blood stasis.
L6710	Anti-Inflammatory Traditional Chinese Medicine Compound Library	1246 compounds
	A collection of 1246 TCM monomers with anti-inflammatory activity or targeting molecular therapeutic targets in inflammation, a powerful tool for drug discovery and mechanism study；
L7110	Anti-Hypertension Compound Library	678 compounds
	678 hypertension-related small molecules for high-throughput and high-content screening.
L9410	Covalent Inhibitor Library	1920 compounds
	A unique collection of 1920 covalent Inhibitors and other molecules with common warheads like chloroacetyl，2-Chloropropionyl，Acryloyl，sulfonyl fluoride, alkyne，acrylamide, ketocarbonyl，disulfide bond, etc.