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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T26396 | 6-Hydroxy-DOPA | 6-Hydroxy-DL-DOPA | DNA/RNA Synthesis |
6-Hydroxy-DOPA is an allosteric inhibitor of RAD52, it inhibits proliferation of BRCA-deficient cancer cells in vitro and also inhibits APE1. | |||
T9318 | TP0586532 | Others | |
TP0586532 is effective against carbapenem-resistant Klebsiella pneumoniae and does not pose a cardiovascular risk. | |||
T8055 | TFEB activator 1 | (1E,4E)-1,5-Bis(2-Methoxyphenyl)penta-1,,Curcumin analog compound C1,Curcumin analog C1,RPN77612 | Others , Autophagy |
TFEB activator 1 (Curcumin analog compound C1) is an activator of transcription factor EB (TFEB) with promise for the prevention or treatment of Alzheimer's disease. | |||
T10718L | CCT241533 hydrochloride | Chk | |
CCT241533 hydrochloride is an effective and selective ATP competitive inhibitor of CHK2 (Ki: 1.16 nM; IC50: 3 nM). | |||
T26360 | Benperidol | R4584,R-4584,Anquil,McN-JR-4584,R 4584 | |
Benperidol (Anquil) is a butanone analog with antipsychotic and stabilizing properties, and has been shown to be effective in blocking D2 receptors.Benperidol can be used in positron emission tomography (PET) scanning to... | |||
T16557 | PNU-159682 | Topoisomerase | |
PNU-159682 is a highly effective metabolite of the anthracycline nemorubicin. PNU-159682 has outstanding cytotoxicity. PNU-159682 is an effective ADCs cytotoxin. | |||
T3453 | WAY-100635 maleate | 5-HT Receptor | |
WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM). | |||
T15649 | KDM5-IN-1 | Histone Demethylase | |
KDM5-IN-1 is an effective and selective inhibitor of KDM5 with an IC50 of 15.1 nM. | |||
T14522 | Beaucage reagent | DNA/RNA Synthesis | |
Beaucage reagent, which is found to be effective in causing DNA cleavage. | |||
T15628 | JT010 | TRP/TRPV Channel | |
JT010 is an effective agonist of TRPA1 (EC50 = 0.65 nM). | |||
T3434 | BAY1217389 | Kinesin | |
BAY 1217389 is an effective and selective inhibitor of the monopolar spindle 1 (MPS1) kinase (IC50<10 nM). | |||
T4044 | DprE1-IN-2 | Antibacterial , DprE1 | |
DprE1-IN-2 is an effective DprE1 inhibitor. | |||
T24918 | UBP710 | UBP-710,UBP 710 | NMDAR |
UBP710 is an effective and selective NMDA receptor modulator. | |||
T17247 | VU0661013 | VU661013 | BCL |
VU0661013 is an effective and selective inhibitor of MCL-1. | |||
T15820 | Mibampator | LY451395 | iGluR |
Mibampator (LY451395) is an effective and selective AMPA receptor potentiator. | |||
T1918 | NVP-TAE 226 | TAE226 | Apoptosis , FAK , c-Met/HGFR , PYK2 , IGF-1R |
NVP-TAE 226 (TAE226) is an effective FAK inhibitor (IC50: 5.5 nM) and most effective to Pyk2(IC50: 3.5 nM); 10- to 100-fold less effective against IGF-1R, InsR, c-Met, and ALK. | |||
T6821 | Dp44mT | Apoptosis , Others , Ferroptosis | |
Dp44mT, a effective iron chelator, has selective antitumor activity. | |||
T4083 | BAR501 | BAR 501 | GPCR19 |
BAR501 is an effective and specific GPBAR1 agonist (EC50: 1 μM). | |||
T15481 | HI-TOPK-032 | TOPK | |
HI-TOPK-032 is an effective and specific inhibitor of TOPK. | |||
T22415 | Resorantel | Parasite | |
Resorantel is a safe, hydroxybenzanilide cestocide moderately effective against Paramphistomum spp and highly effective against Thysaniezia spp. and Moniezia. Resorantel has been used for the research of G. aegypticus an... | |||
T60029 | SOS1-IN-11 | Raf | |
SOS1-IN-11 is an effective inhibitor of SOS1 (IC50 = 30 nM). | |||
T4173 | R162 | Dehydrogenase | |
R162 is an effective glutamate dehydrogenase 1 (GDH1) inhibitor. | |||
T11123 | DuP 105 | Antibacterial , Antibiotic | |
DuP 105 is an oral oxazolidinone, a novel synthetic antimicrobial compound effective against gram-positive bacteria. | |||
T3645 | Endoxifen E-isomer hydrochloride | E-Endoxifen hydrochloride | Estrogen Receptor/ERR , Estrogen/progestogen Receptor |
Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM). | |||
T15796 | LX-1031 | Hydroxylase , LPA Receptor | |
LX-1031 is an effective inhibitor of tryptophan 5-hydroxylase. LX-1031 decreases serotonin (5-HT) synthesis peripherally. | |||
T14863 | Carabersat | SB 204269 | Others |
Carabersat(SB 204269) is a novel and effective anticonvulsant and antiepileptic agent. | |||
T23917 | CRT-0105950 | CRT 0105950 | |
CRT-0105950 is an effective LIMK inhibitor that acts by suppressing cofilin phosphorylation and increasing αTubulin acetylation in cells. | |||
T2704 | MLN0905 | PLK1 Inhibitor | PLK |
MLN0905 (PLK1 Inhibitor) is an effective PLK1 inhibitor(IC50=2 nM). | |||
T10314 | AM103 | AM 103 | FLAP |
T13387L | Zatebradine hydrochloride | UL-FS-49CL,UL-FS-49 | Others , HCN Channel |
Zatebradine hydrochloride (UL-FS-49CL) is a highly effective and effective HCN Channel inhibitor (IC50:1.96 µM). HCN Channel is an effective hyperpolarization activated loop nucleotide gated channel. Zatebradine hydrochl... | |||
T3361 | Cambendazole | Bonlam,MK-905,Novazole | Others |
Cambendazole (Novazole) is one of the most effective agents for the therapy of human strongyloidiasis. Cambendazole is a nematocide effective against a variety of gastrointestinal parasites in cattle, sheep, and horses. | |||
T16120 | MLT-748 | Others | |
MLT-748 is an effective, selective, and allosteric MALT1 inhibitor. It binds MALT1 in the allosteric Trp580 pocket (IC50: 5 nM). | |||
T2439 | O4I1 | OCT | |
O4I1 is an effective Oct3/4 inducer. | |||
T15806 | LY2562175 | FXR , Autophagy | |
LY2562175 is an effective and selective FXR agonist (EC50: 193 nM). | |||
T2418 | A66 | PI3K | |
A66 is a specific and effective p110α inhibitor(IC50=32 nM). | |||
T15673 | KU 59403 | ATM/ATR | |
KU 59403 is an effective ATM inhibitor (IC50: 3 nM, 9.1 μM, and 10 μM for ATM, DNA-PK, and PI3K, respectively). | |||
T14349 | Auristatin F | Microtubule Associated | |
Auristatin F is an effective inhibitor of microtubule and vascular damaging agent. Auristatin F can be used in antibody-drug conjugates. | |||
T9755 | MRTX0902 | UNII-CRG69FR93G | Raf |
MRTX0902 is an effective and high selective inhibitor of SOS1 with an IC50 of 46 nM and a Ki of 2 nM. | |||
T17042 | TES-1025 | Others | |
TES-1025 is an effective and selective inhibitor of human α-amino-β-carboxymuconate-ε-semialdehyde decarboxylase (IC50: 13 nM). | |||
T2657 | Elacridar | GW0918,GW120918,GF120918,GG918 | BCRP , P-gp |
Elacridar (GG918) (GF120918) is an effective BCRP and P-gp (MDR-1) inhibitor. | |||
T4499 | Mequitazine | Metaplexan,Virginan,Primalan,LM-209 | Histamine Receptor |
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist. | |||
T1780 | Parecoxib | SC 69124,Vorth-P,Valus-P | COX |
Parecoxib (SC 69124) is an effective and selective COX-2 inhibitor. | |||
T15582 | InS3-54A18 | STAT | |
T2647 | IDO5L | INCB024360 analogue,INCB14943 | IDO , Indoleamine 2,3-Dioxygenase (IDO) |
IDO5L (INCB024360 analogue) is an effective IDO1 inhibitor(IC50=10 nM). | |||
TQ0187 | SR-3677 | ROCK , Autophagy | |
SR-3677 is an effective and specific inhibitor of ROCK2 (IC50: 3 nM). | |||
T6325 | PCI-34051 | PCI 34051 | Apoptosis , HDAC |
PCI-34051 is an effective and selective HDAC8 inhibitor (IC50: 10 nM). | |||
T3499 | Remodelin | Histone Acetyltransferase | |
Remodelin is an effective and specific inhibitor of the acetyl-transferase protein NAT10. | |||
T24410 | LIMK-IN-22j | LIMK IN 22j,LIMK inhibitor-22j,LIMK inhibitor 22j | LIM Kinase |
LIMK-IN-22j (LIMK inhibitor 22j) is an effective and selective inhibitor of LIMK. | |||
T10336 | Antimalarial agent 1 | Parasite | |
Antimalarial agent 1 is an effective antimalarial agent. | |||
T15372 | GB1107 | (2R,3R,4S,5R,6R)-2-(3,4-dichlorophenyl)sulfanyl-6-(hydroxymethyl)-4-[4-(3,4,5-trifluorophenyl)triazol-1-yl]oxane-3,5-diol | Galectin |
GB1107 is an effective and selective Galectin-3 inhibitor with a Kd of 37 nM. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T0131 | Cepharanthine | NSC-623442 | Apoptosis , TNF , HIV Protease , Autophagy |
Cepharanthine (NSC-623442), a biscoclaurine alkaloid, suppresses tumor necrosis factor (TNF)-α-mediated NFκB stimulation, plasma membrane lipid peroxidation and platelet aggregation and inhibits cytokine production. | |||
T15643 | Kainic acid | Others | |
In the CNS, Kainic acid is an effective agonist at excitatory amino acid receptor subtypes. | |||
T4902 | Isotrifoliin | Isoquercetin,Isoquercitroside | Reactive Oxygen Species |
T2890 | Hordenine | Antibacterial , Antibiotic | |
Hordenine, an effective phenylethylamine alkaloid, has antibacterial activities. | |||
Fr12339 | Anisylacetone | Others | |
Anisylacetone (Anisylacetone) is an effective lure for the male melon fly. | |||
T3233 | Sophoricoside | Genistein sophoricoside | Others |
Sophoricoside (Genistein sophoricoside) is effective against inflammation and can reduce the GPT. | |||
T13669 | (E)-Cinnamamide | trans-Cinnamamide | Others |
(E)-Cinnamamide (trans-Cinnamamide) is the less active isomer of Cinnamamide which is an effective non-lethal chemical repellent suitable for reducing avian pest damage. | |||
T0295 | Digitoxin | Digitoxoside,Unidigin,Digitoxinum | ATPase , Others |
Digitoxin (Digitoxinum) is an effective Na+/K+-ATPase inhibitor (EC50 value: 0.78 μM). | |||
T5S1287 | Ligustilide | Apoptosis , Autophagy | |
3-Butylidene-4,5-dihydrophthalide is an effective constituent extracted from Angelica sinensis. | |||
TN7022 | Cymen-ar-ol | Antibacterial | |
Cymen-ar-ol is a broad spectrum and highly effective bactericide that can contact mucous membrane. | |||
T8201 | Gambogenic acid | Histone Methyltransferase | |
Gambogenic acid is a natural product,is an effective inhibitor of EZH2,with anticancer activity. | |||
T1436 | 4-Aminohippuric Acid | p-Aminohippuric acid | Amino Acids and Derivatives , Endogenous Metabolite |
4-Aminohippuric Acid is the glycine amide of 4-aminobenzoic acid. Its sodium salt is used as a diagnostic aid to measure effective renal plasma flow (ERPF) and excretory capacity. | |||
T6S0105 | Peiminine | Zhebeinone,Fritillarine,Raddeanine,Verticinone | Others , Autophagy |
1. Peiminine (Raddeanine) is an effective inhibitor for lung inflammation and pulmonary fibrosis in a rat model of bleomycin-induced lung injury. | |||
T19125 | 3-Phenylbutyric acid | Others , Endogenous Metabolite | |
3-Phenylbutyric acid undergoes metabolism through initial oxidation processes involving both its benzene ring and side chain. It serves as an effective agent for the isolation of Rhodococcus rhodochrous PB1 from compost ... | |||
T6000 | Delta-Tocopherol | D-DELTA-TOCOPHEROL | Endogenous Metabolite |
Delta-Tocopherol is an isomer of Vitamin E,has antioxidant activity,and might be useful as effective ingredients in whitening cosmetics with lower skin toxicity. | |||
T3251 | Stachydrine Hydrochloride | NF-κB | |
Stachydrine Hydrochloride is an effective component that mainly extracted from the leaf of Leonurussibiricus. | |||
T20326 | 1,2-Dimethoxybenzene | Veratrole,AI302281,AI3 02281,AI3-02281 | Others |
1,2-Dimethoxybenzene (Veratrole), a natural product secreted by Silene latifolia, is an effective pollinator attractant for the nocturnal moth Hadena bicruris. | |||
T5888 | 5-Methoxysalicylic acid | 5-MeOSA | Others |
5-Methoxysalicylic acid (5-MeOSA), a natural product, serves as an effective matrix for oligonucleotide analysis in MALDI MS when used alongside spermine. | |||
TN2232 | Soyasaponin Ab | NOS , NF-κB , COX | |
Soyasaponin Ab may represent a viable candidate for effective vaccine adjuvant, TLR4 receptor dependent pathway may be involved in immune stimulatory effects of soyasaponin Ab. | |||
T0268 | Lobeline hydrochloride | α-Lobeline hydrochloride,L-Lobeline hydrochloride | AChR |
Lobeline hydrochloride (α-Lobeline hydrochloride) is a nicotinic receptor agonist, acting as an effective antagonist at both α4β2 and α3β2 neuronal nicotinic receptor subtypes. | |||
T5037 | Midecamycin | Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,Platenomycin B1,Espinomycin A | Antibacterial , Antibiotic |
Midecamycin (Medecamycin A1), an acetoxy-substituted macrolide antibiotic, has effective on gram-positive and gram-negative bacteria acts by inhibiting bacterial protein synthesis. | |||
T16685 | Purpurogallin | Xanthine Oxidase | |
Purpurogallin is a naturally phenol extracted from the plants of Quercus spp. It has effective xanthine oxidase inhibitory activity (IC50: 0.2 µM). Purpurogallin also has antioxidant and anti-inflammatory effects. | |||
TQ0215 | Salinomycin sodium salt | Sodium salinomycin,Salinomycin sodium | Apoptosis , Wnt/beta-catenin , Antibacterial , Antibiotic , Autophagy |
T3924 | Astragaloside II | Astrasieversianin VIII | TGF-beta/Smad |
Astragaloside II (Astrasieversianin VIII) is an effective MDR reversal agent and may be a potential adjunctive agent for hepatic cancer chemotherapy. Astragaloside II also induces osteogenic activities, differentiation, ... | |||
T0122 | Bergenin | Cuscutin,Bengenin | Apoptosis , IL Receptor , Virus Protease , TNF , NF-κB , Antibacterial , NOD , Autophagy , Antifungal |
Bergenin (Bengenin) is a polyphenol, which is an effective antinarcotic agent with antioxidant action. | |||
T1400 | Demeclocycline hydrochloride | Declomycin,Clortetrin,Detravis,Demeclocycline HCl | ribosome , Antibacterial , Antibiotic |
Demeclocycline hydrochloride (Declomycin) is a TETRACYCLINE analog having a 7-chloro and a 6-methyl. Because it is excreted more slowly than TETRACYCLINE, it maintains effective blood levels for longer periods of time. | |||
T9605 | Sangivamycin | BA-90912,NSC 65346 | Nucleoside Antimetabolite/Analog , PKC |
Sangivamycin (NSC-65346) is an effective inhibitor of protein kinase C (PKC, Ki = 10 μM). Sangivamycin exhibits antiproliferative activity against a variety of human cancers. | |||
T6S0234 | Toosendanin | Others | |
1. Toosendanin possesses hepatotoxicity. 2. Toosendanin has effects on the growth, cell cycle arrest, induction of apoptosis and the involved signaling pathway in human promyelocytic leukemia HL-6 cells. 3. Toosendanin i... | |||
TN2211 | Silybin B | Silibinin B | Apoptosis , Beta Amyloid , Bcr-Abl |
Silybin B (Silibinin B) is an effective inhibitor of raloxifene 4 '- and 6-glucosalylation, an effective anti-fibrinogenic and anti-oligomeric component of Silymarin, with free radical scavenging activity of 1, 1-dipheny... | |||
T6S1684 | 8-Gingerol | Antioxidant , Antibacterial , TRP/TRPV Channel | |
1. 8-Gingerol has antioxidant activity. 2. 8-Gingerol has antimycobacterial activity. 3. 8-Gingerol could be used as an effective skin-whitening agent. 4. 8-Gingerol shows antipyretic and anti-inflammation characteristic... | |||
T21552 | 5-deoxy Thymidine | 5'-Deoxythymidine,Thymidine, 5'-deoxy-1-[(2R,4S,5R)-4-hydroxy-5-methyloxolan-2-yl]-5-methylpyrimidine-2,4-dione | Others |
5-deoxy Thymidine (5'-Deoxythymidine) is a thymidine form which 5' position replaced with hydrogen.5'-deoxy Thymidine was effective against the activity of Bacillus subtilis and Staphylococcus aureus. | |||
TN2230 | Soyasaponin Ba | Others | |
Soyasaponin Ba may represent viable candidates for effective vaccine adjuvants due to their higher and lower or non-haemolytic effects.Soyasaponins Ab and Bb prevent scopolamine-induced memory impairment in mice without ... | |||
TQ0209 | Ailanthone | Δ13-Dehydrochaparrinone | Androgen Receptor |
Ailanthone (Δ13-Dehydrochaparrinone) is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) and constitutively active truncated AR splice variants (IC50: 309 nM). | |||
T6654 | Saponins | Sapogenins Glycosides,Saponin | Others |
Saponins (Sapogenins Glycosides) are a mixture of triterpene and steroid saponins isolated from medicinal plants such as Aesculus hippocastanum L., Hedera helix L. and Ruscus aculeatus L., which are claimed to be effecti... | |||
T60237 | L-Cysteine S-sulfate | S-Sulfo-L-cysteine | NMDAR |
L-Cysteine S-sulfate (S-Sulfo-L-cysteine) is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist. L-Cysteine S-sulfate is the substrate for cystine lyase [1]. | |||
T8255 | (±)-Catechin | (±)-Catechin hydrate | ROS , COX |
(±)-Catechin ((±)-Catechin hydrate) hydrate is a natural product,has antioxidant activity and is effective in reducing oxidative stress. | |||
T5003 | Rifamycin sodium | Rifamycin sodium salt | Antibacterial , Antibiotic |
Rifamycin sodium (Rifamycin sodium salt) salt is an antibiotic that inhibits bacterial DNA-dependent RNA polymerase. It is effective against Gram-positive bacteria. | |||
T4S0094 | Hydroxygenkwanin | Luteolin 7-methylether,7-O-Methylluteolin | Antioxidant |
1. Hydroxygenkwanin (Luteolin 7-methylether) possesses significant the antioxidative activity . 2. Hydroxygenkwanin has cytotoxicity, may be an effective natural product to treat glioma, and the combination of Apigenin a... | |||
T1003 | Tylosin | Fradizine,Tylosin A,Tylosine,Tylocine | Antibacterial , Antibiotic |
Tylosin (Tylosine) is a macrolide antibiotic obtained from cultures of Streptomyces fradiae. The drug is effective against many microorganisms in animals but not in humans. | |||
T21855 | AMI-193 | Espiramida,Spiramide | Dopamine Receptor , 5-HT Receptor |
AMI-193 (Spiramide) is an effective and selective antagonist of 5-HT2 and D2 receptor with Kis of 2, 3, 50, 2530, and 4300 nM for 5-HT2, D2 Receptor, 5-HT1A, D1 Receptor, and 5-HT1C Receptor. AMI-193 shows antipsychotic ... | |||
T19384 | Isovalerylcarnitine | Apoptosis , Cysteine Protease | |
Isovalerylcarnitine (3-methylbutyrylcarnitine) is a small molecule compound produced by the catabolism of L-leucine and the accumulation of isovaleric acid. Isovalerylcarnitine is also a selective and effective calpain a... | |||
T7056 | Dronedarone | SR 33589 | P450 , Potassium Channel , Calcium Channel , Sodium Channel , Adrenergic Receptor , AChR , Autophagy |
Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation. | |||
T2S1200 | Sinapine | Antioxidant , P-gp , AChE | |
1. Sinapine, an alkaloid from seeds of the cruciferous species, can be used as an effective natural compound for chemo-resistance. 2. Sinapine has antioxidant and radio-protective activities. | |||
T14853 | Cabergoline | FCE-21336 | Dopamine Receptor , 5-HT Receptor , Autophagy |
Cabergoline (FCE-21336) is an ergot derived-dopamine D2-like receptor agonist. It has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respectively).Cabergoline permits rapid and effective hormonal a... | |||
TN2256 | Taccalonolide B | Microtubule Associated | |
Taccalonolide B is effective in vitro against cell lines that overexpress P-glycoprotein (Pgp) and multidrug-resistance protein (MRP7). Taccalonolide B inhibits growth of SK-OV-3 cells with an IC50 of 208 nM. | |||
T5055 | For-Met-OH | fMet,N-Formyl-L-methionine | Others , Endogenous Metabolite |
For-Met-OH (N-Formyl-L-methionine) is effective in the initiation of protein synthesis. The initiating methionine residue enters the ribosome as N-formyl methionyl tRNA. This process occurs in Escherichia coli and other ... | |||
T1261 | Medroxyprogesterone Acetate | Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,Farlutin,Medroxyprogesterone (acetate) | Glucocorticoid Receptor , Estrogen/progestogen Receptor , Progesterone Receptor , Androgen Receptor , Endogenous Metabolite |
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective both orally or by intramuscular injection and has also been... | |||
T8678 | Naphthazarin | 5,8-Dihydroxy-1,4-naphthoquinone,DHNQ | Apoptosis |
Naphthazarin (5,8-Dihydroxy-1,4-naphthoquinone) is effective by various cellular mechanisms including oxidative stress, activation of mitochondrial apoptosis-inducing factor (AIF), depolymerization of microtubules, inter... | |||
T3404 | Cucurbitacin B | Cuc B,DATISCACIN,Amarine | Apoptosis , PTEN , Integrin , Endogenous Metabolite , HIF , STAT , Autophagy |
Cucurbitacin B (Cuc B) has profound in vitro and in vivo antiproliferative effects against human pancreatic Y cells. It inhibited AKT signaling activation through up-regulation of PTEN. Cucurbitacin B is an effective inh... | |||
TN1658 | Ganoderenic acid D | Apoptosis , Others | |
Ganoderenic acid D is a natural product isolated from the effective compounds of Ganoderma lucidum extract (GLE). Ganoderenic acid D induces cell cycle arrest and apoptosis and inhibits the proliferation of cancer cells. | |||
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カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPY-02904 | TLR4 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
TLR4, also known as TLR-4, is a member of the Toll-like receptor (TLR) family, which plays a fundamental role in pathogen recognition and activation of innate immunity. TLRs are highly conserved from Drosophila to humans... | |||
TMPY-02481 | ACOX1 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
Peroxisomal acyl-coenzyme A oxidase 1(ACOX1 or AOX) is the first enzyme of the fatty acid beta-oxidation pathway and belongs to the Acyl-CoA oxidase family. Human liver peroxisomes contain two acyl-CoA oxidases, namely, ... | |||
TMPH-00603 | Cytidylate kinase Protein, E. coli, Recombinant (His & SUMO) | E. coli | E. coli |
ATP, dATP, and GTP are equally effective as phosphate donors. CMP and dCMP are the best phosphate acceptors. | |||
TMPH-02773 | Lysozyme C-2 Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
Lysozymes have primarily a bacteriolytic function; those in tissues and body fluids are associated with the monocyte-macrophage system and enhance the activity of immunoagents. Lyz2 is active against a range of Gram-posi... | |||
TMPK-01028 | BSPII Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Osteopontin (OPN), bone sialoprotein (BSPII), and osteonectin (ON) belong to a family of glycoproteins, which have been linked to cancer metastasis and progression. Here, we report on the selection of antisense oligonucl... | |||
TMPH-01703 | CDC25C Protein, Human, Recombinant (His) | Human | E. coli |
Functions as a dosage-dependent inducer in mitotic control. Tyrosine protein phosphatase required for progression of the cell cycle. When phosphorylated, highly effective in activating G2 cells into prophase. Directly de... | |||
TMPK-00127 | CLEC4A Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
Clec4a has been reported to be an immune suppressor of dendritic cells (DCs), but its potential role in cancer therapy remains to be elucidated. silencing of Clec4a2 expression via skin delivery of shRNA produces an effe... | |||
TMPK-00483 | PCSK9 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
Proprotein convertase subtilisin/kexin type 9 (PCSK9) is an enzyme encoded by the PCSK9 gene in humans on chromosome 1.The first two PCSK9 inhibitors, alirocumab and evolocumab, were approved as once every two week injec... | |||
TMPK-01049 | CLEC7A Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
Dendritic cell-associated C-type lectin-1 (Dectin-1), also known as β-glucan receptor is an emerging pattern recognition receptor (PRR) which belongs to the family of C-type lectin receptor (CLR). Dectin-1 signaling axis... | |||
TMPK-00126 | CLEC4A Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Clec4a has been reported to be an immune suppressor of dendritic cells (DCs), but its potential role in cancer therapy remains to be elucidated. silencing of Clec4a2 expression via skin delivery of shRNA produces an effe... | |||
TMPK-01222 | APLN Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
Macrophages play key roles during cardiovascular diseases (CVD) and their related complications.Apelin (APLN) is a key molecule, whose roles during CVD have been documented previously. Therefore, it has been hypothesized... | |||
TMPK-01236 | APLN Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Macrophages play key roles during cardiovascular diseases (CVD) and their related complications.Apelin (APLN) is a key molecule, whose roles during CVD have been documented previously. Therefore, it has been hypothesized... | |||
TMPJ-00787 | GUSB Protein, E. coli, Recombinant (His) | E. coli | E. coli |
Beta-D-glucuronidase from E.coli is a highly specific enzyme in hydrolyzing glucuronides. Beta-D-glucuronidase (GLUase) activity can be measured as the rate of production of fluorescent methylumbelliferone (MU), resulti... | |||
TMPK-00931 | CD164 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
CD164 was found to play a role in many malignant diseases. CD164 was associated with clinical and pathological features of patients. High level of CD164 was related to the distant metastasis and vascular invasion of blad... | |||
TMPK-01220 | CD164 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
CD164 was found to play a role in many malignant diseases. CD164 was associated with clinical and pathological features of patients. High level of CD164 was related to the distant metastasis and vascular invasion of blad... | |||
TMPH-00430 | VxXIIC Protein, Conus vexillum, Recombinant (His & Myc & SUMO) | Conus vexillum | E. coli |
Alpha-conotoxins act on postsynaptic membranes, they bind to the nicotinic acetylcholine receptors (nAChR) and thus inhibit them. This toxin specifically blocks mammalian neuronal nAChR of the alpha-7/CHRNA7, alpha-3-bet... | |||
TMPJ-00710 | ALDH1A2 Protein, Human, Recombinant (His) | Human | E. coli |
Aldehyde dehydrogenase 1 family member A2 (ALDH1A2), also known as retinaldehyde dehydrogenase 2 (RALDH2), belongs to the aldehyde dehydrogenase family which contains two members, the ALDH1 s (ALDH1A1, ALDH1A2 and ALDH1A... | |||
TMPH-01624 | GBA Protein, Human, Recombinant | Human | E. coli |
Glucosylceramidase that catalyzes, within the lysosomal compartment, the hydrolysis of glucosylceramide/GlcCer into free ceramide and glucose. Thereby, plays a central role in the degradation of complex lipids and the tu... | |||
TMPJ-00130 | SLAMF2 Protein, Human, Recombinant (hFc & His) | Human | HEK293 Cells |
CD48 antigen, also known as B-lymphocyte activation marker BLAST-1, BCM1 surface antigen, Leukocyte antigen MEM-102, TCT.1, CD48, BCM1,and BLAST1, CD48 contains one Ig-like C2-type domain and one Ig-like V-type domain, b... | |||
TMPH-01623 | GBA Protein, Human, Recombinant (His & Myc & SUMO) | Human | E. coli |
Glucosylceramidase that catalyzes, within the lysosomal compartment, the hydrolysis of glucosylceramide/GlcCer into free ceramide and glucose. Thereby, plays a central role in the degradation of complex lipids and the tu... | |||
TMPH-01517 | FCGRT Protein, Human, Recombinant (GST) | Human | E. coli |
Cell surface receptor that transfers passive humoral immunity from the mother to the newborn. Binds to the Fc region of monomeric immunoglobulin gamma and mediates its selective uptake from milk. IgG in the milk is bound... | |||
TMPH-01516 | FCGRT Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Cell surface receptor that transfers passive humoral immunity from the mother to the newborn. Binds to the Fc region of monomeric immunoglobulin gamma and mediates its selective uptake from milk. IgG in the milk is bound... | |||
TMPJ-00789 | Flagellin Protein, Salmonella Typhimurium, Recombinant | Salmonella typhimurium | E. coli |
Flagellin is the major structural protein monomer of bacterial flagella. Flagellin through binding to its receptor and activation of antigen presenting cells stimulates the innate and adaptive immune responses. Flagellin... | |||
TMPY-02387 | NF-kB p65 Protein, Human, Recombinant (aa 1-306, GST) | Human | E. coli |
RELA (v-rel reticuloendotheliosis viral oncogene homolog A), also known as Nuclear factor NF-kappa-B p65 subunit, or Transcription factor p65, is a transcription factor expressed in growth plate chondrocytes where it fac... | |||
TMPY-00975 | FSTL3 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Follistatin-like 3 (FLRG/Fstl3) is a secreted glycoprotein of the follistatin-module-protein family. It may have a role in leukemogenesis. FLRG/Fstl3 is a recently described member of the FST family having an overall str... | |||
TMPY-04394 | Glucokinase Protein, Human, Recombinant | Human | E. coli |
Glucokinase belongs to the bacterial glucokinase family. Hexokinases phosphorylate glucose to produce glucose-6-phosphate, the first step in most glucose metabolism pathways. Alternative splicing of this gene results in ... |
カタログ番号 | 製品名 | ||
---|---|---|---|
L4520 | Anti-Bacterial Compound Library | 904 compounds | |
A unique collection of 904 antibacterial bioactive compounds, a powerful tool for antibacterial drug development; | |||
L3900 | DNA Damage & Repair Compound Library | 910 compounds | |
A unique collection of 910 DNA Damage & Repair related compounds for high throughput screening (HTS) and high content screening (HCS); | |||
L2700 | Adrenergic Receptor-Targeted Compound Library | 193 compounds | |
A unique collection of 193 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification; | |||
L3980 | DNA Damage and Repair Compound Library Plus | 667 compounds | |
Well-chosen 667 compounds with unique structures targeting DNA damage & repair; | |||
L7100 | Anti-Obesity Compound Library | 2247 compounds | |
A unique collection of 2247 anti-obesity compounds for high throughput and high content screening; | |||
L4200 | FDA-Approved Drug Library | 1729 compounds | |
A unique collection of 1729 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS); | |||
L4500 | Anti-Fungal Compound Library | 252 compounds | |
A unique collection of 252 antifungal compounds effective for drug repurposing screening, combination screening and biological investigation. | |||
L1900 | Anti-Diabetic Compound Library | 683 compounds | |
A unique collection of 683 diabetes related compounds; | |||
L9500 | Target-Focused Phenotypic Screening Library | 1796 compounds | |
A unique collection of 1796 annotated bioactive compounds with clear targets, suitable for phenotypic screening; | |||
L3400 | Clinical Compound Library | 3404 compounds | |
A unique collection of 3404 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS); | |||
L6100 | Polyphenolic Natural Product Library | 635 compounds | |
A unique collection of 635 natural polyphenolic compounds for high throughput screening (HTS) and high content screening (HCS); | |||
L6810 | Traditional Chinese Medicine Monomer Library | 2755 compounds | |
A unique collection of 2755 compounds (TCM monomers) sourcing from traditional Chinese Medicines, is a powerful tool for drug discovery and research in mechanism; | |||
L5800 | Drug Metabolite/Impurity Library | 197 compounds | |
A unique collection of 197 drug isomers/metabolites for high throughput screening (HTS) and high content screening (HCS); | |||
L2000 | Inhibitor Library | 8328 compounds | |
A unique collection of 8328 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs; | |||
L4700 | Immunology/Inflammation Compound Library | 4720 compounds | |
A unique collection of 4720 anti-inflammation compounds effective for high throughput screening and high content screening. | |||
L9200 | Drug Repurposing Compound Library | 4630 compounds | |
A unique collection of 4630 approved and clinical drugs for high throughput screening (HTS) and high content screening (HCS); | |||
L2192 | Anti-Pancreatic Cancer Compound Library | 2238 compounds | |
A unique collection of 2238 pancreatic cancer related compounds can be used in HTS and HCS; | |||
L6150 | Covalent Natural Product Library | 583 compounds | |
Detialed biological information and pharmacological information of the products, providing theoretical direction and research basis for screening. | |||
L6600 | Anti-Gastroenteritis Natural Product Library | 219 compounds | |
A unique collection of 219 natural products related to gastroenteritis for high throughput screening (HTS) and high content screening (HCS); | |||
L8200 | Anti-Aging Compound Library | 3279 compounds | |
A unique collection of 3279 anti-aging compounds for high throughput screening (HTS) and high content screening (HCS); | |||
L6230 | Miao medicine Compound Library | 534 compounds | |
A unique collection of 534 compounds featuring natural product molecules derived from Miao medicine that can be used for high-throughput and high-content screening. | |||
L8110 | Reprogramming Compound Library | 1813 compounds | |
A unique collection of 1813 reprogramming signaling pathway-related bioactive small molecule compounds for high-throughput, high-content screening. | |||
L8400 | Hematonosis Compound Library | 514 compounds | |
A unique collection of 514 compounds related to hematologic diseases for high throughput screening (HTS) and high content screening (HCS); | |||
L7400 | Sodium Channel Blocker Library | 118 compounds | |
A unique collection of 118 sodium channel blockers and agonists for high throughput and high content screening; | |||
L2140 | Cancer Cell Differentiation Compound Library | 406 compounds | |
A unique collection of 406 cancer cell differentiation inducing compounds for high throughput and high content screening; | |||
L2500 | Human Endogenous Metabolite Library | 499 compounds | |
A collection of 499 selected human endogenous metabolites for high throughput and high content screening. | |||
L6700 | Anti-Tumor Natural Product Library | 1772 compounds | |
A unique collection of 1772 natural products with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS); | |||
L1110 | Microtubule-Targeted Compound Library | 142 compounds | |
A unique collection of 142 microtubule-targeted compounds can be used in HTS and HCS; | |||
L1000 | Approved Drug Library | 2808 compounds | |
A unique collection of 2808 approved drugs for high throughput screening (HTS) and high content screening (HCS); | |||
L2540 | Gut Microbial Metabolite Library | 614 compounds | |
A unique collection of 614 gut microbial metabolites which can be used for HTS and HCS; | |||
L1010 | FDA-Approved & Pharmacopeia Drug Library | 3158 compounds | |
3158 compounds from marketed drugs for high throughput screening (HTS) and high content screening (HCS); | |||
L6730 | Anti-virus Traditional Chinese Medicine Monomer Library | 268 compounds | |
A collection of 268 TCM monomers with anti-virus activity. An effective tool for drug development and pharmacological studies. | |||
L9700 | Endoplasmic Reticulum Stress Compound Library | 193 compounds | |
A unique collection of 193 endoplasmic reticulum stress (ER stress) related compounds used for high throughput screening (HTS) and high content screening (HCS); | |||
L5100 | Fluorochemical Library | 574 compounds | |
A unique collection of 574 fluorochemicals that can be used for high through-put screening (HTS) and high content screening (HCS); | |||
L6740 | Anti-Colorectal Cancer Traditional Chinese Medicine Compound Library | 382 compounds | |
A collection of 382 TCM monomers with anti-colorectal activity. An effective tool for drug development and pharmacological studies. | |||
L6010 | Natural Product Library | 3840 compounds | |
A unique collection of 3840 natural products for high throughput screening (HTS) and high content screening (HCS); | |||
L5700 | Featured Fragment Library | 246 compounds | |
A unique collection of 246 fragment-like small molecules for FBDD; | |||
L6000 | Natural Product Library for HTS | 4533 compounds | |
A unique collection of 4533 pure natural products and their derivatives with known biological activity for drug discovery, pharmacological study, stem cell differentiation, fingerprint study and quality research, and can... | |||
L1700 | Anti-Viral Compound Library | 1040 compounds | |
A unique collection of 1040 anti-virus compounds effective for new anti-virus drugs high throughput screening and high content screening; | |||
L2010 | Highly Selective Inhibitor Library | 575 compounds | |
L6610 | Anti-infective Natural Product Library | 1060 compounds | |
A unique collection of 1060 species of natural products with anti-infective activity for high throughput screening (HTS) and high content screening (HCS); | |||
L2190 | Anti-Lung Cancer Compound Library | 1702 compounds | |
A unique collection of 1702 compounds with anti-lung cancer therapeutic activity or targeting lung cancer’s major signaling pathways, can be used for anti-lung cancer drug discovery and mechanism study; | |||
L6800 | Chinese Pharmacopoeia Natural Product Library | 2051 compounds | |
A unique collection of 2051 natural products included in Chinese Pharmacopoeia (CP), a powerful tool for drug development and pharmacological study; | |||
DO2200 | Covalent inhibitors Library | 12000 compounds | |
L6200 | The Yao nationality medicine Library | 221 compounds | |
A collection of 221 natural product molecules originated from Yao medicine, which can be used for high-throughput and high-content screening. | |||
L2196 | Anti-Ovarian Cancer Compound Library | 1867 compounds | |
L6820 | Tobacco Monomer Library | 747 compounds | |
L2550 | Glutamine Metabolism Compound Library | 565 compounds | |
A unique collection of 565 glutamine metabolism related compounds can be used for high throughput screening (HTS) and high content screening (HCS), and also is an effective tool for research in glutamine metabolism and ... |